General Information of Drug (ID: DMKTX1A)

Drug Name
MCCG Drug Info
Synonyms MCCG-I
Cross-matching ID
PubChem CID
5311457
ChEBI ID
CHEMBL41013
TTD Drug ID
D0YO8B

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Retinol metabolism 2.22 0.00e+0 41/68 (60.29%) ADH1C;CYP2C8;UGT2B4;...
Complement and coagulation cascades 2.12 0.00e+0 76/85 (89.41%) CLU;C9;CFB;...
ABC transporters 2.10 0.00e+0 37/45 (82.22%) ABCB1;ABCA5;CFTR;...
Metabolism of xenobiotics by cytochrome P450 2.08 0.00e+0 49/77 (63.64%) ADH1C;UGT2B4;ADH1A;...
Drug metabolism 1.95 3.13e-3 78/151 (51.66%) ADH1C;CYP2C8;CES1;...
Sulfur metabolism 1.89 9.14e-3 9/10 (90%) SELENBP1;PAPSS2;MPST;...
Cholesterol metabolism 1.86 7.83e-3 44/50 (88%) ANGPTL3;APOA1;NPC2;...
Primary bile acid biosynthesis 1.83 1.18e-2 15/17 (88.24%) CYP39A1;BAAT;ACOT8;...
Peroxisome 1.75 2.35e-2 72/82 (87.8%) IDH2;ACOX1;SOD1;...
Fat digestion and absorption 1.71 3.06e-2 35/43 (81.4%) FABP1;ACAT2;ACAT1;...
Glyoxylate and dicarboxylate metabolism 1.65 4.91e-2 23/30 (76.67%) GLUL;ACAT2;ACAT1;...
Legionellosis -1.72 3.43e-2 51/57 (89.47%) PYCARD;CASP3;HSPA8;...
Phagosome -1.73 3.26e-2 118/152 (77.63%) HLA-F;PIK3C3;RAB5C;...
Toxoplasmosis -1.75 2.37e-2 103/112 (91.96%) MAPK14;IL10RA;JAK2;...
Tuberculosis -1.76 2.77e-2 159/180 (88.33%) PPP3CB;IFNGR1;PIK3C3;...
Hematopoietic cell lineage -1.77 2.85e-2 90/99 (90.91%) EPOR;CD38;HLA-DRA;...
Epithelial cell signaling in Helicobacter pylori infect... -1.86 2.07e-2 62/70 (88.57%) CHUK;MAPK11;ATP6V1H;...
Asthma -1.89 2.77e-2 25/31 (80.65%) IL9;RNASE3;HLA-DOA;...
Collecting duct acid secretion -1.92 2.96e-2 22/27 (81.48%) ATP6V1E1;CLCNKB;ATP4B;...
Bacterial invasion of epithelial cells -2.07 2.37e-2 59/77 (76.62%) CTNNB1;ACTR3;ILK;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Fibroblast
Nasopharyngeal carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
FIBRNPC CVCL_UK07 Homo sapiens 10uM 6H, 24H