General Information of Drug (ID: DM3BHN1)

Drug Name
Etomoxir
Synonyms
ETOMOXIR; 82258-36-4; rac- Etomoxir; Etomoxirum [Latin]; Ethyl 2-(6-(4-chlorophenoxy)hexyl)oxirane-2-carboxylate; BRN 4496620; Oxiranecarboxylic acid, 2-(6-(4-chlorophenoxy)hexyl)-, ethyl ester; B 807-54; Ethyl 2-(6-(4-chlorophenoxy)hexyl)oxiranecarboxylate; Oxiranecarboxylic acid, 2-[6-(4-chlorophenoxy)hexyl]-, ethyl ester- [CAS]; Etomoxirum; etomoxir[inn]; SMR000449321; Rac-Etomoxir Ethyl Ester; C17H23ClO4; ethyl 2-[6-(4-chlorophenoxy)hexyl]oxirane-2-carboxylate; etoxomir; AC1L3XCY; MLS001424024; MLS000758228; SCHEMBL681359
Indication
Disease Entry ICD 11 Status REF
Heart failure BD10-BD13 Terminated [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 1 Molecular Weight (mw) 326.8
Logarithm of the Partition Coefficient (xlogp) 4.3
Rotatable Bond Count (rotbonds) 11
Hydrogen Bond Donor Count (hbonddonor) 0
Hydrogen Bond Acceptor Count (hbondacc) 4
Chemical Identifiers
Formula
C17H23ClO4
IUPAC Name
ethyl (2R)-2-[6-(4-chlorophenoxy)hexyl]oxirane-2-carboxylate
Canonical SMILES
CCOC(=O)[C@]1(CO1)CCCCCCOC2=CC=C(C=C2)Cl
InChI
InChI=1S/C17H23ClO4/c1-2-20-16(19)17(13-22-17)11-5-3-4-6-12-21-15-9-7-14(18)8-10-15/h7-10H,2-6,11-13H2,1H3/t17-/m1/s1
InChIKey
DZLOHEOHWICNIL-QGZVFWFLSA-N
Cross-matching ID
PubChem CID
9840324
ChEBI ID
CHEBI:95011
CAS Number
124083-20-1
TTD ID
D00UEQ

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Carnitine O-palmitoyltransferase I (CPT1B) TTDL0NY CPT1B_HUMAN Modulator [1]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 149 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 7.5472 9.7881 6.8276 7.3456
MEC1 CTRP2 8.3393 9.7464 7.56 2.6025
JM1 CTRP2 8.4207 12.4706 6.2656 7.8782
MV4-11 CTRP2 6.1594 10.5929 5.0685 17.8668
DEL CTRP2 6.3889 8.6645 6.087 13.3235
Peer CTRP2 6.5121 8.594 6.2443 12.3799
SU-DHL-1 CTRP2 6.9226 9.4791 6.3394 10.8755
THP-1 CTRP2; CTRP1 7.0347 9.8056 6.3105 10.6989
KMS-34 CTRP2 7.0611 8.1967 6.963 8.1139
Ku812 CTRP2; CTRP1 7.1268 10.9899 5.8489 12.3394
NCO2 CTRP2 7.2864 12.5478 5.2412 14.4454
KMS-12-BM CTRP2 7.4224 8.6253 7.2158 6.1195
BL-70 CTRP2; CTRP1 7.4295 8.5435 7.2541 5.9541
EoL-1 CTRP2 7.4677 12.0316 5.661 12.3321
EM-2 CTRP2 7.4977 9.9305 6.712 7.9353
KMS-21-BM CTRP2 7.5137 20.9499 1.263 26.9176
NALM-6 CTRP2 7.559 10.5717 6.4611 8.8243
KE-37 CTRP2 7.5807 8.759 7.3296 5.2463
P12-Ichikawa CTRP2 7.5914 9.7175 6.9039 6.9284
JURL-MK1 CTRP2 7.6182 9.1992 7.1732 5.7703
Pfeiffer CTRP2 7.6639 8.2409 7.609 3.9523
KMS-18 CTRP2 7.6733 9.724 6.9795 6.4259
EB1 CTRP2 7.6882 8.9123 7.374 4.7895
L-1236 CTRP2 7.7068 10.7183 6.5261 8.2246
697 CTRP2 7.723 8.5369 7.5702 3.9274
GA-10 CTRP2 7.7249 8.3943 7.6263 3.7085
SUP-M2 CTRP2 7.7252 8.2441 7.675 3.5277
Ri-1 CTRP2 7.7255 10.874 6.4665 8.4313
KMS-27 CTRP2 7.7534 11.3272 6.2676 9.1994
JVM-3 CTRP2 7.7642 10.2638 6.8022 6.9513
DB CTRP2 7.7649 8.9313 7.4428 4.3197
Daudi CTRP2 7.7677 9.1241 7.3562 4.6623
A3/Kawakami CTRP2 7.7709 8.189 7.7394 3.1568
KMS-26 CTRP2 7.788 8.6795 7.5787 3.7193
Mono-Mac-1 CTRP2 7.804 10.3119 6.8151 6.8101
SKM-1 CTRP2; CTRP1 7.8072 11.2004 6.3785 8.6225
L-540 CTRP2 7.8362 9.42 7.2811 4.8079
MOLT-3 CTRP2 7.8434 8.7138 7.6204 3.4104
SUP-HD1 CTRP2 7.8511 9.1129 7.4428 4.1092
HD-MY-Z CTRP2 7.8617 9.6345 7.2007 5.0817
MOLM-6 CTRP2 7.8705 11.2035 6.4333 8.2599
SUP-T11 CTRP2 7.9147 9.0419 7.5379 3.5699
LP-1 CTRP2; CTRP1 7.922 12.1298 6.0171 9.8908
Karpas-299 CTRP2 7.9489 9.7515 7.2232 4.7955
NB4 CTRP2 7.9592 9.084 7.56 3.3757
KMS-11 CTRP2; CTRP1 7.9594 13.0343 5.598 11.5522
SU-DHL-4 CTRP2; CTRP1 7.9852 12.3987 5.9376 10.0934
MOLM-13 CTRP2 7.9893 10.0271 7.1231 5.1268
SU-DHL-8 CTRP2 7.9923 8.972 7.6455 2.9474
MM1.S CTRP2 7.9996 10.6342 6.8302 6.3307
CA46 CTRP2 8.0115 9.4701 7.4189 3.8445
OCI-AML-2 CTRP2 8.0139 8.9399 7.6814 2.7501
BV-173 CTRP2 8.0227 9.333 7.4968 3.4961
P3HR-1 CTRP2; CTRP1 8.0302 9.0026 7.6661 2.776
JeKo-1 CTRP2 8.032 9.3627 7.4906 3.5016
TF-1 CTRP2 8.0509 9.0416 7.6661 2.7302
SUP-T1 CTRP2 8.0539 9.2476 7.5672 3.1349
KMS-28BM CTRP2 8.054 10.3183 7.035 5.3606
Mino CTRP2 8.0542 9.2693 7.5567 3.1782
Namalwa CTRP2 8.0645 9.0083 7.6949 2.5803
RCH-ACV CTRP2 8.0893 9.7919 7.3282 4.0601
CML-T1 CTRP2 8.1025 9.6447 7.413 3.6773
K-562 CTRP2 8.1263 9.48 7.5159 3.1977
RPMI-8226 CTRP2; CTRP1 8.1382 12.6142 5.9602 9.6941
NU-DUL-1 CTRP2; CTRP1 8.1485 9.7536 7.3986 3.6445
RS4;11 CTRP2 8.1538 11.5453 6.5077 7.3729
SU-DHL-6 CTRP2 8.1562 9.3344 7.6144 2.7236
MOLT-16 CTRP2 8.1585 10.4447 7.0617 5.0383
CMK CTRP2 8.1653 8.8227 7.8774 1.6028
SET-2 CTRP2 8.1726 9.6263 7.4827 3.2432
KHM-1B CTRP2 8.1934 14.9099 4.8587 14.0701
ST486 CTRP2 8.1996 12.0547 6.2914 8.1899
SR CTRP2 8.2087 10.0639 7.2945 3.9624
ME1 CTRP2 8.2099 10.0782 7.2883 3.9861
MC116 CTRP2; CTRP1 8.2185 8.9546 7.8573 1.5803
KM-H2 CTRP2 8.2187 11.9044 6.3826 7.7709
OCI-AML-3 CTRP2; CTRP1 8.219 10.4646 7.1027 4.7479
RL CTRP2 8.2206 9.4858 7.5934 2.6841
Reh CTRP2 8.2269 9.7376 7.4728 3.1784
OCI-Ly3 CTRP2 8.2463 9.9873 7.3641 3.5978
Raji CTRP2 8.2927 9.9571 7.4173 3.2864
ALL-SIL CTRP2 8.3096 12.865 5.9777 9.2889
A4/Fukuda CTRP2 8.3122 10.4934 7.1653 4.308
PF-382 CTRP2 8.3212 12.5904 6.1245 8.6548
Mono-Mac-6 CTRP2 8.3393 21.7345 1.5679 24.504
TALL-1 [Human adult T-ALL] CTRP2 8.3404 10.2414 7.3139 3.6321
