General Information of Drug (ID: DM1LO8K)

Drug Name
RVX-208
Indication
Disease Entry ICD 11 Status REF
Alzheimer disease 8A20 Phase 1/2 [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
Cross-matching ID
PubChem CID
24871506
TTD ID
D0N7WW
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Bromodomain-containing protein 4 (BRD4) TTRA6BO BRD4_HUMAN Modulator [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Alzheimer disease
ICD Disease Classification 8A20
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Bromodomain-containing protein 4 (BRD4) DTT BRD4 3.27E-01 0.02 0.04
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 38 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC2 5.557 7.3365 2.7353 0.4989
TC-71 GDSC2 4.0232 6.7278 2.1621 5.5362
EW-24 GDSC2 4.0377 6.326 2.3664 4.2578
MG-63 GDSC2 4.1784 12.841 -0.7441 20.8951
SK-PN-DW GDSC2 4.4542 6.7178 2.4491 2.9728
ES8 GDSC2 4.4913 7.9288 1.905 6.074
EW-3 GDSC2 4.5068 10.1438 0.841 12.2489
A-673 GDSC2 4.5428 7.1935 2.2843 3.7522
CADO-ES1 GDSC2 4.5476 8.7099 1.5683 7.9533
EW-1 GDSC2 4.7184 7.7959 2.114 4.4099
EW-12 GDSC2 4.814 8.43 1.8785 5.5871
CAL-78 GDSC2 4.8145 6.8683 2.5838 1.7301
NY GDSC2 4.9199 14.6298 -1.0618 20.3151
EW-7 GDSC2 4.9247 6.8369 2.6523 1.2852
U-CH2 GDSC2 5.1694 7.1617 2.6362 1.115
NOS-1 [Human HNSCC] GDSC2 5.2041 8.2213 2.206 3.1155
CAL-72 GDSC2 5.2429 6.75 2.826 0.406
HuO-3N1 GDSC2 5.2441 7.7217 2.4422 1.8903
HuO9 GDSC2 5.3742 10.5637 1.2352 8.1554
MHH-ES-1 GDSC2 5.4007 10.6396 1.2165 8.2067
EW-18 GDSC2 5.461 7.6217 2.586 1.0617
SaOS-2 GDSC2 5.5541 13.3078 0.0446 13.9886
HOS GDSC2 5.5605 7.3184 2.7434 0.4747
ES4 GDSC2 5.5925 8.3234 2.3642 1.8604
EW-16 GDSC2 5.6843 13.0107 0.2768 12.5776
EW-22 GDSC2 5.763 7.4936 2.7584 0.3485
ES7 GDSC2 5.8124 8.0303 2.5803 0.8247
U2OS GDSC2 5.9136 13.0194 0.4257 11.3683
SK-ES-1 GDSC2 5.9171 7.5892 2.782 0.2482
EW-13 GDSC2 6.059 7.8101 2.7568 0.2538
CHSA8926 GDSC2 6.0654 15.9864 -0.8953 17.0639
H-EMC-SS GDSC2 6.0887 8.4587 2.5336 0.8019
ES6 GDSC2 6.1147 8.3222 2.5948 0.607
G-292 clone A141B1 GDSC2 6.1286 8.2302 2.6339 0.4971
CHSA0108 GDSC2 6.4633 8.3691 2.7092 0.2297
CHSA0011 GDSC2 6.4864 10.1945 2.0275 2.4091
ES5 GDSC2 6.4912 8.8972 2.5331 0.5917
EW-11 GDSC2 6.5812 9.036 2.5177 0.5904
⏷ Show the Full List of 38 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 157 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JM1 GDSC2 4.2474 6.5187 2.4133 3.5527
SIG-M5 GDSC2 0.6575 3.7415 0.2896 28.6268
OCI-Ly7 GDSC2 1.4051 4.5793 0.7901 22.5921
GA-10 GDSC2 2.3814 3.0974 2.347 9.6156
CRO-AP2 GDSC2 2.3919 5.7546 1.2643 15.9685
SUP-B8 GDSC2 2.4646 6.4816 0.981 17.3928
NB4 GDSC2 2.7607 7.657 0.6706 18.1666
THP-1 GDSC2 2.7997 7.9432 0.5628 18.6369
Kasumi-1 GDSC2 2.8584 6.2425 1.4594 13.1812
KMS-11 GDSC2 2.9142 10.1367 -0.431 23.2199
OCI-AML-3 GDSC2 2.9298 6.6476 1.322 13.7916
Namalwa GDSC2 3.0914 15.6337 -3.0271 31.3097
BONNA-12 GDSC2 3.1848 7.4425 1.1463 14.0574
Jiyoye GDSC2 3.2241 6.5601 1.6206 11.0365
BC-1 GDSC2 3.2626 5.2711 2.2975 6.6607
GDM-1 GDSC2 3.289 7.9706 0.9701 14.785
MOLM-16 GDSC2 3.3177 7.24 1.3594 12.3708
RCH-ACV GDSC2 3.3569 7.2171 1.4034 11.9861
SR GDSC2 3.3721 5.9042 2.0724 7.7646
SUP-HD1 GDSC2 3.387 5.1524 2.4604 5.2684
H9 GDSC2 3.4045 7.2524 1.425 11.7157
A3/Kawakami GDSC2 3.4066 4.5381 2.7828 3.175
KMS-12-BM GDSC2 3.4112 6.0257 2.0437 7.8347
A4/Fukuda GDSC2 3.4514 5.5861 2.2958 6.1299
L-1236 GDSC2 3.4816 11.712 -0.7407 22.8242
OPM-2 GDSC2 3.492 5.3721 2.4349 5.1404
NCI-H929 GDSC2 3.4931 6.6629 1.7918 9.1886
ST486 GDSC2 3.4997 5.6921 2.2815 6.088
VL51 GDSC2 3.5144 6.025 2.1273 7.0211
L-428 GDSC2 3.5225 4.9839 2.6515 3.6961
AMO1 GDSC2 3.5394 5.4009 2.4576 4.8717
SU-DHL-10 GDSC2 3.5924 4.9907 2.7008 3.2124
MM1.S GDSC2 3.6033 6.2132 2.1035 6.932
RPMI-8226 GDSC2 3.631 5.6717 2.3936 5.0379
SU-DHL-16 GDSC2 3.6338 11.596 -0.5582 21.6021
BL-41 GDSC2 3.6429 5.7461 2.3658 5.1817
CTV-1 GDSC2 3.6619 7.4685 1.5248 10.3827
NALM-6 GDSC2 3.6719 5.934 2.2948 5.5534
JSC-1 GDSC2 3.6963 5.407 2.5725 3.7608
JVM-3 GDSC2 3.7149 9.848 0.3804 16.8361
KY821 GDSC2 3.7187 5.6038 2.4924 4.205
BALL-1 GDSC2 3.7201 5.9925 2.3022 5.3866
MOLT-13 GDSC2 3.7406 6.113 2.2581 5.6115
Karpas-422 GDSC2 3.7611 7.489 1.5921 9.7032
HL-60 GDSC2 3.7638 5.0944 2.7714 2.3912
MOLM-13 GDSC2 3.7859 5.4508 2.615 3.2933
KOPN-8 GDSC2 3.8257 6.7594 2.0028 6.9916
Daudi GDSC2 3.8314 5.5837 2.5824 3.3922
ML-2 GDSC2 3.8399 7.8538 1.4719 10.2326
OCI-AML-5 GDSC2 3.8473 6.7276 2.0346 6.74
NOMO-1 GDSC2 3.8549 6.3818 2.2103 5.631
WSU-NHL GDSC2 3.8569 5.8138 2.4888 3.9077
TALL-1 [Human adult T-ALL] GDSC2 3.89 14.2728 -1.6876 25.2568
MHH-CALL-2 GDSC2 3.9107 5.8377 2.5145 3.6327
SKM-1 GDSC2 3.9139 5.3581 2.7448 2.2488
Raji GDSC2 3.9229 6.2231 2.3366 4.6927
MLMA GDSC2 3.9365 13.1861 -1.1078 23.0195
HAL-01 GDSC2 3.9536 6.2892 2.3261 4.6879
NU-DUL-1 GDSC2 3.9587 6.6861 2.1365 5.8419
P30/OHK GDSC2 3.9649 6.1852 2.3843 4.3071
ME1 GDSC2 3.974 6.1791 2.3935 4.2311
DEL GDSC2 3.9872 7.6985 1.6603 8.7063
OCI-AML-2 GDSC2 4.0029 6.7073 2.1577 5.609
697 GDSC2 4.005 5.7393 2.624 2.7828
CCRF-CEM GDSC2 4.0419 6.3239 2.3703 4.225
MC116 GDSC2 4.0676 11.6513 -0.2388 18.9469
