General Information of Drug (ID: DM734V4)

Drug Name
zebularine
Synonyms
Zebularine; 3690-10-6; Pyrimidin-2-one ribonucleoside; Pyrimidin-2-one beta-ribofuranoside; Pyrimidin-2-one beta-D-ribofuranoside; NSC 309132; 4-Deoxyuridine; CHEBI:46938; 1-beta-D-ribofuranosylpyrimidin-2(1H)-one; 1-beta-D-ribofuranosyl-2(1H)-pyrimidinone; UNII-7A9Y5SX0GY; 7A9Y5SX0GY; 2(1H)-Pyrimidinone, 1-beta-D-ribofuranosyl-; 2-Pyrimidone-1-beta-D-riboside; 1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1,2-dihydropyrimidin-2-one
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
Chemical Identifiers
Formula
C9H12N2O5
Canonical SMILES
C1=CN(C(=O)N=C1)C2C(C(C(O2)CO)O)O
InChI
1S/C9H12N2O5/c12-4-5-6(13)7(14)8(16-5)11-3-1-2-10-9(11)15/h1-3,5-8,12-14H,4H2/t5-,6-,7-,8-/m1/s1
InChIKey
RPQZTTQVRYEKCR-WCTZXXKLSA-N
Cross-matching ID
PubChem CID
100016
ChEBI ID
CHEBI:46938
CAS Number
3690-10-6
UNII
7A9Y5SX0GY
DrugBank ID
DB03068
TTD ID
D0IF3H

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 148 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 7.7123 9.987 7.3113 11.4136
JK1 CTRP2 8.8758 12.0706 7.4891 7.8762
JM1 CTRP2 7.7047 11.4966 6.6536 14.0232
SU-DHL-5 CTRP1 4.8237 7.419 4.7674 61.3093
KE-37 CTRP2 4.8347 6.2296 4.8334 29.1359
EoL-1 CTRP2 4.8399 7.0555 4.8136 29.1849
KMS-21-BM CTRP2 4.9027 6.2526 4.9016 28.6817
KMS-18 CTRP2 4.9227 5.9185 4.9226 28.5451
JURL-MK1 CTRP2 4.9962 7.3225 4.9572 28.186
MV4-11 CTRP2 5.1316 6.1984 5.1314 27.1533
KMS-12-BM CTRP2 5.1321 6.3524 5.1313 27.1517
EM-2 CTRP2 5.2277 6.4509 5.2269 26.5144
Ki-JK CTRP2 5.293 7.336 5.2657 26.1682
697 CTRP2 5.3284 7.7291 5.2672 26.0468
JVM-3 CTRP2 5.3611 6.9068 5.3552 25.6421
THP-1 CTRP2; CTRP1 5.3963 7.166 5.3823 25.4589
MHH-CALL-3 CTRP2 5.5307 10.0636 4.9315 26.577
Mono-Mac-1 CTRP2 5.5406 7.0223 5.5347 24.4455
KMS-27 CTRP2 5.5418 7.2512 5.5279 24.4644
SUP-M2 CTRP2 5.5485 6.2464 5.5485 24.3728
MOLT-3 CTRP2 5.5512 7.8876 5.4848 24.5797
AMO1 CTRP2; CTRP1 5.5966 10.3331 4.9114 26.4685
Peer CTRP2 5.6086 7.3007 5.5943 24.0205
DEL CTRP2 5.6637 6.1533 5.6637 23.6048
KMS-11 CTRP2; CTRP1 5.6665 7.1996 5.6578 23.6403
KM-H2 CTRP2 5.6709 7.2764 5.6594 23.5958
OPM-2 CTRP2 5.6974 8.4274 5.5579 23.8578
KMS-26 CTRP2 5.7428 6.4296 5.7428 23.0776
U-937 CTRP2; CTRP1 5.7458 8.2857 5.6357 23.4581
OCI-AML-2 CTRP2 5.8077 6.4915 5.8077 22.645
SKM-1 CTRP2; CTRP1 5.9384 7.1243 5.9359 21.8074
SR CTRP2 5.9467 7.7591 5.9155 21.8237
RCH-ACV CTRP2 6.0823 7.8186 6.0525 20.9149
BV-173 CTRP2 6.1018 8.5585 5.9704 21.1354
NU-DUL-1 CTRP2; CTRP1 6.1449 9.8582 5.6678 22.115
NCI-H929 CTRP2 6.2198 9.0699 5.9829 20.7228
JJN-3 CTRP2 6.2391 8.8852 6.0496 20.4252
L-540 CTRP2 6.3614 8.8486 6.1912 19.5424
GA-10 CTRP2 6.3951 8.7086 6.2583 19.2002
MOLM-13 CTRP2 6.4322 7.987 6.4046 18.575
RPMI-8226 CTRP2; CTRP1 6.4585 8.6792 6.3336 18.762
ALL-SIL CTRP2 6.538 9.0918 6.3245 18.5205
SU-DHL-8 CTRP2 6.6505 8.7289 6.5312 17.4371
Namalwa CTRP2 6.7208 9.4425 6.4255 17.6006
KCL-22 CTRP2 6.7338 8.5514 6.6543 16.7426
TALL-1 [Human adult T-ALL] CTRP2 6.7399 9.8113 6.3276 17.9047
KMS-34 CTRP2 6.7662 8.3773 6.7153 16.4281
CA46 CTRP2 6.8248 9.4348 6.5411 16.8663
LP-1 CTRP2; CTRP1 6.8298 11.5153 5.7552 19.8478
PF-382 CTRP2 6.9339 9.6856 6.5802 16.3988
SU-DHL-1 CTRP2 6.9757 8.5411 6.9159 15.062
Mino CTRP2 7.0354 9.3734 6.7891 15.329
L-363 CTRP2 7.0792 9.8322 6.6878 15.5744
KYO-1 CTRP2 7.0986 9.9882 6.6531 15.649
AML-193 CTRP2 7.1196 9.864 6.7202 15.3365
PL21 CTRP2; CTRP1 7.1657 9.6001 6.8613 14.7037
Karpas-299 CTRP2 7.1799 9.741 6.8283 14.757
OCI-Ly3 CTRP2 7.2377 10.4061 6.6422 15.2992
RS4;11 CTRP2 7.2635 10.6594 6.5667 15.5199
K-562 CTRP2 7.3446 9.4931 7.0892 13.3064
WSU-DLCL2 CTRP2; CTRP1 7.3454 10.0749 6.8872 14.0891
HH [Human lymphoma] CTRP2 7.3593 11.3914 6.3516 16.1063
MOLT-16 CTRP2 7.3995 9.3344 7.1977 12.7446
LAMA-84 CTRP2 7.4085 9.6366 7.1116 13.0353
Mono-Mac-6 CTRP2 7.4252 12.0134 6.1371 16.7828
A3/Kawakami CTRP2 7.653 9.1416 7.5281 10.7791
HEL CTRP2 7.6913 9.4348 7.485 10.8205
SIG-M5 CTRP2 7.7203 9.4789 7.5023 10.671
Ri-1 CTRP2 7.735 10.8791 6.9622 12.7156
A4/Fukuda CTRP2 7.7464 10.924 6.954 12.7188
NALM-6 CTRP2 7.7743 9.5839 7.5257 10.4259
BL-70 CTRP2; CTRP1 7.7992 8.8195 7.7562 9.5157
F-36P CTRP2 7.9024 11.4683 6.8637 12.6853
CML-T1 CTRP2 7.9098 9.5824 7.673 9.4821
Karpas-620 CTRP2 7.9335 12.0592 6.6167 13.6089
M-07e CTRP2 7.954 11.404 6.9447 12.2313
NCO2 CTRP2 8.0109 11.1698 7.1095 11.4249
HEL 92.1.7 CTRP2 8.0355 10.0438 7.631 9.2899
MOLM-6 CTRP2 8.0585 11.2236 7.132 11.2163
P31/FUJ CTRP2 8.0674 9.6671 7.8123 8.5053
MOLM-16 CTRP2; CTRP1 8.0946 10.5272 7.4874 9.7271
SEM CTRP2 8.1386 10.6631 7.4691 9.6584
DB CTRP2 8.1497 10.782 7.4263 9.8022
NOMO-1 CTRP2; CTRP1 8.1579 11.0338 7.3208 10.2357
L-1236 CTRP2 8.218 11.6569 7.0833 15.031
ME1 CTRP2 8.2272 10.9138 7.4429 9.5422
SUP-T11 CTRP2 8.2763 10.3262 7.7599 8.1448
NU-DHL-1 CTRP2 8.2961 12.862 6.5728 12.9431
SU-DHL-10 CTRP2 8.3029 9.3595 8.1743 6.4682
SU-DHL-6 CTRP2 8.4004 10.6357 7.7435 7.898
CMK CTRP2 8.4914 11.4313 7.4526 8.8727
KE-97 CTRP2; CTRP1 8.5497 10.1052 8.1363 5.942
DND-41 CTRP2 8.5587 11.1146 7.6694 7.823
Jurkat CTRP2 8.5949 10.001 8.229 5.456
L-428 CTRP2 8.6008 12.1088 7.223 9.5776
RPMI-6666 CTRP2 8.6657 9.9492 8.3239 4.8961
Toledo CTRP2 8.7026 11.9841 7.3771 8.7137
