General Information of Drug (ID: DM0LPI9)

Drug Name
Netarsudil Drug Info
Synonyms
UNII-W6I5QDT7QI; W6I5QDT7QI; Netarsudil mesylate; Netarsudil [USAN]; AR-11324 free base; Netarsudil [USAN:INN]; Netarsudil (USAN/INN); GTPL9322; SCHEMBL16036278; ZINC113149554; AR11324; AR-11324; ester 60; 1628418-15-4
Indication
Disease Entry ICD 11 Status REF
Open-angle glaucoma 9C61 Approved [1]
Glaucoma/ocular hypertension 9C61 Phase 2 [2]
Cross-matching ID
PubChem CID
66599893
CAS Number
1254032-66-0
TTD ID
D04WYX
ACDINA ID
D01281

Full List of Drug Formulations Containing This Drug

Netarsudil 0.2mg/ml solution
Company Formulation ID FDA Description
Aerie Pharmaceuticals F23239 Boric Acid; Mannitol; Sodium Hydroxide; Water For Injection
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References

1 2017 FDA drug approvals.Nat Rev Drug Discov. 2018 Feb;17(2):81-85.
2 Effect of 0.04% AR-13324, a ROCK, and norepinephrine transporter inhibitor, on aqueous humor dynamics in normotensive monkey eyes. J Glaucoma. 2015 Jan;24(1):51-4.