MOLT-16 GDSC2 4.0685 6.175 2.4593 3.6342
Karpas-299 GDSC2 4.0718 14.5973 -1.7037 24.8272
RPMI-6666 GDSC2 4.0867 7.3141 1.9217 6.864
ARH-77 GDSC2 4.0869 6.1452 2.4855 3.4408
LP-1 GDSC2 4.1393 6.203 2.4923 3.2973
Loucy GDSC2 4.1455 6.9194 2.1547 5.3088
GR-ST GDSC2 4.1557 6.7633 2.2367 4.7905
BC-3 GDSC2 4.1707 8.8312 1.2386 10.7891
EJM GDSC2 4.2062 6.1994 2.5364 2.9137
KE-37 GDSC2 4.2104 6.3332 2.4767 3.2527
Karpas-1106P GDSC2 4.2305 5.9424 2.6691 2.1204
ALL-PO GDSC2 4.2309 12.3864 -0.4768 19.5973
JJN-3 GDSC2 4.2471 5.9721 2.6654 2.114
MHH-CALL-4 GDSC2 4.2501 10.3107 0.5677 14.3906
P12-Ichikawa GDSC2 4.2534 11.1168 0.171 16.4573
OCI-Ly19 GDSC2 4.2914 6.9981 2.2155 4.6357
MEG-01 GDSC2 4.2963 6.4824 2.4611 3.1834
SUP-T1 GDSC2 4.3152 6.2556 2.5769 2.4922
Ku812 GDSC2 4.3159 6.4776 2.4754 3.0654
MN-60 GDSC2 4.4023 6.2686 2.6218 2.1059
Reh GDSC2 4.406 6.298 2.6107 2.1598
KG-1 GDSC2 4.4126 12.6034 -0.4441 18.9765
CA46 GDSC2 4.4207 6.99 2.3027 3.8697
RPMI-8866 GDSC2 4.441 6.5382 2.523 2.5834
L-363 GDSC2 4.4441 9.6492 1.0378 11.2884
JVM-2 GDSC2 4.4503 9.0212 1.3491 9.4665
OCI-M1 GDSC2 4.4694 5.853 2.8365 0.947
MOLP-8 GDSC2 4.4747 6.9331 2.3626 3.4264
L-540 GDSC2 4.4876 6.9464 2.3644 3.3933
SCC-3 GDSC2 4.5373 6.0229 2.7994 1.0404
VAL GDSC2 4.5403 7.0954 2.328 3.5078
P32/ISH GDSC2 4.5567 6.0536 2.7962 1.034
HEL GDSC2 4.5759 6.6231 2.5621 2.163
Karpas-45 GDSC2 4.5879 9.0521 1.431 8.6731
Ramos.2G6.4C10 GDSC2 4.5915 10.3913 0.7814 12.3761
CESS GDSC2 4.6008 6.7068 2.539 2.2482
EoL-1 GDSC2 4.6064 6.205 2.7579 1.1531
JeKo-1 GDSC2 4.6536 10.1448 0.9465 11.3102
Karpas-620 GDSC2 4.701 6.7181 2.5887 1.8517
DND-41 GDSC2 4.7202 9.4261 1.3419 8.9008
CML-T1 GDSC2 4.7316 6.7702 2.5825 1.8425
KM-H2 GDSC2 4.7714 6.9001 2.5476 1.9648
SU-DHL-6 GDSC2 4.7792 6.5091 2.7167 1.1526
EM-2 GDSC2 4.8381 6.38 2.7962 0.7682
SU-DHL-5 GDSC2 4.8547 5.8039 3.0163 0.123
PL-21 GDSC2 4.87 8.5552 1.8554 5.6135
SK-MM-2 GDSC2 4.8821 7.6503 2.2781 3.2167
DB GDSC2 4.8968 7.4827 2.3611 2.7505
MY-M12 GDSC2 4.9124 12.0753 0.1896 14.7279
SUP-M2 GDSC2 4.915 6.0756 2.943 0.2536
IM-9 GDSC2 4.9402 6.139 2.9299 0.275
HH [Human lymphoma] GDSC2 4.9446 7.1868 2.5155 1.9002
KCL-22 GDSC2 4.9824 7.8504 2.246 3.2342
Karpas-231 GDSC2 4.9837 6.5666 2.7876 0.6864
U266B1 GDSC2 5.0066 7.0394 2.6086 1.3929
LAMA-84 GDSC2 5.0378 11.4021 0.6071 12.2844
K-562 GDSC2 5.0404 6.5593 2.8146 0.5548
DG-75 GDSC2 5.0832 7.6162 2.4041 2.2717
RC-K8 GDSC2 5.1336 6.5015 2.8737 0.3313
TUR GDSC2 5.1891 6.7998 2.7857 0.5546
SU-DHL-4 GDSC2 5.2416 6.9465 2.7521 0.6298
BE-13 GDSC2 5.2422 8.6274 2.0471 3.9005
DoHH2 GDSC2 5.2597 6.8044 2.8127 0.4344
PF-382 GDSC2 5.2692 7.2318 2.6537 0.9599
RS4;11 GDSC2 5.2735 7.3001 2.6286 1.0532
HC-1 GDSC2 5.2854 7.0823 2.7188 0.7121
RL GDSC2 5.3224 6.5796 2.9167 0.1715
Hs 445 GDSC2 5.3291 6.8987 2.8056 0.4192
WIL2 NS GDSC2 5.3373 6.8284 2.8343 0.3409
Jurkat GDSC2 5.3863 7.026 2.7816 0.4568
ROS-50 GDSC2 5.3886 8.3797 2.2368 2.7044
HT GDSC2 5.4127 14.8455 -0.8039 18.1127
ATN-1 GDSC2 5.4321 6.7341 2.9028 0.1666
Granta-519 GDSC2 5.4345 7.0554 2.7899 0.4107
QIMR-WIL GDSC2 5.4507 13.9587 -0.3437 16.0289
MHH-PREB-1 GDSC2 5.4564 7.0205 2.811 0.3477
Farage GDSC2 5.4889 7.1515 2.7762 0.4213
CTB-1 GDSC2 5.4942 7.6461 2.5912 1.0152
ALL-SIL GDSC2 5.5296 7.2364 2.7612 0.4418
HDLM-2 GDSC2 5.5619 7.4663 2.6891 0.6326
SUP-B15 GDSC2 5.5757 7.282 2.7626 0.4164
U-698-M GDSC2 5.6198 7.2839 2.7789 0.3573
NK-92MI GDSC2 5.6482 7.242 2.8046 0.2888
EB2 GDSC2 5.6619 7.555 2.6967 0.5538
SU-DHL-8 GDSC2 5.6745 7.0187 2.8914 0.1299
MOLT-4 GDSC2 5.702 7.0243 2.8991 0.1146
JURL-MK1 GDSC2 5.7537 7.2871 2.8276 0.2115
TK [Human B-cell lymphoma] GDSC2 5.8171 7.4058 2.8094 0.2266
KMOE-2 GDSC2 5.8729 7.5335 2.7853 0.2551
LC4-1 GDSC2 6.2577 8.0908 2.7314 0.2444
SU-DHL-1 GDSC2 6.986 18.9268 -1.6784 18.1888
⏷ Show the Full List of 157 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KYSE-50 GDSC2 4.6431 7.0247 2.4212 2.8161
KYSE-220 GDSC2 4.8405 13.0395 -0.3367 17.4193
FLO-1 GDSC2 5.4966 11.0944 1.0642 8.8535
KYAE-1 GDSC2 5.512 7.2829 2.7371 0.5173
SK-GT-4 GDSC2 5.5195 12.5722 0.3753 12.4317
OACM5.1 C GDSC2 5.6707 8.8228 2.1944 2.556
HCE-4 GDSC2 5.6797 15.4035 -0.8845 17.8487
ESO-51 GDSC2 6.0927 7.902 2.737 0.2808
OACP4 C GDSC2 6.1689 8.334 2.6119 0.5352
ESO-26 GDSC2 6.1984 8.0463 2.7254 0.2715
TE-12 GDSC2 7.0419 9.6004 2.4912 0.4692
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC2 4.2557 6.71 2.3286 4.0356
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SJNB-6 GDSC2 1.371 4.3474 0.8456 22.4313
NB69 GDSC2 3.3828 11.7449 -0.8389 23.5209
CHP-212 GDSC2 3.6638 7.5932 1.4641 10.7498
SK-N-DZ GDSC2 4.0777 7.1362 2.0021 6.3922
NB(TU)1 GDSC2 4.1078 6.2468 2.4511 3.6033
LA-N-6 GDSC2 4.1892 6.6839 2.2972 4.3566
KP-N-RT-BM-1 GDSC2 4.1958 7.8861 1.7208 7.8349
IMR-5 GDSC2 4.3803 8.0699 1.7616 7.1693
KP-N-YN GDSC2 4.4687 16.1037 -2.1402 25.2425
SJNB-10 GDSC2 4.6103 9.1776 1.3859 8.8875
SK-N-BE(2)-M17 GDSC2 4.6805 6.649 2.6076 1.7841
CHP-134 GDSC2 4.9051 7.0935 2.5348 1.8556
SJNB-17 GDSC2 5.0019 8.0717 2.158 3.68
SJNB-13 GDSC2 5.1072 7.8073 2.3342 2.5913
Kelly GDSC2 5.1151 6.754 2.772 0.6474