SET-2 CTRP2 8.7078 11.7536 7.4956 8.2088
MOLT-13 CTRP2 8.7408 10.736 8.0248 5.9371
EB1 CTRP2 8.7895 10.6966 8.0896 5.558
P12-Ichikawa CTRP2 8.8065 11.6521 7.6351 7.4126
MM1.S CTRP2 8.8459 10.9171 8.0337 5.6642
KO52 CTRP2 8.8981 10.5671 8.2536 4.6342
Pfeiffer CTRP2 8.9434 10.8228 8.1686 4.8894
SUP-T1 CTRP2 8.957 11.055 8.0657 5.2909
KMS-20 CTRP2 8.9668 16.9153 5.1493 17.1175
JeKo-1 CTRP2 8.9812 9.8758 8.6685 2.7269
OCI-Ly10 CTRP2; CTRP1 8.995 14.9465 6.1603 13.1642
MHH-CALL-4 CTRP2 9 12.6764 7.2954 8.4325
EHEB CTRP2 9.0346 12.5226 7.4019 7.9159
SK-MM-2 CTRP2 9.0457 10.9047 8.2187 4.464
MOTN-1 CTRP2 9.0679 10.5473 8.4162 3.5899
HL-60 CTRP2 9.0739 11.8883 7.7523 6.3653
GDM-1 CTRP2; CTRP1 9.1064 10.4002 8.5261 3.0785
NB4 CTRP2 9.1169 9.8323 8.815 1.8163
Reh CTRP2 9.1918 10.9266 8.3329 3.6913
ST486 CTRP2 9.2098 10.4428 8.5898 2.5756
RL CTRP2 9.2382 10.0411 8.814 1.5788
EJM CTRP2; CTRP1 9.2578 11.1183 8.295 3.7525
TF-1 CTRP2 9.2722 10.3784 8.6731 2.1083
OCI-M1 CTRP2 9.2955 11.5922 8.0857 4.5333
U266B1 CTRP2 9.2991 10.8763 8.4462 3.012
KHM-1B CTRP2 9.3184 11.9171 7.942 5.0949
RPMI-8402 CTRP2 9.3599 11.0296 8.4181 3.0201
SUP-B15 CTRP2 9.3625 12.8017 7.5359 6.7187
Ku812 CTRP2; CTRP1 9.4026 12.4686 7.7345 5.811
HD-MY-Z CTRP2 9.4721 11.5953 8.2242 3.6347
Granta-519 CTRP2 9.5211 12.8049 7.6609 5.9064
Raji CTRP2 9.5417 10.8454 8.6453 1.7753
Kasumi-1 CTRP2 9.554 10.8159 8.6683 1.6635
MOLP-8 CTRP2 9.7434 11.2865 8.5711 1.7858
SUP-HD1 CTRP2 9.7494 12.2548 8.1062 3.668
MC116 CTRP2; CTRP1 9.8169 10.73 8.8714 0.5717
Hs 611.T CTRP2 9.868 16.1351 6.2755 11.0184
HPB-ALL CTRP2 9.8838 11.6994 8.4676 2.0071
HuT 78 CTRP2 9.9028 12.2244 8.2295 2.9328
Ci-1 CTRP2 9.9335 10.8314 8.8883 0.4231
OCI-AML-5 CTRP2 9.96 11.9513 8.3982 2.1801
MOLP-2 CTRP2 10.0507 12.4899 8.2023 2.8344
Kasumi-2 CTRP2 10.1499 20.9975 4.0762 18.5355
OCI-Ly19 CTRP2 10.3921 12.3919 8.458 1.456
Karpas-422 CTRP2 10.4081 11.9296 8.6662 0.748
OCI-AML-3 CTRP2; CTRP1 10.422 11.531 8.8373 0.2914
SU-DHL-4 CTRP2; CTRP1 10.4725 11.537 8.8561 0.2298
Daudi CTRP2 10.7663 12.0568 8.7772 0.265
REC-1 CTRP2 10.8553 12.892 8.4871 0.9622
HT CTRP2; CTRP1 10.9712 12.1457 8.8243 0.1284
P3HR-1 CTRP2; CTRP1 11.0753 12.6809 8.6703 0.3627
⏷ Show the Full List of 148 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 8.9845 9.877 8.6711 2.7086
TE8 CTRP2 11.3326 12.7208 8.7558 0.1427
TE-11 CTRP2 6.7481 11.3721 5.7297 20.1411
KYSE-150 CTRP2 7.4395 9.3925 7.2238 12.5293
KYSE-510 CTRP2 7.9928 9.6682 7.7318 9.0225
KYSE-30 CTRP2 8.8638 10.3638 8.3212 4.4309
OE19 CTRP2 8.9233 10.361 8.378 4.0607
OE21 CTRP2 9.042 12.6021 7.3685 8.0415
EC-GI-10 CTRP2 9.173 15.5538 6.0036 13.4135
KYSE-520 CTRP2 9.4381 12.1351 7.9291 4.9304
TE-5 CTRP2 9.571 11.3272 8.431 2.6109
KYSE-70 CTRP2 9.6719 11.0675 8.6279 1.6577
OE33 CTRP2 9.9141 11.647 8.5119 1.7943
KYSE-450 CTRP2; CTRP1 9.9724 11.4539 8.6371 1.2486
TE-14 CTRP2 10.1164 11.9154 8.5126 1.5499
COLO 680N CTRP2 10.2843 11.8565 8.6336 0.953
KYSE-180 CTRP2 10.6902 12.6057 8.5244 0.9715
TE-4 CTRP2 10.7608 12.4747 8.6125 0.6632
TE-9 CTRP2 11.0061 12.3026 8.7818 0.1815
KYSE-140 CTRP2; CTRP1 11.2974 13.7733 8.3388 1.0897
TE-1 CTRP2 11.3318 13.4093 8.5006 0.6317
TE-10 CTRP2 11.5667 13.1924 8.6767 0.1985
KYSE-410 CTRP2; CTRP1 11.6254 13.2514 8.6777 0.1838
TE-6 CTRP2 11.8266 13.4657 8.6765 0.1458
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 9.2789 10.2511 8.7419 1.8074
PSN1 CTRP2 7.6193 9.5958 7.3538 11.5183
MIA PaCa-2 CTRP2 8.2182 10.3189 7.7037 8.5186
KP-3 CTRP2; CTRP1 8.7447 10.1732 8.2987 4.8026
HuP-T3 CTRP2 8.9984 13.6944 6.7856 10.5658
L3.3 CTRP2 9.0797 10.3601 8.5197 3.1312
HPAC CTRP2; CTRP1 9.1137 12.2217 7.6197 6.8436
Panc 10.05 CTRP2; CTRP1 9.1242 12.3615 7.5586 7.0795
SNU-213 CTRP2 9.3433 12.9755 7.4334 7.1849
Panc 04.03 CTRP2 9.3476 10.516 8.6639 2.0124
Panc 05.04 CTRP2 9.3479 10.5664 8.6391 2.1154
QGP-1 CTRP2; CTRP1 9.3506 12.0304 7.9114 5.1637
Hs 766T CTRP2 9.5444 11.187 8.4804 2.4491
Panc 08.13 CTRP2 9.5643 11.1941 8.4914 2.3723
PaTu 8988s CTRP2 9.5798 11.0893 8.5536 2.0927
KP-4 CTRP2 9.644 13.1687 7.5757 6.0473
BxPC-3 CTRP2 9.6505 11.2071 8.5462 2.0175
SW1990 CTRP2 9.6796 11.7604 8.2977 2.9891
DAN-G CTRP2 9.6973 11.6447 8.3667 2.6786
Panc 03.27 CTRP2; CTRP1 9.7091 11.0679 8.6524 1.5097
HuP-T4 CTRP2; CTRP1 9.7311 11.3321 8.5411 1.9225
CFPAC-1 CTRP2; CTRP1 9.8867 14.1294 7.285 6.8446
SNU-410 CTRP2 10.0698 12.786 8.0735 3.3229
Panc 02.03 CTRP2 10.2235 11.6633 8.6846 0.8371
HPAF-II CTRP2 10.2568 11.9887 8.5608 1.2276
AsPC-1 CTRP2 10.3645 12.9042 8.2089 2.4065
KP-2 CTRP2 10.3893 11.8205 8.7023 0.6526
Capan-1 CTRP2 10.5827 13.0696 8.2638 1.9561
SUIT-2 CTRP2; CTRP1 10.6108 16.0717 6.8606 7.4291
Capan-2 CTRP2; CTRP1 10.6668 12.6169 8.5078 1.0417
YAPC CTRP2 10.7002 14.4441 7.7017 3.9482
TCC-Pan2 CTRP2 10.849 12.1585 8.7729 0.244
SU.86.86 CTRP2 10.8802 12.1057 8.8043 0.1799
PaTu 8902 CTRP2; CTRP1 10.9312 12.7066 8.5981 0.601
PaTu 8988t CTRP2 11.069 12.2813 8.8128 0.1232
PK-45H CTRP2 11.1497 18.8938 5.8698 10.4949
PK-59 CTRP2 11.8738 13.2859 8.7541 0.0668
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 13.7518 30.4887 2.0726 18.5121
Hs 852.T CTRP2; CTRP1 6.4445 9.1709 6.2016 19.2488
RPMI-7951 CTRP2 7.2767 10.0591 6.8181 14.5181
LOX-IMVI CTRP2 7.84 10.2998 7.32 11.0295