PL21 CTRP2; CTRP1 8.3553 12.5137 6.1909 8.313
SU-DHL-10 CTRP2 8.426 9.8064 7.5977 2.2933
MOLT-13 CTRP2 8.4427 9.8683 7.5798 2.3396
KYO-1 CTRP2 8.4504 9.626 7.7051 1.807
Hs 611.T CTRP2 8.4733 10.8617 7.1102 4.2467
Ci-1 CTRP2 8.4862 10.0352 7.5301 2.4736
HPB-ALL CTRP2 8.5096 9.6506 7.7362 1.5858
HuNS1 CTRP2 8.5294 10.4527 7.3564 3.1234
OCI-M1 CTRP2 8.5499 10.1905 7.501 2.4903
HDLM-2 CTRP2 8.5913 11.5288 6.8704 5.0426
EJM CTRP2; CTRP1 8.6347 11.3008 7.0165 4.3599
MOTN-1 CTRP2 8.6407 10.7401 7.2977 3.1841
HEL 92.1.7 CTRP2 8.6442 10.4438 7.4456 2.5694
MHH-CALL-3 CTRP2 8.7143 11.1536 7.1486 3.6814
MHH-CALL-4 CTRP2 8.7508 11.0417 7.2301 3.2881
MOLP-8 CTRP2 8.7679 10.3625 7.5709 1.8799
RPMI-6666 CTRP2 8.7696 10.7019 7.4088 2.53
NU-DHL-1 CTRP2 8.7851 10.8836 7.3316 2.8205
MOLM-16 CTRP2; CTRP1 8.8143 14.681 5.4768 10.4247
EHEB CTRP2 8.8946 13.3449 6.2022 7.304
NOMO-1 CTRP2; CTRP1 8.9055 13.2211 6.2718 6.9979
Toledo CTRP2 8.9175 10.9773 7.3775 2.4448
HL-60 CTRP2 8.9581 10.4286 7.6609 1.2914
F-36P CTRP2 8.9678 12.0316 6.9026 4.2957
SIG-M5 CTRP2 8.9756 10.3254 7.7181 1.0619
KMS-20 CTRP2 9.0082 11.0555 7.4003 2.2322
Kasumi-1 CTRP2 9.0196 11.0084 7.4298 2.1016
SEM CTRP2 9.028 10.996 7.4411 2.047
SU-DHL-5 CTRP1 9.0282 10.4257 7.6864 2.2146
AMO1 CTRP2; CTRP1 9.1048 11.0777 7.4514 1.9115
Karpas-422 CTRP2 9.1818 10.9818 7.5421 1.4824
JJN-3 CTRP2 9.2091 12.4881 6.8504 4.1486
M-07e CTRP2 9.2249 13.5742 6.3339 6.2258
P31/FUJ CTRP2 9.2327 13.2615 6.4921 5.5681
L-428 CTRP2 9.2745 10.7496 7.6963 0.8541
SUP-B15 CTRP2 9.2928 12.5632 6.8714 3.9453
REC-1 CTRP2 9.3164 15.3955 5.5065 9.4438
KMM-1 CTRP2 9.4018 14.8454 5.8399 7.9599
Ki-JK CTRP2 9.413 16.0834 5.2394 10.35
HuT 78 CTRP2 9.4424 13.4929 6.5267 5.117
WSU-DLCL2 CTRP2; CTRP1 9.444 10.9923 7.6802 0.7693
Kasumi-2 CTRP2 9.4775 11.0844 7.6584 0.8112
L-363 CTRP2 9.5118 10.8908 7.7544 0.5087
Granta-519 CTRP2 9.6215 19.1341 3.8889 15.0669
HT CTRP2; CTRP1 9.6307 12.3059 7.2061 2.2266
MOLP-2 CTRP2 9.6345 16.0229 5.4321 9.2276
Karpas-620 CTRP2 9.645 11.8882 7.401 1.5151
AML-193 CTRP2 9.6904 11.0127 7.7857 0.3384
OCI-AML-5 CTRP2 9.8197 11.2689 7.7427 0.3769
RPMI-8402 CTRP2 9.9251 12.494 7.2889 1.6383
Jurkat CTRP2 9.9511 15.6198 5.8515 7.084
KO52 CTRP2 9.9727 15.1321 6.1 6.071
HEL CTRP2 10.0498 13.957 6.7026 3.6309
U-937 CTRP2; CTRP1 10.0708 11.3889 7.7992 0.1811
OCI-Ly10 CTRP2; CTRP1 10.2387 14.6987 6.476 4.265
KE-97 CTRP2; CTRP1 10.2448 11.756 7.734 0.2379
GDM-1 CTRP2; CTRP1 10.2893 16.963 5.4367 8.224
KCL-22 CTRP2 10.4225 17.3 5.3655 8.3089
LAMA-84 CTRP2 10.4694 19.9536 4.1126 12.8927
SK-MM-2 CTRP2 10.6354 19.9202 4.247 12.1604
U266B1 CTRP2 11.0433 18.2729 5.314 7.6616
OCI-Ly19 CTRP2 12.2525 26.2856 2.294 16.0485
NCI-H929 CTRP2 12.5661 28.3435 1.5166 17.7211
⏷ Show the Full List of 149 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 7.6808 9.8753 6.9138 6.6783
TE8 CTRP2 9.5761 14.8979 5.9395 7.2872
EC-GI-10 CTRP2 7.5399 10.1916 6.6274 8.1828
KYSE-140 CTRP2; CTRP1 8.1293 14.6259 4.947 13.8484
TE-5 CTRP2 8.2958 12.2108 6.2934 7.9965
TE-1 CTRP2 8.4446 11.0402 6.9986 4.7645
KYSE-30 CTRP2 8.5832 9.7746 7.7276 1.5116
TE-11 CTRP2 8.6051 12.0426 6.6257 6.0401
KYSE-70 CTRP2 8.6852 11.9543 6.7314 5.4611
KYSE-410 CTRP2; CTRP1 8.7135 10.8807 7.2819 3.1336
KYSE-520 CTRP2 8.7488 11.2749 7.1144 3.7675
OE19 CTRP2 8.7649 11.6064 6.9633 4.3657
OE33 CTRP2 8.805 10.8337 7.3697 2.6365
OE21 CTRP2 8.8199 12.685 6.4721 6.311
TE-4 CTRP2 8.8539 12.2096 6.7323 5.1768
TE-6 CTRP2 8.8836 10.8236 6.5515 0.8988
KYSE-150 CTRP2 9.4426 11.0883 7.639 0.8997
KYSE-510 CTRP2 9.4812 13.6031 6.5002 5.1677
TE-10 CTRP2 9.7918 14.6732 6.1978 5.9358
TE-9 CTRP2 10.2291 15.9967 5.8587 6.6655
COLO 680N CTRP2 10.3322 15.87 5.9868 6.0287
TE-14 CTRP2 10.6435 12.1578 7.7408 0.136
KYSE-450 CTRP2; CTRP1 10.8187 16.7258 5.8958 5.7588
KYSE-180 CTRP2 10.9786 19.1956 4.8332 9.5334
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 9.049 11.8428 7.0513 3.5694
HuP-T4 CTRP2; CTRP1 7.1244 8.4938 6.942 8.0018
KP-4 CTRP2 7.8071 8.7996 7.5451 3.8033
HPAF-II CTRP2 8.0269 9.8332 7.2527 4.5059
L3.3 CTRP2 8.2346 10.3003 7.1979 4.3182
PSN1 CTRP2 8.2876 9.4054 7.6888 2.1568
DAN-G CTRP2 8.3126 9.4677 7.6778 2.1573
Panc 03.27 CTRP2; CTRP1 8.322 9.5989 7.6198 2.3833
PK-59 CTRP2 8.3353 11.0669 6.8975 5.3886
SNU-410 CTRP2 8.3723 10.1477 7.3862 3.2714
HPAC CTRP2; CTRP1 8.4136 11.4828 6.7531 5.8495
AsPC-1 CTRP2 8.4873 10.4361 7.3325 3.2943
YAPC CTRP2 8.5185 9.9687 7.5869 2.186
MIA PaCa-2 CTRP2 8.5361 9.8741 7.6461 1.9143
SU.86.86 CTRP2 8.5383 10.557 7.3115 3.295
SW1990 CTRP2 8.5444 10.2644 7.4606 2.6664
KP-2 CTRP2 8.5938 10.279 7.4897 2.467
TCC-Pan2 CTRP2 8.6888 10.8356 7.2861 3.1554
PaTu 8988s CTRP2 8.6908 11.3123 7.0531 4.1149
BxPC-3 CTRP2 8.6925 13.8419 5.7987 9.3241
HuP-T3 CTRP2 8.7868 12.8036 6.3882 6.7157
Panc 05.04 CTRP2 8.8307 13.7153 5.9696 8.3749
Panc 04.03 CTRP2 8.8449 11.4923 7.0777 3.7675
PaTu 8988t CTRP2 8.9684 10.4006 7.6798 1.2096
QGP-1 CTRP2; CTRP1 9.1493 12.7271 6.693 4.8754
Capan-1 CTRP2 9.1762 12.1822 6.9751 3.694
PK-45H CTRP2 9.2536 15.2908 5.5113 9.5286
Hs 766T CTRP2 9.586 17.3096 4.7639 11.9133
SNU-213 CTRP2 9.7591 10.8996 7.8556 0.1765
PaTu 8902 CTRP2; CTRP1 9.9534 11.253 7.803 0.2076
CFPAC-1 CTRP2; CTRP1 10.0039 13.8971 6.702 3.6876
SUIT-2 CTRP2; CTRP1 10.176 11.4051 7.8326 0.1128
