General Information of Drug (ID: DMA14PR)

Drug Name
TPCA-1
Synonyms TPCA1
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 279.29
Logarithm of the Partition Coefficient (xlogp) 1.7
Rotatable Bond Count (rotbonds) 3
Hydrogen Bond Donor Count (hbonddonor) 3
Hydrogen Bond Acceptor Count (hbondacc) 4
Chemical Identifiers
Formula
C12H10FN3O2S
IUPAC Name
2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide
Canonical SMILES
C1=CC(=CC=C1C2=CC(=C(S2)NC(=O)N)C(=O)N)F
InChI
InChI=1S/C12H10FN3O2S/c13-7-3-1-6(2-4-7)9-5-8(10(14)17)11(19-9)16-12(15)18/h1-5H,(H2,14,17)(H3,15,16,18)
InChIKey
SAYGKHKXGCPTLX-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
9903786
ChEBI ID
CHEBI:91403
CAS Number
507475-17-4
UNII
9M632G86CC
DrugBank ID
DB17058
TTD ID
D0E0XV
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Inhibitor of nuclear factor kappa-B kinase (IKK) TTRPDBG NOUNIPROTAC Inhibitor [1]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Inhibitor of nuclear factor kappa-B kinase subunit beta (IKBKB) OT9RDS3H IKKB_HUMAN Gene/Protein Processing [2]
Signal transducer and activator of transcription 3 (STAT3) OTAAGKYZ STAT3_HUMAN Gene/Protein Processing [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 42 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1 5.6242 14.1578 0.4426 21.9552
CADO-ES1 GDSC1 0.0163 2.4113 -0.0248 53.6276
EW-13 GDSC1 0.3218 4.2078 -0.0129 50.0016
EW-18 GDSC1 0.5047 5.5336 -0.228 48.3934
NOS-1 [Human HNSCC] GDSC1 0.6429 4.1733 0.3465 46.6058
ES5 GDSC1 0.7128 5.9889 -0.171 46.6713
EW-7 GDSC1 0.8024 5.1864 0.2144 45.4292
TC-71 GDSC1 0.8083 3.1382 0.7339 44.2022
ES8 GDSC1 1.0528 4.831 0.6033 42.5259
H-EMC-SS GDSC1 1.1186 4.721 0.7094 41.6872
SK-PN-DW GDSC1 1.2405 4.1891 0.9944 39.7028
ES7 GDSC1 1.6619 9.2181 -0.5864 41.3064
SK-N-MC CTRP2 1.7718 3.0283 1.7712 28.4666
MHH-ES-1 GDSC1; CTRP2 1.8647 5.5059 1.6179 28.6822
EW-16 GDSC1 2.0015 6.893 0.8133 35.321
EW-1 GDSC1 2.0365 6.0107 1.2261 33.2556
EW-3 GDSC1 2.1319 10.1633 -0.5776 38.8948
ES4 GDSC1 2.1958 11.8314 -1.3245 40.1243
EW-11 GDSC1 2.2614 8.4884 0.3447 35.6152
SK-ES-1 GDSC1; CTRP2 2.3731 5.7217 2.1211 25.3267
ES1 GDSC1 2.5658 7.3957 1.1553 30.5979
Hs 888.T CTRP2 3.4312 16.0356 -1.2669 32.0108
ES6 GDSC1 3.5412 11.4723 0.077 30.6906
A-673 GDSC1; CTRP2 3.7152 5.7232 3.5824 15.9761
CHSA0108 GDSC1 3.8188 9.7293 1.1883 24.5881
U2OS GDSC1; CTRP2 3.9555 6.6604 3.5711 15.2964
TC71 CTRP2 4.0899 7.164 3.5277 15.08
EW-24 GDSC1 4.2692 7.3421 2.7677 12.3907
G-292 clone A141B1 GDSC1; CTRP2 4.4347 6.7392 4.0588 12.0879
NY GDSC1 4.4675 7.5278 2.8386 11.1318
CAL-78 GDSC1; CTRP2 4.4817 8.5068 3.3525 14.7353
SaOS-2 GDSC1; CTRP2 4.5899 6.3323 4.37 10.4733
CHSA8926 GDSC1 4.93 6.9399 3.4785 4.7448
HuO9 GDSC1 5.1199 7.7455 3.2209 6.1739
SJSA-1 GDSC1; CTRP2 5.259 9.0864 3.8279 10.9492
SW1353 CTRP2 5.2715 8.5119 4.1193 9.7177
MG-63 GDSC1; CTRP2 5.4645 7.5382 4.7725 6.5818
HuO-3N1 GDSC1 5.5242 9.3738 2.7141 8.8163
CHSA0011 GDSC1 5.5676 11.6805 1.6221 15.9524
CAL-72 GDSC1 6.3453 7.5533 3.934 0.1711
HOS GDSC1; CTRP2 6.3758 9.9843 4.3434 6.5346
Hs 822.T CTRP2 7.2783 11.842 4.0984 6.0775
⏷ Show the Full List of 42 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 209 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 2.4544 5.0755 2.3421 24.2994
MEC1 CTRP2 3.4145 6.1539 3.1437 18.4713
JM1 GDSC1; CTRP2 2.316 5.8491 2.0271 25.8351
YT GDSC1 -4.5579 3.7348 -5.2151 76.7646
A3/Kawakami GDSC1; CTRP2 -1.7921 -0.252 -1.7921 52.2076
GDM-1 GDSC1; CTRP2 -1.6213 2.2726 -1.6676 51.0395
EB2 GDSC1 -1.4909 2.0014 -1.5709 68.6928
DND-41 GDSC1 -1.4702 3.5293 -1.8018 65.4102
697 GDSC1; CTRP2 -1.4664 1.5752 -1.4785 50.0376
ALL-PO GDSC1 -1.399 1.4837 -1.4321 69.0605
SU-DHL-5 GDSC1 -1.3825 2.5365 -1.5226 66.7623
SU-DHL-16 GDSC1 -1.149 0.8274 -1.1531 67.7556
JSC-1 GDSC1 -1.1 4.8439 -1.7455 61.0213
Pfeiffer CTRP2 -1.0825 2.7162 -1.1376 47.5454
P30/OHK GDSC1 -1.0086 1.1092 -1.0163 65.9471
EoL-1 GDSC1; CTRP2 -0.9836 1.6544 -0.9905 46.834
QIMR-WIL GDSC1 -0.8072 3.3389 -1.0412 60.9624
OCI-M1 GDSC1; CTRP2 -0.7907 0.7157 -0.7907 45.5365
NU-DUL-1 GDSC1 -0.6668 1.5019 -0.6793 61.8672
WSU-NHL GDSC1 -0.6479 3.7655 -0.9606 59.1352
MOLT-16 GDSC1; CTRP2 -0.6143 2.0767 -0.6249 44.3878
ATN-1 GDSC1 -0.6032 3.6989 -0.8966 58.8428
KG-1 GDSC1 -0.5893 2.7958 -0.7115 59.7362
MLMA GDSC1 -0.5802 5.3633 -1.3446 57.0505
CTB-1 GDSC1 -0.4491 10.326 -3.2101 53.7196
NALM-6 GDSC1; CTRP2 -0.4153 1.4905 -0.4164 43.0388
L-1236 GDSC1; CTRP2 -0.3993 4.0048 -0.5542 43.2702
H9 GDSC1 -0.3142 4.8206 -0.8821 55.5012
HuT 78 CTRP2 -0.3131 11.6625 -2.9524 45.4463
HAL-01 GDSC1 -0.3052 3.9852 -0.6399 56.0272
Ri-1 CTRP2 -0.2849 4.0964 -0.4451 42.5415
TUR GDSC1 -0.2446 3.5092 -0.4656 55.8212
BC-3 GDSC1 -0.1429 3.9481 -0.4539 54.587
BE-13 GDSC1 -0.1103 3.2345 -0.2675 54.6673
HEL GDSC1; CTRP2 -0.0711 2.9421 -0.1025 40.8335
RPMI-8866 GDSC1 -0.0699 2.8062 -0.1583 54.4519
MHH-PREB-1 GDSC1 -0.0418 2.9079 -0.1421 54.1027
Karpas-45 GDSC1 -0.0237 3.2058 -0.1692 53.7835
MOLM-16 CTRP2 -0.0201 2.6673 -0.0372 40.4542
MOLM-13 GDSC1; CTRP2 0.1076 3.5639 0.037 39.7569
NB4 GDSC1; CTRP2 0.1136 2.7463 0.0967 39.5643
HC-1 GDSC1 0.1361 4.3213 -0.246 51.815
Hs 611.T CTRP2 0.2189 4.9589 -0.053 39.5425
Namalwa GDSC1; CTRP2 0.22 4.4338 0.0443 39.296
SIG-M5 GDSC1; CTRP2 0.2285 2.2272 0.2254 38.7564
MEG-01 GDSC1 0.2924 5.9373 -0.6026 50.2405
Sc-1 GDSC1 0.3413 4.0562 0.0474 49.7992
Loucy GDSC1 0.3458 3.9356 0.0817 49.749
SR GDSC1; CTRP2 0.3571 4.3854 0.1993 38.3511
KMS-28BM CTRP2 0.3797 6.774 -0.3513 39.5605
F-36P CTRP2 0.4337 3.6834 0.3686 37.5815
KE-37 GDSC1; CTRP2 0.5195 2.9506 0.5046 36.856
KMS-34 CTRP2 0.5374 2.8933 0.5248 36.7294
BL-41 GDSC1 0.5708 2.1583 0.5628 46.9138
OCI-AML-2 GDSC1; CTRP2 0.6639 4.0404 0.5738 36.1307
SET-2 CTRP2 0.7061 3.2826 0.6816 35.6444
RPMI-6666 GDSC1; CTRP2 0.73 4.7388 0.5418 35.9886
NOMO-1 GDSC1; CTRP2 0.7701 4.623 0.6049 35.6559
SU-DHL-6 GDSC1; CTRP2 0.8033 3.4299 0.7738 35.0135
OCI-Ly19 GDSC1; CTRP2 0.8038 3.8218 0.7445 35.1059
KMS-12-BM GDSC1; CTRP2 0.8049 3.9204 0.7362 35.1284
KOPN-8 GDSC1 0.8086 3.5375 0.6699 44.394
CCRF-CEM GDSC1 0.8231 3.5785 0.6778 44.2428
WIL2 NS GDSC1 0.8879 5.4851 0.2027 44.7622
MV4-11 GDSC1; CTRP2 0.9086 3.092 0.8974 34.2526
