General Information of Drug (ID: DME9T0A)

Drug Name
RGFP966 Drug Info
Synonyms RGFP-966
Cross-matching ID
PubChem CID
56650312
ChEBI ID
CHEMBL131163
TTD Drug ID
D00HXX

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
ECM-receptor interaction 2.18 0.00e+0 80/88 (90.91%) COL1A1;COL6A3;FN1;...
Staphylococcus aureus infection 2.10 0.00e+0 72/95 (75.79%) FGG;ITGAM;HLA-DQB1;...
Malaria 2.03 0.00e+0 44/50 (88%) IL1B;CCL2;TLR4;...
Amoebiasis 1.92 0.00e+0 99/102 (97.06%) IL1B;COL1A1;CTSG;...
Focal adhesion 1.92 0.00e+0 180/201 (89.55%) PDGFA;IGF1R;FLNB;...
Pertussis 1.92 1.86e-3 64/76 (84.21%) IL1B;CALML3;IL1A;...
Systemic lupus erythematosus 1.92 1.60e-3 45/135 (33.33%) CTSG;HLA-DQB1;HLA-DRB1;...
Intestinal immune network for IgA production 1.82 1.26e-2 38/48 (79.17%) CXCL12;HLA-DQB1;HLA-DRB1;...
Hematopoietic cell lineage 1.82 1.12e-2 90/99 (90.91%) IL1B;CD44;CD1D;...
MicroRNAs in cancer 1.81 1.01e-2 146/310 (47.1%) MARCKS;HMOX1;PDGFA;...
Graft-versus-host disease 1.80 1.02e-2 32/42 (76.19%) IL1B;IL1A;HLA-DQB1;...
Type I diabetes mellitus 1.76 1.86e-2 38/43 (88.37%) IL1B;IL1A;HLA-DQB1;...
Cytokine-cytokine receptor interaction 1.74 2.23e-2 246/295 (83.39%) IL1B;CCL2;LIF;...
Inflammatory bowel disease 1.73 2.47e-2 58/65 (89.23%) IL1B;IL1A;HLA-DQB1;...
Asthma 1.72 2.61e-2 25/31 (80.65%) RNASE3;HLA-DQB1;HLA-DRB1;...
Arachidonic acid metabolism 1.72 2.51e-2 48/61 (78.69%) AKR1C3;GPX2;PTGIS;...
Proteoglycans in cancer 1.71 2.63e-2 172/205 (83.9%) IGF1R;FLNB;CCND1;...
Regulation of actin cytoskeleton 1.71 2.92e-2 185/218 (84.86%) PDGFA;FGFR3;MYH11;...
Viral protein interaction with cytokine and cytokine re... 1.69 3.12e-2 84/100 (84%) CCL2;CXCL12;CXCL1;...
Complement and coagulation cascades 1.68 3.91e-2 76/85 (89.41%) PLAT;FGG;SERPINB2;...
Protein digestion and absorption 1.66 4.20e-2 78/103 (75.73%) COL1A1;COL11A1;COL6A3;...
Legionellosis 1.66 4.01e-2 51/57 (89.47%) IL1B;CXCL1;ITGAM;...
IL-17 signaling pathway 1.66 4.13e-2 84/94 (89.36%) IL1B;CCL2;CXCL1;...
Antigen processing and presentation 1.66 4.09e-2 60/78 (76.92%) PDIA3;HSPA5;HLA-DQB1;...
PI3K-Akt signaling pathway 1.65 3.98e-2 317/354 (89.55%) PDGFA;IGF1R;MYB;...
Fluid shear stress and atherosclerosis 1.65 3.95e-2 123/139 (88.49%) IL1B;HMOX1;PDGFA;...
Rheumatoid arthritis 1.65 3.89e-2 78/93 (83.87%) IL1B;CCL2;TEK;...
Transcriptional misregulation in cancer 1.64 3.87e-2 158/192 (82.29%) DUSP6;PDGFA;IGF1R;...
Folate biosynthesis 1.63 4.31e-2 23/26 (88.46%) AKR1C3;GGH;FPGS;...
Sulfur metabolism 1.61 4.99e-2 9/10 (90%) SQOR;TST;PAPSS1;...
mRNA surveillance pathway -1.78 3.04e-2 71/98 (72.45%) DDX19A;GLE1;PABPC4;...
Ribosome -2.00 0.00e+0 113/158 (71.52%) RPL36;RPL31;RPL36A;...
Oxidative phosphorylation -2.06 0.00e+0 93/133 (69.92%) ATP12A;NDUFA5;NDUFV2;...
Steroid biosynthesis -2.17 0.00e+0 19/20 (95%) TM7SF2;DHCR24;HSD17B7;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Breast
Breast adenocarcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
MCF7 CVCL_0031 Homo sapiens 3.33uM 6H
Lung
Lung adenocarcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
A549 CVCL_0023 Homo sapiens 3.33uM 6H
Pancreas
Pancreatic carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
YAPC CVCL_1791 Homo sapiens 3.33uM 6H
Prostate
Prostate carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
PC-3 CVCL_0035 Homo sapiens 3.33uM 6H
Skin
Melanoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
A-375 CVCL_0132 Homo sapiens 3.33uM 6H