Details of the Drug

General Information of Drug (ID: DM9SX6Y)

Drug Name
INDISULAM
Synonyms
Indisulam; 165668-41-7; E7070; N-(3-chloro-1H-indol-7-yl)benzene-1,4-disulfonamide; UNII-WJ98J3NM90; E-7070; E 7070; N-(3-Chloro-1H-indol-7-yl)-1,4-benzenedisulfonamide; CHEMBL77517; WJ98J3NM90; N1-(3-chloro-1H-indol-7-yl)benzene-1,4-disulfonamide; 1,4-Benzenedisulfonamide, N-(3-chloro-1H-indol-7-yl)-; ER-35744; N-(3-Chloro-1H-indol-7-yl)benzene-1,4disulfonamide; Indisulam (IND); indisulam (e7070); Indisulam (USAN/INN); AC1Q6VCX; AC1L50QL; SCHEMBL91389; N-(3-chloro-7-indolyl)-1,4-benzenedisulphonamide; Indisulam [USAN:INN:BAN]
Indication
Disease Entry ICD 11 Status REF
Lymphoma 2A80-2A86 Phase 2 [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 385.8
Logarithm of the Partition Coefficient (xlogp) 1.8
Rotatable Bond Count (rotbonds) 4
Hydrogen Bond Donor Count (hbonddonor) 3
Hydrogen Bond Acceptor Count (hbondacc) 6
Chemical Identifiers
Formula
C14H12ClN3O4S2
IUPAC Name
4-N-(3-chloro-1H-indol-7-yl)benzene-1,4-disulfonamide
Canonical SMILES
C1=CC2=C(C(=C1)NS(=O)(=O)C3=CC=C(C=C3)S(=O)(=O)N)NC=C2Cl
InChI
InChI=1S/C14H12ClN3O4S2/c15-12-8-17-14-11(12)2-1-3-13(14)18-24(21,22)10-6-4-9(5-7-10)23(16,19)20/h1-8,17-18H,(H2,16,19,20)
InChIKey
SETFNECMODOHTO-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
216468
ChEBI ID
CHEBI:145431
CAS Number
165668-41-7
UNII
WJ98J3NM90
DrugBank ID
DB06370
TTD ID
D04IIU
INTEDE ID
DR0873
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Carbonic anhydrase IX (CA-IX) TT2LVK8 CAH9_HUMAN Modulator [2]

Drug-Metabolizing Enzyme (DME)
DME Name DME ID UniProt ID MOA REF
Cytochrome P450 2C9 (CYP2C9) DE5IED8 CP2C9_HUMAN Substrate [3]
Mephenytoin 4-hydroxylase (CYP2C19) DEGTFWK CP2CJ_HUMAN Substrate [4]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Retinoblastoma-associated protein (RB1) OTQJUJMZ RB_HUMAN Post-Translational Modifications [5]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Lymphoma
ICD Disease Classification 2A80-2A86
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Carbonic anhydrase IX (CA-IX) DTT CA9 6.08E-15 2.8 7.25
Mephenytoin 4-hydroxylase (CYP2C19) DME CYP2C19 1.02E-01 -2.84E-01 -7.34E-01
Cytochrome P450 2C9 (CYP2C9) DME CYP2C9 1.62E-02 -4.23E-01 -1.25E+00
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 135 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 0.1863 3.2157 0.1072 32.6267
JK1 CTRP2 1.4325 3.6795 1.3743 24.2595
JM1 CTRP2 1.3949 5.8619 0.8117 26.3442
MV4-11 CTRP2 -2.9193 -1.6996 -2.9193 53.0553
NCO2 CTRP2 -2.6432 -0.5168 -2.6439 51.2147
SET-2 CTRP2 -2.593 0.5791 -2.6075 50.8718
OCI-AML-3 CTRP2; CTRP1 -2.2015 0.3287 -2.2057 48.3279
SU-DHL-5 CTRP1 -1.9756 -0.7207 -1.9756 94.5874
NU-DUL-1 CTRP2; CTRP1 -1.7448 1.4155 -1.7699 45.3359
GA-10 CTRP2 -1.518 -0.1207 -1.5181 43.7199
F-36P CTRP2 -1.3727 1.5997 -1.3961 42.8142
L-540 CTRP2 -1.247 3.2544 -1.4287 42.3408
SEM CTRP2 -1.2354 0.5895 -1.2362 41.8395
BV-173 CTRP2 -1.166 2.7054 -1.2669 41.636
OCI-M1 CTRP2 -1.0469 1.1852 -1.0519 40.5969
M-07e CTRP2 -0.8293 2.3676 -0.8798 39.2827
CMK CTRP2 -0.7809 1.5641 -0.7899 38.8378
WSU-DLCL2 CTRP2; CTRP1 -0.4332 1.9074 -0.4454 36.5936
BL-70 CTRP2; CTRP1 -0.4087 1.1195 -0.4093 36.3927
697 CTRP2 -0.1204 1.2535 -0.1207 34.4098
RPMI-8402 CTRP2 -0.1101 1.6519 -0.1127 34.3487
GDM-1 CTRP2; CTRP1 0.0713 3.6399 -0.0728 33.6639
EB1 CTRP2 0.0778 3.708 -0.0781 33.5946
NALM-6 CTRP2 0.0936 1.577 0.0928 32.9856
KMS-11 CTRP2; CTRP1 0.0966 5.9644 -0.6284 35.1977
MOLM-6 CTRP2 0.1367 6.577 -0.7964 35.4379
KMS-21-BM CTRP2 0.1979 3.4279 0.093 32.634
MOLM-16 CTRP2; CTRP1 0.2136 4.758 -0.1499 33.4117
CML-T1 CTRP2 0.2859 1.8053 0.2845 31.7064
MOLM-13 CTRP2 0.2914 3.1136 0.2294 31.8711
SKM-1 CTRP2; CTRP1 0.296 1.5915 0.2956 31.7018
Peer CTRP2 0.388 3.2288 0.3193 31.2506
KHM-1B CTRP2 0.4215 3.2495 0.3525 31.0288
Daudi CTRP2 0.4612 3.1633 0.4034 30.7269
NB4 CTRP2 0.4813 1.8352 0.4806 30.4024
OCI-AML-5 CTRP2 0.5508 1.3807 0.5508 29.9368
Ku812 CTRP2; CTRP1 0.5905 3.0643 0.5487 29.8799
MOLT-3 CTRP2 0.6535 1.6789 0.6535 29.2527
JVM-3 CTRP2 0.6657 3.8603 0.5292 29.6304
NU-DHL-1 CTRP2 0.6736 3.6897 0.5643 29.4864
MOLT-16 CTRP2 0.7357 2.1805 0.7338 28.7115
Ri-1 CTRP2 0.7479 4.8758 0.4005 29.7927
Namalwa CTRP2 0.8044 3.3809 0.743 28.4537
MOLP-8 CTRP2 0.8167 3.5846 0.7318 28.4515
OCI-Ly19 CTRP2 0.8995 2.6776 0.89 27.6456
SUP-M2 CTRP2 0.9119 3.7701 0.8077 27.8833
Granta-519 CTRP2 0.9491 4.4095 0.731 28.025
MOTN-1 CTRP2 0.9506 6.3881 0.1492 29.9593
JJN-3 CTRP2 0.9943 3.3065 0.9504 27.1298
ST486 CTRP2 1.1199 4.4582 0.9061 26.8761
L-363 CTRP2 1.1442 2.4135 1.1429 25.9879
PF-382 CTRP2 1.1452 4.1729 0.9914 26.5006
Reh CTRP2 1.1688 2.601 1.1654 25.8311
JURL-MK1 CTRP2 1.2292 5.6459 0.7023 27.2363
KE-37 CTRP2 1.2366 4.2737 1.071 25.9335
P12-Ichikawa CTRP2 1.2838 4.5685 1.0598 25.8223
U-937 CTRP2; CTRP1 1.2946 6.1549 0.6068 27.4296
SU-DHL-6 CTRP2 1.2974 4.2375 1.1439 25.487
Karpas-299 CTRP2 1.3396 4.8804 1.0448 25.699
EM-2 CTRP2 1.407 5.3718 0.9807 25.7145
RCH-ACV CTRP2 1.4135 5.3691 0.9887 25.6665
OPM-2 CTRP2 1.4917 5.6647 0.9816 25.4512
