General Information of Drug (ID: DMY24S0)

Drug Name
Nadifloxacin Drug Info
Synonyms Acuatim; Nadixa; OPC-7251
Cross-matching ID
PubChem CID
4410
ChEBI ID
CHEMBL31889
CAS Number
CAS 124858-35-1
TTD Drug ID
D0I0RB

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Biosynthesis of unsaturated fatty acids -1.72 1.35e-2 21/27 (77.78%) ELOVL5;ELOVL2;HSD17B4;...
Epithelial cell signaling in Helicobacter pylori infect... -1.73 1.32e-2 62/70 (88.57%) RELA;NFKB1;CHUK;...
Measles -1.73 1.36e-2 133/139 (95.68%) CCND2;MAPK8;CDK4;...
Cytokine-cytokine receptor interaction -1.74 1.28e-2 246/295 (83.39%) IL11;CCL16;IL36RN;...
Retinol metabolism -1.76 1.14e-2 41/68 (60.29%) CYP26B1;ADH1C;CYP2C8;...
B cell receptor signaling pathway -1.78 9.91e-3 71/81 (87.65%) LILRB2;INPPL1;IKBKB;...
Colorectal cancer -1.79 9.81e-3 84/86 (97.67%) BCL2;TGFBR2;MAPK8;...
Influenza A -1.82 5.39e-3 156/172 (90.7%) AKT1;RELA;KPNA6;...
Lipid and atherosclerosis -1.85 3.94e-3 190/215 (88.37%) NLRP3;TANK;NFATC3;...
Pancreatic cancer -1.86 4.13e-3 75/76 (98.68%) TGFBR2;MAPK8;CDK4;...
AGE-RAGE signaling pathway in diabetic complications -1.87 2.48e-3 97/100 (97%) PIM1;BCL2;VEGFB;...
Leishmaniasis -1.88 2.61e-3 67/77 (87.01%) NCF4;C3;HLA-DRA;...
TGF-beta signaling pathway -1.88 2.75e-3 81/94 (86.17%) RPS6KB1;ID2;CDKN2B;...
Osteoclast differentiation -1.90 2.92e-3 117/127 (92.13%) IFNB1;NCF4;SYK;...
Hepatitis B -1.91 3.10e-3 151/162 (93.21%) TGFBR2;ATF2;MAPK8;...
Kaposi sarcoma-associated herpesvirus infection -1.91 3.30e-3 172/193 (89.12%) EP300;MICB;IKBKB;...
Primary bile acid biosynthesis -1.92 2.65e-3 15/17 (88.24%) SCP2;CYP46A1;ACOX2;...
Toll-like receptor signaling pathway -1.96 1.91e-3 94/104 (90.38%) CD86;CXCL9;AKT1;...
Complement and coagulation cascades -1.98 2.06e-3 76/85 (89.41%) C8B;PROC;C6;...
PD-L1 expression and PD-1 checkpoint pathway in cancer -2.01 1.13e-3 79/89 (88.76%) IFNG;IKBKB;ALK;...
Bladder cancer -2.03 1.24e-3 40/41 (97.56%) CDK4;RB1;MYC;...
Viral protein interaction with cytokine and cytokine re... -2.06 0.00e+0 84/100 (84%) IL19;TNFRSF10C;TNFSF14;...
Coronavirus disease -2.09 0.00e+0 215/232 (92.67%) RPS25;RPL6;RPS3;...
NOD-like receptor signaling pathway -2.10 0.00e+0 145/181 (80.11%) MAPK8;CASR;IFNA17;...
NF-kappa B signaling pathway -2.10 0.00e+0 90/104 (86.54%) SYK;TNFSF11;EDAR;...
Malaria -2.15 0.00e+0 44/50 (88%) VCAM1;CD40LG;KLRB1;...
Rheumatoid arthritis -2.15 0.00e+0 78/93 (83.87%) TNFSF11;CD86;HLA-DRA;...
TNF signaling pathway -2.17 0.00e+0 103/112 (91.96%) AKT1;RELA;VCAM1;...
C-type lectin receptor signaling pathway -2.21 0.00e+0 93/104 (89.42%) NLRP3;NFATC3;NFATC4;...
IL-17 signaling pathway -2.38 0.00e+0 84/94 (89.36%) IL5;MMP1;RELA;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Breast
Breast adenocarcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
MCF7 CVCL_0031 Homo sapiens 10uM 6H, 24H
Prostate
Prostate carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
PC-3 CVCL_0035 Homo sapiens 10uM 6H, 24H