KP-3 CTRP2; CTRP1 10.3007 13.9384 6.8599 2.7721
Capan-2 CTRP2; CTRP1 10.3719 15.3137 6.2732 4.8754
Panc 02.03 CTRP2 10.4224 11.9128 7.7454 0.1745
Panc 08.13 CTRP2 10.7482 12.453 7.6761 0.197
Panc 10.05 CTRP2; CTRP1 11.1063 12.8211 7.6782 0.1285
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 49 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 11.8047 26.4706 1.889 17.8119
SK-MEL-5 CTRP2; CTRP1 6.6295 9.5506 6.0041 12.9679
SK-MEL-28 CTRP2; CTRP1 7.2532 8.0516 7.2068 6.6528
G-361 CTRP2; CTRP1 7.375 9.8991 6.6072 8.6572
UACC-62 CTRP2 7.6812 8.4649 7.5535 4.1077
WM115 CTRP2 7.6969 8.4621 7.5713 3.9957
RVH-421 CTRP2 7.7897 12.3461 5.7937 11.0929
CJM [Human melanoma] CTRP2 7.8335 9.4826 7.2482 4.9491
WM266-4 CTRP2 7.8346 8.643 7.6427 3.3448
COLO 741 CTRP2; CTRP1 7.9132 9.8652 7.1347 5.2415
Hs 944.T CTRP2; CTRP1 7.9145 9.1628 7.4796 3.81
SK-MEL-1 CTRP2; CTRP1 8.0855 9.6198 7.4105 3.7232
MeWo CTRP2 8.1192 9.5502 7.4747 3.3845
WM88 CTRP2 8.1919 9.7733 7.4256 3.4448
LOX-IMVI CTRP2 8.2281 9.9522 7.3665 3.6223
SK-MEL-31 CTRP2 8.2321 9.4824 7.6047 2.6144
COLO 792 CTRP2 8.2824 12.1574 6.309 7.9568
HT-144 CTRP2 8.3355 9.2171 7.8206 1.5194
K029AX CTRP2 8.5176 10.9958 7.078 4.3037
WT2-iPS CTRP2 8.5496 9.7685 7.7072 1.6439
SK-MEL-3 CTRP2 8.5555 10.8508 7.1792 3.8167
UACC-257 CTRP2 8.6147 13.1233 6.0953 8.2349
WM983B CTRP2 8.6546 13.1656 6.1057 8.1203
SK-MEL-24 CTRP2 8.6774 10.1978 7.5885 1.9373
SK-MEL-30 CTRP2 8.7596 11.9782 6.7759 5.1508
Mel JuSo CTRP2 8.7637 10.7378 7.3873 2.626
WM793 CTRP2 8.8036 11.5982 6.9958 4.1691
COLO 800 CTRP2 8.8404 11.0459 7.2917 2.9009
Hs 852.T CTRP2; CTRP1 8.9015 11.28 7.2209 3.0978
WM1799 CTRP2 8.9135 13.2642 6.2565 7.0478
Hs 936.T CTRP2; CTRP1 8.9748 10.6679 7.5607 1.6512
A-375 CTRP2; CTRP1 8.9974 11.2679 7.2922 2.6744
A2058 CTRP2 9.0914 10.4733 7.7178 0.9464
Hs 294T CTRP2 9.152 10.6825 7.6591 1.0923
SK-MEL-2 CTRP2 9.1651 11.3399 7.3671 2.1616
A101D CTRP2 9.344 10.7535 7.7301 0.6915
IGR-1 CTRP2 9.3573 15.2564 5.6054 8.9786
IGR-37 CTRP2 9.4989 10.8884 7.7494 0.5301
Hs 839.T CTRP2 9.6228 10.7138 7.8699 0.1937
RPMI-7951 CTRP2 9.7799 11.0412 7.812 0.248
Hs 688(A).T CTRP2 9.7984 10.9581 7.8497 0.1751
Hs 895.T CTRP2 9.9964 11.3693 7.7775 0.2387
IPC-298 CTRP2 10.1497 15.99 5.8088 6.9706
Malme-3M CTRP2 10.1982 12.6629 7.3583 1.1901
COLO 829 CTRP2 10.1986 18.3961 4.6786 11.2522
MDA-MB-435S CTRP2 10.2782 17.697 5.0748 9.6334
Mel Ho CTRP2 10.5522 16.4012 5.8787 6.1589
Hs 940.T CTRP2 10.7231 21.9883 3.3008 15.2504
IGR-39 CTRP2 10.8196 17.5694 5.5009 7.2507
⏷ Show the Full List of 49 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 8.6137 10.6937 7.3006 3.2155
Cancer Drug Sensitivity Data Curated from 13 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Kelly CTRP2 7.6417 9.0821 7.2503 5.4021
NB1 CTRP2 8.0954 9.1819 7.637 2.7549
CHP-212 CTRP2 8.3499 11.191 6.8473 5.572
CHP-126 CTRP2 8.9541 11.6351 7.0857 3.5692
NH-6 CTRP2 9.0242 11.8119 7.0491 3.6142
KP-N-SI9s CTRP2 9.1075 12.4743 6.7863 4.5581
SiMa CTRP2 9.1153 11.4259 7.2949 2.5054
SK-N-DZ CTRP2 9.3148 17.6554 4.3871 13.7962
SK-N-AS CTRP2 9.5958 12.3351 7.1721 2.3915
KP-N-YN CTRP2 9.658 13.5091 6.6636 4.2727
SK-N-SH CTRP2 9.8224 15.3025 5.9159 7.0148
SK-N-FI CTRP2 9.9468 11.6224 7.6612 0.5072
SK-N-BE(2) CTRP2 9.9535 18.4462 4.4765 12.3916
⏷ Show the Full List of 13 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-478 CTRP2 8.1061 10.3558 7.0614 5.1443
HuH-28 CTRP2 8.3043 9.4784 7.6658 2.2226
HuCC-T1 CTRP2 8.5567 9.8959 7.6502 1.8656
SNU-1079 CTRP2 8.7969 17.8692 3.8735 16.6008
SNU-869 CTRP2 8.8841 11.8767 6.918 4.3623
SNU-1196 CTRP2 10.5749 13.5054 7.1941 1.4106
SNU-308 CTRP2 10.5805 12.8506 7.4609 0.6721
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HOS CTRP2 7.799 8.2624 7.7501 3.033
MG-63 CTRP2 7.8895 9.7197 7.1847 5.0861
SK-N-MC CTRP2 8.1083 8.6464 7.9127 1.5795
TC71 CTRP2 8.4413 10.2227 7.403 3.0793
A-673 CTRP2 8.4872 10.0585 7.5194 2.5166
CAL-78 CTRP2 8.7815 10.6214 7.4559 2.3222
SK-ES-1 CTRP2 8.8788 11.2373 7.2258 3.1115
U2OS CTRP2; CTRP1 8.932 11.3698 7.1987 3.1432
Hs 822.T CTRP2 8.9847 22.6204 1.6528 23.0644
SJSA-1 CTRP2 9.0172 11.4501 7.2184 2.9419
Hs 888.T CTRP2 9.5054 14.7573 5.9576 7.3221
SaOS-2 CTRP2 9.5912 14.7432 6.0254 6.9185
G-292 clone A141B1 CTRP2 10.4977 21.3944 3.4278 15.1904
MHH-ES-1 CTRP2 11.5884 18.1787 5.6966 5.5931
SW1353 CTRP2 15.5447 27.8881 3.6188 8.2986
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 72 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-361 CTRP2 2.4086 3.988 -0.2532 0.5021
HCC1143 CTRP2 7.6818 11.1354 6.2978 9.228
DU4475 CTRP2 7.7172 8.3392 7.6369 3.6914
BT-20 CTRP2 7.8339 9.3695 7.3033 4.7216
Hs 578T CTRP2 7.9339 13.0108 5.5878 11.6461
HCC1500 CTRP2 7.9581 10.46 6.8803 6.2072
ZR-75-30 CTRP2 8.1214 9.4463 7.5284 3.155
HCC1569 CTRP2 8.1542 10.5184 7.0212 5.2168
HCC1419 CTRP2 8.1993 13.2751 5.6811 10.7325
HCC1954 CTRP2 8.2631 10.0596 7.3418 3.6592
HCC202 CTRP2 8.4375 10.5338 7.2453 3.7449
MDA-MB-468 CTRP2 8.5065 9.8607 7.6311 2.0224
BT-549 CTRP2 8.5356 10.9038 7.1376 4.0241
ZR-75-1 CTRP2 8.6133 10.23 7.5277 2.2805
HCC1428 CTRP2 8.6218 12.7971 6.2634 7.5224
MDA-MB-231 CTRP2 8.7804 10.8867 7.3268 2.8474
CAL-85-1 CTRP2 8.8226 11.4632 7.0759 3.8097
MDA-MB-453 CTRP2 8.8251 11.2031 7.2045 3.2788
