General Information of Drug (ID: DM6BU7N)

Drug Name
Doramapimod
Synonyms
Doramapimod; 285983-48-4; BIRB-796; BIRB 796; BIRB 796 (Doramapimod); BIRB796; UNII-HO1A8B3YVV; 1-(5-TERT-BUTYL-2-P-TOLYL-2H-PYRAZOL-3-YL)-3-[4-(2-MORPHOLIN-4-YL-ETHOXY)-NAPHTHALEN-1-YL]-UREA; 1-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea; HO1A8B3YVV; CHEMBL103667; 3-[3-tert-butyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]-1-{4-[2-(morpholin-4-yl)ethoxy]naphthalen-1-yl}urea; CHEBI:40953; MVCOAUNKQVWQHZ-UHFFFAOYSA-N; C31H37N5O3; 1-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)-3-(4-(2
Indication
Disease Entry ICD 11 Status REF
Inflammatory bowel disease DD72 Discontinued in Phase 2 [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 2 Molecular Weight (mw) 527.7
Logarithm of the Partition Coefficient (xlogp) 5.7
Rotatable Bond Count (rotbonds) 8
Hydrogen Bond Donor Count (hbonddonor) 2
Hydrogen Bond Acceptor Count (hbondacc) 5
Chemical Identifiers
Formula
C31H37N5O3
IUPAC Name
1-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea
Canonical SMILES
CC1=CC=C(C=C1)N2C(=CC(=N2)C(C)(C)C)NC(=O)NC3=CC=C(C4=CC=CC=C43)OCCN5CCOCC5
InChI
InChI=1S/C31H37N5O3/c1-22-9-11-23(12-10-22)36-29(21-28(34-36)31(2,3)4)33-30(37)32-26-13-14-27(25-8-6-5-7-24(25)26)39-20-17-35-15-18-38-19-16-35/h5-14,21H,15-20H2,1-4H3,(H2,32,33,37)
InChIKey
MVCOAUNKQVWQHZ-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
156422
ChEBI ID
CHEBI:40953
CAS Number
285983-48-4
UNII
HO1A8B3YVV
DrugBank ID
DB03044
TTD ID
D05CDF

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Hematopoietic cell kinase (HCK) TT42OGM HCK_HUMAN Inhibitor [2]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
C-X-C motif chemokine 10 (CXCL10) OTTLQ6S0 CXL10_HUMAN Protein Interaction/Cellular Processes [3]
Mitogen-activated protein kinase 14 (MAPK14) OT5TCO3O MK14_HUMAN Gene/Protein Processing [4]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1; GDSC2 4.6564 7.308 2.3007 3.461
CHSA0011 GDSC1; GDSC2 4.4931 17.7296 -2.9306 27.4716
HuO9 GDSC1; GDSC2 4.6582 7.7788 2.0843 4.6915
NOS-1 [Human HNSCC] GDSC1; GDSC2 4.8166 9.1832 1.5238 7.6396
ES7 GDSC1; GDSC2 4.836 7.326 2.3965 2.6537
EW-1 GDSC1; GDSC2 4.8803 9.5056 1.4126 8.1498
EW-22 GDSC1; GDSC2 4.9155 8.2339 2.0328 4.5198
CHSA0108 GDSC1; GDSC2 4.9785 7.914 2.2153 3.4055
ES1 GDSC1; GDSC2 4.9802 9.4726 1.4945 7.4741
EW-24 GDSC1; GDSC2 5 7.2692 2.5091 1.8628
EW-16 GDSC1; GDSC2 5.0402 8.1014 2.1668 3.5714
EW-12 GDSC2 5.0578 7.5174 2.4332 2.1605
EW-13 GDSC1; GDSC2 5.0864 10.2044 1.2168 8.8352
CAL-72 GDSC1; GDSC2 5.173 10.1185 1.3148 8.1084
H-EMC-SS GDSC1; GDSC2 5.2149 15.1408 -1.0937 19.7417
U-CH2 GDSC2 5.3097 7.0628 2.7365 0.6369
CADO-ES1 GDSC1; GDSC2 5.5455 7.0661 2.8285 0.2739
CHSA8926 GDSC1; GDSC2 5.6227 14.2525 -0.3649 15.7444
HuO-3N1 GDSC1; GDSC2 5.659 14.4698 -0.4448 16.0211
A-673 GDSC1; GDSC2; CTRP2 5.6654 8.9249 4.2773 8.1926
SK-PN-DW GDSC1; GDSC2 5.6767 12.2441 0.6377 10.7622
EW-7 GDSC1; GDSC2 5.7656 7.7308 2.6733 0.566
EW-3 GDSC1; GDSC2 5.7829 8.0511 2.5598 0.9136
ES6 GDSC1; GDSC2 5.8114 7.8252 2.6568 0.5889
ES4 GDSC1; GDSC2 5.9719 8.0887 2.6239 0.5987
EW-18 GDSC1; GDSC2 6.1567 7.9301 2.7505 0.2381
TC-71 GDSC1; GDSC2 6.2635 14.2923 0.0519 12.4941
Hs 822.T CTRP2 6.2711 7.8313 5.3322 2.5837
TC71 CTRP2 6.2743 12.1843 3.1639 11.6096
SK-ES-1 GDSC1; GDSC2; CTRP2 6.2919 9.3677 4.5842 5.6763
NY GDSC1; GDSC2 6.3736 14.2861 0.1267 11.928
CAL-78 GDSC1; GDSC2; CTRP2 6.8747 8.7587 5.301 1.8386
ES8 GDSC1; GDSC2 6.889 16.5879 -0.6258 14.309
EW-11 GDSC1; GDSC2 6.9596 13.7451 0.7391 7.9427
SJSA-1 GDSC1; GDSC2; CTRP2 7.3988 15.3819 2.4507 12.4181
SK-N-MC CTRP2 7.4885 8.6439 5.6633 0.2179
MHH-ES-1 GDSC1; GDSC2; CTRP2 7.6561 20.2666 0.2277 19.4545
ES5 GDSC1; GDSC2 7.7132 18.9873 -1.2232 15.1886
Hs 888.T CTRP2 8.4711 9.9286 5.5761 0.1125
MG-63 GDSC1; GDSC2; CTRP2 8.4739 10.4307 5.3984 0.3756
SW1353 CTRP2 8.5718 9.9819 5.5933 0.0825
G-292 clone A141B1 GDSC1; GDSC2; CTRP2 8.6185 15.6385 3.1856 7.7752
U2OS GDSC1; GDSC2; CTRP2 9.1662 23.5589 -0.267 18.4199
HOS GDSC1; GDSC2; CTRP2 9.21 16.0393 3.374 6.3248
SaOS-2 GDSC1; GDSC2; CTRP2 11.0997 23.2919 1.1817 11.5132
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 213 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 5.4573 11.904 2.612 15.4592
JM1 GDSC1; GDSC2 5.6307 11.3643 1.0235 8.8132
EoL-1 GDSC1; GDSC2; CTRP2 -0.5736 1.2938 -0.5743 44.0918
NU-DUL-1 GDSC1; GDSC2 -0.3235 1.6528 -0.3542 36.7293
ALL-SIL GDSC1; GDSC2 -0.2326 1.5106 -0.2504 35.7575
KOPN-8 GDSC1; GDSC2 0.5039 3.7374 0.1237 30.1952
MY-M12 GDSC1; GDSC2 0.6752 2.1274 0.6515 26.6801
BCP-1 CTRP2 1.1996 7.4052 0.3316 34.8819
BONNA-12 GDSC2 2.404 7.4138 0.4683 20.4975
SU-DHL-5 GDSC1; GDSC2 2.4591 7.574 0.44 20.4572
Daudi GDSC1; GDSC2; CTRP2 3.2608 4.2574 3.2589 18.5512
BC-3 GDSC2 3.3413 6.8301 1.5839 10.9182
JSC-1 GDSC1; GDSC2 3.4632 9.8388 0.1805 18.6019
GA-10 GDSC1; GDSC2; CTRP2 3.7239 5.5732 3.6233 15.8045
KMS-11 GDSC1; GDSC2 3.8615 8.382 1.2263 11.6556
DB GDSC1; GDSC2; CTRP2 3.9463 7.7797 3.1254 17.0242
MOLM-13 GDSC1; GDSC2; CTRP2 4.0165 6.0427 3.8318 14.1562
MOLP-8 GDSC1; GDSC2; CTRP2 4.0224 10.6299 1.9066 21.4687
NK-92MI GDSC2 4.0256 8.3607 1.3622 10.4177
Kasumi-1 GDSC2; CTRP2 4.0936 9.5854 2.4679 19.188
CRO-AP2 GDSC1; GDSC2 4.1308 17.0854 -2.8979 28.2671
KO52 CTRP2 4.1803 5.9471 4.0357 12.9222
MV4-11 GDSC1; GDSC2; CTRP2 4.3509 5.8215 4.252 11.624
L-540 GDSC1; GDSC2; CTRP2 4.3874 8.7476 3.1477 15.7876
SCC-3 GDSC2 4.393 6.1295 2.6783 1.8196
RS4;11 GDSC1; GDSC2; CTRP2 4.4294 5.3145 4.4151 10.8074
KMS-12-BM GDSC2; CTRP2 4.4429 5.9269 4.3273 11.071
MOLT-16 GDSC1; GDSC2; CTRP2 4.4851 5.7695 4.4091 10.6497
Peer CTRP2 4.5317 6.6151 4.2088 11.2447
HAL-01 GDSC1; GDSC2 4.5384 7.0805 2.3336 3.479
KE-97 CTRP2 4.5831 11.1633 2.1843 19.0698
QIMR-WIL GDSC1; GDSC2 4.606 8.3625 1.7747 6.6077
SEM CTRP2 4.617 6.5503 4.3241 10.566
EM-2 GDSC1; GDSC2; CTRP2 4.6273 6.5177 4.3469 10.4506
Ramos.2G6.4C10 GDSC1; GDSC2 4.6518 6.0519 2.8419 0.7478
Pfeiffer CTRP2 4.6647 9.5207 3.0553 15.4769
SK-MM-2 GDSC1; GDSC2; CTRP2 4.718 6.6109 4.4105 9.9519
EB1 CTRP2 4.7285 11.2754 2.2649 18.4238
HC-1 GDSC1; GDSC2 4.7329 10.2391 0.957 11.0681
SUP-T1 GDSC1; GDSC2; CTRP2 4.7825 16.3131 -0.1761 26.2316
MHH-PREB-1 GDSC1; GDSC2 4.7969 6.825 2.5932 1.7067
NALM-6 GDSC1; GDSC2; CTRP2 4.8025 6.0859 4.6775 8.7124
ME1 CTRP2 4.8327 7.9092 3.9776 11.3488
DG-75 GDSC1; GDSC2 4.8424 7.1228 2.4891 2.1648
MLMA GDSC1; GDSC2 4.8876 13.5084 -0.5327 18.1835
Karpas-231 GDSC1; GDSC2 4.8918 6.2971 2.8517 0.5289
WSU-NHL GDSC1; GDSC2 4.9034 7.5287 2.3445 2.8287
BC-1 GDSC1; GDSC2 4.9118 6.9755 2.5882 1.592
JURL-MK1 GDSC1; GDSC2; CTRP2 4.9194 6.2254 4.7629 8.0506
KMS-21-BM CTRP2 4.934 14.75 0.7348 23.261
MOLT-4 GDSC1; GDSC2 4.9379 6.941 2.6157 1.4355
AML-193 CTRP2 4.938 7.5561 4.2441 10.014
P12-Ichikawa GDSC1; GDSC2; CTRP2 4.942 6.214 4.791 7.8799
TALL-1 [Human adult T-ALL] GDSC2; CTRP2 4.9587 11.1713 2.5282 16.8817
Ku812 GDSC1; GDSC2; CTRP2 4.9821 6.6737 4.6683 8.2284
OCI-Ly7 GDSC1; GDSC2 5.0348 7.8465 2.2773 2.989
HDLM-2 GDSC1; GDSC2; CTRP2 5.042 9.3849 3.4796 12.8744
DoHH2 GDSC1; GDSC2 5.0608 6.5931 2.8103 0.5556
H9 GDSC1; GDSC2 5.0921 6.798 2.745 0.7588
KMS-26 CTRP2 5.1396 6.2278 5.0014 6.5204
SUP-B15 GDSC1; GDSC2 5.1518 6.503 2.8802 0.3071
KG-1 GDSC1; GDSC2 5.1964 7.0859 2.6786 0.9244
CML-T1 GDSC1; GDSC2; CTRP2 5.2079 7.218 4.6693 7.6272
Sc-1 GDSC1 5.2119 6.7798 2.8025 0.6098
ALL-PO GDSC1; GDSC2 5.2208 7.731 2.4265 1.9915
RC-K8 GDSC1; GDSC2 5.2508 7.0253 2.7259 0.7117
Farage GDSC1; GDSC2 5.2655 13.2897 -0.1497 15.5537
ST486 GDSC1; GDSC2 5.2782 9.8978 1.4862 6.9415
U-698-M GDSC1; GDSC2 5.2793 7.8084 2.4236 1.9366
SUP-M2 GDSC1; GDSC2; CTRP2 5.2878 6.0772 5.2095 5.3158
OPM-2 GDSC1; GDSC2; CTRP2 5.2967 10.102 3.3631 12.7804
OCI-AML-3 GDSC1; GDSC2 5.3006 6.5363 2.9238 0.1649
MHH-CALL-2 GDSC1; GDSC2 5.3484 6.9718 2.7864 0.4627
WIL2 NS GDSC1; GDSC2 5.3521 6.7866 2.855 0.286
ROS-50 GDSC1; GDSC2 5.3819 7.5608 2.5743 1.1745
P32/ISH GDSC1; GDSC2 5.3869 6.6176 2.9267 0.1391
VAL GDSC1; GDSC2 5.4086 12.282 0.4391 12.3444
MOLT-13 GDSC1; GDSC2 5.4183 6.9414 2.8248 0.33
YT GDSC1; GDSC2 5.4216 6.7517 2.893 0.1864
Hs 445 GDSC2 5.4361 7.1128 2.7695 0.4652
CA46 GDSC1; GDSC2; CTRP2 5.4401 7.1311 4.9412 5.9524
L-428 GDSC1; GDSC2; CTRP2 5.4487 8.8268 4.1302 9.274
IM-9 GDSC1; GDSC2 5.4496 6.9311 2.8404 0.2823
A3/Kawakami GDSC1; GDSC2; CTRP2 5.5138 5.9873 5.4799 3.6524