VAL GDSC1 0.997 3.8599 0.8082 42.34
JURL-MK1 GDSC1; CTRP2 1.0557 4.6975 0.8998 33.7407
ARH-77 GDSC1 1.064 5.9824 0.2068 43.4146
NKM-1 GDSC1 1.1451 4.9742 0.6572 41.6452
OCI-Ly3 CTRP2 1.1464 4.0064 1.0873 32.8266
Reh GDSC1; CTRP2 1.1746 3.2924 1.1624 32.4837
Hs 445 GDSC1 1.2083 6.6174 0.1064 42.6101
PL-21 GDSC1 1.2471 5.6555 0.5267 41.2732
BC-1 GDSC1 1.2697 3.8337 1.1104 38.9742
CMK CTRP2 1.2897 2.9955 1.2863 31.688
SUP-HD1 GDSC1; CTRP2 1.3077 4.921 1.1328 32.1336
SKM-1 CTRP2 1.3195 2.675 1.3189 31.4798
P32/ISH GDSC1 1.3197 2.7184 1.3084 37.5956
Kasumi-1 CTRP2 1.3216 4.0954 1.2631 31.6584
M-07e CTRP2 1.3607 5.9969 0.9458 32.5485
A4/Fukuda GDSC1; CTRP2 1.3713 5.5747 1.0646 32.1381
AML-193 CTRP2 1.4156 3.4087 1.4046 30.8744
RS4;11 GDSC1; CTRP2 1.4538 5.4711 1.1786 31.4935
KMS-26 CTRP2 1.4768 5.2972 1.242 31.21
Ramos.2G6.4C10 GDSC1 1.4993 3.2263 1.4571 35.5366
Peer CTRP2 1.5028 3.2879 1.4968 30.2769
Mono-Mac-6 GDSC1; CTRP2 1.558 8.4215 0.3426 33.6247
MOLM-6 CTRP2 1.5711 5.5356 1.2915 30.734
ALL-SIL GDSC1; CTRP2 1.5751 3.3471 1.5688 29.7963
DEL GDSC1; CTRP2 1.6102 5.5877 1.3219 30.5047
GA-10 CTRP2 1.6295 2.2448 1.6295 29.4123
MOLT-3 CTRP2 1.6502 2.0343 1.6502 29.2746
CESS GDSC1 1.716 5.714 1.0056 36.3009
Jiyoye GDSC1 1.7296 6.76 0.5907 37.8217
SU-DHL-10 GDSC1; CTRP2 1.7327 3.7711 1.7151 28.7841
SU-DHL-8 GDSC1; CTRP2 1.7398 4.4965 1.6611 28.9423
OCI-AML-5 GDSC1; CTRP2 1.7452 3.4963 1.738 28.6659
HH [Human lymphoma] GDSC1 1.7526 6.234 0.8359 36.765
MOLP-8 GDSC1; CTRP2 1.7739 6.4848 1.2565 30.183
VL51 GDSC1 1.7753 5.4748 1.1605 35.2148
TF-1 CTRP2 1.7997 2.9586 1.7993 28.2802
RPMI-8402 GDSC1; CTRP2 1.808 2.9801 1.8077 28.2245
HDLM-2 GDSC1; CTRP2 1.8377 5.1148 1.6698 28.5939
ML-2 GDSC1 1.8508 5.3865 1.2745 34.1742
SUP-M2 GDSC1; CTRP2 1.8511 2.8953 1.851 27.9366
EB1 CTRP2 1.9114 4.3148 1.8625 27.6989
U-937 CTRP2 1.9135 3.2178 1.9124 27.5243
KE-97 CTRP2 1.9642 4.4525 1.9041 27.3852
PF-382 GDSC1; CTRP2 2.0128 4.0606 1.9884 26.9408
MOLT-13 GDSC1; CTRP2 2.0198 5.11 1.8676 27.3293
P31/FUJ GDSC1; CTRP2 2.03 4.5519 1.9625 26.9719
JJN-3 GDSC1; CTRP2 2.0367 7.2248 1.2996 29.1978
ST486 GDSC1; CTRP2 2.0794 5.631 1.8227 27.2926
Mono-Mac-1 CTRP2 2.125 6.9031 1.5051 28.235
JVM-3 GDSC1; CTRP2 2.1273 6.1801 1.7318 27.4542
CTV-1 GDSC1 2.1423 6.4346 1.1577 32.9563
KYO-1 CTRP2 2.1496 5.3138 1.9688 26.5648
JVM-2 GDSC1; CTRP2 2.1517 6.5999 1.6325 27.7184
Karpas-299 GDSC1; CTRP2 2.1686 4.0802 2.1486 25.8882
BV-173 GDSC1; CTRP2 2.176 6.0328 1.8258 26.9758
Daudi GDSC1; CTRP2 2.1921 4.7796 2.106 25.956
NCO2 CTRP2 2.195 4.362 2.156 25.7762
CA46 GDSC1; CTRP2 2.1956 6.5878 1.684 27.4041
SEM CTRP2 2.2094 3.195 2.2092 25.55
BALL-1 GDSC1 2.2192 7.0535 0.964 33.4098
KHM-1B CTRP2 2.2204 5.6225 1.9784 26.3061
P12-Ichikawa GDSC1; CTRP2 2.2397 4.59 2.1804 25.5475
Farage GDSC1 2.2577 5.8361 1.5302 30.3282
LAMA-84 GDSC1; CTRP2 2.2684 5.653 2.0234 25.9977
TALL-1 [Human adult T-ALL] CTRP2 2.2825 4.799 2.1998 25.3425
MOTN-1 CTRP2 2.2986 5.4432 2.1036 25.6231
Ku812 GDSC1; CTRP2 2.3403 5.3334 2.1716 25.2545
Jurkat CTRP2 2.3676 5.6774 2.1258 25.3278
SUP-B15 GDSC1; CTRP2 2.39 4.9075 2.2993 24.6541
RCH-ACV CTRP2 2.3962 4.4235 2.3615 24.4216
BL-70 CTRP2 2.4087 3.1099 2.4087 24.2216
L-363 GDSC1; CTRP2 2.4096 5.2922 2.2548 24.7447
MOLT-4 GDSC1 2.4296 6.2173 1.5484 29.2434
KMS-20 CTRP2 2.4737 5.3097 2.3207 24.3119
EJM GDSC1; CTRP2 2.4816 7.9216 1.5205 27.0853
HL-60 GDSC1; CTRP2 2.486 5.3804 2.3201 24.2753
PL21 CTRP2 2.5141 4.6928 2.4592 23.7046
KM-H2 GDSC1; CTRP2 2.5169 6.836 1.9527 25.4764
EM-2 GDSC1; CTRP2 2.5359 5.4686 2.3559 23.9921
DB GDSC1; CTRP2 2.557 6.586 2.0779 24.9106
LC4-1 GDSC1 2.5639 7.7145 1.0047 31.336
HEL 92.1.7 CTRP2 2.6127 4.1599 2.602 22.898
U-698-M GDSC1 2.6143 9.7671 0.0719 34.7621
TK [Human B-cell lymphoma] GDSC1 2.62 8.113 0.8717 31.6538
KMS-21-BM CTRP2 2.6709 4.6078 2.6333 22.6014
HuNS1 CTRP2 2.6737 3.7455 2.6727 22.4592
NCI-H929 CTRP2 2.7386 4.9386 2.6674 22.265
MHH-CALL-4 CTRP2 2.7464 4.6654 2.7073 22.1032
EHEB CTRP2 2.7815 6.9906 2.1866 23.8452
KMS-11 GDSC1; CTRP2 2.8042 6.4497 2.3898 23.0439
OCI-AML-3 GDSC1; CTRP2 2.8798 6.4546 2.4707 22.5237
MY-M12 GDSC1 2.884 9.3564 0.5248 31.8265
OPM-2 GDSC1; CTRP2 2.9393 6.3703 2.5614 22.0164
Ki-JK CTRP2 2.9746 5.2702 2.8694 20.8108
SU-DHL-4 GDSC1; CTRP2 3.0029 5.1397 2.9212 20.5404
Kasumi-2 CTRP2 3.0186 5.3224 2.9076 20.5377
L-428 GDSC1; CTRP2 3.0983 6.7779 2.6027 21.3917
Karpas-422 GDSC1; CTRP2 3.1502 6.2636 2.8234 20.4306
JeKo-1 CTRP2 3.2256 5.8778 3.012 19.5216
GR-ST GDSC1 3.2553 8.7284 1.1769 27.0894
L-540 GDSC1; CTRP2 3.2645 6.7513 2.7919 20.2064
KCL-22 GDSC1; CTRP2 3.3803 6.9619 2.8433 19.6784
AMO1 GDSC1; CTRP2 3.4358 7.612 2.6564 20.221
SUP-T1 GDSC1; CTRP2 3.4676 7.5702 2.7066 19.9426
NU-DHL-1 CTRP2 3.4795 5.9179 3.2788 17.7865
KO52 CTRP2 3.5118 6.5806 3.1175 18.2771
RPMI-8226 GDSC1; CTRP2 3.5195 6.3425 3.2021 17.9431
SK-MM-2 GDSC1; CTRP2 3.5675 8.5372 2.4089 20.791
THP-1 GDSC1; CTRP2 3.6095 7.7434 2.7871 19.2424
CML-T1 CTRP2 3.6158 7.2669 2.9826 18.4829
HPB-ALL CTRP2 3.6365 6.3526 3.3264 17.139
SUP-T11 CTRP2 3.6548 7.4569 2.9501 18.4965
WSU-DLCL2 GDSC1; CTRP2 3.6558 4.629 3.6518 15.9265
KMS-18 CTRP2 3.7306 6.3758 3.4216 16.5097
KMS-27 CTRP2 3.7541 8.9263 2.4289 20.2155
ROS-50 GDSC1 3.765 12.2064 -0.0935 30.4298
RL GDSC1; CTRP2 3.8179 8.0734 2.8675 18.366
KMOE-2 GDSC1 3.8515 8.3168 1.92 20.1011
MHH-CALL-3 CTRP2 3.8611 8.8647 2.565 19.4146
ME1 GDSC1 3.9003 11.2683 0.4914 27.6113
Granta-519 GDSC1; CTRP2 3.9746 7.6335 3.216 16.5971
K-562 GDSC1; CTRP2 4.0713 7.4575 3.39 15.6608
MM1.S CTRP2 4.0785 5.896 3.9375 13.5867
MN-60 GDSC1 4.0884 9.9815 1.2953 22.9262
Raji GDSC1; CTRP2 4.1472 8.696 2.9305 17.2551
U266B1 GDSC1; CTRP2 4.1633 8.7241 2.9339 17.2001
KY821 GDSC1 4.2717 6.1073 3.3871 7.5559
DG-75 GDSC1 4.6954 9.2074 2.1831 15.1324
OCI-Ly10 CTRP2 4.7437 8.5767 3.5797 13.1737
LP-1 GDSC1; CTRP2 4.771 8.483 3.6504 12.8211
SU-DHL-1 GDSC1; CTRP2 4.929 6.8103 4.5573 8.8023
RC-K8 GDSC1 4.9596 7.5883 3.1849 6.8942
HT GDSC1; CTRP2 5.1694 8.7061 3.9288 10.7374
HD-MY-Z CTRP2 5.196 9.3406 3.645 11.845
KMM-1 CTRP2 5.3571 12.1074 2.4227 16.4115
REC-1 CTRP2 5.4451 12.1569 2.4754 16.0192
SCC-3 GDSC1 5.6039 6.8016 3.9187 0.6197
MOLP-2 CTRP2 5.7324 10.8913 3.3562 11.8866