Hs 578Bst CTRP2 8.9105 10.4439 7.6247 1.4842
HCC1806 CTRP2 9.0292 14.1935 5.8844 8.3866
KPL-1 CTRP2 9.0381 9.7429 7.9938 0.1648
MDA-MB-415 CTRP2 9.051 11.4794 7.2271 2.8602
HCC1937 CTRP2 9.0612 13.4491 6.2757 6.7247
SK-BR-3 CTRP2 9.4113 12.2653 7.0904 2.9236
CAL-148 CTRP2 9.6105 11.5277 7.5388 1.0842
AU565 CTRP2 9.6427 12.1724 7.2735 1.9682
JIMT-1 CTRP2 9.7371 14.1813 6.3963 5.2231
CAMA-1 CTRP2 9.7783 12.7144 7.1079 2.4263
BT-474 CTRP2 9.8779 11.3186 7.7484 0.3393
T-47D CTRP2 9.9396 13.3873 6.8975 3.0259
CAL-120 CTRP2 10.1285 11.4671 7.7932 0.1755
HMC-1-8 CTRP2 10.1763 11.0752 7.9435 0.0232
MCF-7 CTRP2; CTRP1 10.3148 13.5885 7.0228 2.1856
HDQ-P1 CTRP2 10.4828 12.0596 7.716 0.2022
CAL-51 CTRP2 10.6257 15.6395 6.2794 4.5482
HCC38 CTRP2 10.651 12.6528 7.566 0.4105
HCC1395 CTRP2 11.0095 18.976 4.9585 9.0285
MDA-MB-157 CTRP2 12.0408 32.9139 -1.0988 24.2489
BT 112 CTRP2 8.1757 10.0054 7.2959 4.0213
BT 145 CTRP2 8.3386 10.2538 7.3063 3.6675
BT164 CTRP2 8.4884 10.6795 7.2125 3.7929
BT 224 CTRP2 8.7044 10.225 7.5939 1.8768
BT 179 CTRP2 8.7595 10.8096 7.3495 2.7862
BT 231 CTRP2 8.8658 12.1549 6.768 5.0097
BT 422 CTRP2 8.8725 10.5219 7.5641 1.7666
BT 320 CTRP2 9.0573 9.9551 7.9195 0.3364
BT 239 CTRP2 9.0626 10.5567 7.6644 1.1644
BT 330 CTRP2 9.113 10.4016 7.7607 0.7807
BT 139 CTRP2 9.2532 10.8811 7.6277 1.104
BT 245 CTRP2 9.271 11.0283 7.5726 1.2794
BT 286 CTRP2 9.3124 10.5463 7.8002 0.5067
BT 340 CTRP2 9.3136 11.2011 7.5198 1.4242
BT 228 CTRP2 9.3253 11.9589 7.1792 2.6874
BT 271 CTRP2 9.3303 10.8932 7.6639 0.9125
BT 504 CTRP2 9.3966 10.6547 7.7959 0.466
BT 248 CTRP2 9.5916 16.5033 5.1651 10.3501
BT 444 CTRP2 9.6497 10.8841 7.8174 0.2869
BT 498 CTRP2 9.6927 11.1826 7.7208 0.4931
BT 428 CTRP2 9.721 11.1858 7.7321 0.4496
BT 232 CTRP2 9.7445 11.6521 7.5544 0.9294
BT 159 CTRP2 9.7654 11.1942 7.7482 0.3894
BT 359 CTRP2 9.7716 11.3922 7.6734 0.5716
BT 216 CTRP2 9.8131 11.4009 7.6887 0.5091
BT 131 CTRP2 9.8154 10.8987 7.8773 0.1289
BT 333 CTRP2 9.8213 11.0839 7.8128 0.2321
BT147 CTRP2 9.8337 11.1886 7.779 0.2933
BT 482 CTRP2 9.8595 11.012 7.8537 0.1525
BT 440 CTRP2 9.872 11.1707 7.8011 0.2368
BT 416 CTRP2 9.8801 11.1976 7.7944 0.2464
BT 328 CTRP2 10.1445 11.2727 7.8668 0.0809
BT 172 CTRP2 10.3153 11.6835 7.7864 0.1428
BT 187 CTRP2 10.8448 14.6256 6.8576 2.2642
⏷ Show the Full List of 72 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 9.4253 11.6793 7.3693 1.8516
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
GB-1 CTRP2 7.2153 8.9441 6.8697 8.0213
Daoy CTRP2 7.5948 10.6812 6.4411 8.8263
T98G CTRP2 7.6738 17.7824 2.982 21.8362
8-MG-BA CTRP2 7.7033 8.1772 7.6685 3.618
TM-31 CTRP2 7.7976 8.1571 7.7756 2.9458
SNU-466 CTRP2 8.2026 16.4366 4.1031 16.924
KNS-60 CTRP2 8.2536 9.2836 6.8783 0.3559
Becker CTRP2 8.4361 9.5352 7.7393 1.6888
D283 Med CTRP2 8.4431 10.5434 7.2449 3.7368
SF126 CTRP2 8.4962 11.217 6.9513 4.8708
SW1088 CTRP2 8.592 10.865 7.1999 3.6692
GaMG CTRP2; CTRP1 8.6446 11.0086 7.1684 3.7127
SF268 CTRP2 8.8214 12.7593 6.4365 6.4566
KNS-42 CTRP2 8.8842 11.4334 7.1344 3.4755
SF539 CTRP2 8.9889 12.901 6.4919 5.9509
Hs 683 CTRP2 9.0188 10.7997 7.527 1.7268
U-118MG CTRP2 9.0473 11.1756 7.369 2.3039
DK-MG CTRP2 9.0582 12.585 6.6973 4.9969
ONS-76 CTRP2 9.1002 11.7839 7.1145 3.2417
KNS-81 CTRP2 9.1343 10.8527 7.5726 1.4222
KALS-1 CTRP2 9.216 12.7024 6.7518 4.5374
CCF-STTG1 CTRP2 9.2217 13.1874 6.5204 5.4693
YKG-1 CTRP2 9.2731 10.8296 7.661 0.972
DBTRG-05MG CTRP2 9.3255 13.498 6.4428 5.6284
KG-1-C CTRP2 9.441 11.527 7.4468 1.5545
LN-18 CTRP2 9.5486 10.4852 7.9238 0.1255
42-MG-BA CTRP2 9.6097 12.1367 7.2704 2.014
U-251MG CTRP2 9.7057 12.0354 7.3698 1.5655
CAS-1 CTRP2 9.7428 11.0183 7.8054 0.2747
SNU-489 CTRP2 9.8202 11.0173 7.8367 0.1904
SNU-1105 CTRP2 9.8292 14.2633 6.4184 5.0101
NMC-G1 CTRP2 9.8508 11.2196 7.7744 0.296
U-87MG ATCC CTRP2 9.8754 13.2036 6.9429 2.9294
SF295 CTRP2; CTRP1 9.8801 11.2892 7.7603 0.3133
SNU-738 CTRP2 9.9133 11.1276 7.8328 0.1706
SNU-201 CTRP2 10.0996 11.9654 7.5946 0.5922
SW1783 CTRP2 10.4147 20.3064 3.9007 13.7213
SNU-626 CTRP2 10.4412 11.5374 7.8801 0.0391
GOS-3 CTRP2 10.5499 15.5175 6.2893 4.5999
SNB-75 CTRP2 10.6133 12.3958 7.6453 0.2784
A-172 CTRP2 10.9665 18.9161 4.9585 9.0874
LN-229 CTRP2; CTRP1 11.1708 19.0399 5.0346 8.5309
M059K CTRP2 11.4909 19.4031 5.07 7.9871
YH-13 CTRP2 11.547 19.8432 4.8993 8.534
GMS-10 CTRP2 11.7509 18.2397 5.7647 5.1716
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-265 CTRP2; CTRP1 5.7377 9.1788 5.2023 18.5099
HEC-151 CTRP2; CTRP1 6.8317 9.5674 6.2074 11.6341
HEC-50B CTRP2 7.7566 8.8238 7.483 4.1799
KLE CTRP2; CTRP1 7.8042 9.9102 7.0124 5.9903
JHUEM-1 CTRP2 7.8566 9.2758 7.3701 4.3945
AN3-CA CTRP2 7.961 9.1415 7.5337 3.4799
MFE-319 CTRP2; CTRP1 7.9958 11.0069 6.6411 7.1304
EFE-184 CTRP2 8.4637 10.0005 7.5303 2.5101
ESS-1 CTRP2 8.6328 10.2929 7.511 2.319
JHUEM-3 CTRP2 8.8659 12.3608 6.6667 5.4282
EN CTRP2 8.9423 11.2021 7.2865 2.7743
JHUEM-7 CTRP2 9.0856 13.3625 6.3363 6.4363
HEC-1-A CTRP2 9.2285 13.0013 6.6156 5.0713
RL95-2 CTRP2 9.4561 15.1673 5.7217 8.3516
HEC-1-B CTRP2 9.5313 14.6667 6.0202 7.0299
HEC-6 CTRP2; CTRP1 9.7918 13.7291 6.6466 4.1646
HEC-251 CTRP2; CTRP1 10.2754 15.232 6.2505 5.0832
HEC-59 CTRP2; CTRP1 10.3205 15.4186 6.1917 5.2523
MFE-296 CTRP2 10.3487 14.7094 6.5385 3.8994