Jiyoye GDSC1; GDSC2 5.5148 7.3033 2.7307 0.5344
Ri-1 CTRP2 5.5156 19.9765 -1.3671 27.5827
HH [Human lymphoma] GDSC1; GDSC2 5.5216 7.8573 2.52 1.2686
SUP-B8 GDSC1; GDSC2 5.5247 7.476 2.67 0.7164
PF-382 GDSC1; GDSC2; CTRP2 5.5312 9.1245 4.0582 9.3937
MOLT-3 CTRP2 5.5313 9.2192 4.0114 9.5883
SU-DHL-16 GDSC1; GDSC2 5.533 6.8775 2.8896 0.1634
TK [Human B-cell lymphoma] GDSC1; GDSC2 5.5456 7.0406 2.8375 0.2551
DEL GDSC1; GDSC2; CTRP2 5.5476 6.9371 5.1378 4.8921
THP-1 GDSC1; GDSC2; CTRP2 5.5476 6.467 5.3483 4.0522
Ki-JK CTRP2 5.5532 14.9468 1.1775 20.4868
KM-H2 GDSC1; GDSC2; CTRP2 5.5705 8.2152 4.5426 7.291
BL-41 GDSC1; GDSC2 5.5734 6.997 2.8629 0.1982
KY821 GDSC1; GDSC2 5.594 7.1678 2.8106 0.2952
U-937 CTRP2 5.6407 7.3361 5.0375 5.082
ML-2 GDSC1; GDSC2 5.6488 7.0184 2.8825 0.1479
Loucy GDSC1; GDSC2 5.6522 6.9631 2.9024 0.1193
EB2 GDSC1; GDSC2 5.6626 7.3758 2.7623 0.3795
BE-13 GDSC1; GDSC2 5.6706 7.145 2.8468 0.2003
BALL-1 GDSC1; GDSC2 5.6905 7.3752 2.7732 0.3427
GDM-1 GDSC1; GDSC2; CTRP2 5.6979 11.7739 2.886 13.8686
MEG-01 GDSC1; GDSC2 5.7173 8.3539 2.4113 1.5336
697 GDSC1; GDSC2; CTRP2 5.7182 12.9235 2.3294 16.0099
LC4-1 GDSC1; GDSC2 5.7326 7.9349 2.5829 0.8692
KE-37 GDSC1; GDSC2; CTRP2 5.7446 6.3791 5.59 2.5806
PL-21 GDSC1; GDSC2 5.7536 8.1712 2.5005 1.1491
TUR GDSC1; GDSC2 5.7632 7.2529 2.8428 0.1832
ME1 GDSC1; GDSC2 5.7834 6.9228 2.9603 0.045
ATN-1 GDSC1; GDSC2 5.7849 7.1891 2.8722 0.1345
Namalwa GDSC1; GDSC2; CTRP2 5.7858 7.6905 4.997 4.9284
CESS GDSC1; GDSC2 5.7924 7.6005 2.7313 0.4004
VL51 GDSC1; GDSC2 5.8446 8.35 2.4708 1.1881
MN-60 GDSC1; GDSC2 5.8465 7.6178 2.7457 0.3457
NU-DHL-1 CTRP2 5.8584 6.9547 5.4262 2.9812
SUP-T11 CTRP2 5.8798 8.0468 4.903 5.1252
NKM-1 GDSC1; GDSC2 5.9335 8.3011 2.5283 0.9178
OCI-M1 GDSC1; GDSC2; CTRP2 5.9428 6.7989 5.5795 2.1597
MOLM-6 CTRP2 5.9567 13.8097 2.0884 16.4353
RPMI-8866 GDSC1; GDSC2 5.9568 7.4071 2.8583 0.1212
CCRF-CEM GDSC1; GDSC2 5.9571 7.5829 2.7986 0.2079
ARH-77 GDSC1; GDSC2 5.9978 7.6541 2.7887 0.2143
Hs 611.T CTRP2 6.0007 26.941 -4.4404 32.1596
CTV-1 GDSC1; GDSC2 6.0093 7.5444 2.8302 0.1482
LP-1 GDSC1; GDSC2; CTRP2 6.0367 15.4603 1.33 18.9791
HuT 78 CTRP2 6.0544 8.0172 5.0663 4.0918
L-1236 GDSC1; GDSC2 6.0597 8.2381 2.6039 0.6096
RPMI-8226 GDSC1; GDSC2; CTRP2 6.0699 11.0603 3.5577 10.3833
KMS-20 CTRP2 6.0828 19.1761 -0.4894 24.3335
Mono-Mac-6 GDSC1; GDSC2; CTRP2 6.1799 10.2936 4.0316 8.1986
Karpas-45 GDSC1; GDSC2 6.301 8.055 2.7591 0.1896
DND-41 GDSC1; GDSC2; CTRP2 6.4245 10.4118 4.1688 7.1775
MOLP-2 CTRP2 6.4427 8.0481 5.352 2.2257
M-07e CTRP2 6.4733 10.637 4.095 7.3991
P30/OHK GDSC1; GDSC2 6.5095 7.9996 2.8488 0.0616
RCH-ACV GDSC1; GDSC2; CTRP2 6.5293 12.5217 3.2004 10.9889
NCI-H929 GDSC1; GDSC2; CTRP2 6.5432 18.8999 0.0274 22.0408
SUP-HD1 GDSC1; GDSC2; CTRP2 6.5835 13.4228 2.7943 12.5161
CTB-1 GDSC1; GDSC2 6.6181 15.1593 -0.1269 12.64
NCO2 CTRP2 6.6223 9.4016 4.8197 4.1342
GR-ST GDSC1; GDSC2 6.6531 8.5933 2.6998 0.2015
SU-DHL-1 GDSC2; CTRP2 6.7183 8.9373 5.1137 2.7866
SU-DHL-10 GDSC1; GDSC2; CTRP2 6.7889 7.8385 5.6655 0.6078
RPMI-8402 GDSC1; GDSC2; CTRP2 6.7898 10.4984 4.4039 5.5825
JJN-3 GDSC1; GDSC2; CTRP2 6.8417 12.5529 3.4284 9.5105
P31/FUJ GDSC1; GDSC2; CTRP2 6.8919 8.6287 5.3717 1.55
OCI-AML-2 GDSC1; GDSC2; CTRP2 7.0219 9.7573 4.9258 3.1162
OCI-AML-5 GDSC1; GDSC2; CTRP2 7.022 8.8689 5.3397 1.523
BL-70 CTRP2 7.0302 14.2259 2.7433 11.9211
KMOE-2 GDSC1; GDSC2 7.0567 15.9144 -0.2006 12.1647
KCL-22 GDSC1; GDSC2; CTRP2 7.1151 11.5213 4.1388 6.16
KMS-34 CTRP2 7.1466 21.8113 -0.9404 23.4909
JVM-2 GDSC1; GDSC2; CTRP2 7.1784 10.0773 4.8766 3.1029
WSU-DLCL2 GDSC1; GDSC2; CTRP2 7.2138 9.3453 5.2366 1.6933
RPMI-6666 GDSC1; GDSC2; CTRP2 7.2716 9.9177 5.0098 2.4727
TF-1 CTRP2 7.2888 10.1782 4.8996 2.8735
K-562 GDSC1; GDSC2; CTRP2 7.2964 11.4161 4.3168 5.1693
SIG-M5 GDSC2; CTRP2 7.3155 8.1523 5.7737 0.0885
Raji GDSC1; GDSC2; CTRP2 7.321 9.57 5.1975 1.7222
SU-DHL-4 GDSC1; GDSC2; CTRP2 7.3391 8.9129 5.4914 0.725
Reh GDSC1; GDSC2; CTRP2 7.3547 11.6837 4.2279 5.443
MHH-CALL-3 CTRP2 7.3652 10.0366 5.0121 2.355
MC116 GDSC1; GDSC2; CTRP2 7.4652 8.3584 5.7565 0.0809
Jurkat GDSC1; GDSC2; CTRP2 7.4661 10.6786 4.7778 3.1242
HEL 92.1.7 CTRP2 7.4674 8.5804 5.6783 0.1974
OCI-Ly19 GDSC1; GDSC2; CTRP2 7.4734 11.5097 4.3913 4.6246
NB4 GDSC1; GDSC2; CTRP2 7.5259 12.885 3.7662 7.0476
JeKo-1 GDSC1; GDSC2; CTRP2 7.5373 11.3051 4.5299 3.9946
SKM-1 GDSC1; GDSC2; CTRP2 7.5408 13.2558 3.5969 7.7033
RL GDSC1; GDSC2; CTRP2 7.5678 11.4619 4.4757 4.167
HL-60 GDSC1; GDSC2; CTRP2 7.6204 8.7577 5.6734 0.1604
U266B1 GDSC1; GDSC2; CTRP2 7.6356 12.3046 4.1205 5.4764
SU-DHL-8 GDSC1; GDSC2; CTRP2 7.7026 9.6927 5.3468 0.897
REC-1 CTRP2 7.7585 9.8891 5.2929 1.0181
HuNS1 CTRP2 7.8001 9.5697 5.4419 0.5747
BV-173 GDSC1; GDSC2; CTRP2 7.8181 9.913 5.3121 0.9188
CMK GDSC1; CTRP2 7.8204 8.8931 5.6996 0.0845
KMM-1 CTRP2 7.8255 12.6442 4.0846 5.3605
KHM-1B CTRP2 7.8729 13.43 3.7419 6.6443
AMO1 GDSC1; GDSC2; CTRP2 7.8766 9.3285 5.5661 0.2668
P3HR-1 CTRP2 7.9567 9.8265 5.4107 0.5697
MOLM-16 GDSC1; GDSC2; CTRP2 7.9834 16.4832 2.3395 11.8856
Karpas-422 GDSC1; GDSC2; CTRP2 7.9966 9.4662 5.563 0.2344
Karpas-620 GDSC1; GDSC2; CTRP2 8.0039 9.4417 5.5747 0.2129
Karpas-1106P GDSC1; GDSC2 8.0581 21.1895 -2.0401 17.4793
PL21 CTRP2 8.1417 10.1934 5.349 0.6257
KMS-18 CTRP2 8.1565 28.4273 -3.4393 27.0427
KMS-27 CTRP2 8.1783 9.7473 5.5317 0.2338
SU-DHL-6 GDSC1; GDSC2; CTRP2 8.2029 9.892 5.4887 0.3
SR GDSC1; GDSC2; CTRP2 8.2381 9.6049 5.6041 0.1201
L-363 GDSC1; GDSC2; CTRP2 8.2611 10.8967 5.122 1.1692
NOMO-1 GDSC1; GDSC2; CTRP2 8.429 9.6185 5.6658 0.0438
EHEB GDSC1; CTRP2 8.4753 17.471 2.2083 11.6108
OCI-Ly3 CTRP2 8.5941 21.7494 0.2022 17.9832
MHH-CALL-4 GDSC2; CTRP2 8.6245 10.5561 5.412 0.3032
Kasumi-2 CTRP2 8.7415 26.2333 -1.8999 23.089
Granta-519 GDSC1; GDSC2; CTRP2 8.8829 16.2836 3.0531 7.9223
Mono-Mac-1 CTRP2 8.9954 27.4035 -2.2866 23.5333
OCI-Ly10 CTRP2 9.0884 11.4635 5.2632 0.4186
A4/Fukuda GDSC1; GDSC2; CTRP2 9.1425 22.7146 0.129 17.3475
JVM-3 GDSC1; CTRP2 9.2232 21.57 0.7448 15.3956
MM1.S GDSC1; GDSC2; CTRP2 9.2872 25.8395 -1.2978 20.876
LAMA-84 GDSC1; GDSC2; CTRP2 9.3917 20.2268 1.5117 12.6941
F-36P CTRP2 10.0223 22.9817 0.6178 14.6385
EJM GDSC1; GDSC2; CTRP2 10.3962 21.668 1.4935 11.4039
KYO-1 CTRP2 10.6617 20.8017 2.0667 9.1928
HT GDSC1; GDSC2; CTRP2 10.671 21.0131 1.9745 9.4882
HPB-ALL CTRP2 11.0895 23.6727 0.9965 12.0947
Karpas-299 GDSC1; GDSC2; CTRP2 11.1665 23.2575 1.24 11.2514
HEL GDSC1; GDSC2; CTRP2 11.3099 23.9755 0.9951 11.8297
⏷ Show the Full List of 213 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 5.9797 7.9824 5.0209 4.4286
TE8 CTRP2 6.3579 9.2498 4.6949 5.0952
KYSE-450 GDSC1; GDSC2 4.4164 5.7864 2.8381 0.9975
KYSE-270 GDSC1; GDSC2 4.7927 7.6718 2.2161 3.703
T.T GDSC1; GDSC2 4.9505 9.0953 1.6534 6.621
OE33 GDSC1; GDSC2 5.0504 7.0559 2.6231 1.2841
KYSE-520 GDSC1; GDSC2 5.5522 10.734 1.2687 7.6324
KYSE-30 CTRP2 5.5694 8.476 4.4131 7.832
TE-15 GDSC1; GDSC2 5.6382 8.0818 2.4838 1.3103
KYSE-180 GDSC1; GDSC2; CTRP2 5.6784 16.9118 0.3027 22.9614
TE-8 GDSC1; GDSC2 5.8024 7.6848 2.7047 0.4626
TE-6 GDSC1; GDSC2; CTRP2 5.8677 7.9308 3.3687 1.0064
TE-5 GDSC1; GDSC2 5.89 7.4953 2.8047 0.2149
EC-GI-10 GDSC1; GDSC2 6.3337 16.6867 -1.0475 17.1194
KYSE-410 GDSC1; GDSC2; CTRP2 6.4779 8.5502 5.1319 3.0757
KYSE-140 GDSC1; GDSC2; CTRP2 6.5804 15.3573 1.8267 16.1831
TE-11 GDSC1; GDSC2; CTRP2 7.6454 9.8436 5.2548 1.2253
OE19 GDSC1; GDSC2; CTRP2 7.7771 9.9426 5.2798 1.0441
OE21 GDSC1; GDSC2 7.8613 17.7537 -0.5532 12.286
TE-9 GDSC1; GDSC2; CTRP2 7.8748 9.4745 5.5109 0.3775
TE-14 CTRP2 7.9582 9.996 5.3444 0.7387
KYSE-510 GDSC1; GDSC2; CTRP2 8.0353 14.9815 3.1066 8.897
TE-10 GDSC1; GDSC2; CTRP2 8.0913 10.2463 5.3055 0.7641
TE-4 GDSC1; GDSC2; CTRP2 8.167 17.4729 1.988 12.8746
COLO 680N GDSC1; GDSC2; CTRP2 8.4334 10.3407 5.4154 0.3577
KYSE-70 GDSC1; GDSC2; CTRP2 8.6234 14.0588 3.9281 4.9636
TE-1 GDSC1; GDSC2; CTRP2 8.6386 10.2082 5.5399 0.1243
KYSE-150 GDSC1; GDSC2; CTRP2 9.2709 15.6264 3.6005 5.428
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 75 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 5.3051 18.4987 -0.8091 26.7145
MZ-MEL-7 GDSC1; GDSC2 3.5053 5.4256 2.4187 5.2072
CP50-MEL-B GDSC1; GDSC2 3.5955 5.0218 2.6878 3.2864
MZ-MEL-2 GDSC1; GDSC2 3.7186 10.3738 0.1208 18.166
G-mel GDSC1; GDSC2 4.0211 13.788 -1.3404 23.6718
MMAc-SF GDSC1; GDSC2 4.1919 7.5924 1.8611 6.9911