RPMI-6666 CTRP2 1.5232 3.8831 1.4451 23.7233
A4/Fukuda CTRP2 1.5449 6.2838 0.8273 25.8334
JeKo-1 CTRP2 1.5876 6.748 0.7004 26.1484
LP-1 CTRP2; CTRP1 1.6609 7.7372 0.3866 27.0681
OCI-AML-2 CTRP2 1.6754 3.7983 1.618 22.6388
SUP-T1 CTRP2 1.6772 6.7896 0.7801 25.6035
LAMA-84 CTRP2 1.6954 5.261 1.3281 23.5959
Jurkat CTRP2 1.7198 4.7293 1.4972 22.9188
MOLT-13 CTRP2 1.7361 4.9889 1.4489 23.0398
MHH-CALL-4 CTRP2 1.7681 5.8881 1.2074 23.81
DB CTRP2 1.8132 5.8215 1.279 23.4171
SU-DHL-4 CTRP2; CTRP1 1.849 5.3135 1.4831 22.6463
KE-97 CTRP2; CTRP1 1.8944 5.6955 1.4127 22.7638
OCI-Ly3 CTRP2 1.9053 4.5128 1.7478 21.4548
P3HR-1 CTRP2; CTRP1 2.0757 5.2888 1.7376 21.0428
THP-1 CTRP2; CTRP1 2.0889 6.7684 1.2311 22.8582
DND-41 CTRP2 2.2402 5.7005 1.7828 20.3114
HEL 92.1.7 CTRP2 2.2861 7.338 1.2017 22.3363
NOMO-1 CTRP2; CTRP1 2.3033 5.472 1.9295 19.6627
KMS-20 CTRP2 2.3675 6.5461 1.6098 20.588
Hs 611.T CTRP2 2.3853 6.7309 1.5554 20.7421
Mono-Mac-6 CTRP2 2.3993 14.8034 -2.1833 31.9145
MC116 CTRP2; CTRP1 2.4241 6.0671 1.8566 19.5795
KMS-26 CTRP2 2.4507 6.3902 1.7591 19.7923
Ci-1 CTRP2 2.4728 5.2118 2.1905 18.1254
Kasumi-2 CTRP2 2.6081 6.2025 1.999 18.4428
MM1.S CTRP2 2.6199 8.3059 1.1224 21.7195
Pfeiffer CTRP2 2.6596 5.4241 2.3291 17.0605
Kasumi-1 CTRP2 2.7102 6.0126 2.1798 17.4706
TF-1 CTRP2 2.7284 6.5634 1.9855 18.1574
CA46 CTRP2 2.7923 6.3953 2.1203 17.4656
U266B1 CTRP2 2.8591 6.4961 2.1507 17.1646
K-562 CTRP2 2.9074 7.9706 1.5642 19.2969
EHEB CTRP2 2.9473 9.3264 0.977 21.402
KM-H2 CTRP2 3.0046 6.4853 2.3084 16.1583
RPMI-8226 CTRP2; CTRP1 3.0801 7.0751 2.1438 16.6738
PL21 CTRP2; CTRP1 3.2827 6.7908 2.476 14.8394
Karpas-422 CTRP2 3.3206 10.0257 1.0034 20.3746
KCL-22 CTRP2 3.3702 6.702 2.5989 14.0446
HEL CTRP2 3.4411 6.2031 2.8833 12.7436
A3/Kawakami CTRP2 3.4777 6.3606 2.8561 12.7508
KMS-27 CTRP2 3.52 7.4222 2.4297 14.3307
HDLM-2 CTRP2 3.606 9.0395 1.7502 16.8302
P31/FUJ CTRP2 3.6527 7.666 2.4484 13.9258
AMO1 CTRP2; CTRP1 3.7181 7.0772 2.7925 12.4621
HH [Human lymphoma] CTRP2 3.7205 14.4355 -0.7955 25.3222
SUP-B15 CTRP2 3.7805 7.6542 2.5793 13.0854
MHH-CALL-3 CTRP2 3.7841 9.3952 1.7464 16.4259
HL-60 CTRP2 3.9001 7.6979 2.675 12.4092
KO52 CTRP2 4.029 7.7698 2.7646 11.738
Raji CTRP2 4.072 7.4678 2.9505 10.8764
ME1 CTRP2 4.0801 8.4757 2.4712 12.8216
SR CTRP2 4.1842 7.6138 2.9875 10.4618
SU-DHL-1 CTRP2 4.2352 7.4637 3.1083 9.8468
DEL CTRP2 4.3308 8.454 2.7136 11.2612
AML-193 CTRP2 4.3682 9.4177 2.2715 12.9997
Mino CTRP2 4.3697 9.7112 2.1273 13.5845
Ki-JK CTRP2 4.3709 8.7058 2.626 11.5355
RL CTRP2 4.4195 8.458 2.7925 10.7402
SUP-HD1 CTRP2 4.5785 7.3704 3.4735 7.561
L-428 CTRP2 4.6287 8.7434 2.838 10.104
EJM CTRP2; CTRP1 4.6779 9.0006 2.7622 10.3975
SIG-M5 CTRP2 4.7519 6.2322 4.192 4.1903
NCI-H929 CTRP2 5.1631 8.5134 3.4078 6.653
HD-MY-Z CTRP2 5.2251 9.3006 3.065 7.9746
HuT 78 CTRP2 5.4022 7.5785 4.0618 3.489
OCI-Ly10 CTRP2; CTRP1 5.5296 10.0532 2.9423 8.0135
SU-DHL-8 CTRP2 5.9871 7.5646 4.4561 1.1396
HT CTRP2; CTRP1 6.0421 10.8256 2.9482 7.1287
Karpas-620 CTRP2 6.2455 12.1331 2.4444 8.7756
MOLP-2 CTRP2 6.5005 9.433 3.9121 2.5749
Toledo CTRP2 7.4195 19.5352 -0.3295 16.8602
KMM-1 CTRP2 7.9411 10.7629 4.0886 0.8529
⏷ Show the Full List of 135 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 5.8999 10.3885 3.0475 6.8743
EC-GI-10 CTRP2 1.8391 7.8907 0.5026 26.09
OE21 CTRP2 1.9049 6.3292 1.1979 23.4394
TE-11 CTRP2 2.2867 6.8653 1.3972 21.6101
KYSE-140 CTRP2; CTRP1 3.2628 7.2909 2.236 15.8345
KYSE-70 CTRP2 3.8484 7.8248 2.5646 12.9817
KYSE-520 CTRP2 3.9356 9.7371 1.7202 16.1807
TE-9 CTRP2 4.0104 7.7298 2.766 11.7762
KYSE-410 CTRP2; CTRP1 4.1049 7.833 2.8141 11.44
TE-5 CTRP2 4.6061 8.7902 2.7948 10.3314
KYSE-510 CTRP2 5.0227 5.9598 4.5685 2.0425
KYSE-180 CTRP2 5.0478 6.7305 4.2042 3.5249
OE33 CTRP2 5.096 8.0677 3.5756 6.0749
KYSE-450 CTRP2; CTRP1 5.1696 10.5333 2.4134 10.8648
TE-10 CTRP2 5.4043 7.0892 4.3042 2.4819
KYSE-30 CTRP2 5.4354 7.5722 4.0897 3.3184
KYSE-150 CTRP2 5.5421 6.9536 4.4659 1.6221
TE-1 CTRP2 5.5479 9.0453 3.4465 5.8045
OE19 CTRP2 5.6577 7.2222 4.4143 1.6721
TE-14 CTRP2 5.8299 8.3974 3.9688 3.211
COLO 680N CTRP2 6.0647 8.4289 4.1081 2.3472
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 34 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 5.298 8.6163 3.4651 6.1643
KP-4 CTRP2 2.2222 8.1967 0.766 24.091
DAN-G CTRP2 3.3803 9.4765 1.3246 19.0248
QGP-1 CTRP2; CTRP1 3.5391 9.6798 1.3855 18.4823
PSN1 CTRP2 4.2047 10.0353 1.8187 15.1869
L3.3 CTRP2 4.2504 7.0741 3.3104 8.981
Panc 08.13 CTRP2 4.7399 8.1369 3.2376 8.203
Panc 03.27 CTRP2; CTRP1 4.8658 8.9677 2.9414 9.2671
KP-3 CTRP2; CTRP1 4.9183 11.8229 1.5591 14.7875
PaTu 8902 CTRP2; CTRP1 5.0029 7.7646 3.6591 5.9869
PK-59 CTRP2 5.0374 9.0804 3.0205 8.517
Panc 04.03 CTRP2 5.1001 6.8084 4.2084 3.408
SW1990 CTRP2 5.1229 11.2398 2.0118 12.5143
SNU-213 CTRP2 5.1703 6.3787 4.4791 2.1441
BxPC-3 CTRP2 5.2311 7.848 3.7949 4.9025
Capan-2 CTRP2; CTRP1 5.2938 7.5398 4.0083 3.979
HuP-T4 CTRP2; CTRP1 5.3827 9.2889 3.2073 7.1707
MIA PaCa-2 CTRP2 5.4367 9.26 3.2539 6.8004
Panc 05.04 CTRP2 5.4743 7.2678 4.2675 2.5235
Panc 02.03 CTRP2 5.579 7.5101 4.2236 2.5445