P3HR-1 CTRP2 5.7721 9.9676 3.8515 9.7515
Ci-1 CTRP2 5.8535 6.6583 5.5668 2.4093
MC116 GDSC1; CTRP2 5.9103 11.8096 3.0493 12.7808
Karpas-620 GDSC1; CTRP2 6.3864 8.0505 5.3102 2.4854
Toledo CTRP2 7.7829 9.5781 5.4308 0.6125
ME1 CTRP2 8.0508 13.7983 3.6851 6.6213
⏷ Show the Full List of 209 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 3.2039 6.1388 2.9181 19.9256
TE15 CTRP2 3.8074 10.0343 1.9761 21.765
TE-15 GDSC1 1.3908 8.4113 -0.4858 42.6292
T.T GDSC1 3.0107 7.0975 1.7324 25.0969
TE-11 GDSC1; CTRP2 3.3928 7.0065 2.8408 19.6518
TE-8 GDSC1 3.7623 9.0941 1.4548 23.3421
TE-6 GDSC1; CTRP2 4.2434 7.1972 3.6772 14.0812
KYSE-140 GDSC1; CTRP2 4.4272 10.8198 2.204 19.3678
TE-9 GDSC1; CTRP2 4.4289 6.2067 4.2345 11.4492
KYSE-70 GDSC1; CTRP2 4.5719 7.9085 3.2017 9.3286
TE-10 GDSC1; CTRP2 4.6007 8.1528 3.6337 13.3117
KYSE-270 GDSC1 5.0373 10.9684 1.5744 17.902
TE-14 CTRP2 5.1016 8.6188 3.9065 10.987
TE-4 GDSC1; CTRP2 5.1584 8.2875 4.1198 9.9789
OE21 GDSC1; CTRP2 5.257 8.2536 4.2304 9.2939
TE-5 GDSC1; CTRP2 5.3955 8.734 4.1268 9.4061
KYSE-150 GDSC1; CTRP2 5.5926 11.4704 2.9463 13.8445
KYSE-410 GDSC1; CTRP2 5.6355 10.6837 3.3758 12.0056
EC-GI-10 GDSC1; CTRP2 5.6819 9.8906 3.8115 10.1034
OE33 GDSC1; CTRP2 5.8029 7.1426 5.283 3.6993
COLO 680N GDSC1; CTRP2 5.8803 10.9897 3.4337 11.2685
KYSE-520 GDSC1; CTRP2 6.2283 8.6357 4.8986 4.4727
KYSE-180 GDSC1; CTRP2 6.3469 12.5961 3.017 12.0664
TE-1 GDSC1; CTRP2 6.3611 12.0461 3.3032 10.8793
KYSE-30 CTRP2 7.0602 10.4081 4.64 4.2062
KYSE-450 GDSC1; CTRP2 7.2228 11.198 4.3713 5.0559
OE19 GDSC1; CTRP2 7.3973 8.6467 5.6245 0.3355
KYSE-510 GDSC1; CTRP2 8.2396 12.5485 4.3886 3.6892
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 7.656 11.8825 4.3344 4.605
MZ-PC-1 GDSC1 -0.3485 5.0667 -0.9963 55.5994
HuP-T4 GDSC1; CTRP2 1.9439 7.1064 1.2401 29.6874
BxPC-3 GDSC1; CTRP2 2.6794 10.3187 0.7143 29.0777
SNU-213 CTRP2 3.1198 9.0332 1.7321 24.4962
HPAC GDSC1; CTRP2 3.2258 8.0692 2.2501 22.3268
Panc 03.27 GDSC1; CTRP2 3.7795 8.3251 2.7196 19.0381
QGP-1 GDSC1; CTRP2 4.2771 8.9461 2.9463 16.8624
PK-59 CTRP2 4.3518 9.993 2.5283 18.3118
PaTu 8988s CTRP2 4.4614 7.2417 3.8887 12.6679
KP-3 GDSC1; CTRP2 4.4822 10.59 2.3672 18.6156
Panc 08.13 GDSC1; CTRP2 4.5554 8.9809 3.2053 15.1408
KP-4 GDSC1; CTRP2 4.7649 8.0312 3.8539 12.0158
SUIT-2 GDSC1; CTRP2 4.7918 10.5688 2.669 16.7129
L3.3 CTRP2 4.8058 8.9085 3.4835 13.4128
TCC-Pan2 CTRP2 4.997 8.07 3.4919 7.0897
Panc 10.05 GDSC1 5.0515 14.8247 -0.3345 26.8564
PL4 GDSC1 5.0611 8.1803 2.9687 8.2375
YAPC GDSC1; CTRP2 5.1766 9.3793 2.9861 8.9909
MIA PaCa-2 GDSC1; CTRP2 5.1807 6.4605 4.9627 6.5479
CFPAC-1 GDSC1; CTRP2 5.2111 8.3088 4.1601 9.6899
PSN1 GDSC1; CTRP2 5.3313 11.921 2.4925 16.1964
HPAF-II GDSC1; CTRP2 5.3501 12.1277 2.4064 16.4897
SW1990 GDSC1; CTRP2 5.5018 8.266 4.4543 7.8102
Panc 05.04 CTRP2 5.6064 13.2665 1.3918 14.9452
PaTu 8902 GDSC1; CTRP2 5.6545 8.9596 4.2503 8.3283
HuP-T3 GDSC1; CTRP2 5.8139 10.4092 3.667 10.4351
PaTu 8988t GDSC1; CTRP2 5.9459 6.6817 5.6404 1.8985
SU.86.86 GDSC1; CTRP2 6.106 8.7237 4.7558 5.2987
KP-2 GDSC1; CTRP2 6.1726 7.9964 5.173 3.4226
AsPC-1 GDSC1; CTRP2 6.3642 12.0154 3.3211 10.8004
Panc 02.03 GDSC1; CTRP2 6.3762 7.7516 5.4491 1.93
Capan-2 GDSC1; CTRP2 6.5269 13.0355 2.9423 12.0319
Hs 766T GDSC1; CTRP2 6.5829 9.3612 4.8106 4.2347
Capan-1 GDSC1; CTRP2 6.6091 10.9389 4.0503 7.3482
Panc 04.03 GDSC1; CTRP2 6.6322 9.9069 4.5784 5.1159
PANC-1 CTRP2 8.2312 9.8469 5.5161 0.2442
SNU-410 CTRP2 8.2482 10.5045 5.2743 0.7566
DAN-G GDSC1; CTRP2 11.0667 31.5035 -2.7811 21.6498
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 76 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 5.6899 18.3998 -0.4312 24.9676
CHL-1 GDSC1 0.3955 6.6513 -0.7658 49.4431
WM35 GDSC1 1.2074 5.5857 0.51 41.6114
WM278 GDSC1 2.0656 6.9618 0.8487 34.7964
A-431 GDSC1 2.382 5.5248 1.7875 28.0913
M14 GDSC1 2.4513 11.5544 -0.9511 38.2702
Hs 852.T CTRP2 2.5804 6.719 2.0604 24.9015
CP50-MEL-B GDSC1 2.963 8.9502 0.7965 30.2963
MZ-MEL-2 GDSC1 3.1745 7.7931 1.557 25.3609
A-375 GDSC1; CTRP2 3.5063 6.6961 3.0726 18.4593
COLO 792 GDSC1; CTRP2 3.6951 8.1486 2.7079 19.3103
LOX-IMVI GDSC1; CTRP2 3.849 6.4417 3.5293 15.7626
COLO 741 CTRP2 3.8704 19.5453 -2.5936 33.4594
G-mel GDSC1 4.0904 8.7548 1.9097 19.2048
G-361 GDSC1; CTRP2 4.0991 9.3451 2.0631 15.4464
RPMI-7951 GDSC1; CTRP2 4.2531 7.905 3.3901 15.1736
MZ-MEL-7 GDSC1 4.3354 11.3193 0.8345 24.3844
SK-MEL-24 GDSC1; CTRP2 4.3475 9.7154 2.6559 17.8266
WM88 CTRP2 4.4135 6.4775 4.1299 11.881
451Lu GDSC1 4.4757 8.921 2.1492 16.141
DJM-1 GDSC1 4.6793 9.8488 1.8504 17.4049
Mel JuSo GDSC1; CTRP2 4.7762 9.5966 3.1256 14.9299
IPC-298 GDSC1; CTRP2 4.7788 9.8285 3.0162 15.3634
Hs 940.T GDSC1; CTRP2 4.8329 8.0199 3.9269 11.5522
WM115 GDSC1; CTRP2 4.925 8.4442 3.8194 11.7616
MDA-MB-435S CTRP2 4.9255 9.3185 3.4018 13.4616
A-388 GDSC1 4.9408 8.5696 2.6892 10.6906
SK-MEL-1 GDSC1; CTRP2 5.0005 7.9647 4.1188 10.3629
MMAc-SF GDSC1 5.0122 9.1085 2.4767 12.0169
LB2518-MEL GDSC1 5.0668 9.161 2.4917 11.7388
GAK GDSC1 5.113 8.3741 2.9113 8.5167
COLO 679 GDSC1 5.1328 9.9148 2.1691 13.788
Hs 944.T CTRP2 5.2453 9.4978 3.6136 11.8639
WM1799 CTRP2 5.3201 12.0233 2.4318 16.4562
SH-4 GDSC1 5.4875 14.656 0.0912 23.8773
HMCB CTRP2 5.6623 8.9082 4.2828 8.176
COLO 783 GDSC1 5.7344 11.0428 2.0534 12.7698
WT2-iPS GDSC1; CTRP2 5.7918 6.7337 5.4718 2.9432
CP66-MEL GDSC1 5.8395 7.6295 3.6963 1.4694
Hs 938.T GDSC1 5.9347 9.4914 2.9257 6.3051
HMV-II GDSC1 5.9895 15.8999 -0.1429 23.364
WM1552C GDSC1 6.0308 8.0433 3.6188 1.6472
MeWo GDSC1; CTRP2 6.0728 9.1174 4.5315 6.3046
IGR-1 GDSC1; CTRP2 6.0833 11.8939 3.1519 12.0238
SK-MEL-5 GDSC1; CTRP2 6.1239 10.2104 4.0273 8.3227
Hs 294T CTRP2 6.1846 10.5604 3.9022 8.731
Hs 895.T CTRP2 6.1847 10.8055 3.7798 9.2413
WM266-4 CTRP2 6.238 9.2658 4.592 5.7411
VMRC-MELG GDSC1 6.2443 8.3614 3.5907 1.5352
CJM [Human melanoma] CTRP2 6.2545 9.8147 4.3313 6.8043
SK-MEL-2 GDSC1; CTRP2 6.2606 8.2353 5.1235 3.473
LB373-MEL-D GDSC1 6.5147 12.7344 1.7729 12.4581
SK-MEL-3 GDSC1; CTRP2 6.5362 10.8782 4.0241 7.5837
UACC-257 GDSC1; CTRP2 6.5984 10.8953 4.0638 7.3108
Hs 936.T CTRP2 6.6998 10.446 4.363 5.8976
UACC-62 GDSC1; CTRP2 6.7012 9.2103 4.9698 3.3957
IST-MEL1 GDSC1 6.723 18.2893 -0.7758 23.7564