COLO 783 GDSC1; GDSC2 4.4406 6.1435 2.6982 1.6489
LB2518-MEL GDSC1; GDSC2 4.4648 5.981 2.7807 1.2096
DJM-1 GDSC1; GDSC2 4.5264 6.4413 2.6148 1.9592
CP66-MEL GDSC1; GDSC2 4.7329 9.793 1.1735 9.8424
COLO 679 GDSC1; GDSC2 4.9079 8.2118 2.0382 4.5024
A-431 GDSC1; GDSC2 4.9539 11.1013 0.6941 12.0086
CHL-1 GDSC1; GDSC2 5.0683 6.898 2.6951 0.9679
A-388 GDSC1; GDSC2 5.1043 11.3737 0.6673 11.8158
COLO 800 GDSC1; GDSC2 5.1344 14.137 -0.6595 18.1457
WM1552C GDSC1; GDSC2 5.2281 7.3166 2.6012 1.2045
M14 GDSC1 5.2646 7.011 2.7372 0.8269
SH-4 GDSC1; GDSC2 5.3579 7.3787 2.6355 0.9574
451Lu GDSC1; GDSC2 5.3681 11.31 0.8775 10.123
VMRC-MELG GDSC2 5.3765 6.9573 2.8028 0.4037
UACC-257 GDSC1; GDSC2 5.4119 7.7603 2.508 1.4193
WM278 GDSC1; GDSC2 5.446 7.4822 2.6339 0.8952
GAK GDSC1; GDSC2 5.5262 6.9835 2.8504 0.2355
WM35 GDSC1; GDSC2 5.7579 12.3727 0.6301 10.6385
RVH-421 GDSC1; GDSC2; CTRP2 5.7859 9.7524 3.9708 9.2249
WM88 CTRP2 5.8523 8.9929 4.4072 7.2612
HMV-II GDSC1; GDSC2 6.0045 7.9549 2.6853 0.4235
SK-MEL-5 GDSC1; GDSC2; CTRP2 6.0101 11.7927 3.1416 12.2087
IST-MEL1 GDSC1; GDSC2 6.1172 7.8004 2.781 0.1975
COLO 829 GDSC1; GDSC2; CTRP2 6.2881 10.2617 4.1353 7.564
MeWo GDSC1; GDSC2; CTRP2 6.3443 8.2992 5.1562 3.1932
Hs 938.T GDSC1; GDSC2 6.3686 17.0752 -1.2109 17.6853
Hs 934.T CTRP2 6.3711 13.9746 2.3482 14.6448
WM115 GDSC1; GDSC2; CTRP2 6.4027 8.113 5.2914 2.537
WM983B CTRP2 6.5602 9.8702 4.5425 5.3845
Hs 688(A).T CTRP2 6.5683 8.651 5.1477 2.87
Mel Ho GDSC1; GDSC2; CTRP2 6.663 9.5464 4.7784 4.2399
WM266-4 CTRP2 6.6809 10.5184 4.3131 6.1357
HT-144 GDSC1; GDSC2; CTRP2 6.7208 9.2635 4.9577 3.4157
SK-MEL-28 GDSC1; GDSC2; CTRP2 6.7495 8.4857 5.3494 1.8076
Hs 895.T CTRP2 6.8539 9.4621 4.9541 3.236
IGR-37 GDSC1; GDSC2; CTRP2 6.9232 11.042 4.2347 6.0665
RPMI-7951 GDSC1; GDSC2; CTRP2 7.0308 8.4941 5.5111 0.909
WT2-iPS GDSC1; GDSC2; CTRP2 7.0893 10.4979 4.6168 4.2582
Hs 839.T CTRP2 7.3356 8.5221 5.6459 0.3151
Hs 940.T GDSC1; GDSC2; CTRP2 7.3532 9.3779 5.3005 1.3287
SK-MEL-2 GDSC1; GDSC2; CTRP2 7.4085 8.3103 5.7526 0.0967
SK-MEL-24 GDSC1; GDSC2; CTRP2 7.4261 10.1563 4.9939 2.354
COLO 741 CTRP2 7.505 9.9177 5.1469 1.7163
LB373-MEL-D GDSC1; GDSC2 7.5888 16.7667 -0.2648 11.5242
UACC-62 GDSC1; GDSC2; CTRP2 7.5911 13.1569 3.6801 7.2954
IGR-39 CTRP2 7.6042 9.4182 5.412 0.7744
IGR-1 GDSC1; GDSC2; CTRP2 7.6561 9.896 5.238 1.2708
A101D GDSC1; GDSC2; CTRP2 7.6838 10.3021 5.0767 1.7882
SK-MEL-30 GDSC1; GDSC2; CTRP2 7.7593 12.0889 4.3039 4.5897
Hs 294T CTRP2 7.7597 9.0944 5.6056 0.2335
Hs 944.T CTRP2 7.7832 11.0602 4.7946 2.6955
A2058 GDSC1; GDSC2; CTRP2 7.8156 9.5694 5.4489 0.5488
WM1799 CTRP2 7.8678 9.4626 5.5124 0.3771
K029AX CTRP2 7.9315 9.7061 5.4464 0.4966
SK-MEL-1 GDSC1; GDSC2; CTRP2 7.979 10.8512 4.9974 1.786
LOX-IMVI GDSC1; GDSC2; CTRP2 7.9945 9.713 5.4706 0.4137
HMCB CTRP2 8.0941 12.4779 4.3329 4.0647
MDA-MB-435S CTRP2 8.1228 9.3505 5.6504 0.0892
Hs 852.T CTRP2 8.1342 9.7553 5.5116 0.2811
SK-MEL-31 GDSC1; GDSC2; CTRP2 8.1694 9.4723 5.6252 0.1082
IPC-298 GDSC1; GDSC2; CTRP2 8.2561 9.3465 5.6976 0.0381
A-375 GDSC1; GDSC2; CTRP2 8.4994 14.3281 3.726 5.8761
WM793 GDSC1; GDSC2; CTRP2 8.5044 9.9214 5.5903 0.0937
COLO 792 GDSC1; GDSC2; CTRP2 8.616 10.3357 5.4874 0.1916
Mel JuSo GDSC1; GDSC2; CTRP2 9.5665 17.2778 3.0211 7.1832
Hs 936.T CTRP2 9.8052 17.6351 3.0026 6.9686
G-361 GDSC1; GDSC2; CTRP2 10.9371 21.1956 2.0539 8.9148
SK-MEL-3 GDSC1; GDSC2; CTRP2 11.7162 23.9823 1.2461 10.5876
EquiPSC Line K2 GDSC1; GDSC2 3.5262 11.3565 -0.5264 21.774
⏷ Show the Full List of 75 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ESO-51 GDSC1; GDSC2 4.1606 7.1794 2.0395 5.9758
OACM5.1 C GDSC1; GDSC2 4.4052 7.2896 2.1519 4.784
TE-12 GDSC1; GDSC2 4.7091 8.3171 1.8642 5.8732
HCE-4 GDSC1; GDSC2 5.0457 8.5544 1.9645 4.6766
KYSE-50 GDSC1; GDSC2 5.2601 7.5644 2.5155 1.5395
KYSE-220 GDSC1; GDSC2 5.4543 7.7155 2.5458 1.2248
KYAE-1 GDSC1; GDSC2 5.6483 7.6345 2.6615 0.6666
ESO-26 GDSC1; GDSC2 5.6591 7.7746 2.613 0.8172
OACP4 C GDSC1; GDSC2 6.5018 15.7174 -0.468 14.3794
SK-GT-4 GDSC1; GDSC2 7.0655 16.6051 -0.5191 13.5309
FLO-1 GDSC1; GDSC2 7.574 23.5196 -3.4902 22.62
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1; GDSC2; CTRP2 5.5336 9.5228 3.8631 10.2006
Cancer Drug Sensitivity Data Curated from 35 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SiMa GDSC1 4.0319 15.3731 -2.1227 29.4856
SK-N-DZ GDSC1; GDSC2 4.1764 7.5 1.895 6.8202
CHP-134 GDSC1 4.3675 6.3592 2.5608 3.107
GOTO GDSC1; GDSC2 4.4717 8.6745 1.5327 8.3329
KP-N-RT-BM-1 GDSC2 4.5488 8.8538 1.4997 8.3563
SJNB-5 GDSC1; GDSC2 4.8594 7.1322 2.4941 2.1167
IMR-5 GDSC1; GDSC2 4.8867 6.6837 2.6968 1.1299
SK-N-MC-IXC GDSC1; GDSC2 5.1075 10.342 1.1653 9.0807
CHP-126 GDSC1; GDSC2 5.22 7.1135 2.6782 0.9066
KP-N-YS GDSC1; GDSC2 5.2411 10.2321 1.3055 8.0251
KP-N-YN GDSC1; GDSC2; CTRP2 5.2859 9.8207 3.492 12.2745
NH-12 GDSC1; GDSC2 5.2984 7.1229 2.7088 0.7372
LA-N-6 GDSC1; GDSC2 5.3256 12.9649 0.0511 14.4604
NB(TU)1 GDSC1 5.4683 7.1565 2.7662 0.5705
SJNB-12 GDSC1; GDSC2 5.5001 8.2473 2.3503 2.0242
SJNB-6 GDSC1; GDSC2 5.5331 7.4558 2.6811 0.6751
SK-N-BE(2)-M17 GDSC1; GDSC2 5.7006 7.3894 2.772 0.3416
SJNB-10 GDSC1; GDSC2 5.7495 8.0268 2.5549 0.9545
SJNB-17 GDSC1; GDSC2 5.7523 8.4894 2.3729 1.6608
SJNB-7 GDSC1; GDSC2 5.8099 7.2144 2.8724 0.1295
SK-N-BE(2) CTRP2 5.8127 7.9389 4.8978 5.2865
GI-ME-N GDSC1; GDSC2 5.823 8.5582 2.3783 1.5713
NB69 GDSC1; GDSC2 5.9001 7.696 2.7381 0.3428
SJNB-14 GDSC1; GDSC2 6.0466 15.0955 -0.478 15.3416
CHP-212 GDSC1; GDSC2; CTRP2 6.1179 8.1621 5.0462 4.0561
TGW GDSC1; GDSC2 6.3689 13.8521 0.3279 10.9718
SK-N-AS GDSC1; GDSC2; CTRP2 6.41 10.1664 4.2796 6.7404
SJNB-13 GDSC1; GDSC2 6.453 8.0004 2.8297 0.0824
MHH-NB-11 GDSC1; GDSC2; CTRP2 7.3262 10.0003 5.0051 2.4262
Kelly GDSC1; GDSC2; CTRP2 7.332 10.4555 4.7974 3.215
SK-N-SH GDSC1; GDSC2; CTRP2 7.3437 10.1994 4.924 2.713
NH-6 CTRP2 7.6603 11.7792 4.3859 4.3977
KP-N-SI9s CTRP2 8.2881 11.6138 4.8325 2.0636
SK-N-FI GDSC1; GDSC2; CTRP2 9.1267 17.7038 2.54 9.4841
NB1 GDSC1; GDSC2; CTRP2 12.0692 22.0025 2.3507 6.7649
⏷ Show the Full List of 35 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-869 CTRP2 6.3528 10.5191 4.0586 7.7668
HuCC-T1 GDSC1; GDSC2; CTRP2 6.4397 8.6601 5.0495 3.478
SNU-478 CTRP2 7.5685 9.4874 5.3659 0.9364
SNU-308 CTRP2 7.8075 9.1832 5.592 0.2424
HuH-28 CTRP2 8.1128 9.6456 5.5431 0.2336
SNU-1196 CTRP2 8.2946 13.6565 3.9104 5.4294
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 86 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
BT-483 GDSC1; GDSC2 3.3349 4.7822 2.6026 4.5012
MFM-223 GDSC1; GDSC2 3.6865 5.9401 2.3029 5.4469
EFM-19 GDSC1; GDSC2 3.7118 6.4909 2.0494 6.9642
Evsa-T GDSC1; GDSC2 3.7994 9.3362 0.7029 14.8011
UACC-893 GDSC1; GDSC2 3.9146 6.7856 2.0557 6.4231
BT-549 GDSC1; GDSC2 4.0713 6.2035 2.4476 3.6855
HCC1428 GDSC1; GDSC2 4.2867 8.0069 1.7266 7.5644
MDA-MB-175-VII GDSC1; GDSC2 4.3264 5.9086 2.7387 1.5944
OCUB-M GDSC1; GDSC2 4.4711 6.5869 2.5185 2.55
HCC1599 GDSC2 4.8401 7.3063 2.4074 2.5811
YMB-1-E GDSC2 4.948 8.0308 2.1449 3.8391
HCC2157 GDSC1; GDSC2 5.0708 6.6567 2.7903 0.6152
MRK-nu-1 GDSC1; GDSC2 5.1459 6.5795 2.8501 0.3867
MDA-MB-330 GDSC1; GDSC2 5.2426 11.3166 0.7899 10.8586
MDA-MB-436 GDSC1; GDSC2 5.2457 8.0243 2.3143 2.4975
CAL-51 GDSC1; GDSC2; CTRP2 5.2817 7.0499 4.8199 6.8372
MDA-MB-453 GDSC1; GDSC2; CTRP2 5.3018 7.3623 4.6969 7.2816
DU4475 GDSC1; GDSC2; CTRP2 5.3585 6.1822 5.2541 4.9415
HCC70 GDSC1; GDSC2 5.4865 7.2401 2.7427 0.513
HCC2218 GDSC1; GDSC2; CTRP2 5.5579 9.5154 3.8885 10.0431
HCC1187 GDSC1; GDSC2 5.5934 12.0837 0.6588 10.7891
EFM-192A GDSC1; GDSC2 5.6404 7.8188 2.588 0.9131
HCC1500 GDSC1; GDSC2; CTRP2 5.6614 6.5822 5.4147 3.4927
MDA-MB-415 GDSC1; GDSC2 5.7336 12.1451 0.722 10.1792
HCC1569 GDSC1; GDSC2 5.7636 15.7876 -1.0118 18.1377
HCC38 GDSC1; GDSC2 5.9 7.8173 2.6947 0.4432
AU565 GDSC1; GDSC2; CTRP2 6.0117 10.1792 3.9496 8.8636
COLO 824 GDSC1; GDSC2 6.3364 8.7118 2.5398 0.6454
CAL-85-1 GDSC1; GDSC2; CTRP2 6.3502 11.0837 3.7748 8.954
BT-20 GDSC1; GDSC2; CTRP2 6.404 7.6547 5.5157 1.6167
HCC202 GDSC1 6.5053 8.3827 2.7194 0.2543
HMC-1-8 CTRP2 6.8697 9.1035 5.1359 2.4887
KPL-1 CTRP2 7.0394 7.8527 5.7754 0.1623
Hs 578T GDSC1; GDSC2; CTRP2 7.1407 9.4955 5.1243 2.1931
Hs 578Bst CTRP2 7.1931 12.8508 3.5446 8.4552
CAL-148 GDSC2; CTRP2 7.2688 9.2827 5.2959 1.4255
ZR-75-1 CTRP2 7.5136 8.8326 5.6029 0.3318
HCC1419 GDSC1; GDSC2; CTRP2 7.7093 9.1159 5.5773 0.3053
