Details of the Drug-Related molecule(s) Activity Atlas

General Information of Drug (ID: DMMPTLH)

• Drug Name: Entrectinib Drug Info
• Synonyms: 1108743-60-7; RXDX-101; UNII-L5ORF0AN1I; Entrectinib (RXDX-101); L5ORF0AN1I; Benzamide, N-[5-[(3,5-difluorophenyl)methyl]-1H-indazol-3-yl]-4-(4-methyl-1-piperazinyl)-2-[(tetrahydro-2H-pyran-4-yl)amino]-; Benzamide, N-(5-((3,5-difluorophenyl)methyl)-1H-indazol-3-yl)-4-(4-methyl-1-piperazinyl)-2-((tetrahydro-2H-pyran-4-yl)amino)-; Entrectinib [USAN:INN]; YMX; Kinome_2659; Entrectinib(rxdx-101); Entrectinib (USAN/INN); SCHEMBL3512601; GTPL8290; CHEMBL1983268; KS-00000TSK
• Cross-matching ID:
  PubChem CID: 25141092
  ChEBI ID: CHEMBL1983268
  CAS Number: CAS 1108743-60-7
  TTD ID: D0O0LS
  INTEDE Drug ID: DR0582
  ACDINA Drug ID: D01050

Molecule-level Activity Landscape of This Drug

IC50 (36) Kd (6) Ki (103) Download

Molecule Name	Gene Name	UniProt ID	Type	IC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Kd (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Ki (nM)	Details
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Cytotoxic Activity Landscape of This Drug

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Cell Line	Disease	Value (nM)	ChEMBL Assay ID	Details
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