SK-N-MC-IXC GDSC2 5.1594 6.2593 2.9686 0.1263
CHP-126 GDSC2 5.1761 7.1215 2.6553 1.0321
SJNB-7 GDSC2 5.2953 7.2298 2.666 0.8927
MHH-NB-11 GDSC2 5.3247 6.976 2.7753 0.5075
TGW GDSC2 5.5526 6.9269 2.8796 0.1749
SiMa GDSC2 5.5673 7.6926 2.6052 0.9086
SJNB-14 GDSC2 5.6448 7.3447 2.7667 0.3764
NH-12 GDSC2 5.7533 7.7339 2.6672 0.5899
SK-N-AS GDSC2 5.8463 17.6374 -1.8565 21.1245
GOTO GDSC2 5.9963 8.131 2.618 0.6024
SJNB-5 GDSC2 6.0186 7.9889 2.6785 0.4342
KP-N-YS GDSC2 6.1518 8.2727 2.6274 0.5031
GI-ME-N GDSC2 6.7064 9.3728 2.444 0.7264
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuCC-T1 GDSC2 5.6348 7.2961 2.7803 0.348
Cancer Drug Sensitivity Data Curated from 46 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-453 GDSC2 3.5478 6.0508 2.1409 6.8447
Hs 578T GDSC2 3.7989 8.4769 1.1304 12.3918
HCC2157 GDSC2 4.0031 6.2922 2.359 4.3774
HCC2218 GDSC2 4.3543 8.5585 1.5062 8.7585
EFM-192A GDSC2 4.437 8.0128 1.8281 6.6473
Evsa-T GDSC2 4.4528 9.775 0.9825 11.5831
DU4475 GDSC2 4.5383 6.4621 2.6122 1.9554
CAL-85-1 GDSC2 4.6023 10.3337 0.8174 12.1512
BT-474 GDSC2 4.6608 7.2406 2.3339 3.268
HDQ-P1 GDSC2 4.7059 6.4021 2.7251 1.1928
COLO 824 GDSC2 4.7327 7.473 2.2709 3.4984
OCUB-M GDSC2 4.7664 7.7151 2.1805 3.9471
BT-549 GDSC2 4.769 10.8343 0.6928 12.441
MDA-MB-468 GDSC2 4.7707 8.8694 1.6428 7.0425
HCC1569 GDSC2 4.779 9.5447 1.3252 8.8694
MFM-223 GDSC2 4.8587 7.0609 2.5245 1.9654
MDA-MB-361 GDSC2 4.8966 10.7168 0.8404 11.343
HCC1500 GDSC2 4.9081 7.7726 2.2382 3.3924
CAL-120 GDSC2 4.9856 6.3707 2.8628 0.4364
HCC1806 GDSC2 5.0083 9.467 1.5155 7.2978
HCC1428 GDSC2 5.0396 6.5707 2.8099 0.5706
YMB-1-E GDSC2 5.0602 7.5726 2.4107 2.2685
HCC1599 GDSC2 5.1792 7.3448 2.5666 1.3986
T-47D GDSC2 5.2701 7.7577 2.4402 1.8696
HCC38 GDSC2 5.3015 8.601 2.0925 3.5679
MCF-7 GDSC2 5.3347 8.2759 2.253 2.6949
BT-20 GDSC2 5.3653 8.0106 2.3819 2.0318
MDA-MB-157 GDSC2 5.4333 8.4763 2.2189 2.7353
MRK-nu-1 GDSC2 5.4447 7.0182 2.8073 0.3616
HCC1937 GDSC2 5.4707 7.9025 2.4781 1.4892
MDA-MB-436 GDSC2 5.4921 7.2693 2.7341 0.5366
CAL-51 GDSC2 5.5763 7.2046 2.7908 0.3468
CAMA-1 GDSC2 5.5782 8.5627 2.2572 2.3687
MDA-MB-415 GDSC2 5.5921 7.5535 2.6687 0.6781
ZR-75-30 GDSC2 5.6358 8.3459 2.376 1.7635
HCC1187 GDSC2 5.6815 7.1681 2.8427 0.2045
HCC70 GDSC2 5.7271 7.9225 2.5853 0.8648
HCC1419 GDSC2 5.7393 9.2424 2.0508 3.1687
EFM-19 GDSC2 5.7552 7.733 2.6683 0.5858
MDA-MB-330 GDSC2 5.8066 12.6738 0.5193 11.1091
JIMT-1 GDSC2 5.8119 7.172 2.8874 0.1102
HCC1954 GDSC2 5.8796 7.5699 2.775 0.273
MDA-MB-231 GDSC2 5.9904 7.8414 2.7204 0.3487
UACC-893 GDSC2 6.1195 15.2121 -0.4841 15.2175
AU565 GDSC2 6.2607 8.5589 2.5659 0.6137
HCC1143 GDSC2 6.3876 8.7057 2.5622 0.5639
⏷ Show the Full List of 46 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 51 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D283 Med GDSC2 3.5686 5.3367 2.512 4.4538
CAS-1 GDSC2 3.6864 7.3643 1.5958 9.8791
LN-229 GDSC2 3.9127 7.1237 1.8881 7.4876
AM-38 GDSC2 4.1555 11.5928 -0.1411 18.2489
NMC-G1 GDSC2 4.4337 5.8708 2.8114 1.1014
LN-18 GDSC2 4.4963 8.9432 1.4197 8.9454
42-MG-BA GDSC2 4.5481 7.0412 2.3576 3.3266
U-87MG ATCC GDSC2 4.5725 7.9928 1.9284 5.7691
LN-405 GDSC2 4.5988 6.7661 2.5115 2.3973
PFSK-1 GDSC2 4.697 7.1923 2.377 2.9718
8-MG-BA GDSC2 4.7342 9.5558 1.2891 9.1755
GI-1 GDSC2 4.7619 6.7944 2.588 1.7759
Hs 683 GDSC2 4.7936 13.397 -0.5479 18.479
SF126 GDSC2 4.8143 6.5299 2.725 1.0806
DK-MG GDSC2 4.9076 7.268 2.4611 2.2185
D-336MG GDSC2 4.9169 6.9807 2.5886 1.5843
KINGS-1 GDSC2 4.9331 10.3781 1.0296 10.2128
SW1088 GDSC2 4.9602 7.143 2.5422 1.7525
A-172 GDSC2 4.9777 7.4608 2.4151 2.3569
Onda 10 GDSC2 4.9782 10.5156 0.9943 10.311
SF295 GDSC2 4.9945 6.4855 2.8233 0.5558
M059J GDSC2 4.9958 6.8706 2.6725 1.1266
GaMG GDSC2 5.0124 9.0842 1.6983 6.2447
KS-1 [Human Krukenberg tumour] GDSC2 5.1308 10.9136 0.9073 10.4606
D-542MG GDSC2 5.159 10.5197 1.1149 9.2552
YH-13 GDSC2 5.2093 7.5639 2.4908 1.7052
KNS-42 GDSC2 5.2458 6.5649 2.8937 0.2396
D-263MG GDSC2 5.2853 6.7906 2.8278 0.3807
ONS-76 GDSC2 5.3145 7.0825 2.731 0.6517
D-245MG GDSC2 5.3187 10.5721 1.1953 8.4851
U-118MG GDSC2 5.3315 7.0717 2.7422 0.605
D-566MG GDSC2 5.349 7.2159 2.6948 0.7506
YKG-1 GDSC2 5.3523 12.898 0.1023 14.1518
DBTRG-05MG GDSC2 5.4021 10.3308 1.3623 7.3986
KNS-81-FD GDSC2 5.422 13.9549 -0.3623 16.1772
Daoy GDSC2 5.461 7.2748 2.7194 0.5986
D-502MG GDSC2 5.5155 7.5563 2.6354 0.8396
KALS-1 GDSC2 5.5605 10.883 1.2044 7.9679
GB-1 GDSC2 5.576 7.1964 2.7936 0.3402
U-251MG GDSC2 5.6285 7.6813 2.6356 0.7621
SNB-75 GDSC2 5.6481 13.2891 0.1185 13.4303
D-392MG GDSC2 5.6899 17.2043 -1.7583 21.1263
SK-MG-1 GDSC2 5.7299 7.5829 2.7135 0.4734
Onda 11 GDSC2 5.7739 8.2656 2.4724 1.2393
Becker GDSC2 5.8064 7.8412 2.6489 0.6146
T98G GDSC2 5.896 7.9635 2.6397 0.5933
D-247MG GDSC2 6.1277 8.3865 2.5763 0.6522
H4 GDSC2 6.1864 24.762 -5.1145 28.8261
SF539 GDSC2 6.1903 14.5269 -0.1081 13.3851
SF268 GDSC2 6.2805 8.3371 2.6535 0.3899
D-423MG GDSC2 6.4254 9.2083 2.3905 1.0513
⏷ Show the Full List of 51 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TGBC24TKB GDSC2 4.0745 7.7429 1.703 8.2318
ETK-1 GDSC2 5.0259 8.5074 1.9741 4.6574
