General Information of Drug (ID: DM3RUT8)

Drug Name
MG-101 Drug Info
Synonyms 110044-82-1
Cross-matching ID
PubChem CID
443118
ChEBI ID
CHEMBL304784
CAS Number
CAS 110044-82-1
TTD Drug ID
D06FFP

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Proteasome 2.39 0.00e+0 44/46 (95.65%) PSMD2;PSMC2;PSMC1;...
Protein processing in endoplasmic reticulum 2.32 0.00e+0 127/171 (74.27%) HSPA6;HSPH1;HSPA8;...
Epithelial cell signaling in Helicobacter pylori infect... 2.14 0.00e+0 62/70 (88.57%) CXCL8;ATP6V0E1;RELA;...
Parkinson disease 2.13 0.00e+0 176/249 (70.68%) UCHL1;DDIT3;PSMD2;...
Phagosome 2.06 2.29e-3 118/152 (77.63%) TUBB2A;TAP1;HLA-DQA1;...
Epstein-Barr virus infection 2.06 1.91e-3 189/202 (93.56%) CDKN1A;PSMD2;PSMC2;...
Collecting duct acid secretion 2.06 1.64e-3 22/27 (81.48%) ATP6V0E1;SLC12A7;TCIRG1;...
Herpes simplex virus 1 infection 2.05 1.43e-3 165/498 (33.13%) TAP1;HLA-DQA1;RELA;...
IL-17 signaling pathway 2.04 1.27e-3 84/94 (89.36%) CXCL8;CEBPB;HSP90AA1;...
Antigen processing and presentation 2.00 1.15e-3 60/78 (76.92%) HSPA6;HSPA8;HSPA1A;...
Prion disease 1.99 1.04e-3 209/273 (76.56%) HSPA6;HSPA8;HSPA1A;...
Legionellosis 1.98 1.91e-3 51/57 (89.47%) HSPD1;HSPA6;HSPA8;...
Ferroptosis 1.94 4.41e-3 36/41 (87.8%) HMOX1;SLC7A11;GCLM;...
Amyotrophic lateral sclerosis 1.92 4.09e-3 267/364 (73.35%) SQSTM1;DDIT3;PSMD2;...
Measles 1.92 3.82e-3 133/139 (95.68%) HSPA6;HSPA8;HSPA1A;...
Alzheimer disease 1.90 3.58e-3 279/369 (75.61%) DDIT3;PSMD2;DKK1;...
Apoptosis 1.90 3.37e-3 126/168 (75%) DDIT3;CTSK;RELA;...
Autophagy 1.90 3.18e-3 113/169 (66.86%) SQSTM1;DDIT4;GABARAPL1;...
Hepatitis C 1.90 3.02e-3 139/157 (88.54%) CDKN1A;RELA;CXCL10;...
Toll-like receptor signaling pathway 1.86 3.44e-3 94/104 (90.38%) CXCL8;SPP1;CTSK;...
Pathways of neurodegeneration 1.86 3.28e-3 354/475 (74.53%) UCHL1;SQSTM1;DDIT3;...
Lipid and atherosclerosis 1.86 3.13e-3 190/215 (88.37%) HSPD1;HSPA6;HSPA8;...
TNF signaling pathway 1.82 4.98e-3 103/112 (91.96%) CEBPB;RELA;DNM1L;...
Human papillomavirus infection 1.81 4.78e-3 284/331 (85.8%) SPP1;CDKN1A;GNAS;...
Mitophagy 1.79 5.96e-3 56/68 (82.35%) SQSTM1;RELA;GABARAPL1;...
Spinocerebellar ataxia 1.79 5.73e-3 128/143 (89.51%) PSMD2;PSMC2;PSMC1;...
Salmonella infection 1.77 6.37e-3 198/249 (79.52%) CXCL8;HSP90AA1;HSP90AB1;...
Staphylococcus aureus infection 1.76 6.96e-3 72/95 (75.79%) KRT14;KRT17;KRT13;...
Estrogen signaling pathway 1.74 7.51e-3 119/137 (86.86%) HSPA6;HSPA8;KRT14;...
Inflammatory bowel disease 1.73 9.55e-3 58/65 (89.23%) HLA-DQA1;RELA;STAT4;...
Valine, leucine and isoleucine degradation -1.66 4.93e-2 42/48 (87.5%) ACADSB;OXCT1;HMGCL;...
Mismatch repair -1.68 4.66e-2 22/23 (95.65%) POLD4;RFC3;SSBP1;...
Morphine addiction -1.69 4.43e-2 80/91 (87.91%) GNB1;PDE4D;GABRD;...
Dilated cardiomyopathy -1.70 4.25e-2 86/96 (89.58%) MYL2;ITGA2;IGF1;...
Fat digestion and absorption -1.73 2.93e-2 35/43 (81.4%) MTTP;APOA4;PLPP3;...
Synthesis and degradation of ketone bodies -1.73 3.35e-2 9/10 (90%) OXCT1;BDH2;HMGCL;...
Drug metabolism -1.73 3.91e-2 78/151 (51.66%) ADH1B;TK2;ADH6;...
Fanconi anemia pathway -1.79 2.61e-2 36/54 (66.67%) TELO2;RAD51C;BRCA1;...
Sulfur metabolism -1.82 2.82e-2 9/10 (90%) TST;PAPSS2;MPST;...
Purine metabolism -1.82 3.48e-2 102/129 (79.07%) ENPP4;GART;NT5C2;...
Butanoate metabolism -1.86 3.04e-2 23/28 (82.14%) OXCT1;L2HGDH;BDH2;...
DNA replication -2.28 0.00e+0 34/36 (94.44%) RFC5;MCM6;MCM3;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Fibroblast
Nasopharyngeal carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
FIBRNPC CVCL_UK07 Homo sapiens 10uM 6H, 24H