G-361 CTRP2; CTRP1 7.9975 9.9852 7.6148 9.4565
A-375 CTRP2; CTRP1 8.2579 10.1331 7.8275 7.9544
CJM [Human melanoma] CTRP2 8.3322 10.0624 7.9329 7.3135
Hs 944.T CTRP2; CTRP1 8.4464 10.026 8.0664 6.4864
Hs 936.T CTRP2; CTRP1 8.6492 10.7076 7.9517 6.4504
WM88 CTRP2 8.9537 11.5752 7.8042 6.3932
WT2-iPS CTRP2 9.0522 9.6107 8.8639 1.7572
Hs 294T CTRP2 9.1209 10.3694 8.551 2.9148
SK-MEL-1 CTRP2; CTRP1 9.1745 10.3433 8.6131 2.5757
HMCB CTRP2 9.1794 10.2139 8.6787 2.2609
MDA-MB-435S CTRP2 9.2253 10.4278 8.6102 2.4604
WM983B CTRP2 9.3316 19.6656 4.0795 20.0797
COLO 741 CTRP2; CTRP1 9.3414 12.183 7.8278 5.5317
RVH-421 CTRP2 9.7841 11.7791 8.3624 2.567
IPC-298 CTRP2 9.7942 11.2255 8.633 1.4752
K029AX CTRP2 9.9817 11.972 8.4025 2.1347
WM115 CTRP2 10.0602 11.9769 8.45 1.8517
WM793 CTRP2 10.0658 12.597 8.1613 2.9768
MeWo CTRP2 10.2171 11.5049 8.7484 0.6391
SK-MEL-2 CTRP2 10.2214 11.0845 8.9178 0.1897
Hs 839.T CTRP2 10.2289 11.3605 8.8135 0.4403
Hs 940.T CTRP2 10.2339 14.6481 7.2856 6.2826
WM1799 CTRP2 10.2889 11.6334 8.7305 0.6405
SK-MEL-28 CTRP2; CTRP1 10.3145 10.9858 8.9936 0.054
SK-MEL-24 CTRP2 10.3252 12.0882 8.5548 1.1826
SK-MEL-31 CTRP2 10.3723 14.2854 7.5592 4.9628
Hs 688(A).T CTRP2 10.4366 11.4109 8.8837 0.1782
UACC-62 CTRP2 10.4972 11.4527 8.8922 0.1447
WM266-4 CTRP2 10.5201 11.5819 8.854 0.205
Mel JuSo CTRP2 10.5923 12.3344 8.5889 0.8467
IGR-1 CTRP2 10.6313 13.894 7.9154 3.2068
SK-MEL-30 CTRP2 10.6462 11.7349 8.8478 0.1753
HT-144 CTRP2 10.7029 12.2093 8.6919 0.4869
IGR-37 CTRP2 10.7191 11.8771 8.8246 0.193
A101D CTRP2 10.7644 11.7999 8.8694 0.1127
A2058 CTRP2 10.805 11.67 8.9283 0.0447
Hs 895.T CTRP2 10.8173 12.754 8.5256 0.8744
SK-MEL-5 CTRP2; CTRP1 10.8443 11.7664 8.9143 0.0563
IGR-39 CTRP2 10.9541 12.0723 8.8437 0.1073
SK-MEL-3 CTRP2 10.9839 12.2394 8.7959 0.1656
UACC-257 CTRP2 11.0088 12.2868 8.7885 0.1705
COLO 800 CTRP2 11.0124 12.6955 8.6383 0.4607
COLO 792 CTRP2 11.2057 13.0827 8.5724 0.5225
Mel Ho CTRP2 11.3259 12.6827 8.7667 0.1305
COLO 829 CTRP2 11.6162 18.0875 6.5763 7.1194
Malme-3M CTRP2 11.7096 13.8713 8.4848 0.4949
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 8.7127 12.1867 7.2861 9.0711
Cancer Drug Sensitivity Data Curated from 13 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-BE(2) CTRP2 7.4992 11.6631 6.3714 15.668
KP-N-SI9s CTRP2 8.4603 11.6737 7.3057 9.5503
NB1 CTRP2 8.7432 10.3079 8.2333 5.0733
SK-N-AS CTRP2 9.2045 10.3295 8.6421 2.3659
IMR-32 CTRP2 9.3465 10.6642 8.5894 2.326
SK-N-DZ CTRP2 9.5216 12.4893 7.8183 5.2464
SK-N-FI CTRP2 9.5616 17.9529 5.1242 16.0326
CHP-212 CTRP2 9.8973 12.5142 8.0855 3.5254
Kelly CTRP2 10.1287 11.4623 8.721 0.7985
KP-N-YN CTRP2 10.1927 14.0483 7.5486 5.2714
NH-6 CTRP2 10.9618 12.7059 8.6121 0.5489
CHP-126 CTRP2 11.4136 13.0888 8.6554 0.2729
SK-N-SH CTRP2 11.44 13.2237 8.6164 0.3342
⏷ Show the Full List of 13 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1196 CTRP2 8.8405 12.1163 7.4352 8.1759
SNU-478 CTRP2 8.8565 9.8957 8.5387 3.5544
HuCC-T1 CTRP2 9.0673 11.9635 7.7091 6.56
SNU-869 CTRP2 9.663 14.4925 6.9323 8.695
SNU-308 CTRP2 10.2489 13.0566 8.0639 3.1158
HuH-28 CTRP2 10.9681 12.4029 8.7304 0.283
SNU-1079 CTRP2 11.4906 13.1912 8.6482 0.2623
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U2OS CTRP2; CTRP1 8.2918 11.6144 7.177 10.4988
MHH-ES-1 CTRP2 8.8836 10.461 8.2923 4.5055
SK-N-MC CTRP2 9.1164 10.1936 8.6348 2.5725
HOS CTRP2 9.3287 10.1936 8.8093 1.4378
TC71 CTRP2 9.4582 12.5532 7.7367 5.7011
SJSA-1 CTRP2 9.7208 11.7192 8.3471 2.7232
MG-63 CTRP2 9.752 13.733 7.3788 6.6826
SW1353 CTRP2 9.9724 11.7195 8.5148 1.7102
CAL-78 CTRP2 10.0561 11.7664 8.5445 1.499
SK-ES-1 CTRP2 10.073 11.8124 8.5337 1.5202
Hs 822.T CTRP2 10.1182 11.403 8.741 0.7419
Hs 888.T CTRP2 10.3405 12.3198 8.4608 1.4983
SaOS-2 CTRP2 10.4184 13.9575 7.7477 4.1414
A-673 CTRP2 11.1044 12.5637 8.7255 0.2464
G-292 clone A141B1 CTRP2 11.2056 12.9609 8.6189 0.4181
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 75 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 CTRP2 4.7065 5.2587 4.7065 29.9861
MDA-MB-157 CTRP2 5.0372 6.6057 5.033 27.7957
HCC2218 CTRP2 8.0726 12.2343 6.6671 13.0727
HMC-1-8 CTRP2 8.1729 11.4474 7.1393 10.9078
MDA-MB-468 CTRP2 8.357 9.854 8.0469 6.8008
MDA-MB-453 CTRP2 8.7282 10.3282 8.2091 5.2079
BT-549 CTRP2 8.8271 9.9324 8.4926 3.8136
CAL-148 CTRP2 9.0564 11.2789 8.0415 5.1861
HCC1143 CTRP2 9.2651 12.1265 7.7937 5.8183
JIMT-1 CTRP2 9.3482 13.1206 7.365 7.4628
CAL-120 CTRP2 9.4881 10.8774 8.5911 2.0818
BT-20 CTRP2 9.6012 11.4383 8.3986 2.6966
MDA-MB-415 CTRP2 9.6687 15.3814 6.4939 10.4906
MDA-MB-361 CTRP2 9.9114 11.9915 8.347 5.241
HCC1954 CTRP2 9.9851 12.4838 8.161 3.0912
T-47D CTRP2 10.0175 13.1901 7.8419 4.3387
EFM-192A CTRP2 10.0298 12.2451 8.3048 2.4559
ZR-75-30 CTRP2 10.0976 13.8321 7.5863 5.2625
AU565 CTRP2 10.1156 15.0609 6.9966 7.6561
KPL-1 CTRP2 10.123 10.8633 8.9602 0.1425
Hs 578Bst CTRP2 10.1513 15.4331 6.8397 8.2401
HCC1428 CTRP2 10.1625 12.2118 8.4045 1.903
HDQ-P1 CTRP2 10.1957 12.7347 8.1813 2.7238
HCC38 CTRP2 10.2063 12.0383 8.5098 1.4617
BT-474 CTRP2 10.2869 11.7247 8.6912 0.7636
HCC1395 CTRP2 10.3492 11.9573 8.6244 0.9272
MCF-7 CTRP2; CTRP1 10.401 12.1165 8.5877 1.0236
UACC-812 CTRP2 10.4183 12.1008 8.5991 0.9515