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RL95-2 GDSC2 3.9304 6.1214 2.3911 4.3418
ESS-1 GDSC2 4.3749 7.893 1.8432 6.6911
MFE-296 GDSC2 4.5229 6.8705 2.4205 3.0164
EN GDSC2 4.5395 11.7087 0.0949 16.1068
MFE-280 GDSC2 4.8288 9.2763 1.4876 7.8246
MFE-319 GDSC2 4.8689 7.4661 2.3528 2.8361
KLE GDSC2 5.8339 8.0395 2.5859 0.7927
AN3-CA GDSC2 5.8934 11.3479 1.1957 7.4075
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 32 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CAL-54 GDSC2 3.8966 7.4691 1.7056 8.6548
UO-31 GDSC2 3.9074 6.1267 2.3725 4.5072
KTCTL-26A GDSC2 4.0481 6.6474 2.2186 5.1344
NCC021 GDSC2 4.222 7.2608 2.0428 5.8208
769-P GDSC2 4.4348 6.7075 2.4422 3.0451
ACHN GDSC2 4.4811 6.7915 2.4316 3.025
KTCTL-13 GDSC2 4.6402 10.515 0.7562 12.3988
LB996-RCC GDSC2 4.666 8.7524 1.6287 7.3426
A-498 GDSC2 4.7013 6.2753 2.775 0.9785
SW13 GDSC2 4.8338 6.6618 2.6803 1.2569
HA7-RCC GDSC2 4.9259 7.3114 2.4521 2.2395
KTCTL-140 GDSC2 5.0293 7.6685 2.3525 2.6056
SN12C GDSC2 5.0365 7.2228 2.5472 1.6399
BFTC-909 GDSC2 5.0558 14.3688 -0.8315 19.0563
LB2241-RCC GDSC2 5.0972 7.5931 2.4214 2.1683
KMRC-20 GDSC2 5.0977 10.6531 1.0099 9.9669
VMRC-RCW GDSC2 5.1502 9.7389 1.4791 7.226
KTCTL-195 GDSC2 5.2906 10.6685 1.1313 8.8954
786-O GDSC2 5.3342 11.5211 0.7539 10.8573
A-704 GDSC2 5.3343 8.0488 2.35 2.2196
NCC010 GDSC2 5.3789 11.7694 0.6651 11.2332
RCC10RGB GDSC2 5.38 6.7874 2.8652 0.2535
TK-10 GDSC2 5.4408 7.8982 2.4656 1.5722
Caki-1 GDSC2 5.5207 12.2228 0.5437 11.5686
VMRC-RCZ GDSC2 5.5245 7.3393 2.7212 0.5567
OS-RC-2 GDSC2 5.7512 7.7533 2.6592 0.6146
KTCTL-21 GDSC2 5.8704 14.2834 -0.2078 14.4998
BB65-RCC GDSC2 5.911 16.3287 -1.1704 18.4857
SW156 GDSC2 6.1088 8.2778 2.6088 0.5717
LB1047-RCC GDSC2 6.1157 9.3231 2.2062 2.0132
KTCTL-1M GDSC2 6.2523 8.3551 2.6364 0.4393
RXF 393L GDSC2 6.2899 10.3486 1.865 3.3712
⏷ Show the Full List of 32 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KM12 GDSC2 3.8295 6.556 2.106 6.3403
SNU-175 GDSC2 3.9211 6.4356 2.2318 5.3421
SW626 GDSC2 3.9862 7.716 1.6509 8.7662
CL-11 GDSC2 4.0319 6.4186 2.3179 4.565
SW48 GDSC2 4.073 8.3245 1.4156 9.9779
RKO GDSC2 4.1162 10.6116 0.316 16.0753
SNU-C5 GDSC2 4.1586 6.6608 2.2878 4.4766
CCK-81 GDSC2 4.3667 10.3997 0.6116 13.8568
HT-29 GDSC2 4.3802 6.7864 2.3722 3.5427
RCM-1 [Human ESC] GDSC2 4.4273 6.5672 2.5017 2.724
SW1116 GDSC2 4.4297 10.1332 0.7897 12.7224
NCI-H508 GDSC2 4.468 9.8869 0.9386 11.7947
C2BBe1 GDSC2 4.5425 11.5173 0.1916 15.6153
SNU-61 GDSC2 4.5948 7.6257 2.1158 4.6281
SNU-283 GDSC2 4.6409 6.5483 2.63 1.7242
COLO205 GDSC2 4.7395 6.6199 2.6508 1.4996
LS411N GDSC2 4.9113 6.0987 2.9333 0.2791
HCT 15 GDSC2 4.9139 7.9876 2.1444 3.8987
LS123 GDSC2 4.953 7.3471 2.4511 2.2079
HT-55 GDSC2 4.9986 6.3934 2.8597 0.4386
NCI-H747 GDSC2 5.0452 7.3723 2.4885 1.9066
SNU-1040 GDSC2 5.121 6.4682 2.8808 0.3188
SK-CO-1 GDSC2 5.1365 6.9672 2.6985 0.8971
GP5d GDSC2 5.1552 6.6531 2.8266 0.4497
SNU-81 GDSC2 5.161 6.6928 2.8142 0.4832
LoVo GDSC2 5.2062 7.2787 2.6062 1.2041
DiFi GDSC2 5.2732 7.9424 2.3638 2.2283
SW620 GDSC2 5.3334 8.3216 2.2325 2.7993
HT115 GDSC2 5.3405 6.797 2.8469 0.3093
LS513 GDSC2 5.4077 7.0421 2.7841 0.439
NCI-H716 GDSC2 5.4741 7.6449 2.5827 1.0634
HCT 116 GDSC2 5.5082 7.2027 2.7651 0.4416
CaR-1 GDSC2 5.5405 7.172 2.7888 0.3663
SW1417 GDSC2 5.5431 7.2599 2.7579 0.444
SW948 GDSC2 5.5808 7.2858 2.7632 0.4127
LS180 GDSC2 5.6623 7.1366 2.8466 0.2028
SW837 GDSC2 5.6629 7.855 2.5838 0.9151
LS1034 GDSC2 5.6745 6.9945 2.8995 0.1189
MDST8 GDSC2 5.7329 7.0276 2.9086 0.098
SW1463 GDSC2 5.7893 7.9562 2.5987 0.7793
SNU-C1 GDSC2 5.7942 7.6828 2.7022 0.4729
COLO 678 GDSC2 5.8376 7.8702 2.6507 0.5925
CW-2 GDSC2 5.8716 7.8715 2.6638 0.5386
HCC2998 GDSC2 5.8901 14.1694 -0.1395 14.1437
SNU-407 GDSC2 5.8996 7.8459 2.6841 0.4715
T84 GDSC2 5.9125 7.8898 2.6732 0.4938
SNU-C2B GDSC2 6.2358 13.9647 0.1889 11.8964
COLO 320HSR GDSC2 6.2515 7.9278 2.785 0.1628
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC2 5.665 7.4027 2.7536 0.3999
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Hep 3B2.1-7 GDSC2 3.896 5.947 2.4516 4.0484
JHH-6 GDSC2 4.083 11.7155 -0.2587 18.9981
JHH-2 GDSC2 4.2678 6.4838 2.4426 3.3432
SNU-398 GDSC2 4.7003 7.7587 2.12 4.4086
Hep-G2/C3A GDSC2 4.7638 6.1677 2.8464 0.6385
JHH-1 GDSC2 4.8997 6.4151 2.8098 0.669
HuH-1 GDSC2 5.0656 6.533 2.8349 0.475
SNU-423 GDSC2 5.1074 14.1065 -0.6643 18.2295
HLE GDSC2 5.1675 13.284 -0.2173 16.0939
SK-HEP-1 GDSC2 5.4139 6.7304 2.8976 0.1804
Huh-7 GDSC2 5.678 7.3655 2.7719 0.3504
JHH-7 GDSC2 5.7677 7.9879 2.5776 0.8633
SNU-387 GDSC2 6.0187 16.8322 -1.3389 18.8996
SNU-449 GDSC2 6.6377 8.1713 2.8351 0.0603
JHH-4 GDSC2 6.9995 16.8046 -0.6561 14.2288
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 166 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H526 GDSC2 3.4263 6.977 1.5806 10.6935
SBC-3 GDSC2 3.4632 5.5935 2.3016 6.0605
HCC44 GDSC2 3.6809 5.5605 2.4859 4.3363
COR-L303 GDSC2 3.6978 11.5334 -0.4749 21.0514
NCI-H1793 GDSC2 3.8035 5.7761 2.4694 4.1483
IST-SL2 GDSC2 3.8776 6.795 2.0239 6.7325
RERF-LC-KJ GDSC2 4.053 6.8885 2.105 5.818
NCI-H2171 GDSC2 4.1293 6.4551 2.3663 4.066