HDQ-P1 GDSC1; GDSC2; CTRP2 7.7319 10.2732 5.1155 1.6105
ZR-75-30 GDSC1; GDSC2; CTRP2 7.7589 12.9551 3.8924 6.2093
HCC1954 GDSC1; GDSC2; CTRP2 7.867 12.7247 4.0737 5.348
HCC1937 GDSC1; GDSC2; CTRP2 7.9283 10.7012 5.0352 1.7046
SK-BR-3 CTRP2 7.9633 11.0772 4.89 2.1686
CAL-120 GDSC1; GDSC2; CTRP2 8.0146 9.2646 5.6412 0.1169
CAMA-1 GDSC1; GDSC2; CTRP2 8.037 10.0505 5.3586 0.6572
MDA-MB-231 GDSC1; GDSC2; CTRP2 8.2067 13.9427 3.7192 6.2789
BT-474 GDSC1; GDSC2; CTRP2 8.2169 9.791 5.5308 0.2247
MDA-MB-157 GDSC1; GDSC2; CTRP2 8.2915 9.8234 5.5474 0.1815
MCF-7 GDSC1; GDSC2; CTRP2 8.3552 10.0979 5.4734 0.2793
HCC1806 GDSC1; GDSC2; CTRP2 8.4508 10.1087 5.506 0.2029
HCC1143 GDSC1; GDSC2; CTRP2 8.5913 10.9079 5.2675 0.6009
T-47D GDSC1; GDSC2; CTRP2 8.7573 15.9836 3.1131 7.8635
MDA-MB-468 GDSC1; GDSC2; CTRP2 8.8055 17.5156 2.4148 10.3816
HCC1395 GDSC1; GDSC2; CTRP2 9.1075 11.3379 5.3163 0.323
JIMT-1 GDSC1; GDSC2; CTRP2 10.2417 18.2667 2.9757 6.5716
MDA-MB-361 GDSC1; GDSC2; CTRP2 12.9922 31.0959 -1.2723 15.9521
BT 416 CTRP2 5.0295 7.2755 4.4627 8.9078
BT 172 CTRP2 6.0621 6.9339 5.6143 1.774
BT 245 CTRP2 6.216 8.0333 5.1891 3.2771
BT147 CTRP2 6.273 7.4152 5.5389 1.722
BT 286 CTRP2 6.4303 7.6295 5.5458 1.4575
BT 216 CTRP2 6.4767 8.0124 5.3932 2.0068
BT 248 CTRP2 6.5227 9.0627 4.913 3.9083
BT 428 CTRP2 6.7137 9.0512 5.0556 3.0283
BT 482 CTRP2 6.7182 8.3037 5.4147 1.5937
BT 228 CTRP2 6.8782 8.3022 5.5113 1.0531
BT 333 CTRP2 7.0761 8.6348 5.4743 0.992
BT 187 CTRP2 7.1427 8.6833 5.4888 0.8856
BT 504 CTRP2 7.2359 8.809 5.4834 0.827
BT 320 CTRP2 7.2934 8.9087 5.4705 0.8225
BT 131 CTRP2 7.4385 8.6478 5.6415 0.2801
BT 330 CTRP2 7.4483 10.9371 4.6457 3.6572
BT 139 CTRP2 7.5704 8.9223 5.5927 0.3296
BT 179 CTRP2 7.6587 10.3526 5.0404 1.9395
BT 444 CTRP2 7.7011 9.2542 5.5213 0.4316
BT 340 CTRP2 7.7237 9.0706 5.6 0.2556
BT 359 CTRP2 7.8707 9.1345 5.6338 0.1569
BT 232 CTRP2 7.8718 9.2986 5.5751 0.2519
BT 239 CTRP2 7.8856 9.1941 5.6182 0.1762
BT 422 CTRP2 7.9046 9.0755 5.6669 0.1066
BT 328 CTRP2 7.9161 9.9841 5.3297 0.8043
BT 271 CTRP2 7.9811 9.3617 5.5946 0.1877
BT 159 CTRP2 8.0703 9.259 5.663 0.0842
BT 224 CTRP2 8.5667 9.9903 5.5887 0.0871
BT 440 CTRP2 10.0191 18.3171 2.8191 7.3691
BT 231 CTRP2 10.447 22.7996 0.9906 12.9296
⏷ Show the Full List of 86 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 7.5897 9.2969 5.4544 0.6638
Cancer Drug Sensitivity Data Curated from 69 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MOG-G-UVW GDSC1; GDSC2 4.3631 6.5356 2.4776 2.9692
KNS-60 CTRP2 4.616 7.1529 4.0875 11.4764
SK-MG-1 GDSC1; GDSC2 4.7083 8.4096 1.82 6.1334
PFSK-1 GDSC1; GDSC2 4.9912 12.3389 0.1176 14.9007
D-566MG GDSC1; GDSC2 4.9978 6.8276 2.6908 1.0484
LN-405 GDSC1; GDSC2 5.0599 6.8875 2.6954 0.9739
Onda 10 GDSC1; GDSC2 5.0878 10.2066 1.2167 8.8331
D-263MG GDSC1; GDSC2 5.0986 6.6264 2.8135 0.5221
LNZTA3WT4 GDSC1; GDSC2 5.3973 10.3213 1.3636 7.3999
GI-1 GDSC1; GDSC2 5.4707 9.5195 1.7779 4.9895
DK-MG GDSC1; GDSC2 5.4989 6.8458 2.8883 0.174
D-245MG GDSC2 5.5192 9.8658 1.6492 5.6087
KS-1 [Human Krukenberg tumour] GDSC1; GDSC2 5.569 7.9727 2.4957 1.3243
Onda 11 GDSC1; GDSC2 5.6176 10.0591 1.6197 5.6031
Daoy GDSC1; GDSC2; CTRP2 5.652 6.4818 5.4499 3.3761
M059J GDSC1; GDSC2 5.7519 7.5053 2.75 0.3724
SF126 GDSC1; GDSC2; CTRP2 5.8251 6.7245 5.5079 2.7174
KINGS-1 GDSC1; GDSC2 5.9146 7.8199 2.6993 0.4271
D-392MG GDSC1; GDSC2 6.0006 8.101 2.6308 0.5651
H4 GDSC1; GDSC2 6.0389 7.75 2.7703 0.2351
D-247MG GDSC1; GDSC2 6.0516 7.8253 2.7488 0.2709
GB-1 GDSC1; GDSC2; CTRP2 6.1495 7.5019 5.4012 2.5074
D-502MG GDSC1; GDSC2 6.4089 16.0896 -0.7086 15.5884
SNU-626 CTRP2 6.4614 12.03 3.3916 10.3329
SW1783 GDSC1; GDSC2; CTRP2 6.4841 10.8189 4.0129 7.722
Hs 683 GDSC1; GDSC2; CTRP2 6.5016 8.5003 5.1735 2.8668
D-336MG GDSC1; GDSC2 6.5759 8.7316 2.6242 0.3508
SF539 GDSC1; GDSC2; CTRP2 6.6868 9.9148 4.615 4.8761
D-423MG GDSC1; GDSC2 6.7207 8.8605 2.6321 0.2936
SNU-738 CTRP2 6.756 10.5795 4.3391 5.9047
SW1088 GDSC1; GDSC2; CTRP2 6.7588 8.5425 5.3287 1.8764
42-MG-BA GDSC1; GDSC2; CTRP2 6.9349 11.7539 3.8935 7.4504
U-251MG GDSC1; GDSC2; CTRP2 6.9746 8.515 5.4711 1.099
KNS-81-FD GDSC1; GDSC2 6.9878 14.9088 0.2238 10.3539
SNU-489 CTRP2 7.0464 8.8026 5.3837 1.3371
MOG-G-CCM GDSC1; GDSC2 7.088 15.9381 -0.1919 12.0704
SNU-1105 CTRP2 7.1964 8.7278 5.4976 0.8135
SNU-466 CTRP2 7.2114 8.2525 5.6962 0.2581
GaMG GDSC1; GDSC2; CTRP2 7.2131 10.3353 4.7773 3.4476
YKG-1 GDSC1; GDSC2; CTRP2 7.2606 8.6524 5.5605 0.5774
GMS-10 CTRP2 7.3106 8.6345 5.591 0.463
KNS-81 CTRP2 7.3746 9.2951 5.348 1.1496
SF295 GDSC1; GDSC2; CTRP2 7.4171 8.8058 5.5713 0.4545
NMC-G1 GDSC1; GDSC2; CTRP2 7.5257 9.8177 5.2024 1.5044
LN-18 GDSC1; GDSC2; CTRP2 7.552 8.5774 5.7118 0.1206
U-118MG GDSC1; GDSC2; CTRP2 7.6605 9.2124 5.5199 0.4548
YH-13 GDSC1; GDSC2; CTRP2 7.8432 9.1822 5.6063 0.2068
D283 Med GDSC1; GDSC2; CTRP2 7.8732 9.8745 5.3539 0.7645
D-542MG GDSC1; GDSC2 7.9154 22.8484 -2.929 20.4769
T98G GDSC1; GDSC2; CTRP2 7.9159 12.3529 4.28 4.4834
ONS-76 GDSC1; GDSC2; CTRP2 7.9171 14.1064 3.4472 7.741
KNS-42 GDSC1; GDSC2; CTRP2 7.9195 9.2376 5.6156 0.1717
SF268 GDSC1; GDSC2; CTRP2 7.9342 13.9538 3.5322 7.3827
CCF-STTG1 CTRP2 7.9432 9.6312 5.4801 0.415
U-87MG ATCC GDSC1; GDSC2; CTRP2 7.953 9.2859 5.611 0.1702
KG-1-C CTRP2 7.9805 9.2782 5.624 0.1456
8-MG-BA GDSC1; GDSC2; CTRP2 7.9845 10.4141 5.1862 1.1754
KALS-1 GDSC1; GDSC2; CTRP2 8.0297 10.2107 5.2914 0.8393
AM-38 GDSC1; GDSC2; CTRP2 8.0779 27.6215 -3.0999 26.5509
CAS-1 GDSC1; GDSC2; CTRP2 8.085 9.2714 5.664 0.0812
M059K CTRP2 8.1159 9.5776 5.5686 0.1927
Becker GDSC1; GDSC2; CTRP2 8.1795 9.6642 5.5618 0.1871
GOS-3 CTRP2 8.2892 9.527 5.6487 0.0692
LN-229 GDSC1; GDSC2; CTRP2 8.3708 9.5995 5.6524 0.0577
DBTRG-05MG GDSC1; GDSC2; CTRP2 8.3852 10.7031 5.2573 0.7254
A-172 GDSC1; GDSC2; CTRP2 8.7644 17.8643 2.219 11.1472
SNB-75 GDSC1; GDSC2; CTRP2 9.0137 10.9157 5.4305 0.1838
SNU-201 CTRP2 10.3451 23.4666 0.6044 14.2385
TM-31 CTRP2 11.9027 22.191 2.1726 7.4912
⏷ Show the Full List of 69 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TGBC1TKB GDSC1; GDSC2 5.0267 6.5782 2.8016 0.607
TGBC24TKB GDSC1; GDSC2 5.7038 8.5905 2.3083 1.9915
ETK-1 GDSC1; GDSC2 6.4572 8.3566 2.7113 0.2277
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-2 CTRP2 5.3384 14.0975 1.4153 20.1404
MFE-280 GDSC1; GDSC2 5.6968 7.8075 2.6164 0.781
JHUEM-1 CTRP2 5.8501 6.5101 5.6348 2.1374
HEC-151 CTRP2 6.0458 7.1052 5.5151 2.222
HEC-1-A CTRP2 6.1526 8.0401 5.1352 3.6178
AN3-CA GDSC1; GDSC2; CTRP2 6.1955 12.0314 3.1758 11.7106
MFE-319 GDSC1; GDSC2; CTRP2 6.568 8.0687 5.4283 1.7361
KLE GDSC1; GDSC2; CTRP2 6.8606 16.7769 1.3423 17.3562
MFE-296 GDSC1; GDSC2; CTRP2 6.8877 10.2715 4.5857 4.6821
EFE-184 CTRP2 6.9563 8.6087 5.4189 1.3045
HEC-6 CTRP2 7.424 11.553 4.3377 4.9055
HEC-265 CTRP2 7.6268 8.8903 5.6277 0.237
ESS-1 GDSC1; GDSC2; CTRP2 7.7812 10.172 5.1851 1.3378
RL95-2 GDSC1; GDSC2; CTRP2 7.8763 9.0751 5.6568 0.1244
HEC-59 CTRP2 8.0986 9.3724 5.6342 0.1101
HEC-108 CTRP2 8.1209 9.4104 5.6291 0.1121
EN GDSC1; GDSC2; CTRP2 8.1709 9.3294 5.6743 0.0617
HEC-251 CTRP2 8.2288 9.9355 5.483 0.3019
HEC-1-B CTRP2 8.4433 9.8792 5.5832 0.1094
HEC-50B CTRP2 8.5444 10.5728 5.3742 0.3969
Ishikawa (Heraklio) 02 ER- CTRP2 7.7959 8.6994 5.7565 0.0385
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KTCTL-140 GDSC1; GDSC2 3.7404 11.9013 -0.6242 21.5847
LB2241-RCC GDSC1; GDSC2 4.4059 9.4227 1.121 10.9018
KTCTL-195 GDSC1; GDSC2 4.6656 8.0122 1.9798 5.2841
NCC021 GDSC1; GDSC2 4.8723 8.5384 1.8648 5.5555
BB65-RCC GDSC1; GDSC2 5.1807 10.1824 1.2896 8.2344
KTCTL-1M GDSC1; GDSC2 5.2811 15.019 -0.985 19.1553
SW156 GDSC1; GDSC2 5.3808 13.6045 -0.2209 15.6243
SN12C GDSC1; GDSC2 5.3848 7.8399 2.4625 1.6432
UO-31 GDSC1; GDSC2; CTRP2 5.4412 9.8146 3.6356 11.3432
A-704 GDSC1; GDSC2 5.5046 12.0478 0.6166 11.2241
BFTC-909 GDSC1; GDSC2 5.5537 8.4592 2.2884 2.2503
LB996-RCC GDSC1; GDSC2 5.6976 8.3173 2.4169 1.5288
KTCTL-13 GDSC1; GDSC2 5.7026 14.0683 -0.2199 14.9119
CAL-54 GDSC1; GDSC2; CTRP2 5.8129 8.7926 4.4729 7.0664
NCC010 GDSC1; GDSC2 5.826 17.3251 -1.7183 20.6903
SW13 GDSC1; GDSC2 5.8436 7.4218 2.8134 0.2122
LB1047-RCC GDSC1; GDSC2 6.1181 17.615 -1.6496 19.8256
VMRC-RCZ GDSC1; GDSC2; CTRP2 6.3684 7.9086 5.3666 2.2812
TK-10 GDSC1; GDSC2 6.4394 8.5289 2.645 0.3531
KTCTL-26A GDSC1; GDSC2 6.6537 16.45 -0.7161 15.1366
RXF 393L GDSC1; GDSC2 6.7319 17.068 -0.959 15.9744