IGR-39 CTRP2 6.7387 9.8922 4.6639 4.5919
Hs 934.T CTRP2 6.7637 9.2478 4.9953 3.1994
Mel Ho GDSC1; CTRP2 6.9233 13.9271 2.8094 11.8485
SK-MEL-31 CTRP2 6.9675 9.6965 4.9186 3.2191
Hs 688(A).T CTRP2 6.9785 11.6568 3.9735 7.0515
A2058 GDSC1; CTRP2 7.0315 10.3322 4.657 4.1793
A101D GDSC1; CTRP2 7.0469 8.3448 5.5832 0.6619
K029AX CTRP2 7.2118 11.3155 4.3069 5.332
SK-MEL-28 GDSC1; CTRP2 7.2461 8.0798 5.7735 0.1043
HT-144 GDSC1; CTRP2 7.2805 11.6788 4.179 5.7482
COLO 829 GDSC1; CTRP2 7.3079 15.0824 2.5303 12.2684
WM983B CTRP2 7.4284 15.0621 2.6305 11.6838
COLO 800 GDSC1; CTRP2 8.0311 13.9892 3.5809 7.0557
Hs 839.T CTRP2 8.667 16.9932 2.5714 10.0057
IGR-37 GDSC1; CTRP2 8.7019 19.0026 1.6242 13.3219
SK-MEL-30 GDSC1; CTRP2 8.7141 15.4689 3.328 7.1113
WM793 GDSC1; CTRP2 8.9759 16.3558 3.0792 7.7044
RVH-421 GDSC1; CTRP2 10.0651 24.5233 -0.0967 16.6421
EquiPSC Line K2 GDSC1 5.897 9.7418 2.7853 7.3694
⏷ Show the Full List of 76 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OACP4 C GDSC1 0.105 4.5083 -0.3324 52.0619
OACM5.1 C GDSC1 0.3769 5.8826 -0.4916 49.5442
FLO-1 GDSC1 1.3438 8.4477 -0.5497 43.0135
ESO-26 GDSC1 1.4931 7.8007 -0.1078 41.2603
KYAE-1 GDSC1 3.9417 8.9083 1.7046 21.1073
KYSE-50 GDSC1 4.1379 6.2585 3.1963 9.5631
KYSE-220 GDSC1 4.1752 10.5438 1.0879 23.707
ESO-51 GDSC1 4.8448 7.4137 3.1872 7.2149
TE-12 GDSC1 5.2011 13.7859 0.3012 23.8763
SK-GT-4 GDSC1 6.8608 13.9847 1.4074 13.713
HCE-4 GDSC1 7.0129 9.433 3.5116 1.1463
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1; CTRP2 4.9772 11.3887 2.438 17.1899
Cancer Drug Sensitivity Data Curated from 35 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IMR-5 GDSC1 0.3346 3.7628 0.1094 49.8643
NB69 GDSC1 0.3845 3.7385 0.1689 49.3244
SJNB-14 GDSC1 1.2559 4.2109 1.0055 39.5393
KP-N-YS GDSC1 1.5253 4.4373 1.2376 36.5293
NB(TU)1 GDSC1 1.6255 4.9688 1.1802 36.1173
CHP-134 GDSC1 1.6395 3.6934 1.539 34.1357
NH-12 GDSC1 1.661 5.7853 0.9193 37.0256
Kelly GDSC1; CTRP2 1.9189 4.6124 1.837 27.761
CHP-212 GDSC1; CTRP2 1.973 3.6876 1.9646 27.1523
IMR-32 CTRP2 1.9788 2.939 1.9787 27.086
SJNB-6 GDSC1 2.0076 5.7141 1.3155 32.9831
MHH-NB-11 GDSC1; CTRP2 2.0945 6.4179 1.6262 27.9201
SK-N-MC-IXC GDSC1 2.162 4.0933 2.023 27.8878
SK-N-FI GDSC1; CTRP2 2.509 5.6379 2.2891 24.3112
SiMa GDSC1; CTRP2 2.5288 9.5399 0.9028 28.9488
SJNB-7 GDSC1 2.589 4.8486 2.2646 23.8192
SJNB-13 GDSC1 2.5965 8.1103 0.8501 31.871
TGW GDSC1 2.7053 5.2151 2.2531 23.2592
SJNB-10 GDSC1 2.7742 5.8046 2.0826 24.0455
KP-N-SI9s CTRP2 2.7964 5.4302 2.6466 22.153
GI-ME-N GDSC1 2.9291 8.8647 0.8061 30.4151
NH-6 CTRP2 3.3612 6.4502 2.9961 19.1692
SJNB-12 GDSC1 3.4174 6.152 2.5755 17.3898
GOTO GDSC1 3.491 6.6824 2.3937 18.3806
SJNB-5 GDSC1 3.5079 7.5965 1.9651 21.2778
SK-N-BE(2) CTRP2 3.6052 9.106 2.1972 21.4819
SK-N-SH GDSC1; CTRP2 3.6685 6.8536 3.1928 17.5408
NB1 GDSC1; CTRP2 3.8672 5.7976 3.7309 14.9764
SJNB-17 GDSC1 3.9061 7.7262 2.2619 17.5428
SK-N-DZ GDSC1; CTRP2 4.2585 7.6977 3.4852 14.7866
CHP-126 GDSC1; CTRP2 4.5581 6.5291 4.2683 10.9449
LA-N-6 GDSC1 4.6999 10.2213 1.681 18.3984
SK-N-AS GDSC1; CTRP2 4.7256 8.7295 3.4901 13.5795
SK-N-BE(2)-M17 GDSC1 4.8111 7.1466 3.2937 6.4961
KP-N-YN GDSC1; CTRP2 6.3825 9.7256 4.4774 5.9618
⏷ Show the Full List of 35 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 1.1672 5.0241 0.9616 33.1615
SNU-478 CTRP2 2.8579 6.9514 2.2829 23.2699
SNU-308 CTRP2 3.3936 7.5497 2.6361 20.4159
HuH-28 CTRP2 4.2041 7.9306 3.3285 15.5445
HuCC-T1 GDSC1; CTRP2 4.6588 13.5486 1.0831 22.7784
SNU-1196 CTRP2 5.5951 7.9581 4.6914 6.6182
SNU-245 CTRP2 6.2266 16.8727 0.7813 20.3995
SNU-869 CTRP2 6.3557 10.0513 4.2941 6.7764
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 89 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Evsa-T GDSC1 1.7421 5.8147 0.994 36.1803
MFM-223 GDSC1 2.6524 5.9299 1.9026 25.8724
HCC1599 GDSC1 2.8968 7.2271 1.5601 26.6978
CAL-148 GDSC1 2.9076 5.6905 2.2697 22.0762
OCUB-M GDSC1 2.9083 6.819 1.7623 25.4232
HCC1187 GDSC1 3.5232 8.4389 1.565 23.7228
CAL-85-1 GDSC1; CTRP2 3.603 9.9194 1.826 22.8446
MDA-MB-468 GDSC1; CTRP2 3.6222 6.1094 3.383 16.9757
COLO 824 GDSC1 3.8021 8.8789 1.597 22.338
BT-549 GDSC1; CTRP2 3.9833 8.1426 3.0088 17.3771
HMC-1-8 CTRP2 4.0357 7.0777 3.5036 15.3233
DU4475 GDSC1; CTRP2 4.0531 6.2444 3.8135 14.1122
MDA-MB-157 GDSC1; CTRP2 4.3071 6.9803 3.8304 13.3165
EFM-19 GDSC1 4.3102 10.3774 1.2845 22.1364
HCC1806 GDSC1; CTRP2 4.7133 8.1985 3.7255 12.6608
HCC1143 CTRP2 4.7817 8.4147 3.693 12.6227
MRK-nu-1 GDSC1 4.9904 8.6533 2.685 10.5674
CAL-51 GDSC1; CTRP2 5.0143 7.0267 4.5559 8.5788
MCF-7 GDSC1; CTRP2 5.0608 7.4584 4.4121 9.0302
Hs 578T GDSC1; CTRP2 5.1142 6.7976 4.757 7.5242
HCC70 GDSC1 5.3167 8.7475 2.8733 8.2243
HCC1954 GDSC1; CTRP2 5.3754 6.8123 5.0211 5.7952
UACC-812 GDSC1 5.4625 7.6998 3.4623 3.592
HCC1569 GDSC1 5.4845 10.1396 2.3158 11.7267
HCC1395 GDSC1; CTRP2 5.5546 10.2264 3.5323 11.5289
BT-474 GDSC1 5.8653 10.8986 2.214 11.3555
EFM-192A GDSC1; CTRP2 5.9045 10.8992 3.4995 10.9483
BT-20 GDSC1; CTRP2 5.942 8.9197 4.5205 6.6057
MDA-MB-330 GDSC1 6.0484 10.7114 2.426 9.4642
MDA-MB-361 GDSC1; CTRP2 6.0681 7.8597 5.1564 3.687
MDA-MB-415 GDSC1 6.0774 7.7458 3.7589 0.8964
BT-483 GDSC1 6.1131 11.899 1.9022 12.6991
MDA-MB-436 GDSC1 6.1158 11.257 2.2114 10.718
HCC2218 GDSC1; CTRP2 6.131 7.7421 5.2666 3.1058
CAL-120 GDSC1; CTRP2 6.1581 11.4517 3.4349 10.7209
MDA-MB-231 GDSC1; CTRP2 6.2023 9.1597 4.6163 5.7047
MDA-MB-453 GDSC1; CTRP2 6.2073 8.4783 4.9604 4.2516
HDQ-P1 GDSC1; CTRP2 6.3343 12.8373 2.8864 12.6131
UACC-893 GDSC1 6.3723 12.6891 1.6991 13.2593
MDA-MB-175-VII GDSC1 6.464 8.1206 3.7776 0.5346
HCC1500 GDSC1; CTRP2 6.478 13.398 2.7224 12.9937
HCC38 GDSC1; CTRP2 6.5006 11.5924 3.6409 9.2365
HCC2157 GDSC1 6.6305 8.1222 3.8401 0.2785
AU565 GDSC1 6.6951 9.2086 3.4593 1.6905
YMB-1-E GDSC1 6.7969 8.8601 3.638 0.8122
ZR-75-1 CTRP2 6.8327 7.9904 4.6704 0.1242
HCC1419 GDSC1; CTRP2 6.9765 9.2929 5.1157 2.4285
ZR-75-30 GDSC1; CTRP2 6.9812 15.3077 2.1684 14.1986
CAMA-1 GDSC1; CTRP2 7.2179 9.7847 5.0383 2.4284
HCC202 GDSC1; CTRP2 7.3118 9.521 5.2142 1.6719
T-47D GDSC1; CTRP2 7.6291 13.3994 3.5892 7.6015
HCC1428 GDSC1; CTRP2 7.6793 11.156 4.6885 3.209
Hs 578Bst CTRP2 7.7742 9.1996 5.5725 0.2905