PK-45H CTRP2 5.6071 8.447 3.7862 4.2965
HPAC CTRP2; CTRP1 5.6525 7.7945 4.1486 2.8183
YAPC CTRP2 5.7185 9.1108 3.542 5.1269
TCC-Pan2 CTRP2 5.7202 10.3825 2.9155 7.7171
Capan-1 CTRP2 5.7253 11.9141 2.1592 10.8042
KP-2 CTRP2 5.7968 8.6252 3.8357 3.7991
AsPC-1 CTRP2 5.9022 9.8724 3.3026 5.8207
HPAF-II CTRP2 6.0503 8.204 4.2034 1.9999
HuP-T3 CTRP2 6.1724 11.3997 2.7508 7.6518
Panc 10.05 CTRP2; CTRP1 6.2379 11.8412 2.5931 8.2615
PaTu 8988s CTRP2 6.3985 8.9784 4.0585 2.1458
Hs 766T CTRP2 6.472 8.5128 4.3057 1.2052
CFPAC-1 CTRP2; CTRP1 6.5851 9.2148 4.0728 1.9624
SUIT-2 CTRP2; CTRP1 6.8275 8.0784 4.6517 0.1659
⏷ Show the Full List of 34 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 47 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 2.4833 7.089 1.512 23.8003
WM266-4 CTRP2 4.4717 5.9098 4.0749 5.3346
A-375 CTRP2; CTRP1 4.5492 9.1538 2.5726 11.4531
LOX-IMVI CTRP2 4.5901 7.1737 3.5809 7.0885
CJM [Human melanoma] CTRP2 5.0019 9.4344 2.8139 9.4501
SK-MEL-5 CTRP2; CTRP1 5.1185 7.3916 3.9419 4.577
G-361 CTRP2; CTRP1 5.1192 10.1507 2.5631 10.3439
MDA-MB-435S CTRP2 5.2764 8.3359 3.5878 5.6893
Hs 852.T CTRP2; CTRP1 5.2851 9.9347 2.8068 9.0196
WM115 CTRP2 5.3186 8.6169 3.4812 6.0596
RVH-421 CTRP2 5.3307 7.558 4.0175 3.7945
UACC-62 CTRP2 5.3344 6.7493 4.4199 2.1155
MeWo CTRP2 5.3497 8.7388 3.4451 6.1555
SK-MEL-1 CTRP2; CTRP1 5.3781 10.9521 2.3739 10.6346
Mel Ho CTRP2 5.4702 7.2608 4.2679 2.528
WT2-iPS CTRP2 5.4955 6.7124 4.5497 1.3528
COLO 800 CTRP2 5.4999 8 3.9269 3.888
WM88 CTRP2 5.5453 9.5495 3.1944 6.859
WM983B CTRP2 5.5574 7.265 4.3271 2.1572
SK-MEL-3 CTRP2 5.5684 8.5574 3.7032 4.7031
Hs 934.T CTRP2 5.6805 7.7396 4.183 2.5615
Hs 294T CTRP2 5.7813 7.094 4.5491 1.0175
Mel JuSo CTRP2 5.7944 7.583 4.3324 1.8168
WM793 CTRP2 5.8032 8.4971 3.9022 3.5192
SK-MEL-2 CTRP2 5.8551 7.294 4.5018 1.1108
WM1799 CTRP2 5.8815 8.132 4.13 2.4961
IGR-39 CTRP2 5.9323 10.2471 3.1408 6.4383
UACC-257 CTRP2 5.9411 8.2591 4.1089 2.5009
IGR-37 CTRP2 5.9998 7.3141 4.5721 0.7347
SK-MEL-28 CTRP2; CTRP1 6.0266 6.8913 4.7696 0.2149
K029AX CTRP2 6.2045 10.1446 3.3844 5.0295
HT-144 CTRP2 6.2482 9.9316 3.5166 4.4357
Hs 936.T CTRP2; CTRP1 6.3542 8.7889 4.1308 1.9953
Hs 688(A).T CTRP2 6.3975 7.4828 4.6863 0.2061
SK-MEL-30 CTRP2 6.4074 7.7409 4.5924 0.4068
SK-MEL-24 CTRP2 6.4572 11.3443 2.98 6.2906
IPC-298 CTRP2 6.4788 11.066 3.1289 5.6624
IGR-1 CTRP2 6.7771 8.4734 4.4694 0.5182
SK-MEL-31 CTRP2 6.9254 8.8498 4.3876 0.6444
Hs 839.T CTRP2 7.0071 13.8024 2.1735 8.679
Hs 944.T CTRP1 7.1649 8.8414 4.5062 0.6687
COLO 741 CTRP2; CTRP1 7.1682 14.9412 1.7461 10.1474
RPMI-7951 CTRP2 7.3399 8.7566 4.5884 0.1204
Hs 940.T CTRP2 7.4399 9.0948 4.5068 0.2044
Malme-3M CTRP2 7.652 10.6109 4.0172 1.2088
Hs 895.T CTRP2 9.341 19.8164 0.8585 10.2758
COLO 829 CTRP2 10.0974 24.2825 -0.7596 14.3124
⏷ Show the Full List of 47 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 2.3555 8.8253 0.6207 24.2354
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MHH-NB-11 CTRP2 -2.4756 3.2519 -2.7517 50.0886
SiMa CTRP2 -1.7536 1.2086 -1.7709 45.3267
SK-N-DZ CTRP2 -1.4766 2.8612 -1.6167 43.7413
NH-6 CTRP2 -1.373 1.8457 -1.4092 42.8473
IMR-32 CTRP2 -0.8303 1.0024 -0.8318 39.1431
SK-N-FI CTRP2 -0.0541 4.0274 -0.2787 34.678
CHP-126 CTRP2 0.8787 8.0192 -0.5562 32.2994
NB1 CTRP2 2.2708 7.8432 0.9703 23.2246
CHP-212 CTRP2 2.351 6.8645 1.4654 21.1755
Kelly CTRP2 2.4842 7.0558 1.5268 20.5745
SK-N-BE(2) CTRP2 2.9566 14.3207 -1.431 28.8133
SK-N-AS CTRP2 3.5594 9.2415 1.6086 17.497
KP-N-SI9s CTRP2 4.7096 10.6646 1.9507 13.5847
KP-N-YN CTRP2 7.3571 9.352 4.3802 0.456
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 3.5831 7.7081 2.3601 14.4521
SNU-478 CTRP2 5.1336 6.4927 4.3931 2.5702
SNU-869 CTRP2 5.5214 7.7553 4.063 3.2908
SNU-308 CTRP2 5.5498 7.6335 4.1431 2.9173
HuH-28 CTRP2 5.6961 9.9797 3.0966 7.0083
SNU-1196 CTRP2 5.7166 7.8665 4.1467 2.6562
HuCC-T1 CTRP2 6.1088 8.7303 3.995 2.7297
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-673 CTRP2 -1.2851 0.7393 -1.287 42.174
SK-ES-1 CTRP2 0.4618 6.1527 -0.298 32.9405
MHH-ES-1 CTRP2 0.7018 3.4299 0.6289 29.1759
SK-N-MC CTRP2 1.4592 3.8583 1.3802 24.1529
TC71 CTRP2 1.8792 7.6325 0.6533 25.4561
HOS CTRP2 4.7175 7.7633 3.4037 7.5543
U2OS CTRP2; CTRP1 5.618 11.751 2.1665 11.04
CAL-78 CTRP2 5.7244 18.3213 -1.0362 21.8792
SW1353 CTRP2 5.8775 8.1155 4.1352 2.4809
SaOS-2 CTRP2 5.8963 9.5947 3.4342 5.2896
Hs 822.T CTRP2 6.2534 7.0873 4.7736 0.1024
G-292 clone A141B1 CTRP2 6.7208 12.4562 2.6255 7.3221
Hs 888.T CTRP2 7.0026 11.6354 3.2028 4.6722
MG-63 CTRP2 7.4618 15.0778 1.8713 9.1792
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 71 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 CTRP2 -1.0535 0.9169 -1.0555 40.6317
BT-474 CTRP2 0.3792 1.8975 -3.4252 0.08
HCC1806 CTRP2 1.4957 5.6554 0.989 25.4126
HCC1954 CTRP2 2.0285 6.1309 1.4034 22.3279
CAL-148 CTRP2 2.7325 5.4095 2.413 16.5357
MDA-MB-157 CTRP2 2.8382 6.8102 1.9996 17.8023
MDA-MB-468 CTRP2 2.9851 7.8457 1.6992 18.5746
HCC202 CTRP2 3.0068 8.4567 1.4416 19.5098
HCC1143 CTRP2 3.0176 7.5542 1.863 17.8543
