Details of the Drug-Related molecule(s) Activity Atlas

General Information of Drug (ID: DMB920Z)

• Drug Name: Ceritinib Drug Info
• Synonyms: ceritinib; LDK378; 1032900-25-6; ZYKADIA; NVP-LDK378-NX; LDK-378; UNII-K418KG2GET; LDK378(Ceritinib); LDK 378; Eritinib (LDK378); 5-chloro-N2-(2-isopropoxy-5-methyl-4-(piperidin-4-yl)phenyl)-N4-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine; K418KG2GET; CHEMBL2403108; CHEBI:78432; AK174337; ceritinib; C28H36ClN5O3S; 5-Chloro-N2-[2-isopropoxy-5-Methyl-4-(4-piperidyl)phenyl]-N4-(2-isopropylsulfonylphenyl)pyriMidine-2,4-diaMine; 5-Chloro-N2-(5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl)-N4-(2-(propane-2-sulfonyl)phenyl)pyrim
• Cross-matching ID:
  PubChem CID: 57379345
  ChEBI ID: CHEMBL78432
  CAS Number: CAS 1032900-25-6
  TTD ID: D04LVK
  VARIDT Drug ID: DR00228
  ACDINA Drug ID: D00115

Molecule-level Activity Landscape of This Drug

IC50 (70) EC50 (3) Kd (25) Ki (2) Download

Molecule Name	Gene Name	UniProt ID	Type	IC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	EC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Kd (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Ki (nM)	Details
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Cytotoxic Activity Landscape of This Drug

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Cell Line	Disease	Value (nM)	ChEMBL Assay ID	Details
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