HCC1937 CTRP2 10.5513 12.5344 8.4828 1.2206
CAMA-1 CTRP2 10.5791 12.2943 8.5991 0.8255
HCC1806 CTRP2 10.7254 12.5817 8.5519 0.8615
ZR-75-1 CTRP2 10.8318 16.3092 6.8999 6.944
SK-BR-3 CTRP2 10.846 12.7604 8.5368 0.8218
HCC1500 CTRP2 10.9829 12.2697 8.7847 0.1831
HCC1419 CTRP2 10.9984 12.483 8.7129 0.306
CAL-85-1 CTRP2 11.0341 18.0254 6.2102 9.3629
MDA-MB-231 CTRP2 11.2279 12.979 8.6213 0.4038
Hs 578T CTRP2 11.2677 13.6369 8.3804 0.9895
CAL-51 CTRP2 11.2942 12.7777 8.7215 0.1993
HCC1569 CTRP2 12.111 14.0754 8.5677 0.2265
HCC202 CTRP2 13.9789 26.5652 4.1078 12.5888
BT 416 CTRP2 7.4928 10.1986 6.995 13.237
BT 428 CTRP2 7.959 10.5862 7.3205 10.7126
BT 145 CTRP2 8.5302 10.4628 7.9522 6.7333
BT164 CTRP2 8.8849 11.4183 7.8212 6.4667
BT 172 CTRP2 9.158 11.6652 7.9352 5.4296
BT 245 CTRP2 9.1704 12.3213 7.6177 6.7406
BT 112 CTRP2 9.4169 12.0454 7.957 4.8513
BT 179 CTRP2 9.4441 15.1181 6.4449 11.106
BT 328 CTRP2 9.4656 12.8629 7.5881 6.3108
BT 159 CTRP2 9.5349 11.4133 8.362 2.9549
BT 216 CTRP2 9.5761 13.7142 7.2514 7.5218
BT 440 CTRP2 9.5791 11.7199 8.2437 3.3731
BT 224 CTRP2 9.6112 14.6905 6.7927 9.3664
BT147 CTRP2 9.7205 15.7322 6.3601 10.9415
BT 320 CTRP2 9.7985 10.8067 8.8276 0.7409
BT 286 CTRP2 9.857 12.691 7.9706 4.0574
BT 482 CTRP2 9.8627 12.6581 7.9908 3.9658
BT 239 CTRP2 9.8801 12.446 8.1065 3.4659
BT 248 CTRP2 9.966 13.8406 7.4865 5.8807
BT 330 CTRP2 10.0253 11.7342 8.5407 1.5486
BT 340 CTRP2 10.0528 11.9403 8.4624 1.8134
BT 422 CTRP2 10.0752 14.0937 7.4422 5.8891
BT 231 CTRP2 10.1162 15.814 6.6254 9.1724
BT 271 CTRP2 10.1444 11.9056 8.5336 1.4413
BT 232 CTRP2 10.1586 12.6335 8.2051 2.6789
BT 359 CTRP2 10.2225 13.2976 7.9316 3.6778
BT 498 CTRP2 10.4495 11.5631 8.832 0.278
BT 187 CTRP2 10.5024 15.5082 7.0579 6.7976
BT 444 CTRP2 10.6234 11.5885 8.8915 0.1135
BT 333 CTRP2 10.6337 11.8848 8.7872 0.2966
BT 139 CTRP2 10.691 11.8538 8.822 0.2065
BT 228 CTRP2 10.7663 16.3053 6.8565 7.2131
BT 504 CTRP2 10.7707 11.9025 8.8354 0.1604
BT 131 CTRP2 10.7755 12.3919 8.6524 0.5478
⏷ Show the Full List of 75 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 8.9118 9.7906 8.6423 2.9986
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D283 Med CTRP2 5.6451 7.6832 5.606 23.8608
ONS-76 CTRP2 8.6899 11.6442 7.5331 8.0918
SF539 CTRP2 8.8892 9.7998 8.6158 3.1615
SF268 CTRP2 9.0861 13.0437 7.1854 8.721
SNU-738 CTRP2 9.2551 10.9927 8.3523 3.4885
Hs 683 CTRP2 9.3278 10.8408 8.4868 2.7893
SF295 CTRP2; CTRP1 9.3299 11.2656 8.2765 3.6679
8-MG-BA CTRP2 9.3707 10.622 8.6291 2.1178
SW1783 CTRP2 9.4225 12.5334 7.7181 5.8436
SF126 CTRP2 9.4347 10.6819 8.6479 1.9328
DK-MG CTRP2 9.4535 11.1285 8.4414 2.7602
LN-18 CTRP2 9.4854 10.509 8.769 1.3556
CCF-STTG1 CTRP2 9.5053 10.8806 8.6021 2.0091
Daoy CTRP2 9.621 13.2318 7.5266 6.2925
GMS-10 CTRP2 9.6385 11.3466 8.4701 2.3451
M059K CTRP2 9.6939 11.0376 8.6568 1.5126
CAS-1 CTRP2 9.7216 11.9415 8.2394 3.1636
SNU-489 CTRP2 9.9387 12.1235 8.3023 2.5895
SNU-466 CTRP2 10.0233 11.3204 8.7259 0.8778
U-118MG CTRP2 10.0538 12.3598 8.2661 2.5768
T98G CTRP2 10.0736 12.2895 8.3123 2.3691
U-87MG ATCC CTRP2 10.1295 14.0424 7.5065 5.5403
A-172 CTRP2 10.1552 16.373 6.3785 10.1051
YH-13 CTRP2 10.2031 15.8607 6.6676 8.8562
TM-31 CTRP2 10.2088 14.2137 7.4796 5.5286
LN-229 CTRP2; CTRP1 10.2657 14.0397 7.6079 4.9466
U-251MG CTRP2 10.2735 12.0716 8.5334 1.3075
KNS-60 CTRP2 10.4084 13.6101 7.9062 3.5266
KNS-81 CTRP2 10.4879 11.5196 8.8641 0.1972
GOS-3 CTRP2 10.4952 13.5298 7.9996 3.0505
SNU-626 CTRP2 10.6047 12.2399 8.6341 0.7036
KNS-42 CTRP2 10.6227 12.5012 8.5343 0.9931
SNU-1105 CTRP2 10.625 11.8328 8.8032 0.2666
NMC-G1 CTRP2 10.7296 17.9507 6.0282 10.5443
Becker CTRP2 10.829 12.3331 8.6989 0.4066
GB-1 CTRP2 10.8569 12.797 8.5271 0.8428
SW1088 CTRP2 11.0341 12.4731 8.7309 0.2594
KALS-1 CTRP2 11.1206 15.8892 7.2923 5.0022
SNU-201 CTRP2 11.1612 12.3011 8.839 0.0787
YKG-1 CTRP2 11.1872 12.5258 8.7706 0.1538
GaMG CTRP2; CTRP1 11.2335 13.0159 8.6097 0.4262
SNB-75 CTRP2 11.5144 14.7875 8.0218 1.9104
DBTRG-05MG CTRP2 11.6076 13.1047 8.7224 0.1316
KG-1-C CTRP2 13.1059 32.4982 0.6275 22.6698
42-MG-BA CTRP2 13.1565 45.0455 -5.5383 31.588
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-151 CTRP2; CTRP1 5.9087 9.0692 5.6445 22.9151
KLE CTRP1 6.6903 8.8636 4.419 2.8503
RL95-2 CTRP2 7.6059 9.9109 7.2266 12.0355
HEC-265 CTRP2; CTRP1 7.824 9.4893 7.6115 9.9614
JHUEM-2 CTRP2; CTRP1 8.1716 11.4126 7.1569 10.8672
HEC-6 CTRP2; CTRP1 8.5835 9.6703 8.3605 4.9668
HEC-251 CTRP2; CTRP1 8.8153 10.9558 7.9866 5.928
ESS-1 CTRP2 9.0371 10.9724 8.1775 4.6546
HEC-108 CTRP2; CTRP1 9.2233 10.9162 8.3643 3.498
EN CTRP2 9.5508 10.7736 8.6865 1.5943
JHUEM-1 CTRP2 9.6098 10.7405 8.7424 1.2864
JHUEM-7 CTRP2 9.6931 11.7574 8.3088 2.9224
JHUEM-3 CTRP2 9.8771 13.0838 7.7929 4.7579
HEC-1-B CTRP2 10.0361 13.7571 7.5786 5.3896
HEC-1-A CTRP2 10.2668 12.9481 8.1267 2.8456
MFE-296 CTRP2 10.4199 13.0707 8.1661 2.5033
EFE-184 CTRP2 11.0473 12.4387 8.7486 0.2239
AN3-CA CTRP2 11.2106 12.7858 8.6862 0.2826
HEC-59 CTRP2; CTRP1 11.3063 12.5728 8.7975 0.099
MFE-319 CTRP2; CTRP1 11.3966 12.8275 8.742 0.1473
HEC-50B CTRP2 18.7007 40.2988 0.6788 15.9245
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 9.5222 10.8386 8.6347 1.8485
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