CAL-51 CTRP2 3.1337 6.4101 2.4751 15.162
HCC2218 CTRP2 3.4048 7.2264 2.4027 14.7304
HCC1428 CTRP2 3.489 10.5866 0.89 20.3843
MCF-7 CTRP2; CTRP1 4.6763 11.9928 1.2681 16.4008
HMC-1-8 CTRP2 4.787 5.9983 4.339 3.5023
HCC1419 CTRP2 5.1551 6.7891 4.2625 3.0792
KPL-1 CTRP2 5.2155 7.151 4.1301 3.5253
ZR-75-1 CTRP2 5.2636 7.6725 3.9083 4.3689
MDA-MB-453 CTRP2 5.2649 7.3021 4.0937 3.5904
MDA-MB-231 CTRP2 5.2793 9.4577 3.0304 8.0189
JIMT-1 CTRP2 5.3908 6.6496 4.509 1.6633
HDQ-P1 CTRP2 5.4241 7.3478 4.1918 2.9143
HCC38 CTRP2 5.5324 9.1021 3.4065 5.9976
BT-20 CTRP2 5.5636 9.4691 3.2485 6.6024
HCC1395 CTRP2 5.5737 8.7482 3.613 5.0689
Hs 578T CTRP2 5.5922 16.1109 -0.0393 19.121
ZR-75-30 CTRP2 5.7548 9.6893 3.2841 6.1341
EFM-192A CTRP2 5.8219 12.7021 1.8426 11.8962
T-47D CTRP2 5.8317 9.5674 3.4008 5.5283
MDA-MB-361 CTRP2 5.8506 12.3981 2.0159 11.1583
BT-549 CTRP2 5.8681 10.5472 2.9457 7.3455
HCC1500 CTRP2 6.0607 21.5777 -2.3913 24.7196
HCC1937 CTRP2 6.1678 9.9747 3.441 4.8539
CAL-85-1 CTRP2 6.2128 9.627 3.6384 3.9982
SK-BR-3 CTRP2 6.2376 8.7808 4.0521 2.3524
CAL-120 CTRP2 6.7021 7.9997 4.6175 0.2306
Hs 578Bst CTRP2 6.7392 8.0011 4.6315 0.195
AU565 CTRP2 7.9208 10.1762 4.3022 0.4029
CAMA-1 CTRP2 8.6404 27.6496 -3.4193 22.8616
BT 145 CTRP2 0.9542 5.2221 0.5308 28.6898
BT 239 CTRP2 1.1941 5.7776 0.6216 27.6226
BT 286 CTRP2 2.3107 7.9504 0.9647 23.1345
BT164 CTRP2 2.3819 7.1643 1.3746 21.4285
BT 112 CTRP2 2.9495 7.647 1.7522 18.4622
BT 271 CTRP2 4.0279 10.5718 1.3937 17.2467
BT 231 CTRP2 4.7046 11.1719 1.6931 14.623
BT 131 CTRP2 4.8996 10.2206 2.3346 11.6379
BT 428 CTRP2 4.9067 9.5887 2.6565 10.2929
BT 504 CTRP2 5.5774 11.6781 2.1606 11.0629
BT 172 CTRP2 5.6071 12.3515 1.8486 12.258
BT 422 CTRP2 5.7161 9.4644 3.3662 5.8577
BT 248 CTRP2 5.7571 8.482 3.8773 3.6891
BT 444 CTRP2 5.7682 7.6645 4.2773 2.0659
BT 139 CTRP2 5.7689 12.0793 2.1109 10.9213
BT 330 CTRP2 5.8493 12.6137 1.9079 11.5898
BT 440 CTRP2 5.8844 8.4873 3.9627 3.158
BT 216 CTRP2 5.8886 10.7449 2.8634 7.6501
BT 416 CTRP2 5.9627 9.067 3.7374 3.9536
BT 245 CTRP2 5.985 11.6089 2.5092 8.9392
BT 232 CTRP2 6.0659 9.865 3.4232 5.0763
BT147 CTRP2 6.0999 14.0073 1.4093 13.0853
BT 320 CTRP2 6.3467 7.462 4.6734 0.2504
BT 328 CTRP2 6.4297 9.3137 3.924 2.6118
BT 228 CTRP2 6.5117 7.8896 4.5802 0.3843
BT 359 CTRP2 6.6186 13.4588 2.0661 9.6876
BT 482 CTRP2 6.6263 11.7495 2.901 6.3623
BT 340 CTRP2 6.7131 11.0741 3.281 4.7395
BT 333 CTRP2 6.9165 13.2128 2.3955 7.9449
BT 224 CTRP2 7.1016 12.3243 2.9429 5.5503
BT 159 CTRP2 7.1401 11.1637 3.5046 3.3711
BT 187 CTRP2 7.2673 13.1005 2.6841 6.3347
BT 179 CTRP2 7.3464 16.4361 1.1343 12.0722
⏷ Show the Full List of 71 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 5.341 6.489 4.5519 1.5631
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-172 CTRP2 2.0456 4.9546 1.7958 20.8487
D283 Med CTRP2 3.0381 5.9967 2.537 15.1891
Daoy CTRP2 3.4202 8.4605 1.8472 16.8972
GB-1 CTRP2 4.6935 6.5432 3.9857 5.1771
T98G CTRP2 5.0352 6.27 4.4239 2.626
Becker CTRP2 5.1013 12.1053 1.5612 14.3442
SNU-738 CTRP2 5.1926 6.4419 4.465 2.1642
SNU-626 CTRP2 5.2358 6.5242 4.4573 2.1221
SNU-466 CTRP2 5.3314 6.7292 4.4276 2.0885
SF295 CTRP2; CTRP1 5.3336 9.1915 3.2168 7.2197
42-MG-BA CTRP2 5.4351 7.3122 4.2173 2.7911
ONS-76 CTRP2 5.5177 9.2829 3.3055 6.4436
SF539 CTRP2 5.5362 8.6205 3.6478 4.9865
SF268 CTRP2 5.5477 7.9629 3.9804 3.5895
DK-MG CTRP2 5.5638 11.1022 2.4368 9.9632
Hs 683 CTRP2 5.6208 9.7813 3.1375 6.9664
SF126 CTRP2 5.8017 8.2649 4.0132 3.0725
U-251MG CTRP2 5.8277 9.3884 3.4856 5.1858
LN-18 CTRP2 5.9652 7.1104 4.6404 0.5479
SNU-201 CTRP2 5.9989 8.9058 3.8395 3.4915
SNB-75 CTRP2 6.0423 8.8306 3.9044 3.1733
U-87MG ATCC CTRP2 6.0694 9.9016 3.4079 5.1332
SW1088 CTRP2 6.1224 10.1934 3.3036 5.4779
YKG-1 CTRP2 6.2399 8.8587 4.0176 2.4808
GaMG CTRP2; CTRP1 6.2762 8.2046 4.3472 1.3028
SW1783 CTRP2 6.3217 12.8176 2.1641 9.7739
DBTRG-05MG CTRP2 6.3315 9.1318 3.9478 2.6372
SNU-489 CTRP2 6.7114 7.7938 4.6946 0.1095
U-118MG CTRP2 6.7631 13.8588 1.9745 9.8197
LN-229 CTRP2; CTRP1 6.8282 10.3404 3.7064 3.0385
SNU-1105 CTRP2 6.8565 8.0932 4.6431 0.147
NMC-G1 CTRP2 6.8639 8.1043 4.642 0.1469
KNS-42 CTRP2 6.9822 11.7017 3.1588 4.8677
KG-1-C CTRP2 7.0577 8.2541 4.6602 0.0889
CCF-STTG1 CTRP2 7.1703 12.1608 3.0634 4.9986
CAS-1 CTRP2 7.2146 8.7531 4.5434 0.2057
KALS-1 CTRP2 7.9428 18.1565 0.7185 12.6419
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-2 CTRP2; CTRP1 -0.9382 3.8106 -1.1923 40.5664
JHUEM-7 CTRP2 -0.9007 4.1846 -1.2307 40.4418
ESS-1 CTRP2 0.0832 2.9913 0.0223 33.2528
HEC-108 CTRP2; CTRP1 0.5235 4.8084 0.1754 31.3363
HEC-50B CTRP2 2.8141 10.2246 0.4222 23.7075
HEC-6 CTRP2; CTRP1 3.155 8.634 1.5128 18.935
HEC-265 CTRP2; CTRP1 3.2472 6.046 2.7458 13.8897
HEC-151 CTRP2; CTRP1 3.4271 6.1722 2.8863 12.8536
AN3-CA CTRP2 3.5793 9.0488 1.7203 17.0115
HEC-251 CTRP2; CTRP1 4.0146 9.0845 2.121 14.4744
JHUEM-1 CTRP2 4.3109 8.8002 2.5249 12.084
HEC-1-A CTRP2 4.5185 9.7302 2.25 12.7666
JHUEM-3 CTRP2 4.7422 14.4137 0.1056 20.3303
HEC-59 CTRP2; CTRP1 4.8018 8.693 3.0234 9.054
MFE-319 CTRP2; CTRP1 4.9838 7.9996 3.5255 6.5853
RL95-2 CTRP2 5.0537 6.489 4.3298 2.9858