SNU-1272 CTRP2 6.7677 8.8686 5.1801 2.4511
TUHR4TKB CTRP2 7.053 13.2575 3.24 9.9141
KMRC-2 CTRP2 7.0773 10.2875 4.7097 3.9015
KMRC-3 CTRP2 7.2771 15.9196 2.0927 13.9596
RCC10RGB GDSC1; GDSC2; CTRP2 7.3602 8.6164 5.6202 0.3633
TUHR10TKB CTRP2 7.5861 8.7436 5.6653 0.1832
A-498 GDSC1; GDSC2; CTRP2 7.7849 9.4815 5.4697 0.5135
Caki-2 CTRP2 7.966 11.3933 4.7508 2.66
OS-RC-2 GDSC1; GDSC2; CTRP2 8.0244 11.1494 4.892 2.1032
KMRC-1 GDSC1; GDSC2; CTRP2 8.109 10.3907 5.2558 0.8878
769-P GDSC1; GDSC2; CTRP2 8.2444 9.8257 5.5288 0.2203
Caki-1 GDSC1; GDSC2; CTRP2 8.3218 15.889 2.8665 9.3983
TUHR14TKB CTRP2 8.3252 16.6378 2.507 10.7414
KTCTL-21 GDSC1; GDSC2 8.3265 24.4111 -3.3997 21.0807
786-O GDSC1; GDSC2; CTRP2 8.3654 13.8762 3.8524 5.5621
HA7-RCC GDSC1; GDSC2 8.5425 22.038 -2.1251 16.9416
VMRC-RCW GDSC1; GDSC2; CTRP2 8.9107 18.3504 2.0853 11.4123
KMRC-20 GDSC1; GDSC2; CTRP2 9.2108 15.6381 3.5591 5.6467
ACHN GDSC1; GDSC2; CTRP2 10.0921 17.8642 3.07 6.4072
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 57 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H716 GDSC1; GDSC2 4.0607 6.8855 2.112 5.7579
C2BBe1 GDSC1; GDSC2 4.1823 7.3212 1.986 6.253
SNU-175 GDSC2 4.3378 9.2104 1.1754 10.7501
GP5d GDSC1; GDSC2 4.6222 6.9608 2.4379 2.7588
SW1116 GDSC1; GDSC2 5.0061 8.688 1.8788 5.2291
SNU-283 GDSC2 5.1022 6.6674 2.7995 0.5643
SNU-81 GDSC1; GDSC2 5.1686 6.9655 2.7134 0.816
SW1463 GDSC1; GDSC2 5.3303 7.4813 2.5824 1.1878
KM12 GDSC1; GDSC2; CTRP2 5.4596 8.0569 4.5171 7.6455
NCI-H747 GDSC1; GDSC2; CTRP2 5.4747 7.3829 4.8565 6.2137
LS1034 GDSC1; GDSC2 5.5041 7.0397 2.8223 0.3023
SNU-C1 GDSC1; GDSC2; CTRP2 5.5065 7.4121 4.8732 6.07
RCM-1 [Human ESC] GDSC1; GDSC2 5.5978 6.9596 2.8845 0.1562
HCC2998 GDSC1; GDSC2 5.6332 7.8041 2.5906 0.9123
SW626 GDSC1; GDSC2 5.6754 7.6797 2.6557 0.6685
COLO 320 CTRP2 5.7392 10.9395 3.3381 11.9473
SW837 GDSC1; GDSC2 5.803 7.8089 2.6595 0.5857
DiFi GDSC1; GDSC2 5.8096 7.9332 2.6158 0.7126
LS180 GDSC1; GDSC2; CTRP2 5.9458 6.8898 5.537 2.3311
COLO 320HSR GDSC1; GDSC2 6.1488 7.7865 2.7969 0.1667
CL-11 GDSC1; GDSC2; CTRP2 6.1621 8.1125 5.1067 3.72
CaR-1 GDSC1; GDSC2 6.1863 7.8307 2.7951 0.1617
T84 GDSC1; GDSC2; CTRP2 6.1915 8.6111 4.8815 4.6113
COLO 678 GDSC1; GDSC2 6.414 7.8704 2.8594 0.0624
SNU-1033 CTRP2 6.5839 8.8953 5.0397 3.2886
SNU-61 GDSC1; GDSC2; CTRP2 6.7158 8.5543 5.2952 2.0648
SNU-C2B GDSC1; GDSC2 6.9809 8.9772 2.6841 0.1611
HCT 8 CTRP2 7.2471 11.6685 4.1606 5.8719
SNU-C4 CTRP2 7.269 9.0137 5.4133 1.0253
HCT 116 GDSC1; GDSC2; CTRP2 7.2696 10.4692 4.7508 3.4774
HT115 GDSC1; GDSC2; CTRP2 7.4485 8.9757 5.518 0.5768
HCC-56 CTRP2 7.5076 8.6236 5.6783 0.1847
COLO205 GDSC1; GDSC2; CTRP2 7.6133 8.9122 5.6142 0.2678
RKO GDSC1; GDSC2; CTRP2 7.6334 10.5883 4.9203 2.3974
SW948 GDSC1; GDSC2; CTRP2 7.6425 20.0671 0.3163 19.2176
DLD-1 CTRP2 7.6617 8.6822 5.7154 0.0937
OUMS-23 CTRP2 7.7397 9.1809 5.5655 0.3178
LS411N GDSC1; GDSC2; CTRP2 7.7521 9.1067 5.598 0.2497
HT-55 GDSC1; GDSC2; CTRP2 7.7523 9.0224 5.6288 0.1956
SK-CO-1 GDSC1; GDSC2; CTRP2 7.7704 9.9288 5.2822 1.0418
LS123 GDSC1; GDSC2; CTRP2 7.787 9.4352 5.4886 0.4671
HT-29 GDSC1; GDSC2; CTRP2 7.8035 8.829 5.7155 0.0709
SNU-407 GDSC1; GDSC2; CTRP2 7.9332 10.3184 5.2006 1.1695
MDST8 GDSC1; GDSC2; CTRP2 7.9701 9.2042 5.646 0.1194
LS513 GDSC1; GDSC2; CTRP2 8.0214 9.5091 5.5571 0.2369
SW620 GDSC1; GDSC2; CTRP2 8.1339 9.985 5.4259 0.4513
LoVo GDSC1; GDSC2; CTRP2 8.1525 17.8742 1.7811 13.6291
NCI-H508 GDSC1; GDSC2; CTRP2 8.179 9.5947 5.5862 0.1535
CW-2 GDSC1; GDSC2; CTRP2 8.2168 9.989 5.4585 0.3518
HCT 15 GDSC1; GDSC2; CTRP2 8.305 9.9595 5.504 0.2433
SW1417 GDSC1; GDSC2; CTRP2 8.3259 10.0924 5.4639 0.3048
SNU-C5 GDSC1; GDSC2; CTRP2 8.4405 17.8014 2.0233 12.3267
COLO201 CTRP2 8.814 18.2223 2.0805 11.5686
SNU-503 CTRP2 9.4971 19.3065 2.0231 10.8133
SNU-C2A CTRP2 9.6429 22.9484 0.3711 15.9068
SW48 GDSC1; GDSC2; CTRP2 9.9871 21.4868 1.3103 12.5318
CCK-81 GDSC1; GDSC2; CTRP2 10.1275 22.9986 0.6814 14.3023
⏷ Show the Full List of 57 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1; GDSC2 5.2779 6.9016 2.784 0.5078
Cancer Drug Sensitivity Data Curated from 25 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-182 CTRP2 4.4577 19.3617 -1.9788 31.0669
SNU-449 GDSC1; GDSC2 4.8611 8.2321 2.0003 4.8008
SNU-761 CTRP2 4.9301 7.9134 2.8231 4.4747
JHH-7 GDSC1; GDSC2 5.0669 8.2621 2.11 3.8373
Li-7 CTRP2 5.0853 7.4865 4.424 8.9207
SNU-878 CTRP2 5.3733 9.7874 3.5879 11.6877
HuH-6 CTRP2 5.9578 9.579 4.2044 7.9017
HLE GDSC1; GDSC2 6.2545 7.9344 2.7838 0.1639
JHH-2 GDSC1; GDSC2; CTRP2 6.4974 8.665 5.0898 3.2183
HLF CTRP2 6.8904 10.1668 4.6386 4.4622
Huh-7 GDSC1; GDSC2 7.0116 18.6974 -1.5506 17.6835
JHH-6 GDSC1; GDSC2; CTRP2 7.3713 8.4602 5.6841 0.2195
SNU-423 GDSC1; GDSC2; CTRP2 7.5558 12.5283 3.9592 6.2312
Hep-G2/C3A GDSC1; GDSC2 7.6662 18.2315 -0.8981 14.0133
SK-HEP-1 GDSC1; GDSC2; CTRP2 7.7785 9.2472 5.5565 0.3209
SNU-475 CTRP2 7.7863 8.9646 5.6624 0.1361
JHH-1 GDSC1; GDSC2; CTRP2 7.8578 8.9048 5.7088 0.0699
Hep 3B2.1-7 GDSC1; GDSC2; CTRP2 7.9029 13.797 3.5862 7.2151
HuH-1 GDSC1; GDSC2; CTRP2 7.9089 9.9334 5.3467 0.7621
Hep-G2 CTRP2 7.9147 9.0436 5.6816 0.0887
PLC/PRF/5 CTRP2 8.34 11.0014 5.117 1.1299
JHH-4 GDSC1; GDSC2; CTRP2 10.3458 19.1147 2.651 7.5785
SNU-398 GDSC1; GDSC2; CTRP2 10.4793 21.7905 1.4894 11.3114
JHH-5 CTRP2 11.0629 22.8425 1.3684 10.9751
SNU-387 GDSC1; GDSC2; CTRP2 13.2974 25.8957 1.3131 8.7183
⏷ Show the Full List of 25 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 217 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H748 GDSC2 2.0936 5.6561 1.0212 18.5071
ChaGo-K-1 GDSC1; GDSC2 2.5491 5.9429 1.3225 15.0609
NCI-H2804 GDSC1; GDSC2 3.2266 6.2346 1.7853 9.9995
NCI-H1385 CTRP2 3.3425 6.4678 2.9701 19.3204
LC-2/ad GDSC1; GDSC2 3.6754 7.2692 1.6346 9.6693
NCI-H250 GDSC2 3.6982 7.1201 1.7266 9.0378
NCI-H2171 GDSC2 3.9787 6.299 2.3389 4.5535
NCI-H1437 GDSC1; GDSC2 4.0106 10.2984 0.3897 15.9717
HCC33 GDSC2 4.0209 6.5144 2.264 4.9176
NCI-H146 GDSC1; GDSC2 4.1237 8.4303 1.4012 9.9386
NCI-H720 GDSC1 4.147 5.5278 2.807 1.8715
NCI-H2135 GDSC1; GDSC2 4.1841 6.6837 2.2939 4.3868
NCI-H510A GDSC1; GDSC2 4.2248 7.1438 2.101 5.4622
NCI-H2029 GDSC1; GDSC2 4.2295 6.1556 2.571 2.6734
NCI-H1836 GDSC1; GDSC2 4.2847 5.7649 2.7788 1.4516
NCI-H345 GDSC1; GDSC2 4.3326 5.5168 2.9086 0.7714
Ms-1 GDSC1; GDSC2 4.4108 9.1519 1.2571 10.099
NCI-H1703 GDSC1; GDSC2; CTRP2 4.4151 9.9617 2.6043 17.862
PC-14 GDSC1; GDSC2; CTRP2 4.4375 6.9449 3.9831 12.3685
NCI-H1304 GDSC1 4.4757 6.0799 2.7443 1.7091
SBC-1 GDSC1; GDSC2 4.5572 6.8626 2.4444 2.8273
NCI-H2405 GDSC1; GDSC2; CTRP2 4.5575 9.8252 2.8068 16.7229
NCI-H1781 GDSC1; GDSC2 4.5857 6.4134 2.659 1.6522
COR-L303 GDSC2 4.5969 9.1734 1.3786 8.9603
NCI-H2803 GDSC2 4.6218 7.7416 2.0787 4.7926
A-427 GDSC1; GDSC2 4.6364 7.4106 2.2415 3.8292
EMC-BAC-1 GDSC1; GDSC2 4.6769 11.8024 0.1511 15.4865
COR-L279 GDSC1; GDSC2 4.6804 6.0344 2.8617 0.6471
HCC44 GDSC1; GDSC2; CTRP2 4.6864 6.2952 4.487 9.7567
NCI-H2810 GDSC1; GDSC2 4.6981 9.5358 1.2737 9.3439
NCI-H889 CTRP2 4.7226 9.5048 3.1186 15.0851
NCI-H647 GDSC1; GDSC2 4.7706 7.3827 2.334 3.0891
SBC-3 GDSC1; GDSC2 4.7794 6.9551 2.528 2.0528
NCI-H2170 GDSC1; GDSC2 4.7915 10.5381 0.8531 11.5118
NCI-H1341 GDSC1; GDSC2; CTRP2 4.8111 7.4912 4.1441 10.7381
COR-L321 GDSC1; GDSC2 4.8142 7.7767 2.1811 3.8621
DMS 53 GDSC1; GDSC2; CTRP2 4.8192 7.9506 3.9451 11.5128
NCI-H82 GDSC1; GDSC2 4.8436 8.2783 1.968 5.017
IST-SL1 GDSC1; GDSC2 4.8595 11.8492 0.2619 14.4886
NCI-H1648 GDSC1; GDSC2 4.9623 7.2632 2.4921 1.9925
NCI-H740 GDSC2 5.0034 8.6901 1.8761 5.2488
NCI-H1688 GDSC1; GDSC2 5.0073 6.941 2.6493 1.214
NCI-H596 GDSC1; GDSC2 5.0843 6.55 2.8362 0.4605
NCI-H1650 GDSC1; GDSC2; CTRP2 5.124 7.7545 4.3386 9.1693
NCI-H187 GDSC1 5.1392 6.2437 2.9668 0.1668
Lu-134-A GDSC1; GDSC2 5.1494 12.4027 0.1997 14.1278
NCI-H2369 GDSC1; GDSC2 5.1552 13.737 -0.448 17.1724
NCI-H1963 GDSC2 5.1581 7.6566 2.4259 2.0703
NCI-H810 GDSC1; GDSC2 5.1597 7.0515 2.6756 0.9661
NCI-H2106 CTRP2 5.1857 8.2694 4.1547 9.7718
VMRC-LCD GDSC1; GDSC2 5.194 7.2602 2.608 1.2081
NCI-H211 GDSC1; GDSC2; CTRP2 5.2259 6.3896 5.0378 6.1346
NCI-H2731 GDSC1; GDSC2 5.2368 9.2926 1.7414 5.5892
NCI-H2087 GDSC1; GDSC2; CTRP2 5.2412 11.6873 2.5285 16.252
COR-L23 GDSC1; GDSC2 5.2423 10.7452 1.0629 9.3715
NCI-H1436 GDSC1; GDSC2 5.3152 11.788 0.6128 11.6443
CPC-N GDSC1; GDSC2 5.3171 7.2372 2.6727 0.8515
NCI-H1876 GDSC1; GDSC2 5.3194 7.4745 2.5801 1.207