786-O CTRP2 7.8699 10.6222 7.2133 11.3695
VMRC-RCW CTRP2; CTRP1 8.5694 10.1326 8.1438 5.8622
BFTC-909 CTRP2 8.9291 11.1806 7.9786 5.7147
TUHR4TKB CTRP2 8.9951 11.8939 7.6816 6.8222
KMRC-1 CTRP2 9.1273 11.2137 8.1349 4.6505
CAL-54 CTRP2 9.4075 11.459 8.2417 3.6749
ACHN CTRP2 9.5295 10.5765 8.7669 1.3
769-P CTRP2 9.6344 11.8356 8.2278 3.3491
UO-31 CTRP2 9.6708 44.2872 -7.9497 37.8361
TUHR14TKB CTRP2 9.7079 17.2142 5.6111 25.2128
TUHR10TKB CTRP2 9.7568 12.2724 8.103 3.6694
VMRC-RCZ CTRP2 9.7836 11.2209 8.6285 1.5064
OS-RC-2 CTRP2 9.9664 13.1418 7.8291 4.4694
Caki-1 CTRP2 10.016 11.9398 8.4396 1.9465
KMRC-2 CTRP2 10.47 13.4869 8.0037 3.0659
RCC10RGB CTRP2; CTRP1 10.8845 12.0257 8.8392 0.135
SNU-1272 CTRP2 11.0319 12.1687 8.8384 0.0995
Caki-2 CTRP2 11.0477 12.2538 8.8146 0.1252
KMRC-20 CTRP2 12.1007 21.4795 5.2808 11.2509
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 51 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-81 CTRP1 4.7906 6.7285 4.7789 62.5527
SNU-C4 CTRP2; CTRP1 5.701 7.9904 5.6315 23.6165
SNU-175 CTRP2; CTRP1 6.5672 9.6677 6.1889 18.9523
SW403 CTRP1 6.6101 8.5013 4.5322 2.2046
LS180 CTRP2; CTRP1 6.7384 9.8385 6.318 17.9712
CW-2 CTRP2; CTRP1 7.0442 10.434 6.4274 16.6868
COLO 320 CTRP2; CTRP1 7.2221 11.3323 6.2392 16.933
SNU-1040 CTRP1 7.8666 9.8414 7.5333 21.7597
CCK-81 CTRP2 8.0673 11.2751 7.1167 11.2563
COLO205 CTRP2; CTRP1 8.5337 14.4247 6.0163 14.6796
SW948 CTRP2; CTRP1 8.5393 11.287 7.5703 8.3055
SNU-61 CTRP2; CTRP1 8.6081 10.4057 8.058 6.1431
HT115 CTRP2; CTRP1 8.786 11.3067 7.7899 6.84
COLO 678 CTRP2; CTRP1 8.8147 12.0922 7.4272 8.2922
RKO CTRP2; CTRP1 8.8704 11.2713 7.8839 6.2647
SW48 CTRP2; CTRP1 8.9805 9.8694 8.6709 2.7184
T84 CTRP2 9.0767 12.9785 7.21 8.6366
CL-40 CTRP1 9.0849 10.6431 8.3864 7.9501
SNU-407 CTRP2 9.0971 11.6694 7.8815 5.776
SNU-C1 CTRP2 9.1244 10.0003 8.7381 2.1228
LoVo CTRP2; CTRP1 9.134 10.7855 8.3577 3.7295
SNU-C5 CTRP2; CTRP1 9.169 10.4991 8.5306 2.9335
SW620 CTRP2; CTRP1 9.2498 12.7203 7.4875 7.1618
HCC-56 CTRP2 9.2588 10 8.8511 1.3854
SNU-C2A CTRP2; CTRP1 9.3051 11.0087 8.3849 3.2584
HCT 15 CTRP2 9.3306 10.9627 8.4282 3.0301
GP2d CTRP2; CTRP1 9.3781 10.7457 8.5734 2.338
SK-CO-1 CTRP2; CTRP1 9.5624 11.7537 8.2146 3.5218
KM12 CTRP2; CTRP1 9.6059 18.6916 4.7945 17.1554
HCT 116 CTRP2; CTRP1 9.6081 11.0572 8.593 1.916
HT-55 CTRP2; CTRP1 9.6342 10.8655 8.703 1.4354
COLO201 CTRP2 9.6383 10.8327 8.7174 1.3473
OUMS-23 CTRP2 9.6557 10.9912 8.6535 1.5775
RCM-1 [Human ESC] CTRP2; CTRP1 9.6814 11.397 8.4796 2.2684
CL-34 CTRP1 9.8846 11.2172 8.6969 2.4609
NCI-H747 CTRP2 9.9339 12.4466 8.1438 3.2344
C2BBe1 CTRP2; CTRP1 9.9637 12.9643 7.9137 4.127
NCI-H508 CTRP2; CTRP1 10.0289 11.6819 8.571 1.4544
MDST8 CTRP2; CTRP1 10.0408 11.3428 8.73 0.8681
CL-11 CTRP2 10.107 12.1581 8.395 2.0061
SNU-503 CTRP2 10.5722 12.7606 8.3954 1.4991
DLD-1 CTRP2; CTRP1 10.5769 11.4768 8.9136 0.0941
LS411N CTRP2; CTRP1 10.6627 12.03 8.7441 0.3803
LS513 CTRP2; CTRP1 10.6632 12.6914 8.4743 1.1523
LS123 CTRP2; CTRP1 10.6737 12.2339 8.6735 0.5666
HT-29 CTRP2; CTRP1 10.9783 11.8827 8.9214 0.037
LS1034 CTRP2 11.015 12.096 8.8574 0.0817
HCT 8 CTRP2; CTRP1 11.19 12.1976 8.8886 0.0404
NCI-H716 CTRP2 11.1928 15.4794 7.5286 4.0058
SW1417 CTRP2 11.3963 12.9816 8.6874 0.2253
SW480 CTRP1 11.9715 13.8765 8.5907 0.5017
⏷ Show the Full List of 51 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-398 CTRP2; CTRP1 6.4708 9.5051 6.135 19.4368
SNU-878 CTRP2 8.4147 10.886 7.6402 8.283
JHH-5 CTRP2 8.5913 10.8026 7.8507 7.0015
HLF CTRP2 8.6612 12.3738 7.1471 9.7615
JHH-2 CTRP2 8.9075 13.6338 6.7378 10.9484
SNU-449 CTRP2; CTRP1 8.9755 11.5535 7.8342 6.2221
JHH-4 CTRP2 9.1469 10.0168 8.7495 2.0285
SK-HEP-1 CTRP2 9.3295 10.187 8.8132 1.4203
HuH-1 CTRP2 9.353 10.4484 8.7016 1.8455
JHH-1 CTRP2 9.3689 10.2075 8.8326 1.2744
SNU-423 CTRP2 9.7262 13.6865 7.3821 6.7133
Li-7 CTRP2 9.7301 12.693 7.8766 4.6487
PLC/PRF/5 CTRP2 9.7779 11.0273 8.7152 1.179
SNU-475 CTRP2 9.817 14.0373 7.2777 6.9923
SNU-182 CTRP2 9.8557 11.6827 8.4571 2.0861
Hep-G2 CTRP2; CTRP1 9.894 11.2784 8.6745 1.2206
SNU-387 CTRP2 9.9264 14.8051 6.9808 8.0363
JHH-6 CTRP2; CTRP1 10.2544 10.9146 8.9918 0.06
Hep 3B2.1-7 CTRP2 10.7297 11.9723 8.7938 0.246
SNU-761 CTRP2 10.8494 12.1952 8.7595 0.2693
HuH-6 CTRP2 12.2239 14.5038 8.4575 0.7851
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 158 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1963 CTRP1 4.1533 6.2344 4.1443 70.6604
NCI-H1975 CTRP1 6.0277 8.0178 4.4145 4.3991
NCI-H82 CTRP1 6.463 9.422 4.0337 6.3511
NCI-H1876 CTRP1 6.6764 11.4586 5.6203 40.8798
NCI-H358 CTRP2; CTRP1 6.852 8.468 6.7943 15.8794
NCI-H1781 CTRP1 7.1017 9.2614 6.8948 31.5692
NCI-H1341 CTRP2 7.1764 9.5215 6.8971 14.5124
NCI-H1930 CTRP1 7.2023 8.773 4.6923 0.6099
NCI-H596 CTRP1 7.2565 11.3208 6.2795 34.1169
Lu-99 CTRP2; CTRP1 7.2617 10.1521 6.7668 14.7556
SCLC-21H CTRP1 7.2619 10.9747 6.4346 33.2637
COR-L279 CTRP1 7.2888 8.6476 4.7702 0.3009
NCI-H526 CTRP2 7.471 10.8705 6.6941 14.4662
Sq-1 CTRP2; CTRP1 7.488 9.4501 7.2599 12.2806
NCI-H810 CTRP2; CTRP1 7.5253 10.4339 6.9345 13.3814
NCI-H1048 CTRP1 7.6259 9.0168 4.7638 0.1967
HCC33 CTRP1 7.6751 8.9879 4.7905 0.1366
HCC2108 CTRP2; CTRP1 7.7202 10.3659 7.1689 11.97