JHUEM-2 CTRP2; CTRP1 11.2663 18.7581 5.2292 7.6889
HEC-108 CTRP2; CTRP1 15.527 27.1282 3.9448 7.3613
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 9.1276 10.2639 7.8268 0.5577
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 20 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1272 CTRP2 8.1896 8.8929 7.8635 1.6115
TUHR14TKB CTRP2 8.1998 15.6375 4.5003 15.4465
VMRC-RCZ CTRP2 8.4145 9.4844 7.7483 1.687
786-O CTRP2 8.6007 10.0885 7.5877 2.0541
769-P CTRP2 8.6098 10.6132 7.3373 3.0701
Caki-2 CTRP2 8.6252 9.7772 7.7548 1.3435
ACHN CTRP2 8.6261 9.7391 7.7736 1.2677
KMRC-1 CTRP2 8.9452 10.9723 7.3983 2.3238
Caki-1 CTRP2 9.0474 10.9798 7.461 1.9454
UO-31 CTRP2 9.2396 11.7038 7.2442 2.5436
KMRC-2 CTRP2 9.2631 15.8388 5.2476 10.568
TUHR10TKB CTRP2 9.3727 10.967 7.6545 0.9073
BFTC-909 CTRP2 9.4956 10.9166 7.7364 0.568
VMRC-RCW CTRP2; CTRP1 9.6422 14.3509 6.2506 5.9384
CAL-54 CTRP2 9.6537 13.8699 6.4892 4.9689
TUHR4TKB CTRP2 9.9956 11.2316 7.8269 0.1585
OS-RC-2 CTRP2 10.1744 12.1579 7.5523 0.6587
KMRC-20 CTRP2 10.8445 12.3212 7.7562 0.0904
RCC10RGB CTRP2; CTRP1 11.5192 18.9821 5.2843 7.1712
KMRC-3 CTRP2 14.1921 37.0747 -1.5772 22.3308
⏷ Show the Full List of 20 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 52 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW480 CTRP1 4.6839 12.5082 2.7052 50.1661
SW620 CTRP2; CTRP1 6.9165 10.815 5.7275 13.337
SNU-175 CTRP1 7.5027 15.2011 4.1085 32.3119
CCK-81 CTRP2 7.5349 8.8722 7.234 5.7426
GP2d CTRP2; CTRP1 7.5909 8.7052 7.3626 5.0904
LS123 CTRP2; CTRP1 7.7777 10.4657 6.7153 7.2828
SW403 CTRP1 7.8374 12.7188 3.3529 8.0683
SNU-C1 CTRP2 7.9912 9.3087 7.48 3.6351
KM12 CTRP2; CTRP1 8.0212 10.3849 6.9732 5.6869
SW48 CTRP2; CTRP1 8.1798 13.5074 5.5486 11.3163
SNU-407 CTRP2 8.1968 10.5355 7.0487 5.0177
CW-2 CTRP2; CTRP1 8.1988 12.7763 5.93 9.7009
HCT 15 CTRP2 8.2342 9.6701 7.5126 2.9971
C2BBe1 CTRP2; CTRP1 8.2799 10.3881 7.1915 4.2585
COLO201 CTRP2 8.2982 9.5248 7.6377 2.3515
SNU-C5 CTRP2; CTRP1 8.3321 11.5298 6.6636 6.376
DLD-1 CTRP2; CTRP1 8.4465 9.6251 7.7028 1.8231
SK-CO-1 CTRP2; CTRP1 8.5353 10.2727 7.4497 2.726
SNU-C2A CTRP2; CTRP1 8.665 16.5502 4.4258 14.8296
SNU-61 CTRP2; CTRP1 8.682 10.8025 7.2973 3.1197
SW948 CTRP2; CTRP1 8.7075 15.19 5.1386 11.9803
HT-55 CTRP2; CTRP1 8.761 10.9 7.3066 2.9591
NCI-H508 CTRP2; CTRP1 8.9028 10.8154 7.4449 2.1965
LoVo CTRP2; CTRP1 8.9215 13.476 6.1578 7.4422
LS180 CTRP2; CTRP1 8.973 15.1435 5.3704 10.575
NCI-H716 CTRP2 9.0488 12.1168 6.9185 4.1078
LS1034 CTRP2 9.1056 11.1278 7.4286 1.9981
CL-11 CTRP2 9.1452 11.4441 7.3057 2.4248
T84 CTRP2 9.2104 14.5022 5.8678 8.1542
HT-29 CTRP2; CTRP1 9.213 17.3422 4.4641 13.6874
MDST8 CTRP2; CTRP1 9.2386 13.4625 6.3983 5.9415
SNU-503 CTRP2 9.262 15.6987 5.3161 10.297
SNU-C4 CTRP2; CTRP1 9.2829 13.5081 6.4077 5.8353
COLO 320 CTRP2; CTRP1 9.2944 14.7923 5.7873 8.3454
SNU-81 CTRP1 9.443 12.8635 6.8128 8.1932
LS411N CTRP2; CTRP1 9.4483 10.7927 7.7644 0.5203
NCI-H747 CTRP2 9.5321 12.034 7.2713 2.0948
COLO 678 CTRP2; CTRP1 9.6233 13.0839 6.8418 3.6202
HT115 CTRP2; CTRP1 9.7016 11.0606 7.7722 0.364
HCC-56 CTRP2 9.8086 15.3482 5.8842 7.1613
CL-40 CTRP1 9.9317 11.2547 7.7751 0.4789
COLO205 CTRP2; CTRP1 9.9638 13.1697 7.0107 2.5813
SNU-1033 CTRP2 9.982 15.2009 6.0734 6.1631
SW1417 CTRP2 10.0923 11.6275 7.7207 0.3123
RCM-1 [Human ESC] CTRP2; CTRP1 10.1746 15.5402 6.0398 6.0321
RKO CTRP2; CTRP1 10.1984 12.4789 7.4344 0.965
OUMS-23 CTRP2 10.2181 11.2631 7.8956 0.0479
CL-34 CTRP1 10.3042 16.6649 5.5743 14.6029
HCT 116 CTRP2; CTRP1 10.959 17.4375 5.6522 6.5017
SNU-1040 CTRP1 11.1714 19.8167 4.65 17.3953
HCT 8 CTRP2; CTRP1 11.2719 17.1758 5.965 4.9736
LS513 CTRP2; CTRP1 12.48 21.4409 4.7397 7.9591
⏷ Show the Full List of 52 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 20 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-886 CTRP2 6.1162 7.812 3.6046 0.5438
PLC/PRF/5 CTRP2 7.6598 8.1561 7.626 3.9039
JHH-5 CTRP2 7.803 9.8555 7.0381 5.8867
SNU-761 CTRP2 7.9124 9.5552 6.574 1.7968
JHH-2 CTRP2 7.9323 8.6336 7.7465 2.6805
SNU-878 CTRP2 7.9598 9.3962 7.4082 4.0025
Li-7 CTRP2 8.0319 9.4124 7.4659 3.6047
JHH-4 CTRP2 8.093 8.9431 7.753 2.2767
HuH-6 CTRP2 8.3555 10.5479 7.1731 4.1952
SK-HEP-1 CTRP2 8.4483 9.5936 7.7196 1.7506
SNU-398 CTRP2; CTRP1 8.5765 11.3444 6.9504 4.7342
Hep-G2 CTRP2; CTRP1 8.6361 10.5362 7.3944 2.7923
SNU-182 CTRP2 8.8482 17.5129 4.0923 15.7202
Hep 3B2.1-7 CTRP2 8.9907 14.9188 5.4956 10.0383
JHH-6 CTRP2; CTRP1 9.0055 9.9877 7.8813 0.4822
SNU-475 CTRP2 9.3567 11.4891 7.4151 1.7579
JHH-1 CTRP2 9.7842 10.8931 7.8676 0.1507
SNU-423 CTRP2 9.9575 11.9114 7.551 0.7917
SNU-387 CTRP2 9.9794 15.2897 6.0292 6.341
SNU-449 CTRP2; CTRP1 10.4173 15.7416 6.102 5.4744
⏷ Show the Full List of 20 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 159 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H82 CTRP1 5.3463 7.7918 4.0304 10.0476
NCI-H460 CTRP2; CTRP1 5.7335 7.4966 5.665 16.8409
COR-L279 CTRP1 5.7892 7.9584 4.283 6.2275
NCI-H1963 CTRP1 5.8347 11.3232 4.4043 40.3824
NCI-H1930 CTRP1 6.3625 9.3913 3.9837 7.0345
SK-LU-1 CTRP2; CTRP1 6.4509 8.7294 6.1319 12.9762
NCI-H1048 CTRP1 6.4558 8.7135 4.3548 3.8157
HCC33 CTRP1 6.7697 9.1232 4.3489 3.2
NCI-H1437 CTRP1 6.8465 9.2948 4.3158 3.2897
SBC-5 CTRP2 6.8908 7.9236 6.8392 9.082
