General Information of Drug (ID: DMDJW5K)

Drug Name
Ajmaline Drug Info
Synonyms (17R,21
Cross-matching ID
PubChem CID
6100671
CAS Number
CAS 4360-12-7
TTD Drug ID
D02GUG
VARIDT Drug ID
DR01161
INTEDE Drug ID
DR0054

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Oxidative phosphorylation -1.62 4.85e-2 93/133 (69.92%) ATP6V1E1;NDUFB1;ATP5PB;...
Chemokine signaling pathway -1.66 3.77e-2 163/192 (84.9%) BRAF;PIK3CB;CCL8;...
Nicotinate and nicotinamide metabolism -1.69 3.21e-2 25/35 (71.43%) AOX1;NADK;QPRT;...
Epithelial cell signaling in Helicobacter pylori infect... -1.72 2.40e-2 62/70 (88.57%) ATP6V0B;CCL5;CXCR2;...
Pertussis -1.88 3.02e-3 64/76 (84.21%) CASP1;IL1A;GNAI1;...
TNF signaling pathway -1.92 8.38e-4 103/112 (91.96%) BAG4;VEGFD;MAP3K7;...
Malaria -1.95 0.00e+0 44/50 (88%) GYPC;TGFB3;CSF3;...
Rheumatoid arthritis -2.02 0.00e+0 78/93 (83.87%) ATP6V1D;IL15;TGFB3;...
IL-17 signaling pathway -2.10 0.00e+0 84/94 (89.36%) CHUK;TBK1;DEFB4A;...
NF-kappa B signaling pathway -2.11 0.00e+0 90/104 (86.54%) CXCL12;NFKBIA;GADD45A;...
Cytokine-cytokine receptor interaction -2.14 0.00e+0 246/295 (83.39%) IL15;IL16;CCL8;...
Legionellosis -2.18 0.00e+0 51/57 (89.47%) CASP1;NFKBIA;RAB1B;...
Complement and coagulation cascades -2.22 0.00e+0 76/85 (89.41%) MASP2;F2;C8B;...
Viral protein interaction with cytokine and cytokine re... -2.54 0.00e+0 84/100 (84%) IL18RAP;IL24;IL6ST;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Bone
Osteosarcoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
U-2 OS CVCL_0042 Homo sapiens 10uM 6H