NCI-H2073 CTRP1 7.7344 10.7358 7.0263 26.4393
HCC1195 CTRP2; CTRP1 7.7509 9.5265 7.5211 10.54
NCI-H441 CTRP2; CTRP1 7.7917 10.0864 7.3581 11.0421
NCI-H1373 CTRP2; CTRP1 7.8661 10.4485 7.2843 11.0996
NCI-H1792 CTRP2; CTRP1 7.9077 11.1861 6.999 12.1277
RERF-LC-KJ CTRP1 7.9433 9.3655 4.7561 0.1344
NCI-H1573 CTRP2; CTRP1 7.9807 12.8241 6.2955 14.796
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 8.0033 9.779 7.7017 9.1067
NCI-H446 CTRP2 8.0069 11.6577 6.878 12.3714
NCI-H1437 CTRP1 8.0088 9.7691 4.6421 0.3423
NCI-H647 CTRP2 8.091 11.6481 6.9645 11.8169
HCC44 CTRP2; CTRP1 8.2071 9.6048 7.9854 7.4527
NCI-H2286 CTRP2; CTRP1 8.2071 10.0829 7.7943 8.1903
NCI-H841 CTRP2; CTRP1 8.2165 12.1097 6.8668 11.9467
LCLC-97TM1 CTRP2; CTRP1 8.2265 11.2713 7.2747 10.2268
NCI-H838 CTRP2 8.233 10.9273 7.4423 9.5302
NCI-H650 CTRP2; CTRP1 8.2839 10.9101 7.5006 9.1686
LK2 CTRP2 8.3379 10.3159 7.8271 7.7185
DV-90 CTRP2; CTRP1 8.3771 10.9687 7.5645 8.6824
NCI-H1355 CTRP2; CTRP1 8.3862 11.0913 7.5152 8.8619
DMS 273 CTRP2; CTRP1 8.3892 12.3755 6.8971 11.3992
HCC1438 CTRP2 8.5229 10.8885 7.7439 7.6008
COR-L23 CTRP1 8.6229 10.6419 7.9604 13.9342
HCC827 CTRP2; CTRP1 8.6699 11.4524 7.6117 7.8378
HCC366 CTRP2 8.7803 10.6654 8.0962 5.5518
NCI-H2009 CTRP2; CTRP1 8.9164 12.1042 7.5081 7.7122
NCI-H1703 CTRP2 8.936 11.885 7.6345 7.1415
ChaGo-K-1 CTRP2; CTRP1 8.945 12.4261 7.3727 8.2203
NCI-H520 CTRP2 8.9473 13.2853 6.946 10.0009
NCI-H1694 CTRP2; CTRP1 8.9516 11.1014 8.0408 5.4354
LC-1/sq-SF CTRP2; CTRP1 8.9762 12.5245 7.3507 8.2491
NCI-H1838 CTRP2 9.0615 12.0459 7.663 6.7657
SBC-5 CTRP2 9.0838 13.5205 6.9452 9.7306
HOP-62 CTRP2 9.086 11.6804 7.8666 5.8609
NCI-H2170 CTRP2 9.1147 11.0025 8.2297 4.2774
MOR/CPR CTRP2 9.1542 9.8364 8.8457 1.6095
SK-MES-1 CTRP2 9.1627 11.4569 8.0433 4.966
HCC78 CTRP2; CTRP1 9.1636 11.0505 8.2473 4.1061
NCI-H2087 CTRP2 9.1826 10.9433 8.3168 3.7764
NCI-H322 CTRP2 9.1955 10.2153 8.6916 2.175
HCC4006 CTRP2; CTRP1 9.2209 10.6109 8.5182 2.8843
NCI-H2110 CTRP2; CTRP1 9.2419 14.8576 6.4124 11.6511
NCI-H1650 CTRP2 9.2528 10.4482 8.6224 2.3571
COR-L51 CTRP1 9.287 11.1242 8.3159 7.7356
COR-L88 CTRP2; CTRP1 9.3095 10.5623 8.6111 2.3007
NCI-H1693 CTRP2 9.3373 11.6634 8.0839 4.4635
NCI-H1581 CTRP2 9.3581 13.346 7.2603 7.8831
NCI-H1568 CTRP2; CTRP1 9.3609 11.8625 8.0035 4.7579
NCI-H2291 CTRP2 9.3647 11.0909 8.3913 3.1238
NCI-H2030 CTRP2; CTRP1 9.3667 11.1778 8.353 3.3086
NCI-H2081 CTRP2; CTRP1 9.3717 14.662 6.6172 10.5611
HCC1833 CTRP2; CTRP1 9.3822 10.4529 8.7252 1.7262
T3M-10 CTRP2; CTRP1 9.383 11.0204 8.4442 2.8979
NCI-H1666 CTRP2; CTRP1 9.3883 11.3158 8.2979 3.473
PC-14 CTRP2 9.3988 11.5121 8.2084 3.8294
NCI-H2228 CTRP2 9.4382 11.1571 8.4156 2.8938
RERF-LC-MS CTRP2 9.4693 10.8252 8.6029 2.0633
LXF 289 CTRP2; CTRP1 9.5009 11.3721 8.3567 3.0331
NCI-H196 CTRP2 9.5168 10.6895 8.7035 1.5755
NCI-H2023 CTRP2; CTRP1 9.5669 12.3189 7.9417 4.6792
CAL-12T CTRP2; CTRP1 9.6022 11.6428 8.3026 3.1184
LUDLU-1 CTRP2 9.6118 11.8745 8.1919 3.5344
NCI-H1299 CTRP2; CTRP1 9.6253 12.058 8.1116 3.8459
NCI-H522 CTRP2; CTRP1 9.7498 11.745 8.355 2.6476
SHP-77 CTRP2; CTRP1 9.7578 11.101 8.6682 1.3844
NCI-H2141 CTRP2; CTRP1 9.7604 12.4187 8.0377 3.9598
LOU-NH91 CTRP2 9.7958 11.7554 8.3819 2.4714
DMS 53 CTRP2 9.7973 12.2386 8.1487 3.4188
Calu-6 CTRP2; CTRP1 9.8101 12.8883 7.8398 4.6716
NCI-H2126 CTRP2; CTRP1 9.8683 11.3945 8.601 1.5067
Calu-3 CTRP2; CTRP1 9.9035 12.5973 8.0495 3.6632
NCI-H146 CTRP2 9.9174 12.4615 8.1251 3.3344
COR-L95 CTRP2 9.9261 11.6626 8.5122 1.7778
NCI-H1563 CTRP2 9.9319 12.6315 8.0529 3.6068
HCC1588 CTRP2 9.9463 11.4745 8.612 1.3717
RERF-LC-Ad2 CTRP2 9.9515 13.4875 7.6492 5.2326
NCI-H1869 CTRP2 9.9561 11.9339 8.4039 2.1629
NCI-H2106 CTRP2 9.9648 13.2381 7.7809 4.6695
NCI-H1435 CTRP2; CTRP1 9.9866 12.0367 8.3751 2.2358
NCI-H1155 CTRP2 9.9896 13.2872 7.7748 4.6562
VMRC-LCD CTRP2; CTRP1 10.0203 11.8952 8.4631 1.8503
HOP-92 CTRP2 10.0375 14.2154 7.3549 13.0824
NCI-H2029 CTRP2; CTRP1 10.0401 11.547 8.6346 1.1846
NCI-H69 CTRP2 10.0473 12.618 8.1389 3.0923
NCI-H1793 CTRP2; CTRP1 10.0604 12.28 8.3082 2.4024
RERF-LC-A1 CTRP2 10.0689 12.2681 8.3193 2.3477
NCI-H1944 CTRP2; CTRP1 10.0947 13.0833 7.9476 3.7948
HCC15 CTRP2; CTRP1 10.1033 13.3944 7.8069 4.3786
EPLC-272H CTRP2; CTRP1 10.1178 12.0245 8.4635 1.7322
SK-LU-1 CTRP2; CTRP1 10.1483 11.9876 8.5029 1.5733
A-549 CTRP2; CTRP1 10.1609 13.0145 8.0256 3.3876
HCC1359 CTRP1 10.1743 11.2496 8.8373 0.9113
NCI-H2196 CTRP2 10.1775 11.7085 8.6403 1.0272
RERF-LC-Ad1 CTRP2 10.215 11.1 8.9093 0.2101
SW1573 CTRP2 10.2172 12.7098 8.2069 2.5961
NCI-H2405 CTRP2; CTRP1 10.239 11.9623 8.5625 1.239
COLO 668 CTRP2; CTRP1 10.3228 13.1788 8.0542 3.0571
DMS 114 CTRP2 10.335 14.9659 7.203 6.4637
NCI-H1836 CTRP1 10.3457 11.832 8.6803 1.6519
NCI-H23 CTRP2; CTRP1 10.3479 13.0212 8.1441 2.6751
DMS 79 CTRP2 10.3627 12.1977 8.5273 1.242
NCI-H1339 CTRP2 10.3731 12.5473 8.3774 1.7661
BEN CTRP2; CTRP1 10.3803 11.069 8.9836 0.0485
NCI-H1755 CTRP2; CTRP1 10.389 12.0274 8.6196 0.9292
NCI-H2342 CTRP2; CTRP1 10.4386 13.2211 8.112 2.7113
NCI-H2444 CTRP2 10.5099 11.8668 8.7403 0.4695
HCC2935 CTRP2; CTRP1 10.5102 12.808 8.3438 1.7653
HCC1171 CTRP2 10.5174 14.4288 7.5889 4.6379
NCI-H1395 CTRP2 10.5205 13.0707 8.2269 2.1588
KNS-62 CTRP2; CTRP1 10.6006 11.9797 8.7365 0.4296