DMS 53 GDSC2 4.1335 6.3688 2.4102 3.7953
NCI-H2170 GDSC2 4.1683 6.4545 2.3924 3.8313
UMC-11 GDSC2 4.1882 8.14 1.5911 8.6388
SHP-77 GDSC2 4.2575 7.3908 2.0046 5.9745
NCI-H345 GDSC2 4.2719 4.9627 3.0964 0.1501
Ms-1 GDSC2 4.2833 6.7327 2.3358 3.939
IA-LM GDSC2 4.2886 9.1152 1.1861 10.8072
NCI-H810 GDSC2 4.3176 7.5128 1.987 5.9502
NCI-H720 GDSC2 4.3563 6.0543 2.6911 1.8059
Lu-165 GDSC2 4.3636 6.9408 2.2895 4.0554
NCI-H82 GDSC2 4.3745 5.8983 2.7691 1.3793
NCI-H1092 GDSC2 4.3881 6.4787 2.5187 2.6948
NCI-H838 GDSC2 4.4067 8.6181 1.5144 8.5887
NCI-H358 GDSC2 4.4193 6.7899 2.3948 3.3418
BEN GDSC2 4.4226 11.8667 -0.0714 17.2167
NCI-H2227 GDSC2 4.4281 8.4607 1.6058 7.9957
EMC-BAC-2 GDSC2 4.4301 13.0267 -0.6407 19.7959
NCI-H2081 GDSC2 4.435 6.5914 2.4952 2.7471
NCI-H446 GDSC2 4.4376 7.397 2.1223 4.8945
NCI-H522 GDSC2 4.4381 10.5309 0.6001 13.7402
NCI-H2030 GDSC2 4.4457 7.02 2.3045 3.813
NCI-H2023 GDSC2 4.4579 7.1371 2.2575 4.0625
NCI-H2369 GDSC2 4.4885 9.2595 1.2603 9.8981
NCI-H1755 GDSC2 4.4971 13.0642 -0.6078 19.4822
EPLC-272H GDSC2 4.551 8.9937 1.4336 8.7406
Lu-134-A GDSC2 4.561 7.5056 2.1506 4.4898
SBC-1 GDSC2 4.5748 6.2933 2.7047 1.4409
NCI-H2029 GDSC2 4.5822 7.0284 2.3839 3.1211
NCI-H2122 GDSC2 4.6132 8.3538 1.7837 6.5399
NCI-H596 GDSC2 4.6236 8.9259 1.5166 8.0923
NCI-H1048 GDSC2 4.6677 6.8962 2.4926 2.3948
NCI-H460 GDSC2 4.7236 6.63 2.6383 1.5785
COR-L311 GDSC2 4.7266 6.7091 2.6061 1.732
NCI-H1915 GDSC2 4.7559 7.2041 2.4055 2.7257
NCI-H196 GDSC2 4.7664 6.8071 2.5849 1.7853
EBC-1 GDSC2 4.8759 7.7381 2.2351 3.4612
NCI-H1666 GDSC2 4.88 11.2451 0.5718 12.8317
NCI-H290 GDSC2 4.9143 7.5788 2.3284 2.8978
NCI-H1563 GDSC2 4.9184 8.0892 2.1008 4.1335
RERF-LC-MS GDSC2 4.9273 9.6823 1.3597 8.3553
SW1271 GDSC2 4.9327 8.0179 2.1418 3.8818
NCI-H1581 GDSC2 4.9336 10.8834 0.7856 11.5594
KNS-62 GDSC2 4.9366 7.7241 2.2763 3.1421
NCI-H1944 GDSC2 4.977 8.2374 2.0681 4.2162
LB647-SCLC GDSC2 4.9808 6.9544 2.6312 1.3201
HOP-92 GDSC2 4.9818 8.1759 2.099 4.0367
NCI-H3122 GDSC2 4.9823 7.6412 2.3387 2.7436
A-427 GDSC2 4.9843 11.7759 0.3875 13.5545
NCI-H2795 GDSC2 4.9988 18.4777 -2.9078 26.2312
COR-L23 GDSC2 5.0145 6.4336 2.8512 0.4552
NCI-H2110 GDSC2 5.0197 7.8123 2.2839 2.9764
LC-1/sq GDSC2 5.0315 12.9064 -0.131 16.0067
NCI-H1781 GDSC2 5.0542 6.802 2.7267 0.8568
NCI-H2444 GDSC2 5.058 6.2525 2.9341 0.2194
DMS 273 GDSC2 5.0717 16.6754 -1.9585 23.205
CPC-N GDSC2 5.0757 6.9655 2.6716 1.0559
NCI-H2087 GDSC2 5.0927 7.8634 2.3018 2.7774
VMRC-LCD GDSC2 5.0982 7.0654 2.6418 1.1575
NCI-H1155 GDSC2 5.1128 7.1817 2.6015 1.3145
NCI-H524 GDSC2 5.1171 6.848 2.7366 0.7707
NCI-H1869 GDSC2 5.1171 10.3945 1.1466 9.1654
HCC33 GDSC2 5.1264 11.6267 0.5603 12.3333
NCI-H1975 GDSC2 5.1489 7.2171 2.6042 1.2672
NCI-H211 GDSC2 5.1567 7.0485 2.6755 0.9693
CAL-12T GDSC2 5.1849 17.3601 -2.2115 23.7604
SK-MES-1 GDSC2 5.1969 7.5481 2.4913 1.7168
LOU-NH91 GDSC2 5.2165 6.9304 2.7476 0.6611
SBC-5 GDSC2 5.2376 6.0975 3.0492 0.0293
SW1573 GDSC2 5.2481 7.5254 2.5257 1.5069
NCI-H1963 GDSC2 5.2551 6.9922 2.7404 0.6597
NCI-H2591 GDSC2 5.2648 9.3714 1.7222 5.6467
ChaGo-K-1 GDSC2 5.2659 8.472 2.1296 3.4253
NCI-H2135 GDSC2 5.2784 6.9144 2.7794 0.5212
NCI-H1876 GDSC2 5.287 6.959 2.7662 0.5566
NCI-H250 GDSC2 5.2878 7.0707 2.7243 0.6918
NCI-H1836 GDSC2 5.3075 6.6716 2.8791 0.2493
DMS 79 GDSC2 5.3169 7.1321 2.7132 0.7097
NCI-H1792 GDSC2 5.3211 11.8625 0.581 11.7985
NCI-H292 GDSC2 5.3416 7.0799 2.7433 0.5953
NCI-H322M GDSC2 5.3469 10.7843 1.1133 8.8814
NCI-H1650 GDSC2 5.3608 7.4946 2.591 1.1264
NCI-H1770 GDSC2 5.3621 6.8902 2.8216 0.3619
NCI-H1437 GDSC2 5.3658 8.0529 2.3644 2.1135
NCI-H1651 GDSC2 5.3683 11.2597 0.9016 9.9927
NCI-H1734 GDSC2 5.3753 7.3641 2.6489 0.8942
NCI-H1623 GDSC2 5.3833 7.5134 2.5938 1.0963
NCI-H1993 GDSC2 5.3881 7.4174 2.6337 0.9401
NCI-H2196 GDSC2 5.3988 7.0191 2.7891 0.4299
NCI-H1105 GDSC2 5.4092 7.323 2.6794 0.7615
NCI-H2810 GDSC2 5.4099 11.9285 0.6098 11.4583
PC-14 GDSC2 5.4101 7.3202 2.6809 0.756
NCI-H513 GDSC2 5.4172 9.515 1.7483 5.2398
NCI-H650 GDSC2 5.4359 14.0069 -0.3777 16.2154
EKVX GDSC2 5.4671 8.7229 2.1302 3.1356
NCI-H841 GDSC2 5.468 7.5742 2.6077 0.9741
NCI-H2141 GDSC2 5.4846 7.2637 2.7331 0.5436
NCI-H2405 GDSC2 5.4979 8.3406 2.3101 2.2138
HOP-62 GDSC2 5.4984 7.671 2.5833 1.0416
NCI-H2818 GDSC2 5.5055 7.5979 2.6149 0.9192
Calu-3 GDSC2 5.5228 13.9201 -0.2739 15.5513
Lu-139 GDSC2 5.5382 7.1947 2.7797 0.3898
LK-2 GDSC2 5.5525 7.607 2.6317 0.8262
NCI-H226 GDSC2 5.5538 14.6168 -0.5909 16.8919
COR-L321 GDSC2 5.556 6.9499 2.8729 0.1854
NCI-H2461 GDSC2 5.5693 10.6901 1.2999 7.4301
SK-LU-1 GDSC2 5.5714 8.1122 2.4406 1.5501
NCI-H1436 GDSC2 5.5967 6.9551 2.8857 0.1546
NCI-H146 GDSC2 5.6021 7.3253 2.7572 0.4185
NCI-H2595 GDSC2 5.6232 7.8108 2.5836 0.9443
LC-2/ad GDSC2 5.6281 7.7693 2.6018 0.8768
IST-SL1 GDSC2 5.6596 7.1519 2.8404 0.2147
NCI-H740 GDSC2 5.6721 13.0035 0.272 12.6266
HCC15 GDSC2 5.688 8.0347 2.5249 1.1098
NCI-H1435 GDSC2 5.7071 7.3531 2.7873 0.3051
A-549 GDSC2 5.718 22.3526 -4.2778 28.0264
HCC78 GDSC2 5.7199 13.5493 0.0424 13.6449
Lu-65 GDSC2 5.7256 7.8027 2.6302 0.7183
NCI-H1694 GDSC2 5.7333 7.3956 2.7821 0.3071
COR-L32 GDSC2 5.778 7.861 2.6299 0.6876