KPL-1 CTRP2 8.5946 20.9967 0.5724 16.8827
JIMT-1 GDSC1; CTRP2 9.0858 16.404 3.1268 7.3879
HCC1937 GDSC1; CTRP2 9.475 18.0324 2.6114 8.7695
BT 416 CTRP2 2.0736 14.3708 -1.7602 36.5136
BT147 CTRP2 2.821 13.7572 -0.7436 32.4619
BT 286 CTRP2 3.1026 9.158 1.6601 24.7965
BT 239 CTRP2 4.056 6.7521 3.647 14.7219
BT 504 CTRP2 4.2414 9.5078 2.6499 18.1132
BT 440 CTRP2 4.5618 8.3911 3.4857 14.0019
BT 145 CTRP2 4.9474 7.9667 4.0653 10.7098
BT 172 CTRP2 5.1579 8.5695 3.9838 10.5381
BT 112 CTRP2 5.2541 8.5407 4.0889 9.8831
BT 428 CTRP2 5.3061 8.146 4.3291 8.7739
BT 482 CTRP2 5.573 8.5891 4.3606 8.0433
BT 330 CTRP2 5.7746 12.0159 2.8309 13.9319
BT 139 CTRP2 5.8288 10.0829 3.8428 9.6727
BT 228 CTRP2 6.0326 9.887 4.1132 8.1379
BT 179 CTRP2 6.1461 6.9696 5.6636 1.4147
BT164 CTRP2 6.1905 9.5274 4.4231 6.5374
BT 340 CTRP2 6.217 17.0387 0.6904 20.7034
BT 248 CTRP2 6.2312 10.3242 4.0581 7.9921
BT 131 CTRP2 6.3366 10.1038 4.2527 6.9843
BT 328 CTRP2 6.3377 10.7396 3.9365 8.3036
BT 245 CTRP2 6.3568 11.2964 3.674 9.3604
BT 333 CTRP2 6.518 11.46 3.7205 8.8765
BT 359 CTRP2 6.7738 11.0976 4.0969 6.8771
BT 231 CTRP2 6.9057 11.9703 3.7651 8.0257
BT 444 CTRP2 7.0835 14.3535 2.7209 11.9164
BT 224 CTRP2 7.2005 10.302 4.7848 3.4345
BT 422 CTRP2 7.2633 14.1572 2.9536 10.7023
BT 159 CTRP2 7.2979 11.2821 4.3822 4.9041
BT 232 CTRP2 7.5817 10.5779 4.8946 2.5487
BT 498 CTRP2 7.634 18.6991 0.9881 17.1566
BT 320 CTRP2 7.6469 20.0375 0.3343 19.1567
BT 216 CTRP2 8.4638 16.2442 2.7928 9.472
BT 187 CTRP2 8.6358 11.2329 5.1609 0.8335
⏷ Show the Full List of 89 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 4.4531 7.6477 3.708 13.3972
Cancer Drug Sensitivity Data Curated from 68 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D283 Med GDSC1; CTRP2 2.2912 3.8789 2.2832 25.031
AM-38 GDSC1 2.6703 5.6216 2.0517 24.8046
MOG-G-CCM GDSC1 2.8181 5.6231 2.2056 22.9826
M059J GDSC1 2.9997 7.0982 1.7214 25.2192
KS-1 [Human Krukenberg tumour] GDSC1 3.6291 6.8683 2.4335 17.4789
GI-1 GDSC1 3.7664 8.4886 1.7593 21.4884
D-566MG GDSC1 3.9903 10.3075 1.0485 24.6298
GB-1 GDSC1; CTRP2 4.0786 10.201 2.1643 20.3759
KNS-60 CTRP2 4.2307 7.4922 3.5429 14.6359
H4 GDSC1 4.2593 7.12 2.8704 11.6401
D-502MG GDSC1 4.411 8.8921 2.1107 16.641
D-336MG GDSC1 4.4247 6.3292 3.4026 6.8854
SF539 GDSC1; CTRP2 4.4491 6.7887 4.0557 12.059
DBTRG-05MG GDSC1; CTRP2 4.4522 9.6189 2.8033 16.9918
D-392MG GDSC1 4.562 7.1973 3.0791 8.9505
D-423MG GDSC1 4.6184 12.0906 0.6818 24.0987
SNU-1105 CTRP2 4.706 10.4497 2.6466 17.0013
PFSK-1 GDSC1 4.768 12.0277 0.8342 22.8472
LN-18 GDSC1; CTRP2 4.8179 5.9577 4.7285 8.4816
MOG-G-UVW GDSC1 4.8266 8.238 2.7669 10.4723
LN-405 GDSC1 5.0809 7.7467 3.1934 6.4875
SNU-201 CTRP2 5.1008 10.7985 2.8414 15.3266
42-MG-BA GDSC1; CTRP2 5.1065 9.0198 3.7175 11.7511
8-MG-BA GDSC1; CTRP2 5.1237 9.1192 3.6854 11.8431
SNU-466 CTRP2 5.1489 7.4465 4.5059 8.4319
LNZTA3WT4 GDSC1 5.1669 8.183 3.0422 7.385
M059K CTRP2 5.1733 7.9151 4.3114 9.1605
SNU-738 CTRP2 5.2162 7.5527 4.5237 8.1934
ONS-76 GDSC1; CTRP2 5.2318 9.8804 3.4132 12.718
YH-13 GDSC1; CTRP2 5.2654 8.8945 3.9275 10.5232
T98G GDSC1; CTRP2 5.3342 9.4234 3.7318 11.1785
SF126 GDSC1; CTRP2 5.4206 8.9024 4.0672 9.5976
KG-1-C CTRP2 5.4413 9.613 3.7355 10.929
SK-MG-1 GDSC1 5.5149 8.3302 3.2033 5.3097
A-172 GDSC1; CTRP2 5.5626 10.0482 3.628 11.1159
DK-MG GDSC1; CTRP2 5.6054 9.0685 4.1525 8.8413
Hs 683 GDSC1; CTRP2 5.6315 8.0608 4.6743 6.6088
D-263MG GDSC1 5.7079 7.2915 3.7715 1.2291
U-118MG GDSC1; CTRP2 5.8156 9.0288 4.3575 7.5448
SW1783 GDSC1; CTRP2 5.8209 9.7834 3.9855 9.092
Onda 11 GDSC1 5.8418 11.0401 2.1297 11.9749
Onda 10 GDSC1 5.8889 8.9434 3.1496 4.8587
KNS-81-FD GDSC1 5.908 9.5892 2.8636 6.7977
KINGS-1 GDSC1 5.9501 13.3739 1.0707 17.9368
TM-31 CTRP2 6.1031 9.883 4.1738 7.7486
GMS-10 CTRP2 6.1671 8.6933 4.8207 4.9117
SNU-626 CTRP2 6.2121 8.3215 5.0424 3.8988
SF268 GDSC1; CTRP2 6.2523 11.6718 3.402 10.6777
NMC-G1 GDSC1; CTRP2 6.2935 11.0558 3.7431 9.1904
LN-229 GDSC1; CTRP2 6.3158 9.6858 4.4447 6.2179
GOS-3 CTRP2 6.407 10.2791 4.2211 6.9904
CAS-1 GDSC1; CTRP2 6.4191 12.9757 2.8858 12.4567
SNU-489 CTRP2 6.4273 9.3447 4.7014 4.9477
U-251MG GDSC1; CTRP2 6.5223 7.9937 5.4335 1.7785
D-542MG GDSC1 6.5558 8.4388 3.6969 0.7624
GaMG GDSC1; CTRP2 6.6342 11.5252 3.7787 8.4309
U-87MG ATCC GDSC1; CTRP2 6.6527 8.813 5.1284 2.8226
Becker GDSC1; CTRP2 6.6653 12.1928 3.4711 9.6425
SW1088 GDSC1; CTRP2 6.7198 10.8441 4.1815 6.6165
KNS-81 CTRP2 6.8131 11.302 4.0255 7.1069
SF295 GDSC1; CTRP2 6.8504 11.0238 4.1903 6.3658
D-247MG GDSC1 6.8957 9.1543 3.5682 1.0095
CCF-STTG1 CTRP2 7.2267 11.2527 4.3476 5.1459
SNB-75 GDSC1; CTRP2 7.3476 10.1713 4.9394 2.6498
YKG-1 GDSC1; CTRP2 7.4606 12.7803 3.7713 7.1248
Daoy GDSC1; CTRP2 8.0627 18.2383 1.5368 14.6188
KNS-42 GDSC1; CTRP2 8.5589 15.4614 3.2305 7.685
KALS-1 GDSC1; CTRP2 8.9231 18.806 1.8742 12.1338
⏷ Show the Full List of 68 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TGBC24TKB GDSC1 5.118 10.5512 1.8433 15.9787
TGBC1TKB GDSC1 5.4188 9.6959 2.4851 10.7376
ETK-1 GDSC1 5.4665 11.3555 1.7075 15.7393
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-2 CTRP2 1.3132 4.4855 1.2081 31.8687
RL95-2 GDSC1; CTRP2 2.1292 7.0071 1.4747 28.3242
JHUEM-7 CTRP2 3.5749 5.5252 3.4713 16.8072
MFE-280 GDSC1 3.6144 10.6671 0.542 28.5384
JHUEM-1 CTRP2 3.6997 5.895 3.5247 16.229
HEC-151 CTRP2 4.1717 7.7761 3.3616 15.5009
JHUEM-3 CTRP2 4.1836 7.0503 3.6717 14.268
KLE GDSC1; CTRP2 4.2028 9.2587 2.7279 17.9062
AN3-CA GDSC1; CTRP2 4.4623 8.1026 3.5166 14.1307
HEC-59 CTRP2 4.8023 9.3726 3.2583 14.3329
ESS-1 GDSC1; CTRP2 4.82 6.0661 4.7022 8.5699
HEC-265 CTRP2 4.9927 7.3798 4.3787 9.3369
HEC-1-B CTRP2 5.1519 10.0125 3.275 13.4611
EN GDSC1; CTRP2 5.2394 9.3545 3.6785 11.6095
HEC-108 CTRP2 5.5352 8.6678 4.2875 8.4299
HEC-6 CTRP2 5.5438 11.9622 2.6586 15.0931
MFE-319 GDSC1; CTRP2 5.9925 6.9884 5.5285 2.2709
EFE-184 CTRP2 6.5147 11.4642 3.7158 8.9016
HEC-50B CTRP2 6.5837 8.7766 5.0975 3.0522
HEC-1-A CTRP2 6.6837 10.13 4.5068 5.3286
HEC-251 CTRP2 6.7612 11.2247 4.0247 7.1967
MFE-296 GDSC1; CTRP2 6.9319 11.0117 4.2559 5.9658
Ishikawa (Heraklio) 02 ER- CTRP2 7.9521 13.0924 3.9553 5.6982
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TUHR10TKB CTRP2 1.7593 12.4798 -1.1919 36.4213