NCI-H2106 CTRP2 6.9623 9.1094 6.5358 10.0026
RERF-LC-KJ CTRP1 7.1268 9.2479 4.4762 1.772
NCI-H1975 CTRP1 7.28 9.1269 4.5918 0.9809
NCI-H1581 CTRP2 7.2873 8.8045 7.002 7.3133
NCI-H1184 CTRP2 7.3276 12.6342 5.2364 14.373
HCC44 CTRP2; CTRP1 7.3438 12.5597 5.2878 14.1292
NCI-H1155 CTRP2 7.3738 9.4832 6.7985 7.8879
NCI-H211 CTRP2 7.4344 10.9147 6.1775 10.2779
NCI-H647 CTRP2 7.5193 9.7888 6.8001 7.5243
NCI-H1568 CTRP2; CTRP1 7.5641 11.6068 5.9583 10.8938
NCI-H146 CTRP2 7.588 8.8264 7.3086 5.3089
SW1573 CTRP2 7.5931 8.7063 7.3644 5.0773
HCC2108 CTRP2; CTRP1 7.6478 13.2752 5.2065 13.7978
LCLC-103H CTRP2; CTRP1 7.6882 8.1361 7.6613 3.6908
COR-L51 CTRP1 7.7178 21.954 0.9233 38.8525
NCI-H1944 CTRP2; CTRP1 7.8035 10.125 6.9065 6.4314
NCI-H1755 CTRP2; CTRP1 7.8087 11.1079 6.4258 8.422
COR-L88 CTRP2; CTRP1 7.8629 10.3612 6.8442 6.561
RERF-LC-A1 CTRP2 7.8634 11.1788 6.4393 8.2499
LXF 289 CTRP2; CTRP1 7.8712 10.8353 6.6167 7.4923
DV-90 CTRP2; CTRP1 7.8756 10.4991 6.7873 6.7707
COLO 668 CTRP2; CTRP1 7.8874 11.0972 6.501 7.9417
RERF-LC-MS CTRP2 7.9071 8.6017 7.7351 2.7908
NCI-H810 CTRP2; CTRP1 7.9238 9.4697 7.3388 4.3703
NCI-H446 CTRP2 7.926 9.7449 7.2056 4.9186
IA-LM CTRP2 7.9478 9.5364 7.3282 4.3613
NCI-H1915 CTRP2; CTRP1 7.968 11.2933 6.4741 7.8868
PC-14 CTRP2 7.9722 8.951 7.6366 3.0306
NCI-H358 CTRP2; CTRP1 7.9779 9.174 7.5337 3.4416
NCI-H1341 CTRP2 8.046 9.3979 7.4857 3.4918
NCI-H2087 CTRP2 8.047 16.8799 3.7509 18.4991
Lu-65 CTRP2; CTRP1 8.0507 13.161 5.6128 11.3079
EPLC-272H CTRP2; CTRP1 8.1731 9.708 7.4423 3.4117
NCI-H1373 CTRP2; CTRP1 8.2063 11.4227 6.6131 6.8281
NCI-H2029 CTRP2; CTRP1 8.2247 10.7134 6.9831 5.2393
NCI-H841 CTRP2; CTRP1 8.2465 12.5825 6.0667 9.039
NCI-H1703 CTRP2 8.2467 10.1605 7.2778 3.9592
NCI-H2141 CTRP2; CTRP1 8.2607 14.348 5.1958 12.5949
Calu-3 CTRP2; CTRP1 8.265 12.5335 6.1066 8.8366
HCC1195 CTRP2; CTRP1 8.271 12.3803 6.1882 8.4843
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 8.2745 9.7123 7.5248 2.8694
ChaGo-K-1 CTRP2; CTRP1 8.2958 10.6855 7.0559 4.7979
NCI-H1105 CTRP2; CTRP1 8.2984 10.7454 7.028 4.9101
NCI-H2023 CTRP2; CTRP1 8.3013 9.9961 7.4048 3.3231
SCLC-21H CTRP1 8.3278 16.2115 4.3066 28.0855
NCI-H1666 CTRP2; CTRP1 8.3372 14.2329 5.3166 11.9584
NCI-H1355 CTRP2; CTRP1 8.3527 12.0143 6.4383 7.2821
NCI-H1092 CTRP2 8.3568 10.1523 7.3715 3.3609
NCI-H2342 CTRP2; CTRP1 8.3633 13.2123 5.8483 9.7249
Calu-6 CTRP2; CTRP1 8.4049 10.2364 7.3678 3.2903
NCI-H838 CTRP2 8.4052 10.6789 7.1475 4.2121
NCI-H889 CTRP2 8.4232 13.2447 5.8809 9.477
NCI-H322 CTRP2 8.4383 10.1366 7.4434 2.9157
NCI-H2170 CTRP2 8.4502 11.8333 6.6076 6.3925
NCI-H650 CTRP2; CTRP1 8.4876 12.6622 6.2239 7.9294
LUDLU-1 CTRP2 8.494 10.1301 7.4891 2.631
NCI-H1693 CTRP2 8.4988 10.5896 7.2652 3.5551
NCI-H2122 CTRP2; CTRP1 8.5153 10.2262 7.4576 2.7262
NCI-H2286 CTRP2; CTRP1 8.5436 12.0418 6.5779 6.3482
COR-L105 CTRP2 8.5451 10.4437 7.3726 3.0299
Lu-99 CTRP2; CTRP1 8.5855 13.5283 5.8701 9.2222
NCI-H23 CTRP2; CTRP1 8.6013 14.2548 5.5203 10.6327
NCI-H522 CTRP2; CTRP1 8.603 11.2344 7.0253 4.3768
LK2 CTRP2 8.6141 10.0146 7.6331 1.8491
NCI-H2126 CTRP2; CTRP1 8.6311 10.3873 7.4637 2.5155
NCI-H1339 CTRP2 8.6337 10.245 7.535 2.2193
NCI-H1836 CTRP1 8.65 18.3192 3.5168 29.8699
NCI-H1573 CTRP2; CTRP1 8.6524 13.5905 5.8923 9.0096
NCI-H3255 CTRP1 8.6655 14.2899 5.5404 20.2998
NCI-H520 CTRP2 8.7114 10.526 7.4533 2.4354
NCI-H2228 CTRP2 8.7201 11.2229 7.1189 3.7951
SK-MES-1 CTRP2 8.7442 12.1343 6.6872 5.5449
Sq-1 CTRP2; CTRP1 8.7543 10.7611 7.3694 2.7129
NCI-H2196 CTRP2 8.7835 10.5205 7.5058 2.1186
NCI-H1650 CTRP2 8.7927 10.994 7.2833 3.006
NCI-H1435 CTRP2; CTRP1 8.8172 11.6785 6.9664 4.2689
NCI-H196 CTRP2 8.8422 12.1751 6.7406 5.1611
LOU-NH91 CTRP2 8.8547 10.616 7.5078 2.0122
NCI-H2110 CTRP2; CTRP1 8.8935 13.487 6.131 7.6002
HCC366 CTRP2 8.9102 11.0582 7.3338 2.6297
NCI-H1838 CTRP2 8.9234 12.5095 6.6362 5.4612
NCI-H292 CTRP2 8.932 16.1898 4.818 12.836
LC-1/sq-SF CTRP2; CTRP1 8.933 12.4785 6.6584 5.354
VMRC-LCD CTRP2; CTRP1 8.9426 12.8852 6.4654 6.1356
DMS 273 CTRP2; CTRP1 9.0068 11.169 7.3455 2.4499
HOP-62 CTRP2 9.026 10.6962 7.5792 1.5197
NCI-H661 CTRP2; CTRP1 9.0345 15.8861 5.0492 11.7483
NCI-H1734 CTRP2 9.0395 16.0468 4.9732 12.0385
EBC-1 CTRP2; CTRP1 9.0653 14.4846 5.7677 8.8037
NCI-H1793 CTRP2; CTRP1 9.0917 11.5249 7.2326 2.783
NCI-H2172 CTRP2; CTRP1 9.1327 10.8043 7.5936 1.3472
NCI-H226 CTRP2 9.1507 11.346 7.3551 2.2255
A-549 CTRP2; CTRP1 9.1579 14.0355 6.0587 7.4592
NCI-H2081 CTRP2; CTRP1 9.1741 14.0411 6.0679 7.3952
RERF-LC-Ad1 CTRP2 9.2109 10.2016 7.8915 0.322
NCI-H2030 CTRP2; CTRP1 9.2156 13.2844 6.4687 5.6894
NCI-H1869 CTRP2 9.2513 14.4829 5.9076 7.9255
NCI-H596 CTRP1 9.2591 15.7034 5.2972 19.602
HCC15 CTRP2; CTRP1 9.3026 12.8034 6.7628 4.3675
DMS 114 CTRP2 9.3144 11.6104 7.3343 2.1071
LCLC-97TM1 CTRP2; CTRP1 9.3515 11.2288 7.5289 1.3535
BEN CTRP2; CTRP1 9.3539 10.2582 7.9304 0.1725
HCC1359 CTRP1 9.3706 10.4346 7.8523 0.6019
DMS 53 CTRP2 9.3827 12.6856 6.8732 3.8142
SW1271 CTRP2 9.4449 12.1749 7.1537 2.6383
NCI-H1781 CTRP1 9.4626 11.5721 7.4219 3.2878
NCI-H2291 CTRP2 9.4634 17.2931 4.6799 12.439
DMS 454 CTRP2 9.4964 14.3743 6.1377 6.6081
KNS-62 CTRP2; CTRP1 9.4971 12.3313 7.1135 2.7284
NCI-H1651 CTRP2 9.5427 13.0784 6.7922 3.9195
HCC2935 CTRP2; CTRP1 9.6026 13.2623 6.7442 4.0289