NCI-H3255 GDSC1; GDSC2 5.343 7.7709 2.4707 1.651
NCI-H1581 GDSC1; GDSC2; CTRP2 5.4328 8.7088 4.1735 9.1292
Lu-139 GDSC1; GDSC2 5.437 7.0419 2.7958 0.3941
Lu-165 GDSC1; GDSC2 5.4371 7.1547 2.7544 0.5075
NCI-H1770 GDSC1; GDSC2 5.4411 7.1591 2.7544 0.5053
NCI-H2444 GDSC1; GDSC2; CTRP2 5.4427 7.4993 3.3347 1.514
DMS 79 GDSC1; GDSC2; CTRP2 5.47 7.9017 4.6023 7.2694
RERF-LC-A1 CTRP2 5.474 6.1541 5.3888 4.1031
NCI-H1155 GDSC1; GDSC2; CTRP2 5.482 8.9293 4.1101 9.2846
NCI-H2795 GDSC1; GDSC2 5.494 7.5577 2.6255 0.8897
NCI-H524 GDSC1; GDSC2 5.5161 7.1015 2.8048 0.338
EMC-BAC-2 GDSC1; GDSC2 5.5221 17.5762 -2.065 22.5298
HCC2279 CTRP2 5.5356 6.7673 5.2039 4.6557
COR-L32 GDSC2 5.5365 7.5019 2.6651 0.7247
NCI-H2227 GDSC1; GDSC2 5.5654 7.0998 2.8239 0.2766
NCI-H1048 GDSC1; GDSC2 5.5928 7.4496 2.7079 0.5583
NCI-H2722 GDSC1; GDSC2 5.5975 20.1984 -3.303 25.9664
HCC1588 CTRP2 5.6186 6.3723 5.4621 3.417
PaCa-3 GDSC1; GDSC2 5.6328 8.5263 2.2999 2.1069
RERF-LC-KJ GDSC1; GDSC2 5.6329 7.7248 2.6209 0.8081
Lu-135 GDSC1; GDSC2 5.6959 7.8581 2.5967 0.8473
ABC-1 GDSC1; GDSC2 5.6972 11.6747 0.9203 9.2368
NCI-H847 GDSC1 5.7036 7.1265 2.8649 0.2021
NCI-H1993 GDSC1; GDSC2 5.7169 7.4426 2.7591 0.3649
NCI-H522 GDSC1; GDSC2; CTRP2 5.7541 8.611 4.5118 7.0249
RERF-LC-Sq1 GDSC1; GDSC2 5.8035 12.7246 0.4931 11.2483
NCI-H2066 GDSC1; GDSC2 5.8057 7.9107 2.6227 0.6938
Calu-3 GDSC1; GDSC2; CTRP2 5.8132 6.8032 5.4585 2.9484
NCI-H513 GDSC1; GDSC2 5.839 7.5724 2.759 0.3192
IST-SL2 GDSC1; GDSC2 5.8393 14.6633 -0.4125 15.4893
Lu-99A GDSC1; GDSC2 5.8573 9.2846 2.0943 2.8072
EBC-1 GDSC1; GDSC2; CTRP2 5.8951 10.6282 3.6269 10.4389
NCI-H290 GDSC1; GDSC2 5.9084 16.9246 -1.4629 19.596
UMC-11 GDSC1; GDSC2 5.9133 8.2436 2.5417 0.8863
NCI-H1944 GDSC1; GDSC2; CTRP2 5.971 8.0571 4.9762 4.6335
NCI-H1694 GDSC1; GDSC2; CTRP2 6.0009 7.5534 5.2534 3.4098
SW1573 GDSC1; GDSC2 6.0453 13.4943 0.287 11.7936
COLO 668 GDSC1; GDSC2 6.0496 7.7581 2.7714 0.2304
NCI-H1573 GDSC1; GDSC2; CTRP2 6.0787 8.1176 5.0362 4.1722
SBC-5 GDSC1; GDSC2; CTRP2 6.0902 6.8667 5.6708 1.4842
NCI-H835 GDSC1; GDSC2 6.0966 8.2167 2.6263 0.5311
SK-MES-1 GDSC1; GDSC2; CTRP2 6.1008 8.6615 4.7825 5.1962
NCI-H1693 GDSC1; GDSC2; CTRP2 6.1115 8.9313 4.6565 5.7054
HCC15 GDSC1; GDSC2; CTRP2 6.1368 8.7411 4.7722 5.1716
COR-L311 GDSC2 6.1414 7.9981 2.7213 0.2963
SW1271 GDSC1; GDSC2; CTRP2 6.1587 8.907 4.7072 5.4041
EPLC-272H GDSC1; GDSC2; CTRP2 6.168 7.4694 5.4321 2.345
HARA [Human squamous cell lung carcinoma] GDSC1; GDSC2; CTRP2 6.195 8.6116 4.884 4.5943
NCI-H2347 GDSC1; GDSC2 6.2336 8.4801 2.584 0.5782
NCI-H1623 GDSC1; GDSC2 6.2496 8.3655 2.6317 0.4514
NCI-H209 GDSC1; GDSC2 6.2561 8.1662 2.7046 0.2935
DMS 454 CTRP2 6.3566 16.382 1.1334 19.0081
NCI-H2595 GDSC1; GDSC2 6.3817 8.2269 2.7289 0.2176
NCI-H2591 GDSC1; GDSC2 6.3904 8.9526 2.4724 0.8132
LCLC-97TM1 GDSC1; GDSC2; CTRP2 6.3975 9.0415 4.829 4.4663
NCI-H322M GDSC1; GDSC2 6.398 8.6932 2.5708 0.5374
NCI-H1666 GDSC1; GDSC2; CTRP2 6.4294 18.9466 -0.0887 22.5832
LC-1/sq GDSC1; GDSC2 6.4297 15.3306 -0.3318 13.9231
Sq-1 CTRP2 6.4498 14.4047 2.1971 15.067
NCI-H2110 GDSC1; GDSC2; CTRP2 6.4548 8.5068 5.1363 3.0943
LK-2 GDSC1; GDSC2 6.4641 14.601 0.0368 12.1782
NCI-H1355 GDSC1; GDSC2; CTRP2 6.4881 9.1026 4.8675 4.154
RERF-LC-Ad1 CTRP2 6.4956 7.9195 5.451 1.7461
Calu-6 GDSC1; GDSC2; CTRP2 6.5 8.2935 5.2732 2.4608
COR-L51 CTRP2 6.5003 9.9948 4.435 5.9337
NCI-H322 CTRP2 6.5254 8.4074 5.2358 2.5752
NCI-H3122 GDSC1; GDSC2 6.5874 8.5691 2.6848 0.2391
NCI-H1105 GDSC1; GDSC2; CTRP2 6.5963 14.6035 2.2156 14.7228
NCI-H226 GDSC1; GDSC2; CTRP2 6.63 8.6811 5.1765 2.6609
HCC1171 CTRP2 6.6756 8.9742 5.0664 3.0407
LB647-SCLC GDSC1; GDSC2 6.8068 16.2363 -0.5131 13.9863
NCI-H1838 GDSC1; GDSC2; CTRP2 6.8174 9.1914 5.0591 2.8656
NCI-H1651 GDSC1; GDSC2; CTRP2 6.8426 10.2667 4.5558 4.874
NCI-H2869 GDSC1; GDSC2 6.8981 16.4567 -0.5577 14.0047
LUDLU-1 CTRP2 6.9089 10.9094 4.2893 5.865
NCI-H2228 GDSC1; GDSC2; CTRP2 6.9533 15.5958 2.0034 14.8568
NCI-H1793 GDSC1; GDSC2; CTRP2 6.9845 9.1015 5.2102 2.0532
Lu-99 CTRP2 7.0422 9.6609 4.9848 2.8562
NCI-H1092 GDSC1; GDSC2; CTRP2 7.0898 14.9675 2.4213 13.0572
NCI-H196 GDSC1; GDSC2; CTRP2 7.1097 9.3696 5.1634 2.0816
NCI-H292 GDSC1; GDSC2; CTRP2 7.1112 9.5851 5.0645 2.4577
KNS-62 GDSC1; GDSC2; CTRP2 7.1173 11.9137 3.9487 6.9322
Lu-65 GDSC1; GDSC2; CTRP2 7.1254 10.2272 4.7708 3.5911
HCC1438 CTRP2 7.1316 9.1488 5.2774 1.6326
BEN GDSC1; GDSC2; CTRP2 7.1879 8.1249 5.7344 0.1882
NCI-H2286 CTRP2 7.2046 8.8681 5.442 0.9865
HCC4006 CTRP2 7.2341 9.9146 4.9881 2.6006
NCI-H358 GDSC1; GDSC2; CTRP2 7.2598 13.5842 3.2332 9.5993
NCI-H520 GDSC1; GDSC2; CTRP2 7.307 12.8692 3.6185 7.9759
NCI-H2461 GDSC1; GDSC2 7.358 15.6886 0.0908 10.338
NCI-H69 GDSC1; GDSC2; CTRP2 7.3583 10.0436 5.0047 2.3905
HOP-62 GDSC1; GDSC2; CTRP2 7.364 11.3695 4.3851 4.7997
HCC827 GDSC1; GDSC2; CTRP2 7.4158 10.4881 4.8349 2.9666
NCI-H1373 CTRP2 7.4535 11.0237 4.6083 3.7965
NCI-H1755 GDSC1; GDSC2; CTRP2 7.4574 18.1344 1.1328 16.9896
HCC2935 CTRP2 7.469 11.314 4.4813 4.2747
MOR/CPR CTRP2 7.5322 8.7864 5.6281 0.2707
NCI-H1734 GDSC2; CTRP2 7.6049 9.6976 5.2959 1.1266
NCI-H1869 GDSC1; CTRP2 7.6651 10.253 5.0879 1.7671
NCI-H441 GDSC1; GDSC2; CTRP2 7.6855 9.6975 5.3364 0.9399
NCI-H727 GDSC1; GDSC2; CTRP2 7.6918 9.9994 5.2124 1.3241
NCI-H2818 GDSC1; GDSC2 7.7043 22.3813 -2.849 20.6176
SHP-77 GDSC1; GDSC2; CTRP2 7.7382 15.6974 2.5464 11.5004
NCI-H526 GDSC1; GDSC2; CTRP2 7.7526 9.3762 5.4965 0.4651
NCI-H2291 GDSC1; GDSC2; CTRP2 7.7639 9.544 5.4357 0.6104
NCI-H2126 CTRP2 7.825 9.5271 5.4695 0.4939
NCI-H1339 CTRP2 7.8916 9.1351 5.6414 0.1415
COR-L95 GDSC1; GDSC2; CTRP2 7.8992 9.4046 5.547 0.2949
IA-LM GDSC1; GDSC2; CTRP2 7.9178 11.0556 4.8741 2.269
HCC1195 CTRP2 7.9263 9.7793 5.4157 0.573
SK-LU-1 GDSC1; GDSC2; CTRP2 7.941 9.8172 5.4074 0.5859
NCI-H1975 GDSC1; GDSC2; CTRP2 7.9725 10.5434 5.1259 1.3722
NCI-H1435 GDSC1; GDSC2; CTRP2 7.9771 10.1571 5.2884 0.8809
HCC78 GDSC1; GDSC2; CTRP2 7.9809 11.4313 4.7423 2.6749
NCI-H460 GDSC1; GDSC2; CTRP2 7.984 9.2154 5.6472 0.1155
NCI-H2085 GDSC1; GDSC2; CTRP2 7.9991 10.7839 5.0371 1.6368
NCI-H2030 GDSC1; GDSC2; CTRP2 8.0758 12.2732 4.416 3.7731
NCI-H2196 GDSC2; CTRP2 8.1536 9.5909 5.5781 0.17
NCI-H2172 GDSC1; GDSC2; CTRP2 8.1771 13.2582 4.0221 5.1484
NCI-H1299 GDSC1; GDSC2; CTRP2 8.1799 10.6052 5.2023 0.9924
HOP-92 GDSC1; GDSC2; CTRP2 8.1914 19.1715 1.1728 15.6296
LCLC-103H GDSC1; GDSC2; CTRP2 8.1919 9.3965 5.659 0.0719
CAL-12T GDSC1; GDSC2; CTRP2 8.2055 10.2645 5.3493 0.5929
HCC95 CTRP2 8.2307 9.7312 5.5573 0.1815
HCC2108 CTRP2 8.2389 13.4968 3.9498 5.3485
NCI-H2122 GDSC1; GDSC2; CTRP2 8.2684 9.6134 5.6121 0.1064
NCI-H661 GDSC1; GDSC2; CTRP2 8.2982 10.5513 5.2782 0.7194
NCI-H2342 GDSC1; GDSC2; CTRP2 8.2989 13.2588 4.0981 4.709
NCI-H64 GDSC1; GDSC2 8.3013 16.4344 0.303 7.9492
NCI-H650 GDSC1; GDSC2; CTRP2 8.3244 10.418 5.3413 0.5551
NCI-H446 GDSC1; GDSC2; CTRP2 8.3621 10.1346 5.4627 0.2955
COR-L88 GDSC1; GDSC2; CTRP2 8.381 15.8777 2.9124 9.1392
NCI-H1395 CTRP2 8.419 11.0121 5.15 0.9867
NCI-H1568 GDSC1; GDSC2; CTRP2 8.4984 17.1343 2.3875 10.925
NCI-H2373 GDSC1; GDSC2 8.5166 21.5002 -1.8885 16.1987
RERF-LC-MS GDSC1; GDSC2; CTRP2 8.5748 10.0413 5.5743 0.0993
NCI-H1915 GDSC1; GDSC2; CTRP2 8.6021 15.424 3.2765 7.4526
COR-L105 GDSC1; GDSC2; CTRP2 8.6048 11.4398 5.0643 1.107
NCI-H23 GDSC1; GDSC2; CTRP2 8.6056 17.0223 2.5155 10.2993
NCI-H841 GDSC1; GDSC2; CTRP2 8.6403 16.6052 2.7393 9.4216
NCI-H2023 GDSC1; GDSC2; CTRP2 8.6596 10.4624 5.4589 0.2211
HCC366 GDSC1; GDSC2; CTRP2 8.7207 10.2705 5.5476 0.1046
DMS 114 GDSC1; GDSC2; CTRP2 8.8161 14.4106 3.8833 4.907
NCI-H2009 GDSC1; GDSC2; CTRP2 8.8987 10.5391 5.5188 0.1076
A-549 GDSC1; GDSC2; CTRP2 9.0617 15.3085 3.6201 5.5947
HCC1833 CTRP2 9.1191 29.1196 -3.0417 24.8599
NCI-H1184 CTRP2 9.1265 21.707 0.6095 15.9533
NCI-H838 GDSC1; GDSC2; CTRP2 9.3367 16.3617 3.303 6.4346
NCI-H2141 GDSC1; GDSC2; CTRP2 9.7088 21.9502 0.8994 14.2156
NCI-H1563 GDSC1; GDSC2; CTRP2 9.7847 24.1916 -0.1326 17.1392
EKVX GDSC1; GDSC2; CTRP2 9.8104 23.1356 0.3974 15.5903
NCI-H1792 GDSC1; GDSC2; CTRP2 10.0148 19.8265 2.1146 9.8219
NCI-H2081 GDSC1; GDSC2; CTRP2 10.2123 22.0807 1.1771 12.6557
LOU-NH91 GDSC1; GDSC2; CTRP2 10.5144 22.5007 1.1768 12.2618
DMS 273 GDSC1; GDSC2; CTRP2 11.5118 24.7664 0.7531 12.3109
Calu-1 CTRP2 11.6419 21.9736 2.1196 7.9285
LXF 289 GDSC1; GDSC2; CTRP2 12.0348 25.1116 0.9203 11.2044