EFE-184 CTRP2 5.3359 7.4874 4.0565 3.6226
HEC-1-B CTRP2 5.338 10.4214 2.5964 9.7162
MFE-296 CTRP2 6.051 11.3117 2.7049 8.0334
KLE CTRP2; CTRP1 6.4519 11.765 2.7839 7.1605
EN CTRP2 7.0382 15.4914 1.3749 11.6687
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 5.1205 6.4541 4.4119 2.6002
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
786-O CTRP2 4.3257 8.0766 2.8943 10.5249
A-498 CTRP2 4.7193 5.7675 4.3858 3.4672
769-P CTRP2 4.867 8.5901 3.1216 8.4294
UO-31 CTRP2 5.2781 8.0894 3.7121 5.1651
RCC10RGB CTRP2; CTRP1 5.6015 8.3554 3.8381 4.1705
OS-RC-2 CTRP2 5.747 9.0993 3.5685 4.972
CAL-54 CTRP2 5.8041 12.1697 2.0934 10.9298
ACHN CTRP2 5.8423 8.0062 4.164 2.414
TUHR4TKB CTRP2 5.8479 7.3841 4.457 1.2821
KMRC-20 CTRP2 6.0375 8.0271 4.2769 1.7382
VMRC-RCW CTRP2; CTRP1 6.1789 10.7644 3.0771 6.3889
TUHR10TKB CTRP2 6.4076 13.5554 1.8647 10.8127
VMRC-RCZ CTRP2 6.4659 12.0419 2.6479 7.6123
KMRC-1 CTRP2 6.6139 10.2196 3.6185 3.5547
Caki-1 CTRP2 6.6187 9.4159 3.9894 2.162
KMRC-2 CTRP2 6.8348 12.4985 2.6832 6.9294
SNU-1272 CTRP2 6.9249 13.0797 2.4654 7.6585
BFTC-909 CTRP2 7.0184 8.3808 4.6019 0.1677
KMRC-3 CTRP2 7.3257 13.7563 2.4115 7.3078
Caki-2 CTRP2 7.9429 53.6815 -16.9029 37.8826
TUHR14TKB CTRP2 8.2382 10.4813 4.3147 0.2915
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 52 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HCT 116 CTRP2; CTRP1 -1.9629 -0.1468 -1.9632 46.7357
SNU-175 CTRP2; CTRP1 -0.5359 3.6519 -0.7283 37.804
SW48 CTRP2; CTRP1 -0.4083 3.558 -0.575 36.8955
LS180 CTRP2; CTRP1 -0.0999 2.7638 -0.1487 34.4947
HT115 CTRP2; CTRP1 0.4714 4.1898 0.2601 31.2346
GP2d CTRP2; CTRP1 0.5531 5.2327 0.093 31.5019
SW948 CTRP2; CTRP1 0.7441 3.7531 0.6315 29.0969
SK-CO-1 CTRP2; CTRP1 1.1732 5.4459 0.7067 27.4654
HCC-56 CTRP2 1.6039 4.0362 1.5091 23.2436
SNU-C2A CTRP2; CTRP1 1.7572 7.1921 0.7111 25.6783
CL-11 CTRP2 1.7739 9.3622 -0.2094 28.5749
T84 CTRP2 1.7964 6.6921 0.9448 24.6691
SW620 CTRP2; CTRP1 1.8162 7.3311 0.7171 25.4851
SNU-81 CTRP1 1.9112 12.587 -1.568 48.2626
LS513 CTRP2; CTRP1 2.2867 5.555 1.8849 19.8754
CCK-81 CTRP2 2.8392 6.7975 2.0059 17.7754
SNU-407 CTRP2 2.9854 6.1787 2.4107 15.8186
SW480 CTRP1 3.8944 7.8397 2.6093 26.4477
COLO201 CTRP2 4.0167 7.9912 2.6463 12.251
SNU-C5 CTRP2; CTRP1 4.0615 10.5066 1.4649 16.9692
RKO CTRP2; CTRP1 4.5543 7.0943 3.5952 7.1941
SNU-C4 CTRP2; CTRP1 4.605 7.2887 3.5463 7.2848
HCT 15 CTRP2 4.7182 8.2067 3.1838 8.4732
COLO205 CTRP2; CTRP1 4.7661 7.0725 3.7988 5.8845
KM12 CTRP2; CTRP1 4.8163 8.8516 2.9568 9.3027
NCI-H747 CTRP2 4.9213 7.8777 3.5239 6.6328
LoVo CTRP2; CTRP1 4.9949 9.1674 2.9511 8.9707
LS411N CTRP2; CTRP1 5.1363 7.243 4.0306 4.1711
SW1417 CTRP2 5.1485 8.1698 3.5676 6.0094
SNU-C1 CTRP2 5.1941 6.4978 4.4384 2.2727
CL-40 CTRP1 5.2136 9.0509 3.1903 15.8012
DLD-1 CTRP2; CTRP1 5.2581 7.6559 3.9225 4.4016
NCI-H508 CTRP2; CTRP1 5.3297 6.6448 4.4788 1.9609
CW-2 CTRP2; CTRP1 5.3451 11.8452 1.9012 12.6076
LS1034 CTRP2 5.3546 11.0529 2.2946 10.9264
SNU-1040 CTRP1 5.4388 9.7472 3.0233 16.1918
COLO 678 CTRP2; CTRP1 5.5008 8.7477 3.5686 5.4558
OUMS-23 CTRP2 5.5133 7.7368 4.0662 3.2904
RCM-1 [Human ESC] CTRP2; CTRP1 5.5147 6.8384 4.5143 1.5429
SNU-1033 CTRP2 5.5165 10.1265 2.8852 8.1959
HCT 8 CTRP2; CTRP1 5.636 7.5363 4.2619 2.3841
COLO 320 CTRP2; CTRP1 5.6367 11.0713 2.5092 9.5367
CL-34 CTRP1 5.6446 11.7775 2.1744 21.1244
HT-55 CTRP2; CTRP1 5.7158 9.6625 3.279 6.2972
MDST8 CTRP2; CTRP1 5.7596 8.0645 4.0924 2.8898
SNU-61 CTRP2; CTRP1 5.9067 10.0649 3.2225 6.2197
SW403 CTRP1 6.1339 10.5787 3.1355 12.8312
NCI-H716 CTRP2 6.6876 10.7523 3.4161 4.2451
C2BBe1 CTRP2; CTRP1 6.9215 17.9999 0.0675 16.4734
LS123 CTRP2; CTRP1 7.0564 11.9129 3.1192 4.9962
HT-29 CTRP2; CTRP1 7.0645 8.0512 4.745 0.0342
SNU-503 CTRP2 7.1014 15.3212 1.503 11.0947
⏷ Show the Full List of 52 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHH-5 CTRP2 2.8203 6.134 2.2519 16.8857
PLC/PRF/5 CTRP2 4.257 6.3367 3.6643 7.5242
JHH-2 CTRP2 4.8049 7.4731 3.6251 6.4445
SNU-878 CTRP2 4.9964 7.1995 3.9266 4.7917
SNU-398 CTRP2; CTRP1 5.0904 11.7179 1.7556 13.6749
Li-7 CTRP2 5.2858 7.061 4.2295 2.9869
JHH-4 CTRP2 5.3067 7.9054 3.8262 4.6363
SNU-182 CTRP2 5.3948 9.4456 3.1285 7.3988
SNU-423 CTRP2 5.4081 10.6016 2.5628 9.7267
Hep 3B2.1-7 CTRP2 5.4908 9.333 3.2598 6.6813
SNU-475 CTRP2 5.6677 7.9078 4.093 2.9443
JHH-1 CTRP2 5.7113 7.8826 4.1353 2.7098
Hep-G2 CTRP2; CTRP1 5.7375 7.2305 4.473 1.4183
SNU-449 CTRP2; CTRP1 5.9362 9.2984 3.6183 4.5524
SK-HEP-1 CTRP2 6.0887 10.8433 2.9625 6.9209
HuH-6 CTRP2 6.1059 10.1188 3.3282 5.4026
JHH-6 CTRP2; CTRP1 6.2714 7.0982 4.7906 0.0979
HLF CTRP2 6.4733 10.2116 3.5325 4.0675
SNU-387 CTRP2 7.7867 16.7329 1.2975 10.8326
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 153 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H82 CTRP1 -0.4757 1.9474 -0.4902 75.465
NCI-H1930 CTRP1 -0.1098 42.9389 -18.344 52.122
LCLC-97TM1 CTRP2; CTRP1 0.0915 4.5091 -0.2225 34.0574
NCI-H1876 CTRP1 0.2087 25.6032 -9.4906 52.8954
SCLC-21H CTRP1 0.2242 7.3687 -0.9888 59.2751
NCI-H1155 CTRP2 0.2496 4.8353 -0.1327 33.1715
