General Information of Drug (ID: DMKDZLG)

Drug Name
BAZ2-ICR Drug Info
Synonyms inhibitor 13 [PMID: 25719566]
Cross-matching ID
PubChem CID
91654625
ChEBI ID
CHEMBL4296718
TTD Drug ID
D0I4FP

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Type I diabetes mellitus -1.68 3.78e-2 38/43 (88.37%) HLA-DQA1;HLA-DQB1;HLA-DRB1;...
AMPK signaling pathway -1.74 2.07e-2 106/120 (88.33%) IRS2;RAB8A;PPP2R2A;...
Systemic lupus erythematosus -1.75 2.01e-2 45/135 (33.33%) SSB;HLA-DQA1;HLA-DQB1;...
Legionellosis -1.76 1.81e-2 51/57 (89.47%) NFKB1;RAB1A;CASP8;...
PPAR signaling pathway -1.76 1.95e-2 66/74 (89.19%) ACOX3;MMP1;ANGPTL4;...
Rheumatoid arthritis -1.80 1.46e-2 78/93 (83.87%) IFNG;ATP6V1B2;TNFSF11;...
Pertussis -1.81 1.59e-2 64/76 (84.21%) CALML3;PYCARD;MAPK13;...
Asthma -1.82 1.65e-2 25/31 (80.65%) IL10;RNASE3;MS4A2;...
Fatty acid biosynthesis -1.83 1.51e-2 16/18 (88.89%) ACSL4;ACSBG1;ACACA;...
Allograft rejection -1.85 1.09e-2 32/38 (84.21%) HLA-DQA1;HLA-DQB1;HLA-DRB1;...
Graft-versus-host disease -1.92 1.39e-3 32/42 (76.19%) HLA-E;KIR3DL1;IL1B;...
Viral myocarditis -1.94 1.62e-3 53/60 (88.33%) HLA-DQA1;HLA-DQB1;ABL1;...
Intestinal immune network for IgA production -1.94 1.95e-3 38/48 (79.17%) HLA-DQA1;HLA-DQB1;ICOS;...
Complement and coagulation cascades -2.01 0.00e+0 76/85 (89.41%) C3AR1;F13A1;C5AR1;...
Staphylococcus aureus infection -2.05 0.00e+0 72/95 (75.79%) HLA-DPA1;DEFA5;HLA-DPB1;...
Cytokine-cytokine receptor interaction -2.21 0.00e+0 246/295 (83.39%) IL3RA;IL4;TNFRSF10B;...
Viral protein interaction with cytokine and cytokine re... -2.28 0.00e+0 84/100 (84%) TNFRSF10B;CCR9;IL24;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Prostate
Prostate carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
PC-3 CVCL_0035 Homo sapiens 1.11uM - 10uM 24H
Skin
Melanoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
A-375 CVCL_0132 Homo sapiens 1.11uM - 10uM 24H