COLO 699 CTRP2 13.4166 26.9738 0.8978 9.7937
Hs 888.Lu CTRP2 8.7207 14.5407 3.7654 5.4568
⏷ Show the Full List of 217 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1; GDSC2 5.4941 7.6125 2.6043 0.9666
Cancer Drug Sensitivity Data Curated from 31 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 7.104 8.9035 5.3715 1.3221
Aska-SS CTRP2 7.4952 8.9222 5.5604 0.4402
Rh41 GDSC1; GDSC2 3.7403 8.0925 1.2757 11.6844
A-204 GDSC1; GDSC2; CTRP2 4.3052 7.6055 3.5729 14.3192
TE 617.T CTRP2 4.4406 8.6209 3.2591 15.2108
SW684 GDSC1; GDSC2 4.8789 6.0369 2.9431 0.2687
EW-8 GDSC1; GDSC2 4.9191 12.2933 0.0877 15.2177
SW872 GDSC1; GDSC2 4.9413 6.7983 2.6761 1.1647
TE 441.T GDSC2; CTRP2 5.3851 6.2233 5.2691 4.808
VA-ES-BJ GDSC1; GDSC2 5.5415 15.4327 -0.9981 18.6157
GCT GDSC1; GDSC2; CTRP2 6.0677 7.702 5.2349 3.3577
HT-1080 GDSC1; GDSC2; CTRP2 6.2215 7.4908 5.463 2.1228
G-401 GDSC1; GDSC2 6.3174 16.0523 -0.753 15.958
MES-SA GDSC1; GDSC2; CTRP2 6.3688 7.6987 5.4696 1.8573
Rh18 GDSC1; CTRP2 6.4225 7.7521 5.4814 1.7285
KYM-1 GDSC1; GDSC2; CTRP2 6.6088 11.2947 3.8735 8.0824
Rh30 GDSC1; GDSC2 6.9414 17.5042 -1.0268 15.8408
STS-0421 GDSC1; GDSC2 7.1591 18.3122 -1.267 16.3573
G-402 GDSC1; GDSC2; CTRP2 7.1678 15.5807 2.1771 13.8378
BT-12 CTRP2 7.2621 8.2572 5.7153 0.1984
Hs 729.T CTRP2 7.3209 12.0867 4.0096 6.373
TTC-709 CTRP2 7.6164 11.194 4.632 3.4998
BT-16 CTRP2 7.6402 9.4531 5.4149 0.7421
SW982 GDSC1; GDSC2; CTRP2 7.7002 9.0047 5.6149 0.236
MFH-ino GDSC1; GDSC2 7.7733 18.6097 -1.0071 14.2555
Hs 633.T GDSC1; GDSC2 7.9978 20.6643 -1.8306 16.8772
Tm87-16 CTRP2 8.0794 14.1945 3.5151 7.245
RKN GDSC1; GDSC2; CTRP2 8.179 9.263 5.6992 0.0431
SK-UT-1 GDSC1; GDSC2; CTRP2 8.923 14.053 4.1085 3.9708
SK-LMS-1 GDSC1; GDSC2; CTRP2 11.6702 22.3547 1.9637 8.3961
RD GDSC1; GDSC2; CTRP2 12.4933 23.3478 1.9923 7.4694
⏷ Show the Full List of 31 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 43 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 8.4472 22.2281 -0.1427 19.197
EFO-21 GDSC1; GDSC2 4.8468 6.8939 2.5896 1.6624
SNU-119 CTRP2 5.3513 6.3355 5.1924 5.1936
A2780 GDSC1; GDSC2; CTRP2 5.3857 7.6188 4.6581 7.2366
Caov-4 GDSC1; GDSC2 5.4234 17.046 -1.8772 22.1262
ES-2 GDSC1; GDSC2 5.5589 12.9514 0.2199 13.1241
JHOS-4 GDSC1; GDSC2 5.5622 16.8589 -1.6824 21.1431
OVCAR-3 GDSC1; GDSC2 5.8175 7.2195 2.8733 0.1269
OVKATE GDSC1; GDSC2 5.8701 12.3869 0.6964 10.0758
TYK-nu GDSC1; GDSC2; CTRP2 5.9462 8.5663 4.7007 5.8403
HEY A8 CTRP2 6.0179 8.8249 4.632 5.9882
TOV-112D GDSC1; GDSC2; CTRP2 6.3239 7.9437 5.3164 2.5609
SNU-840 CTRP2 6.5891 8.0755 5.439 1.6652
OAW42 GDSC1; GDSC2; CTRP2 6.807 8.0391 5.588 0.8537
OC 314 GDSC1; GDSC2; CTRP2 7.106 9.7304 4.9932 2.7405
OVCAR-5 GDSC1; GDSC2; CTRP2 7.1266 11.2479 4.28 5.5675
Kuramochi GDSC1; GDSC2; CTRP2 7.2416 10.8603 4.5463 4.3259
OV7 CTRP2 7.2546 9.8515 5.03 2.4162
JHOC-5 CTRP2 7.2629 9.6529 5.1261 2.0458
DOV13 GDSC1; GDSC2; CTRP2 7.2693 9.9045 5.0145 2.4574
COV434 CTRP2 7.3566 13.0941 3.5443 8.1974
ES2 CTRP2 7.404 10.728 4.7155 3.4419
JHOS-2 GDSC1; GDSC2; CTRP2 7.5563 9.1707 5.4896 0.5884
COV644 CTRP2 7.6916 10.8439 4.8387 2.6335
FU-OV-1 GDSC1; GDSC2; CTRP2 7.7135 9.3267 5.4986 0.4794
TOV-21G GDSC1; GDSC2; CTRP2 7.7826 8.8863 5.6884 0.1035
SNU-8 CTRP2 7.9281 9.048 5.6848 0.0833
OV56 GDSC1; GDSC2; CTRP2 7.9415 9.0357 5.6937 0.0727
RMG-I GDSC1; GDSC2; CTRP2 7.9718 11.293 4.799 2.4809
Caov-3 GDSC2; CTRP2 8.0002 13.9604 3.5738 7.1264
OVISE GDSC1; GDSC2; CTRP2 8.129 9.1301 5.7262 0.0311
ONCO-DG-1 CTRP2 8.2314 12.3071 4.4933 3.3129
OVSAHO CTRP2 8.3098 9.6385 5.6181 0.094
OVCAR-8 GDSC1; GDSC2; CTRP2 8.3116 10.6847 5.2316 0.8318
MCAS CTRP2 8.3558 10.0315 5.4976 0.2396
OV-90 GDSC1; GDSC2; CTRP2 8.4461 13.165 4.2307 4.0419
OVK18 GDSC1; GDSC2; CTRP2 8.5014 10.1517 5.5096 0.1865
IGROV-1 GDSC1; GDSC2; CTRP2 8.6593 10.6752 5.3823 0.3437
EFO-27 GDSC1; GDSC2 9.4122 21.3936 -1.2842 12.687
OAW28 GDSC1; GDSC2; CTRP2 10.3515 19.9736 2.2583 8.9173
OVCAR-4 GDSC1; GDSC2; CTRP2 11.0328 25.7321 -0.0168 15.1168
SK-OV-3 GDSC1; GDSC2; CTRP2 12.1396 23.1754 1.8673 8.2083
OVTOKO GDSC1; GDSC2; CTRP2 13.5479 25.3459 1.6967 7.3669
⏷ Show the Full List of 43 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 10.3811 21.3554 1.631 10.9759
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KP-1N GDSC1; GDSC2 5.4465 7.6542 2.5666 1.149
MZ-PC-1 GDSC1; GDSC2 5.7258 10.3436 1.5545 5.7745
Panc 10.05 GDSC1; GDSC2; CTRP2 6.0098 8.3665 4.8544 5.0691
MIA PaCa-2 GDSC1; GDSC2; CTRP2 6.037 6.9509 5.585 1.9454
Panc 03.27 GDSC1; GDSC2; CTRP2 6.2105 11.6243 3.3916 10.7993
PL4 GDSC1; GDSC2 6.3694 19.1772 -2.2318 21.2705
Panc 04.03 GDSC1; GDSC2; CTRP2 6.6476 9.8331 4.6263 4.8926
Capan-1 GDSC1; GDSC2; CTRP2 6.6961 8.5854 5.2674 2.2015
KP-4 GDSC1; GDSC2; CTRP2 6.7318 9.1194 5.0352 3.0844
Capan-2 GDSC1; GDSC2; CTRP2 6.9004 9.2944 5.0655 2.7263
Hs 766T GDSC1; GDSC2; CTRP2 6.9068 8.7202 5.3386 1.657
PaTu 8902 GDSC1; GDSC2; CTRP2 6.9557 8.301 5.5545 0.8303
SU.86.86 GDSC1; GDSC2; CTRP2 7.2552 13.6839 3.1808 9.816
KP-3 GDSC1; GDSC2; CTRP2 7.2905 12.0166 4.0223 6.3672
PSN1 GDSC1; GDSC2; CTRP2 7.4093 10.8108 4.68 3.5733
PK-45H CTRP2 7.6249 11.2976 4.5891 3.6543
HPAF-II GDSC1; GDSC2; CTRP2 7.6762 11.2555 4.6406 3.3944
QGP-1 GDSC1; GDSC2; CTRP2 7.8043 9.217 5.5783 0.2687
TCC-Pan2 CTRP2 7.9048 9.4694 5.5252 0.3358
SNU-213 CTRP2 7.9336 9.3067 5.5962 0.1978
KP-2 GDSC1; GDSC2; CTRP2 7.9358 10.5052 5.1232 1.4101
Panc 08.13 GDSC1; GDSC2; CTRP2 7.9602 16.363 2.3815 11.7664
PaTu 8988t GDSC1; GDSC2; CTRP2 7.9661 9.2167 5.6402 0.1275
Panc 05.04 CTRP2 8.0206 9.9445 5.3928 0.5807
SUIT-2 GDSC1; GDSC2; CTRP2 8.0533 15.0998 3.0619 9.0433
HuP-T4 GDSC1; GDSC2; CTRP2 8.0628 12.1071 4.4843 3.5329
HPAC GDSC1; GDSC2; CTRP2 8.1506 9.6825 5.5443 0.2211
L3.3 CTRP2 8.1784 9.5374 5.6059 0.1288
BxPC-3 GDSC1; GDSC2; CTRP2 8.2928 11.397 4.9281 1.7445
YAPC GDSC1; GDSC2; CTRP2 8.301 9.7881 5.5633 0.1579
DAN-G GDSC1; GDSC2; CTRP2 8.3024 9.8926 5.5269 0.2084
HuP-T3 GDSC1; GDSC2; CTRP2 8.3704 10.0879 5.4829 0.2591
CFPAC-1 GDSC1; GDSC2; CTRP2 8.4312 9.9133 5.5671 0.1287
AsPC-1 GDSC1; GDSC2; CTRP2 8.4347 12.3529 4.589 2.7614
SW1990 GDSC1; GDSC2; CTRP2 8.5108 10.5937 5.3528 0.4517
PK-59 CTRP2 8.6179 10.6727 5.3668 0.3853
Panc 02.03 GDSC1; GDSC2; CTRP2 8.8454 16.1064 3.1124 7.7503
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ACC-MESO-1 CTRP2 7.9196 9.5753 5.4914 0.4005
JL-1 CTRP2 8.0225 9.4624 5.5743 0.2084
NCI-H2452 GDSC1; GDSC2; CTRP2 8.2449 19.1947 1.2008 15.4517
NCI-H28 GDSC1; GDSC2; CTRP2 8.4701 17.7564 2.0662 12.129
MSTO-211H GDSC1; GDSC2; CTRP2 8.5677 10.7098 5.3327 0.4707
MPP 89 GDSC1; GDSC2; CTRP2 8.634 10.086 5.5798 0.0866
NCI-H2052 GDSC1; GDSC2; CTRP2 9.0537 16.7625 2.9378 8.1267
IST-Mes1 GDSC1; GDSC2; CTRP2 12.2732 27.2805 0.0599 13.3806
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H660 GDSC2 4.0713 8.5832 1.2867 10.7534
LNCaP clone FGC GDSC1; GDSC2 4.6582 6.9104 2.4809 2.471
PC-3 GDSC1; GDSC2 5.6174 11.1974 1.0934 8.4622
VCaP GDSC1; GDSC2 5.7317 11.9552 0.8105 9.7505
PaCa-3 CTRP2 6.4259 7.551 5.5804 1.3253
DU145 GDSC1; GDSC2; CTRP2 8.0006 11.4871 4.7286 2.7037
22Rv1 GDSC1; GDSC2; CTRP2 8.4317 15.8706 2.9502 8.9239
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 GDSC1; GDSC2; CTRP2 6.4845 10.2042 4.3189 6.4453
YD-15 CTRP2 7.6577 8.964 5.6129 0.2543
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1; GDSC2 7.469 21.5652 -2.6176 20.3551
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-16 GDSC1; GDSC2; CTRP2 3.7242 5.7013 3.5971 15.896
MKN7 GDSC1; GDSC2 4.6108 9.9289 1.0212 10.9886
HSC-39 GDSC1; GDSC2 4.6382 6.1499 2.7961 0.9505
ECC10 GDSC1; GDSC2; CTRP2 4.6387 5.9966 4.523 9.7683
Fu97 GDSC1; GDSC2; CTRP2 4.8316 7.898 3.9816 11.3352
SCH GDSC1; GDSC2 4.9455 6.7787 2.686 1.118
KATO III GDSC1; GDSC2; CTRP2 4.9903 8.2741 3.9635 11.0184
OCUM-1 GDSC1; GDSC2 5.0708 11.4244 0.6194 12.145
HGC-27 GDSC1; GDSC2; CTRP2 5.1425 8.9171 3.8012 11.3241
GCIY GDSC1; GDSC2 5.6085 7.5089 2.6922 0.5961
MKN28 GDSC1; GDSC2 5.609 8.1302 2.451 1.4706
TMK-1 GDSC1; GDSC2 5.697 7.6169 2.6879 0.5604
SK-GT-2 GDSC1; GDSC2 5.7644 12.1296 0.7493 10.007
TGBC11TKB GDSC1; GDSC2 6.0539 7.8837 2.7292 0.3085
RF-48 GDSC1; GDSC2 6.247 8.1076 2.7217 0.2645
Hs 746.T GDSC1; GDSC2; CTRP2 6.5678 8.6929 5.127 2.9558
SNU-620 CTRP2 6.646 9.9309 4.5769 5.0999
RERF-GC-1B GDSC1; GDSC2 6.7881 8.8749 2.6514 0.2446
GSU CTRP2 6.9907 7.7173 5.8058 0.1225
MKN45 GDSC1; GDSC2; CTRP2 7.2475 8.1979 5.7314 0.1732