TK-10 GDSC1 2.6777 6.1291 1.8422 26.1211
LB1047-RCC GDSC1 2.6851 6.143 1.8437 26.0719
HA7-RCC GDSC1 2.7567 7.0453 1.507 27.7188
CAL-54 GDSC1; CTRP2 2.776 6.4779 2.3503 23.2712
KTCTL-1M GDSC1 3.0729 7.8394 1.4382 26.5299
KTCTL-140 GDSC1 3.6938 8.6026 1.638 22.5459
KTCTL-21 GDSC1 3.7253 9.9496 0.9966 25.9651
KTCTL-26A GDSC1 3.8462 7.2484 2.4455 16.4672
A-704 GDSC1 4.1022 7.2915 2.6503 13.9162
LB996-RCC GDSC1 4.143 8.1314 2.2661 16.5703
Caki-1 GDSC1; CTRP2 4.3113 8.3671 3.2448 15.5958
UO-31 GDSC1; CTRP2 4.3717 9.1114 2.9634 16.5577
786-O GDSC1; CTRP2 4.3771 10.7219 2.2036 19.4908
NCC021 GDSC1 4.7213 9.1928 2.2108 14.8518
KTCTL-195 GDSC1 4.8096 9.0642 2.344 13.6203
SN12C GDSC1 5.0074 7.3328 3.3424 5.564
BB65-RCC GDSC1 5.0312 8.087 2.9928 8.1429
TUHR4TKB CTRP2 5.0313 9.7866 3.274 13.7375
ACHN GDSC1; CTRP2 5.128 11.7374 2.4022 16.9911
VMRC-RCW GDSC1; CTRP2 5.1639 9.6318 3.4728 12.6253
769-P GDSC1; CTRP2 5.3563 11.8687 2.5406 15.9553
RXF 393L GDSC1 5.5425 16.0043 -0.5358 26.0957
KMRC-2 CTRP2 5.5441 7.5217 4.8564 6.0513
OS-RC-2 GDSC1; CTRP2 5.5802 11.8214 2.7605 14.6138
KMRC-1 GDSC1; CTRP2 5.6331 7.6015 4.9012 5.6625
A-498 GDSC1 5.6338 7.7148 3.5537 2.6442
KMRC-20 GDSC1; CTRP2 5.7136 8.5036 4.5293 7.0372
TUHR14TKB CTRP2 5.7328 9.5612 4.02 9.1277
KMRC-3 CTRP2 5.8977 11.1096 3.3885 11.4199
VMRC-RCZ GDSC1; CTRP2 5.924 12.1337 2.8989 13.3592
BFTC-909 GDSC1; CTRP2 6.1573 9.5893 4.3651 6.843
LB2241-RCC GDSC1 6.3217 11.7245 2.1251 10.7584
SW13 GDSC1 6.5165 7.9598 3.8551 0.2856
SW156 GDSC1 6.5475 16.6746 -0.1121 21.7395
SNU-1272 CTRP2 6.7748 12.1625 3.5707 9.0439
Caki-2 CTRP2 6.9368 12.0064 3.7705 7.9522
KTCTL-13 GDSC1 6.9816 8.7646 3.7443 0.3755
RCC10RGB GDSC1; CTRP2 7.3243 9.342 5.3005 1.3559
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 57 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 320 CTRP2 0.0854 1.5797 0.0852 39.7004
NCI-H508 CTRP2 1.3945 5.2134 1.1702 31.7195
LoVo GDSC1; CTRP2 1.9226 5.2961 1.7262 28.1266
SW48 GDSC1; CTRP2 1.9453 4.7572 1.8453 27.6469
NCI-H716 GDSC1; CTRP2 2.1493 5.0478 2.0183 26.3951
SNU-407 GDSC1; CTRP2 2.3977 7.7784 1.4859 27.4567
SK-CO-1 CTRP2 2.4313 8.0831 1.404 27.6295
LS513 GDSC1; CTRP2 2.4923 5.9592 2.1908 24.7095
SW620 GDSC1; CTRP2 2.5859 5.157 2.47 23.4364
GP2d CTRP2 2.7469 4.6938 2.705 22.1096
KM12 GDSC1; CTRP2 2.9331 7.6041 2.1245 23.6238
COLO205 GDSC1; CTRP2 3.1608 4.7326 3.1358 19.2948
HCT 15 GDSC1; CTRP2 3.2798 7.8339 2.4026 21.6096
SNU-175 GDSC1 3.3484 6.7545 2.2226 20.2489
SNU-1040 GDSC1 3.4877 14.5576 -1.5067 35.476
COLO201 CTRP2 3.5172 5.3679 3.4372 17.1094
CCK-81 GDSC1; CTRP2 3.5444 6.4932 3.1816 17.9446
HT115 GDSC1; CTRP2 3.6778 4.6593 3.6733 15.7817
DLD-1 CTRP2 3.938 7.2227 3.3431 16.2088
SNU-C1 GDSC1; CTRP2 3.9406 6.5241 3.6016 15.2262
C2BBe1 GDSC1; CTRP2 3.959 9.1052 2.5551 19.1976
MDST8 GDSC1; CTRP2 4.0832 8.2184 3.0785 16.8417
GP5d GDSC1 4.1085 9.0475 1.779 19.9756
COLO 320HSR GDSC1 4.2127 10.4546 1.1641 23.1607
T84 GDSC1; CTRP2 4.2568 8.2721 3.2321 15.786
SW948 GDSC1; CTRP2 4.2727 6.6065 3.9327 13.026
SW837 GDSC1 4.4453 6.319 3.4243 6.6443
SNU-61 GDSC1; CTRP2 4.4563 10.1712 2.5439 17.9967
CL-11 GDSC1; CTRP2 4.4642 7.9895 3.5691 13.9172
SNU-C2A CTRP2 4.5212 9.2953 3.0237 15.9497
CW-2 GDSC1; CTRP2 4.6232 8.7468 3.3816 14.2669
SNU-C5 GDSC1; CTRP2 4.75 9.0142 3.3792 13.9688
LS180 GDSC1; CTRP2 4.8072 7.6771 4.0572 11.0944
HT-55 GDSC1; CTRP2 4.8331 6.9462 4.4007 9.6708
SW1417 GDSC1; CTRP2 4.9715 8.6021 3.7895 11.7723
CaR-1 GDSC1 5.0304 8.5441 2.7682 9.8285
LS411N GDSC1; CTRP2 5.0613 8.9248 3.7208 11.8421
SW626 GDSC1 5.2766 12.3695 1.0634 19.9993
LS1034 GDSC1; CTRP2 5.4204 12.8113 2.1278 17.399
SNU-C2B GDSC1 5.5215 9.8286 2.4929 10.3931
HCC2998 GDSC1 5.6616 9.628 2.6852 8.6591
COLO 678 GDSC1; CTRP2 5.7571 10.3412 3.6522 10.612
LS123 GDSC1; CTRP2 5.925 9.4268 4.2527 7.7637
SW1463 GDSC1 5.9366 7.8028 3.672 1.4781
SNU-81 GDSC1; CTRP2 5.9907 9.6478 4.1977 7.8651
RKO GDSC1; CTRP2 6.0291 7.4939 5.3068 3.1299
HT-29 GDSC1; CTRP2 6.0628 10.9017 3.6311 10.0925
SNU-1033 CTRP2 6.1852 10.7468 3.8095 9.1164
NCI-H747 GDSC1; CTRP2 6.2707 10.7569 3.874 8.6876
HCT 116 GDSC1; CTRP2 6.2769 7.5125 5.494 1.9017
RCM-1 [Human ESC] GDSC1; CTRP2 6.2934 9.5492 4.495 6.0474
SNU-503 CTRP2 6.3151 11.4259 3.5758 9.8442
HCC-56 CTRP2 6.3492 7.5434 5.5312 1.635
SW1116 GDSC1 6.3879 8.4597 3.6171 1.2489
OUMS-23 CTRP2 6.7076 8.0667 5.518 1.2129
HCT 8 CTRP2 6.9451 8.6718 5.3838 1.4451
SNU-C4 CTRP2 7.8278 8.8429 5.7193 0.0642
⏷ Show the Full List of 57 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1 0.4153 6.4132 -0.6514 49.2713
Cancer Drug Sensitivity Data Curated from 26 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Li-7 CTRP2 1.3697 11.6119 -1.1952 37.6375
SNU-878 CTRP2 2.3355 17.4368 -2.9762 37.6539
JHH-4 GDSC1; CTRP2 3.6693 9.105 2.2628 21.0662
JHH-1 GDSC1; CTRP2 3.8962 8.0783 2.9466 17.8506
HuH-6 CTRP2 3.9618 9.1153 2.5534 19.1973
Hep 3B2.1-7 GDSC1; CTRP2 3.967 6.9045 3.4955 15.5479
HLE GDSC1 4.1869 8.5364 2.1011 17.5485
SNU-886 CTRP2 4.3167 6.1727 4.1223 12.1949
Hep-G2 CTRP2 4.337 8.3647 2.7633 11.8266
SNU-449 GDSC1; CTRP2 4.4323 10.9423 2.1497 19.5599
SK-HEP-1 GDSC1; CTRP2 4.5765 8.8677 3.2791 14.7935
JHH-7 GDSC1 4.9506 8.0686 2.9432 8.7571
SNU-182 CTRP2 5.0021 11.3976 2.4562 17.0634
Huh-7 GDSC1 5.1764 8.7252 2.7854 9.2677
SNU-398 GDSC1; CTRP2 5.2246 9.9754 3.3599 12.9524
JHH-5 CTRP2 5.3733 8.8081 4.07 9.6911
HuH-1 GDSC1; CTRP2 5.4385 7.6734 4.6827 7.0117
SNU-761 CTRP2 5.5702 11.1514 3.0857 13.3276
SNU-423 GDSC1; CTRP2 5.6587 10.1631 3.6554 10.8011
HLF CTRP2 5.7677 7.6044 5.0233 4.8577
SNU-475 GDSC1; CTRP2 6.3436 7.5631 5.5176 1.6992
PLC/PRF/5 CTRP2 6.5577 9.2901 4.8269 4.2079
Hep-G2/C3A GDSC1 6.9104 8.5485 3.7937 0.285
JHH-2 GDSC1; CTRP2 6.9659 12.1097 3.7413 8.0239
SNU-387 GDSC1; CTRP2 6.9846 15.2975 2.1761 14.164
JHH-6 GDSC1; CTRP2 7.1148 8.0116 5.7469 0.1906
⏷ Show the Full List of 26 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 211 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H847 GDSC1 -0.3991 1.91 -0.4224 58.5917
NCI-H1048 GDSC1 -0.0809 5.0311 -0.6938 53.5001
LC-2/ad GDSC1 0.6428 5.1767 0.0446 47.0013
NCI-H2227 GDSC1 0.9693 3.8328 0.7841 42.6525
NCI-H1755 GDSC1; CTRP2 1.4008 7.1436 0.639 33.3315