NCI-H810 CTRP2; CTRP1 0.3668 4.5906 0.0581 32.2386
NCI-H1341 CTRP2 0.4055 4.6353 0.0874 31.95
NCI-H211 CTRP2 0.4425 4.1186 0.2413 31.3266
NCI-H1836 CTRP1 0.63 18.3658 -5.5691 52.8297
LK2 CTRP2 0.8877 1.4528 0.8877 27.6922
EBC-1 CTRP2; CTRP1 1.0168 11.4117 -1.8963 35.1192
SHP-77 CTRP2; CTRP1 1.1194 6.2035 0.4004 28.6704
NCI-H1373 CTRP2; CTRP1 1.3846 6.0366 0.745 26.6775
DV-90 CTRP2; CTRP1 1.4634 8.3592 -0.0816 29.1584
NCI-H2081 CTRP2; CTRP1 1.4743 7.695 0.2083 28.2097
NCI-H1963 CTRP1 1.6743 9.8113 -0.5063 49.2743
NCI-H69 CTRP2 1.7161 10.3936 -0.737 30.262
Lu-99 CTRP2; CTRP1 2.0528 5.2391 1.7273 21.1494
COR-L51 CTRP1 2.053 9.0194 0.2337 46.4623
NCI-H1694 CTRP2; CTRP1 2.1147 11.7602 -0.9778 29.8559
EPLC-272H CTRP2; CTRP1 2.2081 6.5201 1.4549 21.6931
HCC4006 CTRP2; CTRP1 2.3637 11.9571 -0.8314 28.7984
NCI-H526 CTRP2 2.5116 6.7852 1.6669 19.9696
NCI-H1184 CTRP2 2.8199 6.7468 2.0068 17.8247
NCI-H596 CTRP1 2.8449 8.3776 1.323 39.1068
LXF 289 CTRP2; CTRP1 2.9623 8.3838 1.4376 19.7129
DMS 273 CTRP2; CTRP1 3.1371 8.3315 1.6357 18.5059
DMS 454 CTRP2 3.2361 13.7121 -0.8754 26.6758
NCI-H2110 CTRP2; CTRP1 3.2792 10.1398 0.9167 20.8636
NCI-H2009 CTRP2; CTRP1 3.3394 10.3873 0.8542 20.9434
NCI-H2286 CTRP2; CTRP1 3.5754 10.4825 1.0295 19.7366
HCC78 CTRP2; CTRP1 3.7595 9.4823 1.6889 16.785
NCI-H1339 CTRP2 3.7624 8.4478 2.184 14.7272
SW1573 CTRP2 3.7772 9.8498 1.5183 17.3364
DMS 79 CTRP2 3.8579 10.2491 1.3973 17.6184
LC-1/sq-SF CTRP2; CTRP1 3.8932 9.9722 1.574 16.9259
COR-L279 CTRP1 3.9666 8.3629 2.4271 27.2099
DMS 114 CTRP2 3.9957 8.2258 2.5131 12.8444
NCI-H841 CTRP2; CTRP1 4.065 9.5194 1.9544 15.0308
NCI-H1703 CTRP2 4.0906 8.0791 2.6738 11.967
HCC44 CTRP2; CTRP1 4.1163 6.9369 3.2526 9.6223
NCI-H2106 CTRP2 4.1331 9.9441 1.7991 15.4234
Calu-6 CTRP2; CTRP1 4.1951 8.1554 2.7426 11.5266
NCI-H1623 CTRP2 4.2754 10.1353 1.8328 14.9761
NCI-H1693 CTRP2 4.2817 9.4477 2.1788 13.5665
NCI-H1048 CTRP1 4.2897 9.9811 1.9307 28.3517
RERF-LC-KJ CTRP1 4.3312 13.7954 0.0703 35.1732
COR-L23 CTRP1 4.379 8.5579 2.7148 23.1588
NCI-H1581 CTRP2 4.38 7.3757 3.2874 8.7762
NCI-H2141 CTRP1 4.3884 7.4528 3.2657 18.9575
HCC33 CTRP1 4.4035 10.7885 1.6312 29.286
HCC1588 CTRP2 4.4277 7.4686 3.2866 8.6716
RERF-LC-MS CTRP2 4.4721 7.3996 3.3614 8.2618
NCI-H2171 CTRP2 4.4794 8.3445 2.9027 10.1526
NCI-H1734 CTRP2 4.5685 9.149 2.5832 11.2892
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 4.5762 9.3872 2.4803 11.7773
NCI-H520 CTRP2 4.5798 7.9716 3.1776 8.7914
VMRC-LCD CTRP2; CTRP1 4.6051 12.5366 0.9355 17.7901
HCC827 CTRP2; CTRP1 4.7577 8.7006 2.9814 9.3195
NCI-H522 CTRP2; CTRP1 4.763 10.0783 2.2985 12.1384
NCI-H292 CTRP2 4.7836 8.7727 2.9587 9.2803
SBC-5 CTRP2 4.7934 5.2672 4.6888 2.0623
SK-MES-1 CTRP2 4.8811 10.5673 2.1457 12.4475
NCI-H2087 CTRP2 4.8889 8.4028 3.2339 7.9149
NCI-H650 CTRP2; CTRP1 4.9062 7.4233 3.7471 5.8103
NCI-H889 CTRP2 4.9161 12.4801 1.2191 16.0265
NCI-H838 CTRP2 4.9474 7.157 3.9062 4.9749
Lu-65 CTRP2; CTRP1 4.9572 6.5086 4.2476 3.6082
HCC95 CTRP2 4.9634 8.5175 3.2398 7.7419
NCI-H1355 CTRP2; CTRP1 5.0051 10.2376 2.4245 11.1371
NCI-H1092 CTRP2 5.0233 10.6387 2.2297 11.8237
NCI-H1975 CTRP1 5.0309 7.4423 3.8437 11.0409
HCC2108 CTRP2; CTRP1 5.0416 8.0671 3.5404 6.4099
NCI-H647 CTRP2 5.0467 8.081 3.5281 6.369
NCI-H727 CTRP2; CTRP1 5.0784 10.0819 2.5636 10.4203
HCC366 CTRP2 5.1008 8.9493 3.1387 7.8999
NCI-H358 CTRP2; CTRP1 5.1406 7.9758 3.6679 5.6854
COR-L105 CTRP2 5.1541 10.4785 2.4182 10.7972
NCI-H2170 CTRP2 5.1664 7.2142 4.0594 3.9105
NCI-H1666 CTRP2; CTRP1 5.1733 12.6674 1.3496 15.0908
MOR/CPR CTRP2 5.1837 6.1006 4.6274 1.5016
Calu-3 CTRP2; CTRP1 5.2277 8.6692 3.3924 6.6787
NCI-H1755 CTRP2; CTRP1 5.2635 8.0525 3.729 5.2024
NCI-H1915 CTRP2; CTRP1 5.2677 9.8076 2.8562 8.8461
NCI-H23 CTRP2; CTRP1 5.2785 7.9783 3.7779 4.9703
NCI-H1105 CTRP2; CTRP1 5.3143 9.2319 3.1812 7.404
EKVX CTRP2 5.3148 8.1218 3.7249 5.046
NCI-H1437 CTRP1 5.3191 10.0708 2.7664 18.5523
NCI-H2342 CTRP2; CTRP1 5.3427 8.8422 3.3983 6.4443
NCI-H1568 CTRP2; CTRP1 5.3524 7.1547 4.2444 2.8944
HCC1438 CTRP2 5.3995 6.7909 4.4465 1.9051
NCI-H661 CTRP2; CTRP1 5.4151 8.2266 3.7612 4.7998
NCI-H1299 CTRP2; CTRP1 5.4349 8.0605 3.8588 4.3596
LCLC-103H CTRP2; CTRP1 5.4413 7.2363 4.2701 2.6439
NCI-H1944 CTRP2; CTRP1 5.443 7.5387 4.1228 3.2495
NCI-H1838 CTRP2 5.4502 8.2389 3.7715 4.6164
NCI-H2029 CTRP2; CTRP1 5.4649 7.8191 4.0008 3.7189
HOP-92 CTRP2 5.4676 9.13 3.3427 6.3754
NCI-H1573 CTRP2; CTRP1 5.4758 11.2827 2.2873 10.8084
NCI-H1793 CTRP2; CTRP1 5.4872 7.5925 4.1289 3.1528
NCI-H2122 CTRP2; CTRP1 5.5071 7.4981 4.1896 2.8715
NCI-H460 CTRP2; CTRP1 5.5142 6.565 4.643 1.0391
NCI-H3255 CTRP1 5.5185 7.1505 4.3669 4.5713
COLO 699 CTRP2; CTRP1 5.5333 6.8847 4.5046 1.5559
RERF-LC-Ad2 CTRP2 5.5379 10.7288 2.6023 9.3292
COR-L95 CTRP2 5.582 10.1827 2.9084 7.9847
NCI-H322 CTRP2 5.6009 7.3444 4.3186 2.1291
NCI-H2405 CTRP2; CTRP1 5.6049 7.8929 4.0671 3.2225
NCI-H2073 CTRP1 5.605 10.3875 2.8349 16.9404
KNS-62 CTRP2; CTRP1 5.6391 8.528 3.7809 4.3459
RERF-LC-A1 CTRP2 5.6599 9.111 3.4985 5.4018
DMS 53 CTRP2 5.6622 8.4798 3.8104 4.1092
HCC1195 CTRP1 5.7382 7.7169 4.2445 4.9566