EMC-BAC-1 GDSC2 5.778 9.3864 2.0092 3.3242
NCI-H3255 GDSC2 5.7843 7.7131 2.6873 0.5174
NCI-H2731 GDSC2 5.7859 8.0269 2.5704 0.8754
HARA [Human squamous cell lung carcinoma] GDSC2 5.788 9.0557 2.1558 2.5987
NCI-H748 GDSC2 5.8379 7.9094 2.6363 0.6343
NCI-H1693 GDSC2 5.8747 7.8406 2.6763 0.5033
NCI-H647 GDSC2 5.8977 7.858 2.679 0.4857
NCI-H2172 GDSC2 5.9121 8.3261 2.5096 0.9969
NCI-H2291 GDSC2 5.9171 7.9932 2.6372 0.5895
ABC-1 GDSC2 5.9172 8.952 2.2629 1.9684
NCI-H2373 GDSC2 5.9258 7.5351 2.8039 0.2071
NCI-H510A GDSC2 5.9376 7.7099 2.7472 0.3101
HCC827 GDSC2 5.9395 7.9182 2.6734 0.4809
COLO 668 GDSC2 5.9607 8.0015 2.6514 0.5286
DMS 114 GDSC2 5.9684 7.2829 2.9037 0.0715
Lu-99A GDSC2 5.9821 8.1757 2.5958 0.6744
Lu-135 GDSC2 5.9915 7.7835 2.7413 0.3044
NCI-H661 GDSC2 6.0051 7.8444 2.7249 0.3339
NCI-H2803 GDSC2 6.0278 7.7438 2.7685 0.2414
NCI-H23 GDSC2 6.0423 7.8914 2.7222 0.3268
LCLC-97TM1 GDSC2 6.0693 9.1599 2.2506 1.8702
RERF-LC-Sq1 GDSC2 6.1123 10.4064 1.746 4.1875
NCI-H2869 GDSC2 6.1154 9.2953 2.2174 1.9659
NCI-H2228 GDSC2 6.1211 9.0917 2.3022 1.6104
NCI-H209 GDSC2 6.1323 8.0324 2.7059 0.3301
Calu-6 GDSC2 6.1383 7.6633 2.8349 0.1194
NCI-H727 GDSC2 6.1453 9.264 2.2442 1.8248
NCI-H2804 GDSC2 6.168 8.838 2.4226 1.1189
NCI-H2722 GDSC2 6.2105 8.1049 2.7093 0.2983
COR-L105 GDSC2 6.3248 18.6497 -2.0064 20.6252
NCI-H520 GDSC2 6.3504 14.8769 -0.1684 13.3443
NCI-H2085 GDSC2 6.382 8.5716 2.6083 0.4535
LCLC-103H GDSC2 6.4735 15.1174 -0.2015 13.2544
NCI-H441 GDSC2 6.6103 18.809 -1.8818 19.6289
NCI-H1568 GDSC2 6.6335 16.9487 -0.9683 16.204
HCC366 GDSC2 6.694 17.667 -1.2721 17.2678
LXF 289 GDSC2 7.0358 19.5437 -1.9413 19.0022
NCI-H1355 GDSC2 7.0742 18.9993 -1.6531 17.931
NCI-H1299 GDSC2 7.1048 16.0698 -0.2427 12.265
⏷ Show the Full List of 166 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC2 3.9292 6.5069 2.2028 5.5019
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OE19 GDSC2 4.0566 5.6381 2.7038 2.2226
TE-5 GDSC2 4.5199 7.5147 2.1201 4.7463
EC-GI-10 GDSC2 4.6216 6.9642 2.436 2.7697
TE-8 GDSC2 4.7646 9.2014 1.4802 8.0023
KYSE-140 GDSC2 4.846 7.653 2.2561 3.3944
OE33 GDSC2 5.1047 8.0209 2.2392 3.0868
TE-10 GDSC2 5.2496 7.2337 2.6441 1.013
TE-11 GDSC2 5.3377 11.9505 0.55 11.9245
TE-4 GDSC2 5.4244 7.113 2.7647 0.4845
KYSE-450 GDSC2 5.4856 15.2037 -0.9265 18.4521
OE21 GDSC2 5.6545 7.5821 2.6837 0.5958
COLO 680N GDSC2 5.6613 7.6586 2.6578 0.6704
TE-9 GDSC2 5.7319 7.0538 2.8994 0.109
KYSE-180 GDSC2 5.7692 7.9894 2.5777 0.8622
TE-15 GDSC2 5.8699 10.3824 1.621 5.1886
TE-6 GDSC2 5.8717 7.7226 2.7178 0.4001
TE-1 GDSC2 5.9067 7.5263 2.8 0.2186
KYSE-70 GDSC2 5.9114 14.2103 -0.1447 14.1233
KYSE-520 GDSC2 6.0126 13.5719 0.2286 12.1439
KYSE-270 GDSC2 6.4292 8.4471 2.6699 0.3076
KYSE-410 GDSC2 7.9728 23.5574 -3.2311 21.2259
KYSE-510 GDSC2 8.4426 19.3459 -0.9313 12.8506
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 25 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TOV-112D GDSC2 3.724 5.9919 2.3054 5.3572
OAW42 GDSC2 4.0696 6.8505 2.1352 5.5955
TOV-21G GDSC2 4.1252 6.2748 2.4493 3.5797
OVCAR-8 GDSC2 4.2031 6.3688 2.4554 3.3912
A2780 GDSC2 4.2528 6.5843 2.386 3.7028
DOV13 GDSC2 4.4629 6.2445 2.6663 1.7819
JHOS-2 GDSC2 4.5133 6.0475 2.7773 1.169
OV56 GDSC2 4.628 7.3634 2.2581 3.7499
OV-90 GDSC2 4.7264 8.3536 1.8582 5.8747
JHOS-4 GDSC2 4.7614 8.9662 1.5905 7.3667
TYK-nu GDSC2 4.7947 7.0677 2.4873 2.2398
OVISE GDSC2 4.9184 6.1112 2.9315 0.2804
Kuramochi GDSC2 5.3791 14.2495 -0.5368 17.0491
Caov-3 GDSC2 5.4017 6.9725 2.8072 0.3809
ES-2 GDSC2 5.4204 6.9653 2.817 0.348
OVCAR-4 GDSC2 5.4389 10.1006 1.4923 6.6109
EFO-21 GDSC2 5.5184 11.9152 0.6892 10.8158
OAW28 GDSC2 5.5916 11.4752 0.9461 9.3046
IGROV-1 GDSC2 5.7366 7.7882 2.6402 0.6804
OVTOKO GDSC2 5.7466 14.571 -0.4324 15.7763
OVCAR-3 GDSC2 5.7724 7.8456 2.6334 0.6804
SK-OV-3 GDSC2 5.939 7.32 2.8814 0.0973
OVK18 GDSC2 6.1201 7.7639 2.7945 0.1762
OVCAR-5 GDSC2 7.3891 23.8374 -3.7756 23.6786
EFO-27 GDSC2 7.8795 21.4153 -2.2664 18.5276
⏷ Show the Full List of 25 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 27 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PaTu 8988t GDSC2 4.0628 6.3676 2.3636 4.2214
SUIT-2 GDSC2 4.2707 6.2419 2.5565 2.6835
PaTu 8902 GDSC2 4.3438 6.4185 2.5196 2.7651
YAPC GDSC2 4.4243 6.7948 2.3956 3.3281
MIA PaCa-2 GDSC2 4.4888 6.3776 2.622 1.9754
DAN-G GDSC2 4.5891 8.2533 1.8155 6.4017
HPAC GDSC2 4.6789 7.6269 2.1678 4.1738
QGP-1 GDSC2 4.6907 10.6281 0.7372 12.3829
Capan-2 GDSC2 4.8006 7.4928 2.3019 3.2166
KP-2 GDSC2 4.9228 7.0355 2.5685 1.6719
Panc 08.13 GDSC2 4.9922 12.3305 0.1224 14.8743
HuP-T4 GDSC2 4.9927 8.6636 1.8818 5.236
HuP-T3 GDSC2 5.0669 10.8658 0.8866 10.7123
AsPC-1 GDSC2 5.1553 7.8279 2.3511 2.4414
SU.86.86 GDSC2 5.3306 6.5891 2.9164 0.1698
CFPAC-1 GDSC2 5.5193 7.0634 2.8196 0.3027
KP-3 GDSC2 5.7236 8.3408 2.4195 1.4938
PSN1 GDSC2 5.7341 7.386 2.7858 0.2989
Panc 10.05 GDSC2 5.7613 15.3291 -0.7901 17.2808
KP-1N GDSC2 5.7758 8.3066 2.4571 1.2973
PL4 GDSC2 5.7785 7.638 2.7124 0.4537
KP-4 GDSC2 5.8537 7.165 2.904 0.0855
HPAF-II GDSC2 5.9659 8.2917 2.5456 0.8397
BxPC-3 GDSC2 6.1204 8.709 2.4518 1.0508
Capan-1 GDSC2 6.2911 7.9707 2.7843 0.1562