HCC44 GDSC1; CTRP2 1.6643 6.0326 1.2675 30.5052
NCI-H209 GDSC1 1.7479 9.6259 -0.6932 41.0619
LCLC-97TM1 GDSC1; CTRP2 1.8162 7.8553 0.8342 31.372
NCI-H2795 GDSC1 2.0834 8.7647 0.0404 37.5318
Lu-135 GDSC1 2.1006 4.0091 1.9755 28.5626
NCI-H211 GDSC1; CTRP2 2.243 6.033 1.8989 26.5116
NCI-H1688 GDSC1 2.2961 8.8434 0.2108 35.8853
NCI-H2286 CTRP2 2.3313 5.7646 2.065 25.6546
IST-SL1 GDSC1 2.3824 7.0911 1.112 31.8051
EMC-BAC-1 GDSC1 2.393 8.6011 0.4198 34.6587
EPLC-272H GDSC1; CTRP2 2.4604 6.327 2.0524 25.2969
NCI-H358 GDSC1; CTRP2 2.4733 9.0253 1.0646 28.6085
LK-2 GDSC1 2.5991 4.9632 2.2346 23.9662
NCI-H1734 GDSC1; CTRP2 2.6357 5.3924 2.48 23.243
HCC827 GDSC1; CTRP2 2.6502 6.0934 2.3267 23.7397
PC-14 GDSC1; CTRP2 2.6521 6.222 2.2922 23.8566
DV-90 CTRP2 2.6553 4.5046 2.6258 22.6776
DMS 273 GDSC1; CTRP2 2.6839 7.8779 1.7529 25.6792
EMC-BAC-2 GDSC1 2.913 5.9864 2.1459 22.8989
NCI-H2731 GDSC1 3.016 6.2352 2.1385 22.429
NCI-H446 GDSC1; CTRP2 3.0535 6.616 2.6081 21.5046
NCI-H1975 GDSC1; CTRP2 3.0911 6.5337 2.6756 21.1461
NCI-H2085 GDSC1; CTRP2 3.1299 7.65 2.3164 22.3546
NCI-H1944 GDSC1; CTRP2 3.1325 7.8575 2.2372 22.6386
HCC1588 CTRP2 3.1499 6.2579 2.8247 20.4271
NCI-H292 GDSC1; CTRP2 3.1522 8.1229 2.1506 22.9
NCI-H1436 GDSC1 3.1928 7.5659 1.684 24.5139
SK-MES-1 GDSC1; CTRP2 3.1954 6.6917 2.7372 20.6111
NCI-H1184 CTRP2 3.2069 6.3427 2.8614 20.1222
Lu-99 CTRP2 3.2524 6.5109 2.8584 19.9975
NCI-H1341 CTRP2 3.302 5.9868 3.0671 19.0899
LXF 289 GDSC1; CTRP2 3.3477 6.9024 2.8294 19.8247
NCI-H2141 GDSC1; CTRP2 3.3768 7.3986 2.677 20.31
CAL-12T GDSC1; CTRP2 3.4061 8.6227 2.2053 21.9913
HCC2108 CTRP2 3.4268 7.2224 2.7976 19.7158
NCI-H526 GDSC1; CTRP2 3.4698 7.206 2.8498 19.3973
NCI-H82 GDSC1 3.5049 8.1088 1.7109 22.9192
NCI-H2171 GDSC1; CTRP2 3.5309 6.6855 3.1029 18.275
NCI-H1563 GDSC1; CTRP2 3.5395 6.4729 3.1828 17.9547
NCI-H1876 GDSC1 3.5421 8.4519 1.5758 23.5754
SBC-3 GDSC1 3.5874 5.4176 3.0849 12.7868
LC-1F CTRP2 3.6056 9.5499 1.9975 22.2166
NCI-H2135 GDSC1 3.6196 9.6573 1.0485 26.1455
HCC366 CTRP2 3.7056 6.2549 3.4315 16.548
NCI-H64 GDSC1 3.7509 7.8621 2.0561 19.6143
NCI-H2087 GDSC1; CTRP2 3.7514 10.5959 1.6584 23.0508
NCI-H1770 GDSC1 3.7521 4.3772 3.6842 7.5725
NCI-H2126 CTRP2 3.7539 7.8441 2.4636 14.584
VMRC-LCD CTRP2 3.7895 5.7714 3.6524 15.4966
HCC95 CTRP2 3.8245 7.713 3.0256 17.7396
COR-L47 CTRP2 3.8508 28.9595 -7.2889 38.9587
Lu-134-A GDSC1 3.8594 9.0184 1.5779 22.2159
SK-LU-1 GDSC1; CTRP2 3.8751 9.121 2.4636 19.7659
COR-L105 GDSC1; CTRP2 3.8871 9.6369 2.2393 20.5836
NCI-H1105 CTRP2 3.9093 7.7475 3.1002 17.2215
NCI-H2081 GDSC1; CTRP2 3.9145 6.7054 3.511 15.6399
NCI-H2030 GDSC1; CTRP2 3.9317 7.3958 3.2678 16.5148
NCI-H524 GDSC1 3.9453 6.5374 2.8865 12.7398
NCI-H510A GDSC1 3.9547 7.6623 2.3366 16.8122
ABC-1 GDSC1 3.962 8.1163 2.117 18.3263
NCI-H2009 GDSC1; CTRP2 3.973 7.598 3.2289 16.5514
PaCa-3 GDSC1 3.982 12.6288 -0.1181 29.7026
COR-L311 GDSC1 3.9831 7.7746 2.3057 16.9191
Ms-1 GDSC1 3.9863 9.4164 1.4898 22.2222
CPC-N GDSC1 3.988 5.7055 3.3353 9.0805
NCI-H520 GDSC1; CTRP2 3.9936 8.3361 2.935 17.637
NCI-H2228 GDSC1; CTRP2 4.012 8.2267 3.0018 17.3282
DMS 53 GDSC1; CTRP2 4.0199 6.7734 3.6005 15.0006
A-427 GDSC1 4.0221 8.1916 2.1319 17.983
NCI-H1435 GDSC1; CTRP2 4.0258 9.8519 2.2767 20.0873
Lu-65 GDSC1; CTRP2 4.1079 8.6546 2.9094 17.4386
COR-L51 CTRP2 4.1081 7.3543 3.4708 15.2484
NCI-H2110 GDSC1; CTRP2 4.1541 9.3675 2.6291 18.4135
COR-L303 GDSC1 4.158 5.3544 3.6634 5.8196
NCI-H1581 GDSC1; CTRP2 4.1685 7.7708 3.3605 15.5136
NCI-H2405 GDSC1; CTRP2 4.2008 8.9573 2.8651 17.3745
NCI-H2869 GDSC1 4.2063 11.1912 0.7905 25.0775
HARA [Human squamous cell lung carcinoma] GDSC1; CTRP2 4.2289 7.2812 3.6279 14.311
Calu-6 GDSC1; CTRP2 4.2313 8.1286 3.2697 15.7044
COR-L23 GDSC1 4.236 11.3912 0.7154 25.3219
NCI-H810 GDSC1; CTRP2 4.2453 6.882 3.8022 13.597
NCI-H1437 GDSC1 4.2842 6.3978 3.2524 8.5693
RERF-LC-MS GDSC1; CTRP2 4.2932 7.6506 3.5412 14.4749
UMC-11 GDSC1 4.298 7.3732 2.7763 12.2179
NCI-H1155 GDSC1; CTRP2 4.3467 8.8366 3.0662 16.2132
NCI-H596 GDSC1 4.3494 11.0112 1.0001 23.5053
NCI-H1838 GDSC1; CTRP2 4.3754 8.6069 3.2004 15.6086
HCC15 GDSC1; CTRP2 4.399 9.1729 2.9616 16.497
COR-L321 GDSC1 4.4139 7.9906 2.5636 13.397
NCI-H841 GDSC1; CTRP2 4.439 7.8443 3.6076 13.83
A-549 GDSC1; CTRP2 4.471 6.5949 4.1508 11.6369
HCC33 GDSC1 4.5093 9.0052 2.1346 16.1206
NCI-H1573 GDSC1; CTRP2 4.5279 7.7256 3.751 13.0316
NCI-H1703 GDSC1; CTRP2 4.5399 7.3858 3.9102 12.3729
NCI-H647 GDSC1; CTRP2 4.5457 9.8834 2.7675 16.9063
NCI-H1568 GDSC1; CTRP2 4.5939 12.1779 1.6984 20.8268
NCI-H1781 GDSC1 4.5989 6.1121 3.6459 4.4084
SBC-1 GDSC1 4.6156 7.7752 2.8335 10.6615
NCI-H345 GDSC1 4.6454 6.0319 3.7192 3.7025
NCI-H441 GDSC1; CTRP2 4.6699 10.7982 2.4433 17.8775
NCI-H187 GDSC1 4.6982 7.9869 2.7928 10.6948
NCI-H2122 GDSC1; CTRP2 4.6993 7.0693 4.2095 10.7765
Lu-99A GDSC1 4.7281 11.258 1.1863 21.1641
NCI-H1993 GDSC1 4.772 8.7546 2.4686 12.8532
NCI-H69 GDSC1; CTRP2 4.777 7.8493 3.949 11.6038
COLO 668 GDSC1; CTRP2 4.7938 10.2864 2.8084 16.1577
NCI-H2591 GDSC1 4.811 9.8566 1.9509 16.2985
NCI-H2106 CTRP2 4.8153 8.4138 3.7264 12.4056
NCI-H1648 GDSC1 4.8439 8.8841 2.4599 12.6783
NCI-H23 GDSC1; CTRP2 4.8526 7.9357 3.9853 11.2678
LUDLU-1 CTRP2 4.8559 7.9338 3.9894 11.2432
NCI-H1355 GDSC1; CTRP2 4.8939 10.8035 2.6492 16.5557
NCI-H1869 GDSC1; CTRP2 4.9116 10.4206 2.8529 15.7084
NCI-H1963 GDSC1 4.9144 7.3592 3.2643 6.4183
LOU-NH91 GDSC1; CTRP2 4.9296 8.0789 3.9954 11.0365
NCI-H1650 GDSC1; CTRP2 4.992 9.1167 3.5623 12.652
NCI-H1373 CTRP2 4.997 8.8559 3.6926 12.1076
HCC2279 CTRP2 4.9975 9.2436 3.5062 12.8685
NCI-H2023 GDSC1; CTRP2 5.0033 8.845 3.1097 8.7936
NCI-H838 GDSC1; CTRP2 5.0091 8.2757 3.981 10.9016
IA-LM GDSC1 5.0157 8.4855 2.7862 9.7391
HCC1195 CTRP2 5.0307 10.545 2.9021 15.2412
HCC4006 CTRP2 5.054 8.2317 4.0455 10.531
MOR/CPR CTRP2 5.0652 6.8979 4.6638 8.0201
DMS 454 CTRP2 5.0874 10.366 3.042 14.5512
EBC-1 GDSC1; CTRP2 5.12 8.3336 4.0609 10.3111
NCI-H2029 GDSC1 5.1215 8.4687 2.8712 8.7911
NCI-H1693 GDSC1; CTRP2 5.1343 11.4327 2.5587 16.3692
NCI-H1792 GDSC1; CTRP2 5.1448 10.1546 3.1987 13.7881
NCI-H889 CTRP2 5.1452 10.6438 2.9582 14.7597
NCI-H748 GDSC1 5.1533 10.3728 1.9584 15.1252
