General Information of Drug (ID: DMELYAX)

Drug Name
NU-6027 Drug Info
Cross-matching ID
PubChem CID
398148
ChEBI ID
CHEMBL303958
CAS Number
CAS 220036-08-8
TTD Drug ID
D0U8YN

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Histidine metabolism 1.83 3.34e-2 16/22 (72.73%) HNMT;MAOA;ALDH3A1;...
Malaria -1.67 5.00e-2 44/50 (88%) IL1B;THBS2;TGFB1;...
Vibrio cholerae infection -1.68 4.88e-2 44/50 (88%) ATP6V1D;KCNQ1;TCIRG1;...
ECM-receptor interaction -1.70 4.17e-2 80/88 (90.91%) THBS1;TNN;VWF;...
Gastric acid secretion -1.72 3.34e-2 63/76 (82.89%) ATP1B4;ATP1A1;ADCY1;...
Insulin signaling pathway -1.76 2.03e-2 121/137 (88.32%) FLOT1;ACACA;SREBF1;...
Adipocytokine signaling pathway -1.77 1.97e-2 64/69 (92.75%) STK11;TNFRSF1A;ACSL3;...
Citrate cycle (TCA cycle) -1.78 2.03e-2 30/30 (100%) SUCLA2;IDH3B;DLST;...
Melanoma -1.79 1.96e-2 68/72 (94.44%) FGF5;FGF4;PIK3R1;...
Insulin resistance -1.80 2.20e-2 96/108 (88.89%) PRKAB2;SOCS3;PIK3R1;...
Legionellosis -1.81 2.13e-2 51/57 (89.47%) RAB1A;ARF1;IL1B;...
PPAR signaling pathway -1.85 1.58e-2 66/74 (89.19%) ACOX3;ANGPTL4;APOA1;...
Cardiac muscle contraction -1.89 1.36e-2 64/87 (73.56%) ATP1B4;ATP1A1;ATP1A3;...
Dilated cardiomyopathy -1.91 1.36e-2 86/96 (89.58%) CACNG1;CACNA1S;TGFB3;...
Hypertrophic cardiomyopathy -1.92 1.81e-2 81/90 (90%) PRKAB2;CACNG1;CACNA1S;...
Regulation of lipolysis in adipocytes -1.92 2.03e-2 52/55 (94.55%) NPR1;PLAAT3;PIK3R3;...
AMPK signaling pathway -1.96 2.71e-2 106/120 (88.33%) PPP2R5A;PPP2CA;PPP2R5B;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Breast
Fibrocystic breast disease
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
MCF-10A (Parent) CVCL_0598 Homo sapiens 1.11uM - 10uM 3H, 6H, 12H, 24H