NCI-H69 CTRP2 9.639 13.381 6.7118 4.1083
NCI-H2444 CTRP2 9.6462 10.6936 7.8864 0.1582
NCI-H2085 CTRP2 9.6697 15.674 5.6281 8.3927
NCI-H441 CTRP2; CTRP1 9.7002 15.1326 5.913 7.2068
HCC4006 CTRP2; CTRP1 9.7026 11.9555 7.403 1.4546
NCI-H1876 CTRP1 9.7298 14.7352 6.1102 12.7136
EKVX CTRP2 9.7431 12.1566 7.3371 1.6426
NCI-H1694 CTRP2; CTRP1 9.7474 11.6322 7.5641 0.8979
T3M-10 CTRP2; CTRP1 9.7745 14.4052 6.3144 5.4963
COR-L23 CTRP1 9.8527 11.1577 7.7794 0.5175
NCI-H2405 CTRP2; CTRP1 9.9362 15.818 5.7456 7.5247
NCI-H526 CTRP2 9.9494 11.356 7.7637 0.2804
NCI-H1623 CTRP2 9.9693 12.4546 7.3295 1.464
NCI-H1395 CTRP2 9.977 14.5334 6.3872 4.9363
HCC1171 CTRP2 9.9837 17.5577 4.9337 10.6222
HCC95 CTRP2 10.0482 12.9085 7.1748 1.914
HCC78 CTRP2; CTRP1 10.1967 13.0582 7.1898 1.7286
NCI-H1563 CTRP2 10.2131 16.3872 5.6613 7.4585
DMS 79 CTRP2 10.2258 11.9664 7.6485 0.4077
HCC1438 CTRP2 10.2385 11.7265 7.7422 0.226
MOR/CPR CTRP2 10.2837 21.8492 3.0461 16.7687
SHP-77 CTRP2; CTRP1 10.3183 16.2911 5.7779 6.8584
Calu-1 CTRP2 10.3559 12.5481 7.4798 0.7442
CAL-12T CTRP2; CTRP1 10.3643 12.0082 7.689 0.2789
COR-L95 CTRP2 10.3913 11.5658 7.8536 0.0617
NCI-H2009 CTRP2; CTRP1 10.4418 14.8142 6.5465 3.7636
NCI-H1792 CTRP2; CTRP1 10.4952 16.4542 5.8168 6.4707
RERF-LC-Ad2 CTRP2 10.4971 16.6144 5.7422 6.7554
NCI-H1299 CTRP2; CTRP1 10.7471 12.5328 7.6474 0.2386
HOP-92 CTRP2 10.8089 18.0206 5.2801 8.0995
HCC1833 CTRP2; CTRP1 10.8553 16.169 6.1754 4.6705
NCI-H727 CTRP2; CTRP1 10.8629 16.7305 5.9212 5.6094
COLO 699 CTRP2; CTRP1 10.8654 22.7006 3.0553 15.8129
NCI-H2073 CTRP1 11.4719 21.8343 3.8868 20.1058
HCC827 CTRP2; CTRP1 11.9683 19.5277 5.3079 6.5571
HCC2279 CTRP2 12.2238 23.3315 3.6911 11.8159
HCC1588 CTRP2 16.0643 35.6201 0.3829 16.1726
Hs 888.Lu CTRP2 9.7621 13.5429 6.715 3.9362
⏷ Show the Full List of 159 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 8.2911 9.9188 7.4352 3.2144
SYO-1 CTRP2 9.1794 11.9777 7.0751 3.2891
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 9.0569 11.7148 7.1183 3.2875
Aska-SS CTRP2 9.4081 11.1144 7.6098 1.0237
HT-1080 CTRP2; CTRP1 7.67 10.5106 6.5943 8.0233
SK-UT-1 CTRP2 7.7513 18.4182 2.7309 22.4495
G-401 CTRP2; CTRP1 7.9625 15.5239 4.3571 16.4673
MES-SA CTRP2 8.2712 9.0495 7.8532 1.4972
TE 617.T CTRP2 8.3849 12.1593 6.3921 7.4155
SK-LMS-1 CTRP2 8.3869 9.8662 7.5379 2.6106
Rh18 CTRP2 8.3921 9.955 7.4977 2.7695
G-402 CTRP2 8.4162 13.1053 5.9449 9.2242
TE 441.T CTRP2 8.4736 10.8585 7.112 4.2389
Hs 729.T CTRP2 8.4965 10.7189 7.1992 3.8344
TTC-709 CTRP2 8.8689 10.3376 7.6481 1.4453
A-204 CTRP2 9.1081 12.8803 6.5889 5.3637
BT-12 CTRP2 9.1192 10.2373 7.8337 0.5429
GCT CTRP2 9.2152 11.003 7.552 1.4107
Tm87-16 CTRP2 9.2524 10.8015 7.6621 0.9871
RKN CTRP2; CTRP1 9.2753 12.124 7.0691 3.1829
BT-16 CTRP2 9.4319 11.279 7.5512 1.1991
KYM-1 CTRP2 9.4611 13.6898 6.4446 5.4206
Rh41 CTRP2 9.5718 12.2711 7.187 2.3633
SW982 CTRP2 10.0741 11.3974 7.7975 0.183
RD CTRP2 14.9364 27.747 3.331 9.7479
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 9.0799 10.9777 7.4823 1.8237
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 9.9041 11.5487 7.6711 0.5049
OVMANA CTRP1 6.8431 10.3426 3.8428 6.8712
COV318 CTRP1 6.8591 7.7729 4.9173 0.1114
OVKATE CTRP1 6.8954 16.2736 3.036 38.0895
JHOS-4 CTRP1 7.1086 8.6619 4.6958 0.6654
HEY A8 CTRP2; CTRP1 7.2122 7.8653 7.1934 6.8299
COV434 CTRP2; CTRP1 7.4069 11.0555 6.0832 10.7291
RMUG-S CTRP1 7.6707 15.878 3.9174 32.2635
MCAS CTRP2 7.692 8.4645 7.5652 4.0326
OVISE CTRP2 7.7025 8.2064 7.6604 3.6496
TOV-112D CTRP2 8.091 12.1456 6.1544 8.9765
OV-90 CTRP2; CTRP1 8.1075 11.3241 6.5789 7.1655
ES2 CTRP2 8.117 9.5255 7.4851 3.3458
DOV13 CTRP2 8.1406 10.3346 7.1015 4.9068
SNU-119 CTRP2 8.1842 10.1978 7.207 4.3778
OAW28 CTRP2 8.3237 12.1684 6.3375 7.759
OVCAR-4 CTRP2; CTRP1 8.3778 13.2159 5.8583 9.6562
OV56 CTRP2 8.7036 9.8963 7.7498 1.2593
OV7 CTRP2; CTRP1 8.7571 15.8384 4.8548 13.0108
Kuramochi CTRP2 8.9582 12.2007 6.813 4.6776
OVK18 CTRP2; CTRP1 9.0057 14.7276 5.602 9.5804
A2780 CTRP2; CTRP1 9.007 14.8491 5.5427 9.819
EFO-21 CTRP2; CTRP1 9.0132 11.6421 7.1234 3.3296
OAW42 CTRP2; CTRP1 9.1201 10.2852 7.8141 0.6026
ONCO-DG-1 CTRP2 9.1331 13.412 6.3468 6.3176
COV644 CTRP2; CTRP1 9.1961 11.1832 7.4587 1.7759
SK-OV-3 CTRP2; CTRP1 9.2184 12.6302 6.7883 4.3863
FU-OV-1 CTRP2 9.262 11.2103 7.4857 1.602
RMG-I CTRP2; CTRP1 9.3119 14.7248 5.8333 8.1301
EFO-27 CTRP2; CTRP1 9.4299 11.3083 7.5373 1.2486
OC 314 CTRP2 9.4754 16.342 5.1584 10.5664
IGROV-1 CTRP2; CTRP1 9.4831 15.5949 5.5316 9.0722
SNU-8 CTRP2 9.6018 11.7641 7.4318 1.4499
COV362 CTRP2; CTRP1 9.6437 12.2706 7.2298 2.1256
JHOS-2 CTRP2 9.7606 16.5512 5.2648 9.6891
OVCAR-5 CTRP2 9.7622 11.9462 7.4389 1.2819
JHOM-1 CTRP2; CTRP1 9.9069 11.2182 7.7975 0.2318
OVCAR-8 CTRP2; CTRP1 9.9402 15.3047 5.9955 6.5294
TYK-nu CTRP2; CTRP1 10.0865 15.3173 6.0876 5.9641
OVTOKO CTRP2 10.7106 16.6624 5.8573 6.0387
Caov-3 CTRP2; CTRP1 10.9248 18.5473 5.1064 8.5945
SNU-840 CTRP2; CTRP1 11.1676 17.4131 5.7934 5.7221
OVSAHO CTRP2 13.8193 23.9035 4.4146 7.5749
JHOC-5 CTRP2; CTRP1 14.6896 22.0522 5.671 2.9916
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2; CTRP1 7.8138 9.0408 7.4405 4.2084
NCI-H28 CTRP2; CTRP1 8.2826 11.6469 6.5644 6.8859
NCI-H2452 CTRP2 8.804 11.0905 7.2444 3.148