MZ-PC-1 GDSC2 6.4332 8.6112 2.6136 0.422
Panc 02.03 GDSC2 7.4198 20.62 -2.1962 19.1272
⏷ Show the Full List of 27 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MPP 89 GDSC2 4.1601 8.4591 1.414 9.7722
NCI-H2052 GDSC2 4.6932 10.3095 0.8946 11.5086
NCI-H28 GDSC2 5.5605 14.809 -0.6797 17.2581
MSTO-211H GDSC2 5.992 8.1835 2.5969 0.6656
IST-Mes1 GDSC2 6.1481 17.3147 -1.482 19.1582
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
VCaP GDSC2 4.0157 8.899 1.0884 12.0652
22Rv1 GDSC2 4.1708 7.2215 2.0263 6.0335
LNCaP clone FGC GDSC2 4.2165 6.9352 2.1955 4.9102
NCI-H660 GDSC2 5.068 6.7376 2.758 0.7301
DU145 GDSC2 5.8432 7.7586 2.6938 0.4721
PC-3 GDSC2 6.109 8.4012 2.5634 0.6998
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 GDSC2 5.5596 8.8734 2.1146 3.0889
Cancer Drug Sensitivity Data Curated from 54 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-MEL-2 GDSC2 3.6339 5.7741 2.3452 5.3342
UACC-62 GDSC2 3.7243 5.1608 2.7124 2.8342
G-mel GDSC2 3.9545 5.8025 2.561 3.2593
A2058 GDSC2 4.0438 15.3273 -2.0903 26.1649
HT-144 GDSC2 4.076 9.2032 0.9836 12.5165
Hs 940.T GDSC2 4.1039 6.7389 2.2131 5.0448
LB2518-MEL GDSC2 4.1477 6.2242 2.4878 3.3076
WM115 GDSC2 4.2639 6.8234 2.2803 4.3055
IGR-37 GDSC2 4.2918 8.0607 1.7041 7.7144
A101D GDSC2 4.294 7.0917 2.1726 4.8865
G-361 GDSC2 4.3077 12.8048 -0.6251 20.0464
RVH-421 GDSC2 4.3219 8.4525 1.5347 8.6634
SK-MEL-31 GDSC2 4.3253 31.0511 -9.7156 38.0958
MZ-MEL-7 GDSC2 4.3661 6.7239 2.3924 3.452
RPMI-7951 GDSC2 4.3784 8.6613 1.4732 8.8991
COLO 783 GDSC2 4.3796 9.6803 0.9753 11.8012
M14 GDSC2 4.4557 6.6793 2.4676 2.8667
COLO 792 GDSC2 4.484 7.736 1.992 5.5725
SK-MEL-30 GDSC2 4.5842 6.6628 2.5492 2.2188
A-431 GDSC2 4.5964 8.3773 1.7612 6.7075
CP50-MEL-B GDSC2 4.7258 6.9899 2.4836 2.357
LB373-MEL-D GDSC2 4.8025 6.2114 2.8464 0.6095
A-375 GDSC2 4.8358 10.9399 0.689 12.306
WT2-iPS GDSC2 4.8817 6.2553 2.8633 0.4974
Hs 938.T GDSC2 5.0012 6.5858 2.7877 0.673
CHL-1 GDSC2 5.0075 7.0846 2.5904 1.4742
COLO 800 GDSC2 5.0968 7.2731 2.5561 1.532
451Lu GDSC2 5.1265 7.1355 2.6268 1.1936
IGR-1 GDSC2 5.1443 6.8578 2.7446 0.7219
HMV-II GDSC2 5.2067 9.9287 1.4262 7.415
SK-MEL-28 GDSC2 5.2586 20.2597 -3.5921 27.4128
IPC-298 GDSC2 5.2805 19.2047 -3.0521 25.9911
GAK GDSC2 5.2859 6.7701 2.8355 0.3606
MMAc-SF GDSC2 5.3013 6.8582 2.8094 0.4224
COLO 679 GDSC2 5.304 6.8973 2.7961 0.4582
SK-MEL-3 GDSC2 5.3176 6.907 2.798 0.4459
CP66-MEL GDSC2 5.3201 6.7534 2.8547 0.2991
Mel JuSo GDSC2 5.3353 6.5502 2.9315 0.1436
VMRC-MELG GDSC2 5.3471 6.6347 2.9066 0.1827
SK-MEL-5 GDSC2 5.3518 6.8764 2.8226 0.3638
WM793 GDSC2 5.3913 7.2042 2.7171 0.6481
Mel Ho GDSC2 5.3913 6.9829 2.7993 0.4062
DJM-1 GDSC2 5.4132 13.1514 0.0221 14.4055
WM1552C GDSC2 5.4707 7.7068 2.5567 1.1671
UACC-257 GDSC2 5.5441 6.7992 2.9202 0.116
MZ-MEL-2 GDSC2 5.6762 19.1097 -2.7061 24.1657
WM35 GDSC2 5.6769 8.3788 2.3822 1.6954
COLO 829 GDSC2 5.8627 7.6709 2.733 0.3684
WM278 GDSC2 5.8634 17.1109 -1.5863 20.1413
SH-4 GDSC2 5.9272 7.9622 2.6526 0.5418
A-388 GDSC2 5.9364 8.023 2.6339 0.5887
SK-MEL-24 GDSC2 5.9697 15.0148 -0.492 15.5637
LOX-IMVI GDSC2 6.0169 7.9555 2.6898 0.4079
EquiPSC Line K2 GDSC2 3.9969 10.3335 0.3616 16.1565
⏷ Show the Full List of 54 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC2 4.3218 6.6243 2.411 3.4256
Cancer Drug Sensitivity Data Curated from 20 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Rh41 GDSC2 3.8967 6.7014 2.084 6.3138
SW684 GDSC2 4.0922 6.6247 2.26 4.7855
SW982 GDSC2 4.1612 12.1571 -0.4172 19.515
SK-UT-1 GDSC2 4.2148 7.5804 1.8831 6.8057
G-401 GDSC2 4.2493 12.0385 -0.2897 18.6986
KYM-1 GDSC2 4.287 7.4274 2.0071 5.8949
STS-0421 GDSC2 4.4063 8.1145 1.7581 7.1334
HT-1080 GDSC2 4.4467 6.8517 2.3831 3.3596
G-402 GDSC2 4.4689 7.2419 2.2155 4.2865
GCT GDSC2 4.5441 14.027 -1.0493 21.194
RKN GDSC2 4.9239 6.2719 2.8745 0.4364
MES-SA GDSC2 5.2396 6.7794 2.8138 0.4416
TE 441.T GDSC2 5.249 6.5912 2.8856 0.256
SW872 GDSC2 5.2766 7.3936 2.5927 1.1947
VA-ES-BJ GDSC2 5.3575 14.5466 -0.6977 17.7919
SK-LMS-1 GDSC2 5.4529 11.3858 0.8977 9.8414
Rh30 GDSC2 5.4879 7.3472 2.7033 0.6326
EW-8 GDSC2 5.7 7.2888 2.8073 0.2658
RD GDSC2 6.0837 11.8126 1.0978 7.5908
A-204 GDSC2 6.4838 8.6071 2.6339 0.3611
⏷ Show the Full List of 20 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 25 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-5 GDSC2 3.6452 7.307 1.592 10.0141
NUGC-4 GDSC2 3.8231 6.4788 2.1392 6.1494
MKN1 GDSC2 4.0054 7.1577 1.9395 6.946
MKN45 GDSC2 4.0898 5.585 2.7482 1.9142
GCIY GDSC2 4.2726 6.5723 2.4043 3.5575
KATO III GDSC2 4.3349 6.514 2.4703 3.0608
23132/87 GDSC2 4.5549 11.1663 0.3739 14.6507
AGS GDSC2 4.8341 11.5212 0.404 13.8196
Hs 746.T GDSC2 4.865 8.3198 1.962 5.0122
OCUM-1 GDSC2 5.033 11.0679 0.7656 11.4453
RF-48 GDSC2 5.0429 7.7372 2.3298 2.7032
SCH GDSC2 5.1422 6.4336 2.9014 0.2607
IM95 GDSC2 5.2178 8.4364 2.1185 3.5563
NCI-N87 GDSC2 5.2879 7.9067 2.3865 2.1015
RERF-GC-1B GDSC2 5.4079 14.9014 -0.8348 18.2516
ECC12 GDSC2 5.4334 6.6242 2.9408 0.1094
MKN28 GDSC2 5.5756 10.6901 1.3038 7.3971
ECC10 GDSC2 5.6233 7.358 2.7536 0.4181
TMK-1 GDSC2 5.6274 7.4415 2.7248 0.4926