NCI-H889 CTRP2 10.6797 23.4332 3.2791 20.0154
Calu-1 CTRP2 10.7047 14.1436 7.8452 3.3866
NCI-H1092 CTRP2 10.8092 12.3927 8.6672 0.4923
COR-L105 CTRP2 10.826 13.7054 8.1187 2.2256
NCI-H1623 CTRP2 10.833 13.734 8.1099 2.2503
NCI-H1915 CTRP2; CTRP1 10.8723 12.549 8.6339 0.542
NCI-H226 CTRP2 10.9285 12.2226 8.7808 0.2048
NCI-H2172 CTRP2; CTRP1 10.9402 12.4049 8.723 0.3194
NCI-H661 CTRP2; CTRP1 10.9446 13.4736 8.2863 1.5292
HCC95 CTRP2 10.9731 12.4123 8.7289 0.284
Lu-65 CTRP2; CTRP1 10.9748 13.8899 8.1208 2.0675
NCI-H211 CTRP2 11.0036 12.8046 8.592 0.577
EKVX CTRP2 11.0054 18.6956 5.8633 10.7429
LCLC-103H CTRP2; CTRP1 11.0091 12.2547 8.8 0.1535
NCI-H1734 CTRP2 11.0574 13.3115 8.4125 1.0404
DMS 454 CTRP2 11.0579 16.8786 6.7806 7.0923
COLO 699 CTRP2; CTRP1 11.1069 12.6014 8.7174 0.2703
NCI-H1105 CTRP2; CTRP1 11.1171 12.9922 8.5735 0.5779
NCI-H727 CTRP2; CTRP1 11.2786 12.8779 8.6793 0.273
NCI-H460 CTRP2; CTRP1 11.287 23.4288 3.7482 17.6142
NCI-H292 CTRP2 11.2894 12.8688 8.6868 0.2566
NCI-H3255 CTRP1 11.2944 12.7923 8.7211 0.447
SW1271 CTRP2 11.4983 12.94 8.7399 0.1307
EBC-1 CTRP2; CTRP1 11.594 13.2938 8.6509 0.2298
HCC2279 CTRP2 11.6661 13.3858 8.6454 0.22
NCI-H2085 CTRP2 11.7169 13.3678 8.6706 0.1738
NCI-H1184 CTRP2 11.822 13.5041 8.6615 0.1644
NCI-H2122 CTRP2; CTRP1 12.1619 29.0645 1.6222 21.8952
NCI-H1651 CTRP2 15.1461 59.1026 -10.9823 33.9748
Hs 888.Lu CTRP2 9.9932 13.2248 7.8078 4.5154
⏷ Show the Full List of 158 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 6.4422 11.1667 5.495 21.8691
H-STS CTRP2 8.9988 14.1413 6.5627 11.4879
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Aska-SS CTRP2 8.0594 11.4159 7.0431 11.5738
Yamato-SS CTRP2 9.766 13.8563 7.3285 6.868
SW982 CTRP2 6.662 9.6506 6.2963 18.2498
BT-16 CTRP2 8.1209 10.6675 7.4492 9.783
MES-SA CTRP2 8.6305 11.1694 7.7106 7.4879
TTC-709 CTRP2 8.924 18.6317 4.2552 20.3318
HT-1080 CTRP2; CTRP1 9.2392 11.749 7.9644 5.1781
G-402 CTRP2 9.3122 11.2287 8.2807 3.6827
RKN CTRP2; CTRP1 9.3685 13.0998 7.3952 7.3254
Tm87-16 CTRP2 9.4502 16.0525 5.9831 12.9578
GCT CTRP2 9.4697 12.1238 7.9596 4.7462
KYM-1 CTRP2 9.4772 12.8717 7.593 6.2694
TE 617.T CTRP2 9.5615 12.8895 7.6504 5.8788
RD CTRP2 9.615 14.702 6.79 9.3708
TE 441.T CTRP2 9.65 11.9866 8.1651 3.5834
A-204 CTRP2 9.7122 12.2073 8.1024 3.7428
SK-LMS-1 CTRP2 9.7138 11.2776 8.5556 1.8887
Hs 729.T CTRP2 9.7157 11.7933 8.3075 2.8932
Rh41 CTRP2 9.7668 16.1532 6.187 11.5556
G-401 CTRP2; CTRP1 9.8419 11.9523 8.3187 2.6601
BT-12 CTRP2 10.0625 10.7249 8.987 0.1135
Rh18 CTRP2 11.5023 13.0011 8.7201 0.1539
SK-UT-1 CTRP2 12.4402 23.0622 4.7517 12.5925
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 9.5607 12.455 7.8658 4.9796
JHOC-5 CTRP2; CTRP1 6.6895 9.1383 6.4785 17.53
A2780 CTRP2; CTRP1 6.7695 9.134 6.5669 16.9673
COV318 CTRP1 6.9424 7.787 4.9409 0.0602
OVMANA CTRP1 7.2766 8.4245 4.8424 0.1414
JHOS-4 CTRP1 7.637 9.227 4.6953 0.3548
COV362 CTRP2; CTRP1 8.3342 11.7262 7.1637 10.4545
TYK-nu CTRP2; CTRP1 8.4698 12.2525 7.0347 10.6773
OVCAR-8 CTRP2; CTRP1 8.547 11.0533 7.6904 7.7926
HEY A8 CTRP2; CTRP1 8.609 11.453 7.5523 8.1922
OVKATE CTRP1 8.7387 11.3053 7.7473 15.2035
SNU-8 CTRP2 8.8765 22.5296 2.2667 26.088
COV434 CTRP2; CTRP1 8.9203 11.6408 7.7451 6.7391
JHOM-1 CTRP2; CTRP1 8.9248 10.987 8.0736 5.3554
OVCAR-4 CTRP2; CTRP1 9.1166 11.8497 7.8111 6.0613
OV-90 CTRP2; CTRP1 9.1514 12.1427 7.6942 6.4843
OVK18 CTRP2; CTRP1 9.2781 11.4203 8.1607 4.2789
TOV-112D CTRP2 9.4098 13.1406 7.4048 7.1815
ES2 CTRP2 9.4379 10.8833 8.5508 2.3305
OV7 CTRP2; CTRP1 9.6179 12.0059 8.1353 3.7865
SNU-119 CTRP2 9.6643 14.2236 7.0672 8.1325
OVCAR-5 CTRP2 9.6651 11.7512 8.2916 3.0366
TOV-21G CTRP2 9.672 11.1549 8.5861 1.8249
SNU-840 CTRP2; CTRP1 9.6957 12.2222 8.0866 3.8612
OC 314 CTRP2 9.7304 10.8864 8.751 1.0994
OV56 CTRP2 9.8052 10.97 8.758 0.9868
OVTOKO CTRP2 9.8522 11.9691 8.3177 2.6493
RMG-I CTRP2; CTRP1 9.9759 13.1441 7.8385 4.442
JHOS-2 CTRP2 10.0851 14.0136 7.4886 5.6828
OVSAHO CTRP2 10.1254 12.6904 8.1564 2.915
EFO-21 CTRP2; CTRP1 10.1599 13.1799 7.9457 3.7093
DOV13 CTRP2 10.1906 13.3408 7.8894 3.8923
COV644 CTRP2; CTRP1 10.2881 12.9033 8.1654 2.692
Caov-3 CTRP2; CTRP1 10.3844 12.1502 8.5643 1.1162
OVISE CTRP2 10.4203 11.9825 8.6502 0.788
RMUG-S CTRP1 10.4706 16.809 6.4027 18.2465
OAW42 CTRP2; CTRP1 10.6172 11.6177 8.8836 0.1348
ONCO-DG-1 CTRP2 10.6513 16.8978 6.4869 8.8633
EFO-27 CTRP2; CTRP1 10.6618 12.2012 8.6811 0.5534
FU-OV-1 CTRP2 11.2963 12.9212 8.6705 0.283
SK-OV-3 CTRP2; CTRP1 11.4742 13.042 8.6953 0.1936
Kuramochi CTRP2 11.6048 13.5281 8.5701 0.3644
OAW28 CTRP2 11.7347 13.6146 8.5896 0.289
MCAS CTRP2 12.5073 30.2385 1.2971 22.1005
IGROV-1 CTRP2; CTRP1 15.4656 27.6834 4.5188 9.6168
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 11.1953 12.603 8.7463 0.1869
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2; CTRP1 6.8538 9.0624 6.6765 16.2885
NCI-H2452 CTRP2 9.4428 11.419 8.2891 3.4141
ACC-MESO-1 CTRP2 9.479 10.4886 8.7743 1.3434
NCI-H2052 CTRP2; CTRP1 9.6377 11.3145 8.4852 2.2847
MPP 89 CTRP2 9.895 11.7757 8.4389 2.1057
JL-1 CTRP2 10.1352 12.5891 8.2109 2.6869
NCI-H28 CTRP2; CTRP1 10.4606 12.648 8.3827 1.6548
IST-Mes1 CTRP2 12.874 23.2292 4.9641 11.2769
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