IST-Mes1 CTRP2 9.4517 13.2152 6.6665 4.5428
ACC-MESO-1 CTRP2 9.6726 12.2827 7.2412 2.0536
NCI-H2052 CTRP2; CTRP1 10.3266 14.6106 6.5704 3.8055
MPP 89 CTRP2 10.5555 12.0907 7.7321 0.1636
JL-1 CTRP2 10.9436 17.6005 5.5661 6.8446
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LNCaP clone FGC CTRP2 7.9922 9.3932 7.4393 3.8016
PaCa-3 CTRP2; CTRP1 8.1091 9.2888 7.596 2.8975
DU145 CTRP2 8.6972 10.7172 7.3501 2.879
22Rv1 CTRP2 8.8124 12.5469 6.5347 6.0637
VCaP CTRP2 9.7898 11.3524 7.6974 0.4997
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 CTRP2 8.2574 9.4978 7.618 2.5105
YD-15 CTRP2 10.092 15.3978 6.0529 6.0927
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ECC10 CTRP2 7.2404 8.4073 7.0966 7.0894
GSS CTRP2 7.6668 8.8687 7.3714 4.8547
SNU-16 CTRP2 7.678 8.7481 7.4354 4.5731
SNU-620 CTRP2 7.682 11.437 6.149 9.8465
MKN7 CTRP2; CTRP1 8.0445 10.4726 6.9499 5.737
SNU-1 CTRP2 8.0485 9.6616 7.3571 4.024
NUGC-3 CTRP2 8.1258 10.0983 7.2069 4.4943
SH-10-TC CTRP2; CTRP1 8.239 11.8857 6.4088 7.6218
KATO III CTRP2 8.4075 11.7323 6.6237 6.4035
MKN74 CTRP2; CTRP1 8.4087 12.263 6.3596 7.5076
Hs 746.T CTRP2 8.4522 9.5997 7.7195 1.7446
MKN1 CTRP2 8.6872 10.8355 7.2849 3.1625
Fu97 CTRP2; CTRP1 8.7091 11.0017 7.2194 3.3975
SNU-668 CTRP2 9.0666 10.738 7.5846 1.453
GSU CTRP2 9.0691 9.804 7.9837 0.1735
LMSU CTRP2 9.072 11.8112 7.0823 3.4109
HuG1-N CTRP2 9.2634 28.7212 -1.1684 28.6072
HGC-27 CTRP2 9.3298 11.1743 7.5408 1.333
SNU-5 CTRP2 9.3784 16.3152 5.0991 10.9608
AGS CTRP2; CTRP1 9.3925 11.8116 7.2893 2.1855
SNU-216 CTRP2 9.399 11.8105 7.2938 2.1612
IM95 CTRP2 9.4735 16.9977 4.8335 11.8344
MKN45 CTRP2 9.678 14.6309 6.1402 6.3289
ECC12 CTRP2 9.7836 10.9521 7.8461 0.1853
NUGC-4 CTRP2; CTRP1 9.7964 11.3604 7.6971 0.4968
NCI-N87 CTRP2 10.2074 14.8243 6.398 4.6009
23132/87 CTRP2 10.2534 11.6544 7.7737 0.1737
SNU-601 CTRP2 11.3554 21.7605 3.8581 12.4543
KE-39 CTRP2 12.1034 19.3141 5.4853 5.7805
SNU-719 CTRP2 12.7108 21.9378 4.6517 7.9947
SNU-1077 CTRP2 8.7138 14.0574 5.7081 9.6588
SNG-M CTRP2; CTRP1 8.7499 11.8268 6.8435 4.8866
SNU-685 CTRP2 9.8654 14.4157 6.3699 5.1524
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
B-CPAP CTRP2 5.6923 6.8624 5.6833 16.9122
8505C CTRP2 7.5322 9.2933 7.0441 6.5046
CAL-62 CTRP2 7.9459 8.6895 7.7346 2.694
FTC-133 CTRP2 8.2905 9.672 7.558 2.7002
SW579 CTRP2 8.8357 11.2265 7.2007 3.2783
TT2609-C02 CTRP2 8.9258 10.9359 7.4028 2.3327
ML-1 [Human leukemia] CTRP2 9.3489 14.019 6.2058 6.5566
8305C CTRP2 9.8648 13.9757 6.5776 4.3396
CGTH-W-1 CTRP2 10.0652 11.8678 7.6175 0.5533
BHT-101 CTRP2 10.3116 12.346 7.5394 0.6179
FTC-238 CTRP2 10.6972 17.7156 5.3512 7.9821
TT CTRP2 14.3898 32.899 0.5735 17.668
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-4 CTRP2 7.3824 8.2165 7.3085 5.8915
HSC-2 CTRP2; CTRP1 7.642 8.113 7.6159 3.9953
SCC-4 CTRP2 7.6531 8.7777 7.3969 4.79
FaDu CTRP2 7.8788 8.9981 7.5242 3.7112
PE/CA-PJ34 (clone C12) CTRP2 8.1942 9.9928 7.3178 3.8929
SCC-25 CTRP2 8.2011 10.9818 6.8291 5.9314
PE/CA-PJ15 CTRP2 8.4277 11.4797 6.766 5.7697
YD-10B CTRP2 8.4424 12.815 6.1112 8.4828
PE/CA-PJ49 CTRP2 8.76 11.5148 7.0047 4.2024
BICR 6 CTRP2 8.7718 10.4634 7.5252 2.0572
SCC-9 CTRP2; CTRP1 8.799 11.1462 7.2137 3.281
PE/CA-PJ41 (clone D2) CTRP2 8.8153 12.1625 6.7268 5.2625
YD-8 CTRP2 8.9503 11.526 7.1359 3.371
SNU-899 CTRP2 8.9811 12.7506 6.5601 5.6825
BICR 22 CTRP2 9.27 11.6322 7.2967 2.303
SNU-1214 CTRP2 9.3288 15.4285 5.4995 9.4514
BICR 16 CTRP2 9.5476 14.0864 6.313 5.8249
HSC-3 CTRP2 10.0214 14.9274 6.2298 5.4939
BICR 31 CTRP2 10.1991 12.9927 7.2192 1.6294
BICR 56 CTRP2 10.2023 15.4323 6.1091 5.7251
Detroit 562 CTRP2 10.2477 13.2506 7.1338 1.8703
CAL-33 CTRP2 10.3853 11.9329 7.7243 0.2145
BHY CTRP2 10.4001 12.0457 7.6893 0.2673
BICR 18 CTRP2 10.4046 12.2798 7.6045 0.4274
SNU-1041 CTRP2 11.1606 16.9417 6.0053 4.9507
SNU-1066 CTRP2 11.6024 17.9021 5.8304 5.0971
SNU-1076 CTRP2 12.0987 22.4004 4.0504 10.7869
SNU-46 CTRP2 13.9767 33.4952 0.0057 19.4498
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HT-1197 CTRP2 3.6556 21.9274 -7.8882 30.5603
UM-UC-3 CTRP2; CTRP1 6.1277 8.2593 5.9274 14.6856
UM-UC-1 CTRP2 7.3631 8.0727 7.3216 5.9044
RT-4 CTRP2; CTRP1 7.8478 14.0648 4.9875 14.2579
J82 CTRP2 8.0151 9.0882 7.6102 3.0417
BC-3C CTRP2 8.0261 9.2778 7.5271 3.3626
TCCSUP CTRP2 8.11 10.9335 6.7762 6.3329
RT-112 CTRP2 8.2046 9.6013 7.5223 3.014
T24 CTRP2 8.4776 9.8354 7.6222 2.1058
5637 CTRP2; CTRP1 8.5966 13.7674 5.7598 9.6579
SW1710 CTRP2 8.6835 10.2973 7.5446 2.1058
HT-1376 CTRP2; CTRP1 8.757 11.4655 7.0268 4.1158
253J-BV CTRP2 8.9946 12.6558 6.6166 5.4283
639V CTRP2 9.1357 10.9751 7.5177 1.6242
BFTC-905 CTRP2 9.2726 10.6355 7.7437 0.7039
KMBC-2 CTRP2; CTRP1 9.2922 14.2612 6.0464 7.2943
CAL-29 CTRP2 9.3447 10.767 7.7248 0.7073
KU-19-19 CTRP2 9.5084 12.1824 7.1893 2.4275
VM-CUB-1 CTRP2 9.542 14.0427 6.3301 5.764
JMSU-1 CTRP2 9.8652 12.0609 7.4434 1.182
253J CTRP2 10.2416 11.4234 7.8497 0.0838
U-BLC1 CTRP2 10.3542 11.8756 7.733 0.2092
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 8.5905 10.5942 7.3323 3.1222

References

1 Etomoxir, a carnitine palmitoyltransferase I inhibitor, protects hearts from fatty acid-induced ischemic injury independent of changes in long chain acylcarnitine. Circ Res. 1988 Dec;63(6):1036-43.