SK-GT-2 GDSC2 5.7576 8.3901 2.4155 1.4792
NUGC-3 GDSC2 5.8851 7.4213 2.8284 0.1772
SNU-1 GDSC2 5.8971 7.6574 2.7507 0.3167
MKN7 GDSC2 6.0288 12.7603 0.6229 10.1478
HGC-27 GDSC2 6.1544 7.5752 2.8697 0.0808
SNG-M GDSC2 5.7065 7.7423 2.645 0.6832
⏷ Show the Full List of 25 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
8305C GDSC2 3.8061 5.5323 2.5896 3.4041
K5 GDSC2 4.3874 7.2285 2.1692 4.7171
ASH-3 GDSC2 4.5947 6.2213 2.7453 1.2247
KMH-2 GDSC2 4.8862 8.8503 1.7273 6.3206
WRO GDSC2 5.0378 10.1053 1.2316 8.853
IHH-4 GDSC2 5.143 6.6629 2.818 0.4819
CAL-62 GDSC2 5.2023 6.621 2.8571 0.3429
FTC-133 GDSC2 5.3261 8.662 2.0792 3.6014
BHT-101 GDSC2 5.3429 14.4727 -0.6721 17.7161
B-CPAP GDSC2 5.3821 13.6828 -0.2581 15.793
HTC-C3 GDSC2 5.8082 8.0401 2.5748 0.8456
TT2609-C02 GDSC2 5.9029 14.8786 -0.4725 15.6187
ML-1 [Human leukemia] GDSC2 5.9887 16.5733 -1.2342 18.5658
8505C GDSC2 6.8484 17.5146 -1.0942 16.2827
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 38 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DOK GDSC2 3.5823 8.7267 0.8333 14.7199
Detroit 562 GDSC2 3.806 7.2393 1.7506 8.6075
HO-1-N-1 GDSC2 4.113 6.3361 2.4121 3.8254
BB30-HNC GDSC2 4.4046 8.649 1.4979 8.6919
OSC-19 GDSC2 4.4063 6.5197 2.5109 2.7079
UPCI-SCC-090 GDSC2 4.4152 18.2223 -3.2379 28.4494
HSC-2 GDSC2 4.4822 6.7743 2.4401 2.9755
BICR 31 GDSC2 4.4897 14.8196 -1.485 22.9808
JHU-029 GDSC2 4.5001 7.1784 2.2648 3.9418
KOSC-2 GDSC2 4.6561 8.1912 1.8892 5.8325
SAS GDSC2 4.6648 9.8965 1.0754 10.5559
JHU-022 GDSC2 4.7006 8.4247 1.8077 6.2206
BB49-HNC GDSC2 4.7348 12.9638 -0.3782 17.8667
LB771-HNC GDSC2 4.7658 10.6316 0.7893 11.9221
Ca9-22 GDSC2 4.7769 7.4995 2.285 3.3477
PCI-06A GDSC2 4.8498 11.5984 0.3776 13.9194
SAT [Human HNSCC] GDSC2 4.878 9.5539 1.388 8.2963
SCC-4 GDSC2 5.0519 9.4327 1.56 6.9581
SKN-3 GDSC2 5.0584 10.8469 0.8899 10.7126
KON GDSC2 5.1058 12.6072 0.0689 14.8733
CAL-27 GDSC2 5.1489 6.7383 2.7922 0.5587
HSC-3 GDSC2 5.149 9.3416 1.6643 6.1808
HSC-4 GDSC2 5.2021 6.4678 2.9117 0.2169
BICR 22 GDSC2 5.2484 6.8425 2.794 0.4945
SCC-9 GDSC2 5.2678 10.7716 1.0673 9.2947
PE/CA-PJ15 GDSC2 5.4183 8.7339 2.0987 3.3652
PCI-15A GDSC2 5.4668 7.0722 2.7963 0.3793
PCI-04B GDSC2 5.5172 7.5595 2.6349 0.84
OSC-20 GDSC2 5.5656 7.6626 2.616 0.8716
CAL-33 GDSC2 5.6748 7.6109 2.6811 0.5921
SCC-15 GDSC2 5.7811 7.3773 2.8062 0.2429
SCC-25 GDSC2 5.8865 7.5786 2.7745 0.2718
JHU-011 GDSC2 5.9294 17.4716 -1.7151 20.4565
BICR 78 GDSC2 6.2107 8.3249 2.6314 0.4681
NCI-H3118 GDSC2 6.2713 8.5736 2.5647 0.6118
BHY GDSC2 6.4241 8.502 2.6488 0.3504
FaDu GDSC2 6.6028 15.7321 -0.408 13.922
BICR 10 GDSC2 6.8247 20.0386 -2.3277 20.6712
⏷ Show the Full List of 38 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
BFTC-905 GDSC2 3.6249 5.7527 2.3489 5.334
639V GDSC2 4.2456 5.7899 2.7461 1.6787
J82 GDSC2 4.4819 8.2631 1.7385 7.0858
KU-19-19 GDSC2 4.789 14.0087 -0.8535 19.7912
SW1710 GDSC2 4.8097 7.2978 2.3942 2.7049
647V GDSC2 4.9565 6.2432 2.8983 0.3499
HT-1197 GDSC2 4.9941 6.9658 2.6329 1.2985
RT-4 GDSC2 5.266 9.2869 1.7618 5.4241
SW780 GDSC2 5.4541 16.5713 -1.6207 21.1668
TCCSUP GDSC2 5.6242 7.293 2.7774 0.3592
RT-112 GDSC2 5.6467 7.5273 2.7008 0.55
CAL-29 GDSC2 5.7186 7.2955 2.8119 0.2508
T24 GDSC2 5.7672 7.5588 2.7367 0.398
5637 GDSC2 5.824 7.7424 2.6922 0.4852
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 36 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PA-1 GDSC2 3.2625 4.8284 2.5187 5.2611
NEC8 GDSC2 3.8826 6.379 2.2318 5.4321
CAL-39 GDSC2 3.9212 6.6806 2.1121 6.0812
OV17R GDSC2 3.9799 6.9115 2.0416 6.3773
TC-YIK GDSC2 4.1999 6.2994 2.4858 3.219
SW954 GDSC2 4.2207 7.357 1.9955 6.1103
JEG-3 GDSC2 4.3255 7.4567 2.0193 5.7395
DSH1 GDSC2 4.4456 9.435 1.1438 10.6754
LB831-BLC GDSC2 4.4932 7.6403 2.0435 5.2491
DoTc2 4510 GDSC2 4.5967 6.9845 2.4123 2.9397
JHOS-3 GDSC2 4.6459 11.271 0.3895 14.3461
SKN GDSC2 4.6511 8.7026 1.6425 7.2928
ME-180 GDSC2 4.6593 8.667 1.665 7.1429
MS751 GDSC2 4.8901 12.5257 -0.0475 15.9442
Ca Ski GDSC2 4.97 7.5625 2.3665 2.6167
HT-3 GDSC2 5.0031 7.6076 2.3648 2.5788
SW756 GDSC2 5.0115 7.6792 2.3381 2.705
BPH-1 GDSC2 5.0297 17.3713 -2.3352 24.5028
HEC-1 GDSC2 5.0342 6.8784 2.6873 1.0296
PWR-1E GDSC2 5.0675 10.257 1.1791 9.0865
PEO1 GDSC2 5.139 9.9508 1.372 7.8537
OVMIU GDSC2 5.1902 10.2917 1.244 8.4707
HeLa GDSC2 5.2611 12.4233 0.2685 13.5321
OVCA420 GDSC2 5.2658 7.4695 2.557 1.3537
SiSo GDSC2 5.3593 7.965 2.3981 1.9633
OVCA433 GDSC2 5.4105 15.7184 -1.2336 19.8355
C-4-I GDSC2 5.4941 7.0292 2.8222 0.3062
OMC-1 [Human cervical carcinoma] GDSC2 5.6589 7.43 2.7413 0.4336
ACC-OV7 GDSC2 5.7666 9.9275 1.7653 4.5898
SW962 GDSC2 5.8008 7.6688 2.7099 0.45
JAR GDSC2 5.8364 7.3022 2.8518 0.1527
C-33 A GDSC2 5.8549 7.5697 2.7659 0.2993
HEY GDSC2 6.0167 7.9736 2.6832 0.4235
SKG-IIIa GDSC2 6.1799 18.1054 -1.8445 20.3771
UWB1.289 GDSC2 6.2215 8.8208 2.452 0.9814
SiHa GDSC2 6.3543 19.0899 -2.2 21.1989
⏷ Show the Full List of 36 Cancer Drug Sensitivity Data of This Drug

References

1 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 7034).
2 Targeting bromodomains: epigenetic readers of lysine acetylation.Nat Rev Drug Discov.2014 May;13(5):337-56.