22Rv1 CTRP2 7.8456 10.87 7.0791 11.965
LNCaP clone FGC CTRP2 9.2284 12.074 7.7897 5.9052
DU145 CTRP2 9.3139 10.3746 8.708 1.887
PaCa-3 CTRP2; CTRP1 9.5459 10.8666 8.638 1.7992
VCaP CTRP2 9.5504 10.7719 8.687 1.5927
NCI-H660 CTRP2 10.4433 17.2703 6.1518 10.5263
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 8.6931 10.3656 8.1574 5.5034
A-253 CTRP2 11.1488 13.0453 8.5621 0.5751
Cancer Drug Sensitivity Data Curated from 34 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
GSS CTRP2 5.3925 7.12 5.3802 25.4543
HGC-27 CTRP2 6.9385 9.1729 6.7401 15.8002
SNU-16 CTRP2 7.321 9.4439 7.0789 13.4142
SNU-620 CTRP2 7.3428 9.0682 7.2083 12.879
AGS CTRP2; CTRP1 7.3539 9.1459 7.2014 12.8977
23132/87 CTRP2 8.0084 17.278 4.1323 22.7159
ECC10 CTRP2 8.2561 10.3761 7.717 8.3676
SNU-1 CTRP2 8.4066 10.1115 7.988 6.9011
HuG1-N CTRP2 8.5039 10.6136 7.8558 7.189
NUGC-4 CTRP2; CTRP1 8.8517 10.127 8.4241 4.0345
Hs 746.T CTRP2 8.8665 10.7317 8.1437 5.1609
SNU-719 CTRP2 8.8946 12.0081 7.5368 7.6373
ECC12 CTRP2 9.0054 9.8722 8.693 2.57
GSU CTRP2 9.1531 9.7311 8.8973 1.3953
SNU-601 CTRP2 9.4028 10.976 8.4781 2.6935
KE-39 CTRP2 9.4057 12.3644 7.789 5.5765
NCI-N87 CTRP2 9.4328 12.0386 7.973 4.7558
NCC-StC-K140 CTRP2 9.6179 12.8388 7.7194 11.6334
SNU-216 CTRP2 9.6189 19.9436 4.1763 19.2059
IM95 CTRP2 9.6555 11.3117 8.499 2.2015
SNU-5 CTRP2 9.6588 10.8631 8.7164 1.3239
NUGC-3 CTRP2 9.8556 12.7115 7.9596 4.105
SH-10-TC CTRP2; CTRP1 9.8612 11.1933 8.6895 1.1786
MKN1 CTRP2 9.9716 11.8677 8.445 1.9815
LMSU CTRP2 10.2823 13.3565 7.9435 3.5482
MKN45 CTRP2 10.3697 11.3693 8.872 0.2256
MKN74 CTRP2; CTRP1 10.3939 15.8346 6.8209 7.9256
KATO III CTRP2 10.4516 12.0883 8.6215 0.8534
MKN7 CTRP2; CTRP1 10.8575 12.3813 8.6926 0.4079
SNU-668 CTRP2 11.0754 12.3354 8.7962 0.1436
Fu97 CTRP2; CTRP1 11.2114 12.7144 8.7125 0.2364
SNU-685 CTRP2 9.5035 11.0711 8.5072 2.4039
SNG-M CTRP2; CTRP1 10.3036 13.5262 7.8768 3.7847
SNU-1077 CTRP2 10.8803 12.5614 8.6326 0.5409
⏷ Show the Full List of 34 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CGTH-W-1 CTRP2 7.947 10.6236 7.2918 10.8575
BHT-101 CTRP2 8.6873 12.0923 7.3098 9.0276
ML-1 [Human leukemia] CTRP2 9.0486 11.9882 7.6807 6.7171
CAL-62 CTRP2 9.2258 12.9358 7.3567 7.7299
FTC-238 CTRP2 9.2475 11.0675 8.3086 3.6866
SW579 CTRP2 9.3458 12.4071 7.7194 5.9789
B-CPAP CTRP2 9.4684 12.5777 7.7325 5.7001
FTC-133 CTRP2 10.0698 12.0504 8.4219 1.9482
8505C CTRP2 10.2476 12.187 8.4668 1.5743
8305C CTRP2 10.2621 19.1061 5.1052 14.8128
TT2609-C02 CTRP2 10.6798 12.4235 8.595 0.7662
TT CTRP2 11.5527 12.8417 8.7926 0.0708
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 29 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 8.6108 10.9615 7.7928 7.1939
BICR 22 CTRP2 8.8403 10.5821 8.1928 5.0157
PE/CA-PJ15 CTRP2 8.9399 12.1681 7.4969 7.7104
BICR 6 CTRP2 8.9648 9.4109 8.8676 1.9608
SNU-1214 CTRP2 8.998 11.2513 8.0044 5.4616
HSC-2 CTRP2; CTRP1 9.0595 10.361 8.5014 3.2503
BICR 56 CTRP2 9.1265 9.8523 8.8135 1.8022
PE/CA-PJ34 (clone C12) CTRP2 9.2302 10.3384 8.6589 2.2463
Detroit 562 CTRP2 9.2451 10.8073 8.4367 3.1521
SCC-9 CTRP2; CTRP1 9.6006 12.2326 8.0102 4.336
BHY CTRP2 9.7535 12.8348 7.8242 4.8281
SCC-4 CTRP2 9.7558 11.0619 8.6853 1.3208
SCC-25 CTRP2 9.7742 11.6521 8.4169 2.3612
HSC-4 CTRP2 9.801 11.1939 8.6521 1.3928
SNU-1066 CTRP2 9.8942 11.5864 8.5276 1.7585
BICR 18 CTRP2 9.9702 12.5878 8.1007 3.356
HSC-3 CTRP2 10.0064 11.4169 8.6736 1.0792
BICR 16 CTRP2 10.4545 12.2317 8.562 1.0424
CAL-33 CTRP2 10.4717 12.1757 8.5948 0.9218
YD-8 CTRP2 10.601 12.1858 8.6544 0.6481
PE/CA-PJ49 CTRP2 10.7835 12.4024 8.6519 0.5448
SNU-46 CTRP2 10.8722 12.4131 8.6867 0.4147
FaDu CTRP2 10.959 12.1725 8.8104 0.1505
BICR 31 CTRP2 11.1663 16.5295 7.0196 6.0046
SNU-899 CTRP2 11.4952 12.444 8.9042 0.0143
SNU-1041 CTRP2 11.5208 15.8026 7.5775 3.4532
CAL-27 CTRP2 12.1871 20.384 5.8623 9.0336
PE/CA-PJ41 (clone D2) CTRP2 12.6037 19.2264 6.6631 5.5911
SNU-1076 CTRP2 14.1386 26.4274 4.276 11.8717
⏷ Show the Full List of 29 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JMSU-1 CTRP2 6.4368 8.474 6.3476 18.7557
HT-1376 CTRP2; CTRP1 7.1964 10.7809 6.446 18.647
5637 CTRP2; CTRP1 7.788 9.6971 7.5008 10.4794
UM-UC-3 CTRP2; CTRP1 8.1164 10.0303 7.7216 8.7182
VM-CUB-1 CTRP2 8.9706 10.4054 8.3995 3.8668
253J CTRP2 9.0367 11.257 8.0353 5.2521
T24 CTRP2 9.1613 10.1134 8.7136 2.1502
647V CTRP2 9.187 10.4441 8.5701 2.7028
SCaBER CTRP2 9.2675 10.5049 8.6061 2.3985
BFTC-905 CTRP2 9.6585 11.5086 8.4054 2.5794
BC-3C CTRP2 9.6817 11.5757 8.3893 2.61
TCCSUP CTRP2 9.801 11.2422 8.6295 1.4802
253J-BV CTRP2 9.9183 12.756 7.9828 3.9135
J82 CTRP2 9.9303 17.5395 5.6254 13.4648
UM-UC-1 CTRP2 9.9559 11.7803 8.4761 1.8804
SW1710 CTRP2 10.0764 14.0921 7.4438 5.8805
KU-19-19 CTRP2 10.1157 21.8796 3.6094 20.0497
U-BLC1 CTRP2 10.1277 11.7594 8.5898 1.2547
KMBC-2 CTRP2; CTRP1 10.2527 14.6754 7.2859 6.2524
639V CTRP2 10.3165 19.395 5.0038 15.0825
CAL-29 CTRP2 10.7363 12.4436 8.6137 0.6754
RT-112 CTRP2 10.7622 12.0879 8.764 0.2933
HT-1197 CTRP2 11.022 17.3242 6.5414 8.0858
RT-4 CTRP2; CTRP1 11.6459 13.0852 8.7427 0.1039
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 8.3392 12.4812 6.799 11.9164

References

1 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 4729).