SNU-5 GDSC1; GDSC2; CTRP2 7.3059 9.3731 5.2766 1.4566
SNU-668 CTRP2 7.5859 15.6348 2.4654 12.0529
GSS CTRP2 7.5908 14.3352 3.1065 9.5725
NUGC-3 GDSC1; GDSC2; CTRP2 7.8458 9.7101 5.407 0.6389
MKN1 GDSC1; GDSC2; CTRP2 7.8785 10.0388 5.2896 0.9429
ECC12 GDSC2; CTRP2 7.9238 9.2821 5.6013 0.1924
SNU-601 CTRP2 8.0893 13.9512 3.6379 6.7527
SNU-719 CTRP2 8.099 14.4705 3.3962 7.6807
AGS GDSC1; GDSC2; CTRP2 8.1764 9.462 5.6312 0.1006
23132/87 GDSC1; GDSC2; CTRP2 8.4402 15.4779 3.1439 8.1762
NCI-N87 GDSC1; GDSC2; CTRP2 8.5344 11.6624 4.9389 1.5209
IM95 GDSC1; GDSC2; CTRP2 8.5525 14.8187 3.5299 6.5547
LMSU CTRP2 8.6582 10.912 5.294 0.5147
MKN74 CTRP2 8.805 10.8933 5.3599 0.3377
SNU-1 GDSC1; GDSC2; CTRP2 9.0962 21.2815 0.7951 15.429
SNU-216 CTRP2 9.8786 21.0293 1.456 12.2053
NUGC-4 GDSC1; GDSC2; CTRP2 11.4209 33.1304 -3.3214 22.2519
KE-39 CTRP2 11.8826 25.5932 0.6014 12.3138
SNG-M GDSC1; GDSC2; CTRP2 6.285 7.5765 5.4684 1.9943
SNU-1077 CTRP2 8.764 10.2 5.5863 0.0673
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 18 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HTC-C3 GDSC1; GDSC2 4.5106 10.7563 0.5429 13.8687
IHH-4 GDSC1; GDSC2 4.5181 8.8845 1.4634 8.6386
K5 GDSC1; GDSC2 5.268 9.2336 1.7874 5.2789
TT GDSC1; GDSC2; CTRP2 5.313 6.3426 5.1487 5.4678
ASH-3 GDSC1; GDSC2 5.4208 6.8436 2.8606 0.2493
SW579 CTRP2 5.4578 10.2948 3.4126 12.2285
8505C GDSC1; GDSC2; CTRP2 5.4711 7.625 4.737 6.7121
WRO GDSC1; GDSC2 5.5032 6.906 2.869 0.2069
CGTH-W-1 GDSC1; GDSC2; CTRP2 5.5246 8.6572 4.283 8.4718
KMH-2 GDSC1; GDSC2 6.0878 7.7378 2.792 0.1871
TT2609-C02 GDSC1; GDSC2; CTRP2 6.3124 7.5076 5.5223 1.728
ML-1 [Human leukemia] GDSC1; GDSC2; CTRP2 6.6457 8.9591 5.0527 3.1411
CAL-62 GDSC1; GDSC2; CTRP2 7.3441 8.8509 5.5194 0.6396
8305C GDSC1; GDSC2; CTRP2 7.9797 10.0411 5.3363 0.7479
B-CPAP GDSC1; GDSC2; CTRP2 8.0309 10.4359 5.2 1.1003
BHT-101 GDSC1; GDSC2; CTRP2 8.1727 9.374 5.6599 0.0735
FTC-133 GDSC1; GDSC2 9.3213 21.1434 -1.2244 12.6038
FTC-238 CTRP2 9.751 20.6945 1.5305 12.1336
⏷ Show the Full List of 18 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 54 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PCI-15A GDSC1; GDSC2 3.528 7.2265 1.5386 10.6657
PCI-38 GDSC1 4.273 21.4112 -4.9429 34.9413
SCC-15 GDSC1; GDSC2 4.4766 9.2389 1.2618 9.9167
Ca9-22 GDSC1; GDSC2 4.6119 6.7549 2.5239 2.3117
KOSC-2 GDSC1; GDSC2 4.7844 7.19 2.4278 2.5649
DOK GDSC1; GDSC2 4.8761 8.8839 1.705 6.4692
JHU-022 GDSC1; GDSC2 4.9255 9.3137 1.5339 7.3581
HO-1-N-1 GDSC1; GDSC2 4.9517 7.1769 2.5234 1.853
BB30-HNC GDSC1; GDSC2 4.982 7.5682 2.3706 2.5785
PCI-30 GDSC1; GDSC2 5.2425 7.6076 2.489 1.6765
BICR 78 GDSC1; GDSC2 5.3283 12.5515 0.2534 13.4589
JHU-011 GDSC1; GDSC2 5.377 14.9935 -0.9024 18.6
LB771-HNC GDSC1; GDSC2 5.4205 10.176 1.446 6.9007
PCI-04B GDSC1; GDSC2 5.451 7.5863 2.5955 1.0336
OSC-19 GDSC1; GDSC2 5.518 7.821 2.5328 1.2205
BICR 10 GDSC1 5.541 29.5139 -7.9738 36.2652
PCI-06A GDSC1; GDSC2 5.551 12.5369 0.4137 12.1706
OSC-20 GDSC1; GDSC2 5.5732 7.478 2.6893 0.6252
NCI-H3118 GDSC1; GDSC2 5.5854 8.6454 2.2259 2.5092
JHU-029 GDSC1; GDSC2 5.7671 12.0233 0.8012 9.7303
HO-1-u-1 GDSC1; GDSC2 5.782 7.4862 2.7682 0.3197
UPCI-SCC-090 GDSC1; GDSC2 5.8132 7.7982 2.6675 0.5576
BB49-HNC GDSC1 5.8191 7.5546 2.7579 0.4097
SAT [Human HNSCC] GDSC1; GDSC2 6.166 9.7633 2.049 2.6573
FaDu GDSC1; GDSC2; CTRP2 6.2351 7.4344 5.5012 1.9406
SKN-3 GDSC1; GDSC2 6.2378 7.9302 2.7793 0.1735
PE/CA-PJ34 (clone C12) CTRP2 6.392 9.1701 4.761 4.7599
PE/CA-PJ41 (clone D2) CTRP2 6.5559 8.064 5.4225 1.7759
HSC-2 GDSC1; GDSC2; CTRP2 6.5674 10.0631 4.4526 5.7464
HSC-4 GDSC2; CTRP2 6.6321 9.7329 4.6641 4.7613
PE/CA-PJ49 CTRP2 6.6868 8.6208 5.2443 2.3067
SCC-4 GDSC1; GDSC2; CTRP2 6.7106 13.8975 2.6583 12.818
CAL-33 GDSC1; GDSC2; CTRP2 6.7865 9.9338 4.6781 4.4592
BICR 56 CTRP2 7.4482 11.8707 4.2018 5.4142
KON GDSC1; GDSC2 7.4732 26.5627 -5.0466 26.3939
SAS GDSC1; GDSC2 7.5362 19.8678 -1.7573 17.4413
SNU-899 CTRP2 7.6296 9.4373 5.4163 0.7451
SCC-25 GDSC1; GDSC2; CTRP2 7.736 10.377 5.0725 1.7533
YD-10B CTRP2 7.9164 9.1185 5.6563 0.1171
SNU-1076 CTRP2 7.9225 9.2025 5.6291 0.1515
BHY GDSC1; GDSC2; CTRP2 7.9364 9.7397 5.4356 0.5198
CAL-27 GDSC1; GDSC2; CTRP2 7.9444 9.2214 5.6306 0.1445
SNU-46 CTRP2 7.9764 10.1929 5.2735 0.9235
SCC-9 GDSC1; GDSC2; CTRP2 8.024 13.4915 3.8132 6.1571
BICR 16 CTRP2 8.084 10.1324 5.3473 0.6603
YD-8 CTRP2 8.1014 9.861 5.4592 0.394
HSC-3 GDSC1; GDSC2; CTRP2 8.2294 9.715 5.5625 0.1745
SNU-1066 CTRP2 8.2901 9.5521 5.6406 0.0759
Detroit 562 GDSC1; GDSC2; CTRP2 8.3076 10.161 5.4314 0.3715
SNU-1041 CTRP2 8.4356 10.4031 5.3933 0.3993
SNU-1214 CTRP2 8.5753 21.6822 0.2214 17.9572
BICR 22 GDSC1; GDSC2 8.745 23.7349 -2.7959 18.6905
BICR 31 GDSC2; CTRP2 11.0799 22.909 1.3481 11.0183
PE/CA-PJ15 GDSC1; GDSC2; CTRP2 11.5213 22.1423 1.9722 8.5292
⏷ Show the Full List of 54 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW780 GDSC1; GDSC2 4.824 9.5896 1.3343 8.7197
CAL-29 GDSC1; GDSC2 5.2513 10.2379 1.3093 7.9836
U-BLC1 CTRP2 5.4867 8.8977 4.1299 9.1917
TCCSUP GDSC1; GDSC2; CTRP2 5.6462 7.063 5.1744 4.5058
UM-UC-1 CTRP2 6.0215 8.1227 4.9861 4.4925
SW1710 GDSC1; GDSC2; CTRP2 6.374 8.4854 5.0866 3.433
UM-UC-3 GDSC1; GDSC2; CTRP2 6.3776 8.1949 5.2327 2.8202
253J-BV CTRP2 6.5491 8.1319 5.3854 1.9338
KMBC-2 CTRP2 6.6689 8.2919 5.3887 1.7582
BC-3C CTRP2 6.7989 8.4665 5.3895 1.592
JMSU-1 CTRP2 6.8333 14.0749 2.6661 12.5675
639V GDSC1; GDSC2; CTRP2 6.9866 11.2599 4.1741 6.2154
BFTC-905 GDSC1; GDSC2; CTRP2 7.1041 8.8748 5.3843 1.2768
KU-19-19 GDSC1; GDSC2; CTRP2 7.689 8.9259 5.6393 0.1967
RT-112 GDSC1; GDSC2; CTRP2 7.7643 9.7499 5.353 0.8367
647V GDSC1; GDSC2; CTRP2 8.0197 9.3713 5.6058 0.1619
T24 GDSC1; GDSC2; CTRP2 8.0804 14.1521 3.5361 7.1619
HT-1376 GDSC1; GDSC2; CTRP2 8.4076 10.1417 5.4778 0.2569
SCaBER CTRP2 8.6411 12.0275 4.8394 1.7469
VM-CUB-1 CTRP2 9.5394 16.4088 3.4039 5.8364
5637 GDSC1; GDSC2; CTRP2 10.358 21.7581 1.4261 11.6704
RT-4 GDSC1; GDSC2; CTRP2 10.479 20.8985 1.9076 9.942
HT-1197 GDSC1; GDSC2; CTRP2 11.2604 27.3371 -2.8919 13.6956
J82 GDSC1; GDSC2; CTRP2 13.2703 23.7771 2.2294 6.049
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JAR GDSC1; GDSC2 4.5434 6.3306 2.6722 1.6415
JEG-3 GDSC1; GDSC2 4.6419 12.3046 -0.1224 16.908
HEY GDSC1; GDSC2 4.8024 9.831 1.2033 9.5179
TC-YIK GDSC1; GDSC2 4.823 8.4782 1.8616 5.6671
SKG-IIIa GDSC1; GDSC2 4.927 6.7057 2.7069 1.0479
LB831-BLC GDSC1; GDSC2 4.9373 8.3807 1.9784 4.7882
SW954 GDSC1; GDSC2 5.0392 10.8595 0.8705 10.8604
OVCA420 GDSC1; GDSC2 5.0707 7.1031 2.6134 1.3053
NEC8 GDSC1; GDSC2 5.2614 16.8225 -1.8881 22.5312
NT2-D1 GDSC1; GDSC2 5.303 7.039 2.7427 0.6212
MS751 GDSC1; GDSC2 5.317 6.8188 2.8299 0.3607
PWR-1E GDSC1; GDSC2 5.325 7.6114 2.5274 1.4218
OMC-1 [Human cervical carcinoma] GDSC1; GDSC2 5.3532 7.5759 2.555 1.2788
NCC-IT GDSC2 5.4379 6.9789 2.8188 0.3363
SiSo GDSC1; GDSC2 5.4844 11.7028 0.7678 10.4711
SW962 GDSC1; GDSC2 5.5835 7.691 2.6128 0.8701
CAL-39 GDSC1; GDSC2 5.6144 7.5724 2.6709 0.6579
OVCA433 GDSC1; GDSC2 5.6396 7.732 2.621 0.8034
BPH-1 GDSC1; GDSC2 5.6731 9.0135 2.1143 2.9411
HEC-1 GDSC1; GDSC2 5.7892 7.162 2.8829 0.1197
DSH1 GDSC1; GDSC2 5.8228 7.6546 2.7236 0.4065
C-33 A GDSC1; GDSC2 5.8609 10.7686 1.4414 6.1549
DoTc2 4510 GDSC1; GDSC2 5.8845 7.4388 2.8222 0.1871
ACC-OV7 GDSC1; GDSC2 5.8988 9.4334 2.0524 2.9571
PA-1 GDSC1; GDSC2 6.0454 7.7127 2.7855 0.2075
SKN GDSC1; GDSC2 6.0698 8.5174 2.5035 0.9104
SW756 GDSC1; GDSC2 6.1401 20.5347 -3.0636 24.2031
C-4-I GDSC1; GDSC2 6.2534 16.4497 -0.9885 17.0494
UWB1.289 GDSC1; GDSC2 6.3 8.9676 2.4293 1.0053
KGN GDSC1; GDSC2 6.3185 8.2147 2.7105 0.2647
JHOS-3 GDSC1; GDSC2 6.3237 8.4882 2.616 0.4586
ME-180 GDSC1; GDSC2 6.5216 15.5746 -0.3869 13.9866
HT-3 GDSC1; GDSC2 6.5354 14.2216 0.2608 10.9861
OVMIU GDSC1; GDSC2 6.7999 11.7802 1.5188 4.3803
PEO1 GDSC1; GDSC2 7.3939 20.1528 -1.9895 18.4939
Ca Ski GDSC1; GDSC2 7.5049 19.7425 -1.7184 17.3622
HeLa GDSC1; GDSC2; CTRP2 7.566 8.6767 5.6817 0.162
SiHa GDSC1; GDSC2 7.9772 22.4669 -2.7038 19.7092
OV17R GDSC1; GDSC2 8.131 20.6908 -1.7561 16.3917
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug

References

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4 Differential effect of p38 and MK2 kinase inhibitors on the inflammatory and toxicity biomarkers in vitro. Hum Exp Toxicol. 2018 May;37(5):521-531. doi: 10.1177/0960327117715901. Epub 2017 Jun 20.