NCI-H1651 CTRP2 5.748 7.6356 4.2778 2.0905
NCI-H2291 CTRP2 5.7522 11.5905 2.3409 10.0211
NCI-H1395 CTRP2 5.7618 9.2058 3.5271 5.1191
NCI-H1385 CTRP2 5.7618 17.5343 -0.6133 20.5852
Calu-1 CTRP2 5.7825 8.0515 4.1026 2.7401
NCI-H1792 CTRP2; CTRP1 5.7898 7.9397 4.1727 2.5256
BEN CTRP2; CTRP1 5.814 7.4659 4.4114 1.5616
HOP-62 CTRP2 5.8167 8.699 3.8138 3.8584
A-549 CTRP2; CTRP1 5.8339 9.0062 3.6879 4.4234
NCI-H2030 CTRP2; CTRP1 5.8368 8.1656 4.0962 2.7655
NCI-H441 CTRP2; CTRP1 5.8512 10.179 3.1254 6.7091
NCI-H2196 CTRP2 5.8767 12.0698 2.199 10.3793
HCC1833 CTRP2; CTRP1 5.9136 12.5616 1.9938 11.2089
LUDLU-1 CTRP2 5.9171 10.0486 3.2271 6.1074
COLO 668 CTRP2; CTRP1 5.9272 10.6948 2.9278 7.3981
Sq-1 CTRP2; CTRP1 6.0258 8.6368 3.9973 2.9017
NCI-H196 CTRP2 6.0424 7.8386 4.3653 1.4079
ChaGo-K-1 CTRP2; CTRP1 6.0697 10.6128 3.0727 6.5761
NCI-H1869 CTRP2 6.0869 16.3158 0.2522 17.2481
HCC1171 CTRP2 6.1219 9.7831 3.5018 4.6752
HCC2935 CTRP2; CTRP1 6.1252 12.3564 2.2562 9.8017
LOU-NH91 CTRP2 6.1452 9.2523 3.772 3.5594
HCC15 CTRP2; CTRP1 6.1457 11.4011 2.7416 7.8062
RERF-LC-Ad1 CTRP2 6.1472 7.0055 4.7622 0.1502
NCI-H2085 CTRP2 6.1594 12.0389 2.4273 8.9839
CAL-12T CTRP2; CTRP1 6.1832 8.2357 4.2808 1.6316
NCI-H1563 CTRP2 6.2214 7.8447 4.4608 0.9108
NCI-H1781 CTRP1 6.2221 15.6359 0.7057 26.1896
NCI-H2023 CTRP2; CTRP1 6.369 12.0625 2.5798 8.1084
SK-LU-1 CTRP2; CTRP1 6.3976 11.3793 2.9329 6.6419
IA-LM CTRP2 6.4233 11.4617 2.8996 6.6642
HCC1359 CTRP1 6.5439 7.5933 4.7173 0.2979
NCI-H2126 CTRP2; CTRP1 6.5515 9.9927 3.6972 3.399
HCC2279 CTRP2 6.6907 10.7483 3.4199 4.2261
NCI-H2172 CTRP2; CTRP1 6.9713 12.6889 2.6959 6.7588
T3M-10 CTRP2; CTRP1 7.2078 13.9096 2.271 8.0818
COR-L88 CTRP1 7.4047 9.0037 4.5401 0.4058
NCI-H1435 CTRP2; CTRP1 8.5989 28.627 -3.9208 23.9683
Hs 888.Lu CTRP2 5.5842 12.1252 1.9432 11.9237
⏷ Show the Full List of 153 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 0.9484 3.8476 0.835 27.6717
SYO-1 CTRP2 2.6587 7.2508 1.6265 19.7194
P-STS CTRP2 4.5845 10.393 1.9778 13.7344
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Aska-SS CTRP2 3.9284 8.9308 2.1075 14.6483
Yamato-SS CTRP2 4.3221 13.0381 0.4307 20.1226
KYM-1 CTRP2 -0.4929 1.9141 -0.5068 36.9355
G-402 CTRP2 0.4781 5.4734 -0.0624 32.1759
G-401 CTRP2; CTRP1 1.6585 7.0732 0.654 26.1672
TTC-709 CTRP2 1.8957 6.5504 1.105 23.803
A-204 CTRP2 4.0762 9.8854 1.7762 15.6412
SK-UT-1 CTRP2 4.1093 7.8415 2.8065 11.3793
TE 617.T CTRP2 4.5512 8.6427 2.8193 10.3453
RD CTRP2 4.7005 10.9448 1.8029 14.1955
TE 441.T CTRP2 4.9359 10.4439 2.2537 11.8978
Rh41 CTRP2 5.0959 8.2807 3.469 6.523
GCT CTRP2 5.1094 6.9658 4.1373 3.6891
HT-1080 CTRP2; CTRP1 5.2065 7.674 3.8722 4.7059
RKN CTRP2; CTRP1 5.4741 8.6206 3.6111 5.3242
BT-12 CTRP2 5.6692 7.5591 4.2619 2.2606
SK-LMS-1 CTRP2 5.7033 10.4927 2.848 8.0252
BT-16 CTRP2 6.224 7.8358 4.4659 0.8922
MES-SA CTRP2 6.3851 7.8851 4.5249 0.5972
Tm87-16 CTRP2 6.388 12.4947 2.371 8.8429
SW982 CTRP2 6.6477 8.3383 4.4646 0.6014
Hs 729.T CTRP2 7.237 14.7806 1.8603 9.5454
Rh18 CTRP2 7.2786 8.5629 4.6329 0.0843
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 4.184 9.2258 2.1995 13.6976
OVKATE CTRP1 -5.7544 3.9159 -6.4507 83.1028
OVCAR-4 CTRP1 0.2018 14.5143 -4.1445 55.0697
A2780 CTRP2; CTRP1 0.2834 3.7634 0.1352 32.2727
IGROV-1 CTRP2; CTRP1 1.2818 9.51 -0.7696 31.6824
OVK18 CTRP2; CTRP1 1.8197 7.0791 0.8225 25.1055
SNU-119 CTRP2 2.7894 8.3095 1.2917 20.6407
Caov-3 CTRP2; CTRP1 3.7052 10.5884 1.0984 19.1761
TOV-21G CTRP2 4.5868 11.2725 1.5413 15.4634
OVCAR-8 CTRP2; CTRP1 4.6155 8.1745 3.1177 9.0474
TYK-nu CTRP2; CTRP1 4.7 7.9568 3.3009 8.1041
OV-90 CTRP2; CTRP1 4.9047 7.1469 3.8837 5.2403
JHOM-1 CTRP2; CTRP1 4.9321 7.9069 3.5279 6.6777
MCAS CTRP2 5.1785 9.6228 2.866 8.8935
OC 314 CTRP2 5.1899 6.8645 4.2526 3.0576
COV434 CTRP2; CTRP1 5.24 9.0123 3.231 7.3322
SNU-8 CTRP2 5.2712 8.5349 3.4844 6.1322
ONCO-DG-1 CTRP2 5.3275 7.4898 4.0489 3.6689
HEY A8 CTRP2; CTRP1 5.3936 8.4007 3.6581 5.2677
DOV13 CTRP2 5.4281 9.6391 3.0585 7.6316
OVISE CTRP2 5.4349 7.9852 3.8854 4.1681
OVSAHO CTRP2 5.4366 6.5202 4.6021 1.2243
ES2 CTRP2 5.501 7.2196 4.3098 2.3099
OV56 CTRP2 5.509 7.3026 4.2752 2.4392
RMUG-S CTRP1 5.5453 12.1714 1.8995 23.0703
JHOC-5 CTRP2; CTRP1 5.5781 8.2882 3.8539 4.1429
EFO-27 CTRP2; CTRP1 5.6012 9.7797 3.1338 7.0931
SNU-840 CTRP2; CTRP1 5.6145 7.4236 4.3014 2.2559
EFO-21 CTRP2; CTRP1 5.7074 8.0485 4.064 3.0808
RMG-I CTRP2; CTRP1 5.7324 9.8219 3.2127 6.5444
Kuramochi CTRP2 5.8118 7.743 4.2685 2.0438
OAW42 CTRP2; CTRP1 6.0228 7.1051 4.6838 0.4332
OVTOKO CTRP2 6.0595 8.749 3.9544 2.9528
OVCAR-5 CTRP2 6.07 10.5474 3.0937 6.414
JHOS-2 CTRP2 6.1069 10.9456 2.9256 7.0431
JHOS-4 CTRP1 6.1303 9.9433 3.4417 10.4575
OAW28 CTRP2 6.1534 10.0421 3.3986 5.0465
OV7 CTRP2; CTRP1 6.1732 9.2651 3.7962 3.4991
COV318 CTRP1 6.2115 7.4607 4.6286 1.0047
COV644 CTRP2; CTRP1 6.4189 13.7559 1.7852 11.1732
SK-OV-3 CTRP2; CTRP1 6.5541 12.0386 2.7229 7.2518
FU-OV-1 CTRP2 6.5717 13.8111 1.8596 10.567
OVMANA CTRP1 7.2065 8.3803 4.6838 0.1358
COV362 CTRP2; CTRP1 7.6305 15.0289 2.0198 8.4518
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 5.264 8.3483 3.5717 5.7792
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2; CTRP1 1.0281 6.2827 0.274 29.3748
NCI-H28 CTRP2; CTRP1 5.4041 9.4253 3.1562 7.3457
ACC-MESO-1 CTRP2 5.671 8.7681 3.6755 4.6516
MPP 89 CTRP2 5.7692 9.8388 3.2212 6.3708
NCI-H2052 CTRP2; CTRP1 6.1218 9.3818 3.7062 3.9278
JL-1 CTRP2 6.1947 10.0357 3.4301 4.8592
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LNCaP clone FGC CTRP2 4.7265 8.0926 3.2479 8.1873
DU145 CTRP2 5.1362 10.0666 2.6093 10.0418
22Rv1 CTRP2 5.7489 10.2191 3.0182 7.2441
VCaP CTRP2 5.9382 9.03 3.7383 3.9858
PaCa-3 CTRP2; CTRP1 5.9878 10.2339 3.1988 6.1885
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 3.7725 7.105 2.8275 12.1027
A-253 CTRP2 5.927 7.9672 4.2368 2.0215
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-620 CTRP2 0.7451 1.9401 0.7447 28.6439
HGC-27 CTRP2 1.114 5.7321 0.5493 28.1202
IM95 CTRP2 1.5031 4.6852 1.2715 24.3916
NUGC-4 CTRP2; CTRP1 2.3681 6.7926 1.5174 21.0075
NCC-StC-K140 CTRP2 2.5388 9.3483 0.5642 23.9383
NUGC-3 CTRP2 2.5584 7.3563 1.4773 20.5575
SNU-16 CTRP2 3.3904 7.1351 2.429 14.6628
SNU-668 CTRP2 4.1164 7.2694 3.088 10.2088
SNU-1 CTRP2 4.45 8.5525 2.7733 10.7536
GSS CTRP2 4.8611 7.4498 3.6857 6.0752
Fu97 CTRP2; CTRP1 4.9016 8.0331 3.4388 7.1125
NCI-N87 CTRP2 4.958 10.5262 2.2312 11.9459
GSU CTRP2 5.1427 7.6844 3.8054 5.0213
SNU-5 CTRP2 5.3103 8.3885 3.5884 5.6257
SNU-719 CTRP2 5.3537 8.308 3.6626 5.2379
SNU-216 CTRP2 5.375 8.096 3.7846 4.6905
SNU-601 CTRP2 5.4862 6.8561 4.4751 1.6628
MKN74 CTRP2; CTRP1 5.556 9.9214 3.0284 7.6095
23132/87 CTRP2 5.5655 7.1101 4.4069 1.8248
SH-10-TC CTRP2; CTRP1 5.5707 7.9045 4.0368 3.4002
MKN7 CTRP2; CTRP1 5.6109 7.9744 4.0316 3.3588
ECC12 CTRP2 5.6504 6.7025 4.6493 0.7928
KE-39 CTRP2 5.6738 7.9642 4.07 3.0287
HuG1-N CTRP2 5.7559 9.4763 3.3898 5.6952
Hs 746.T CTRP2 5.991 10.5624 3.029 6.8035
AGS CTRP2; CTRP1 6.0977 7.5525 4.5343 0.8339
MKN1 CTRP2 6.1746 9.6648 3.5947 4.226
MKN45 CTRP2 6.3606 7.3849 4.7076 0.1792
LMSU CTRP2 6.395 9.6273 3.7569 3.2925
KATO III CTRP2 6.7389 8.7397 4.345 0.8769
SNG-M CTRP2; CTRP1 3.5089 9.1995 1.5883 17.772
SNU-1077 CTRP2 5.657 7.7651 4.1546 2.7101
SNU-685 CTRP2 5.6957 10.0862 3.0436 7.2287
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CGTH-W-1 CTRP2 4.2843 10.1298 1.8434 14.9143
SW579 CTRP2 4.3964 8.8371 2.5843 11.6525
TT CTRP2 5.1565 7.8153 3.7512 5.223
B-CPAP CTRP2 5.5444 8.951 3.4906 5.6271
BHT-101 CTRP2 5.6047 10.0814 2.9763 7.6634
8305C CTRP2 5.6771 14.6055 0.7803 16.1687
8505C CTRP2 5.7809 8.3256 3.9697 3.2783
TT2609-C02 CTRP2 5.9766 8.9458 3.8053 3.6602
CAL-62 CTRP2 6.2733 8.2197 4.3261 1.3159
FTC-133 CTRP2 7.267 20.0444 -0.6935 18.2025
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 27 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1214 CTRP2 1.1915 5.4959 0.7081 27.3341
BICR 22 CTRP2 2.1083 5.8227 1.5983 21.3783
PE/CA-PJ34 (clone C12) CTRP2 2.4099 5.968 1.873 19.482
PE/CA-PJ15 CTRP2 2.5045 7.3622 1.4189 20.9247
Detroit 562 CTRP2 2.9698 10.1267 0.6192 22.6292
PE/CA-PJ49 CTRP2 3.7828 7.3632 2.718 12.5191
HSC-4 CTRP2 4.2022 8.6776 2.4857 12.4863
SNU-46 CTRP2 4.7452 8.5626 3.0302 9.0599
SCC-4 CTRP2 4.7459 9.6486 2.4891 11.3108
FaDu CTRP2 4.9143 6.7243 4.0937 4.2544
HSC-2 CTRP2; CTRP1 4.9456 10.1129 2.4369 11.2033
HSC-3 CTRP2 4.9676 7.9662 3.5191 6.5611
BICR 18 CTRP2 5.3104 12.0884 1.7415 13.2334
YD-10B CTRP2 5.4 9.7407 2.9856 7.9858
SNU-1066 CTRP2 5.4472 7.9313 3.9214 3.9977
BHY CTRP2 5.4545 10.7902 2.5057 9.877
BICR 31 CTRP2 5.4734 13.8059 1.0158 15.6962
BICR 16 CTRP2 5.4826 10.7253 2.5604 9.601
SNU-1076 CTRP2 5.7115 8.0768 4.0417 3.0879
SNU-899 CTRP2 5.7154 7.0895 4.5122 1.2257
BICR 6 CTRP2 5.7412 13.0054 1.6286 12.8785
PE/CA-PJ41 (clone D2) CTRP2 5.7623 9.9406 3.1658 6.6114
SCC-9 CTRP2; CTRP1 5.8667 8.6677 3.8753 3.6118
SNU-1041 CTRP2 5.9184 7.3568 4.5097 1.0188
SCC-25 CTRP2 6.4459 15.732 0.8189 14.6594
CAL-33 CTRP2 6.777 9.0929 4.2166 1.2405
BICR 56 CTRP2 7.5953 13.8553 2.5401 6.4611
⏷ Show the Full List of 27 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JMSU-1 CTRP2 3.6846 8.355 2.1537 15.0349
UM-UC-3 CTRP2; CTRP1 3.9504 7.952 2.6095 12.6377
RT-4 CTRP2; CTRP1 3.9939 9.869 1.7173 16.1348
5637 CTRP2; CTRP1 4.3709 10.464 1.7636 15.1197
253J CTRP2 5.0088 6.0439 4.5147 2.2962
T24 CTRP2 5.1335 8.867 3.2068 7.5522
BC-3C CTRP2 5.207 7.2055 4.0962 3.6827
KU-19-19 CTRP2 5.3712 6.5464 4.5452 1.5451
UM-UC-1 CTRP2 5.412 7.5673 4.0746 3.4194
HT-1197 CTRP2 5.416 9.3169 3.2094 7.023
BFTC-905 CTRP2 5.4194 9.8553 2.9439 8.1249
RT-112 CTRP2 5.4454 8.7339 3.5223 5.6644
TCCSUP CTRP2 5.6415 7.5566 4.2444 2.37
KMBC-2 CTRP2; CTRP1 5.6884 7.3135 4.4031 1.75
639V CTRP2 5.7051 7.2562 4.4287 1.5562
VM-CUB-1 CTRP2 5.7799 10.3342 2.9846 7.3309
J82 CTRP2 5.828 8.8791 3.7344 4.1652
U-BLC1 CTRP2 6.2422 8.0814 4.3697 1.1954
HT-1376 CTRP2; CTRP1 6.2456 9.5411 3.7129 3.7314
253J-BV CTRP2 6.5913 8.1794 4.5021 0.5354
CAL-29 CTRP2 7.5005 8.9328 4.585 0.0992
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 5.7547 8.2858 3.9707 3.3126

References

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