NCI-H1694 GDSC1; CTRP2 5.179 7.7616 4.3893 8.8297
NCI-H226 GDSC1; CTRP2 5.2209 10.4076 3.1435 13.8433
NCI-H1623 GDSC1; CTRP2 5.2455 8.0968 4.2948 9.0565
NCI-H727 GDSC1; CTRP2 5.2902 9.0139 3.8922 10.6132
SW1271 GDSC1; CTRP2 5.3192 11.1476 2.8658 14.7489
LK2 CTRP2 5.3327 18.233 -0.6527 26.2713
COLO 699 CTRP2 5.3596 11.6364 2.6591 15.4832
Lu-139 GDSC1 5.3596 14.8644 -0.1115 25.0728
NCI-H1666 GDSC1; CTRP2 5.3604 9.4433 3.7459 11.0625
COR-L95 GDSC1; CTRP2 5.3806 8.309 4.3204 8.6383
NCI-H2373 GDSC1 5.3916 11.8108 1.4272 17.6343
Lu-165 GDSC1 5.4165 11.6591 1.5208 17.0126
RERF-LC-KJ GDSC1 5.4244 8.6549 2.9911 7.0732
NCI-H2818 GDSC1 5.4353 7.6709 3.4592 3.6711
RERF-LC-Sq1 GDSC1 5.441 10.2867 2.2129 12.5542
NCI-H1395 CTRP2 5.4552 9.3104 3.8976 10.2261
NCI-H1836 GDSC1 5.4951 7.1485 3.7251 1.7957
NCI-H720 GDSC1 5.5043 8.1607 3.2756 4.8165
NCI-H2170 GDSC1; CTRP2 5.5127 8.1984 4.4975 7.6065
NCI-H522 GDSC1; CTRP2 5.5246 9.6317 3.801 10.4782
COR-L88 GDSC1; CTRP2 5.5439 9.653 3.8077 10.409
LCLC-103H GDSC1; CTRP2 5.563 10.7999 3.2544 12.655
SHP-77 GDSC1; CTRP2 5.646 8.8593 4.2925 8.1702
HCC1438 CTRP2 5.6465 8.1726 4.6329 6.7487
NCI-H661 GDSC1; CTRP2 5.6497 9.9906 3.7334 10.4955
Calu-3 GDSC1; CTRP2 5.6818 7.3115 5.0881 4.7789
Sq-1 CTRP2 5.6845 8.0339 4.7358 6.2368
HCC78 GDSC1; CTRP2 5.7193 12.7204 2.4318 15.6138
NCI-H3255 GDSC1 5.7238 11.0458 2.0445 12.8575
HCC1833 CTRP2 5.7644 13.8277 1.917 17.4594
NCI-H2804 GDSC1 5.7704 10.9993 2.0998 12.3671
NCI-H3122 GDSC1 5.7878 10.5308 2.3379 10.7338
NCI-H650 GDSC1; CTRP2 5.8117 10.7863 3.4768 11.2281
ChaGo-K-1 GDSC1; CTRP2 5.8508 8.8878 4.4583 7.0503
NCI-H460 GDSC1; CTRP2 5.8744 9.7562 4.045 8.7357
NCI-H2369 GDSC1 5.8985 11.1769 2.1027 11.9972
NCI-H1299 GDSC1; CTRP2 6.0228 12.3325 2.8823 13.2298
NCI-H2595 GDSC1 6.0381 11.1554 2.2079 10.9404
NCI-H2444 GDSC1; CTRP2 6.0452 8.4287 4.8529 5.0066
RERF-LC-A1 CTRP2 6.052 11.7395 3.2032 11.8759
LC-1/sq-SF CTRP2 6.0873 6.8369 5.6833 1.4368
NCI-H2722 GDSC1 6.0975 14.3729 0.6885 19.4434
SW1573 GDSC1 6.1297 8.7054 3.3903 2.8373
HOP-92 GDSC1; CTRP2 6.1437 8.5163 4.8902 4.6631
LC-1/sq GDSC1 6.1524 11.9166 1.9205 12.4817
NCI-H2347 GDSC1 6.1664 15.5632 0.1546 21.6612
NCI-H513 GDSC1 6.1726 8.7677 3.3861 2.7944
NCI-H2342 GDSC1; CTRP2 6.2334 10.6347 3.9048 8.6284
NCI-H1339 CTRP2 6.2385 9.6056 4.4229 6.4497
HCC1171 CTRP2 6.2504 13.8989 2.2875 15.1071
NCI-H2461 GDSC1 6.277 11.9026 2.011 11.5936
NCI-H1092 GDSC1; CTRP2 6.3379 10.7203 3.9463 8.2627
DMS 114 GDSC1; CTRP2 6.444 11.4382 3.6729 9.2061
NCI-H322 CTRP2 6.4657 10.427 4.1935 7.0016
BEN GDSC1; CTRP2 6.489 8.124 5.3478 2.1731
NCI-H1793 GDSC1; CTRP2 6.5232 10.7603 4.0726 7.4047
RERF-LC-Ad1 CTRP2 6.5706 12.4675 3.2601 10.6718
NCI-H2803 GDSC1 6.6033 21.981 -2.6859 29.4168
NCI-H1915 GDSC1; CTRP2 6.6389 13.536 2.7818 12.4642
NCI-H2291 GDSC1; CTRP2 6.6717 10.5915 4.2701 6.3295
NCI-H2172 GDSC1; CTRP2 6.6809 11.4052 3.8742 7.955
NCI-H322M GDSC1 6.7007 16.5607 0.0539 20.6669
T3M-10 CTRP2 6.7816 8.6328 5.3009 1.9556
NCI-H1304 GDSC1 6.8153 8.228 3.8697 0.1646
RERF-LC-Ad2 CTRP2 6.8302 10.1594 4.5993 4.7147
NCI-H2196 GDSC1; CTRP2 6.8571 12.4065 3.5127 9.1406
EKVX GDSC1; CTRP2 7.1807 10.9802 4.4473 4.8102
NCI-H1651 GDSC1; CTRP2 7.2003 11.5178 4.2009 5.7783
HOP-62 GDSC1; CTRP2 7.2109 12.9814 3.4936 8.6328
KNS-62 CTRP2 7.24 11.1784 4.3926 4.9452
SBC-5 GDSC1; CTRP2 7.3091 8.4105 5.6772 0.2577
DMS 79 GDSC1; CTRP2 7.7004 11.3023 4.6339 3.391
Calu-1 CTRP2 7.8759 10.6469 5.0307 1.7667
NCI-H196 GDSC1; CTRP2 7.9552 16.2269 2.4444 11.5399
Hs 888.Lu CTRP2 4.3779 8.3689 3.3112 15.1622
⏷ Show the Full List of 211 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1 4.2599 8.499 2.1815 16.7157
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 1.0322 2.4952 -2.4088 0.108
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 2.0859 8.2698 0.9636 30.1149
A2780 GDSC1; CTRP2 1.682 6.1735 1.2477 30.5121
OVKATE GDSC1 1.7634 7.9652 0.092 39.1607
IGROV-1 GDSC1; CTRP2 3.117 7.1657 2.486 21.7661
OVTOKO GDSC1; CTRP2 3.1189 8.0953 2.1269 23.081
ES-2 GDSC1 3.1743 9.3085 0.8177 29.2179
SNU-840 CTRP2 3.4884 8.1486 2.4924 20.6922
SK-OV-3 GDSC1; CTRP2 3.8933 9.3747 2.3662 20.0889
OC 314 GDSC1; CTRP2 4.2064 7.4363 3.5407 14.7101
Caov-3 GDSC1; CTRP2 4.2357 7.7329 3.4464 14.9992
RMG-I GDSC1; CTRP2 4.3275 11.5939 1.735 21.3326
FU-OV-1 GDSC1; CTRP2 4.3989 10.9463 2.116 19.7667
COV434 CTRP2 4.4007 10.9054 2.1375 19.6816
OAW28 GDSC1; CTRP2 4.5246 10.9598 2.2283 19.0426
SNU-8 CTRP2 4.7205 6.6427 4.4013 9.9797
SNU-119 CTRP2 4.7273 10.2204 2.7779 16.4338
OVCAR-8 GDSC1; CTRP2 4.8001 7.7718 4.0073 11.3117
TOV-21G GDSC1 4.8086 7.8917 2.9246 9.3372
EFO-27 GDSC1; CTRP2 5.1048 8.8412 3.8024 11.4064
MCAS CTRP2 5.1689 8.3096 4.1193 9.9563
OVSAHO CTRP2 5.3127 12.0768 2.3986 16.6004
ONCO-DG-1 CTRP2 5.3448 9.8151 3.5484 11.9128
TOV-112D GDSC1; CTRP2 5.4262 11.5447 2.7635 14.9271
JHOS-2 GDSC1; CTRP2 5.4325 13.3031 1.8933 18.2417
OAW42 GDSC1; CTRP2 5.5461 7.432 4.9015 5.8607
OV7 CTRP2 5.5464 12.543 2.3712 16.2072
DOV13 GDSC1; CTRP2 5.5923 7.4159 4.9531 5.5414
HEY A8 CTRP2 5.8022 10.5926 3.5655 10.8801
COV362 CTRP2 5.8145 10.143 3.8005 9.878
OV-90 GDSC1; CTRP2 5.9346 6.8391 5.5523 2.2906
ES2 CTRP2 5.9944 10.4183 3.8157 9.4571
OV56 GDSC1; CTRP2 6.0386 7.9448 5.0894 4.0254
OVCAR-3 GDSC1 6.4187 8.5641 3.5897 1.3478
JHOM-1 CTRP2 6.423 8.7308 5.0022 3.7022
JHOC-5 CTRP2 6.4305 11.3453 3.7085 9.0832
OVCAR-4 GDSC1; CTRP2 6.4532 11.659 3.5701 9.6144
Caov-4 GDSC1 6.558 9.2882 3.3619 2.3729
OVK18 GDSC1; CTRP2 6.5988 11.5508 3.7385 8.6588
OVCAR-5 GDSC1; CTRP2 6.6087 11.4664 3.7881 8.4361
OVISE GDSC1; CTRP2 6.8061 12.2845 3.5342 9.1398
COV644 CTRP2 7.8304 25.9262 -2.4501 25.6931
TYK-nu GDSC1; CTRP2 8.1059 14.2853 3.4895 7.3081
EFO-21 GDSC1; CTRP2 8.5133 14.5047 3.6522 6.1394
Kuramochi GDSC1; CTRP2 8.5693 17.2718 2.3702 10.8842
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 4.4159 7.8792 3.5686 14.0441
P-STS CTRP2 5.7722 7.6633 4.9982 4.9526
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 5.2962 9.4436 3.6871 11.4474
Aska-SS CTRP2 5.9589 11.8768 3.0567 12.6543
EW-8 GDSC1 1.6156 3.5778 1.5333 34.3256
Hs 633.T GDSC1 3.0919 6.2948 2.1872 21.7185
G-401 GDSC1; CTRP2 3.5768 6.8973 3.0784 18.2336
A-204 GDSC1; CTRP2 3.662 8.287 2.6144 19.7568
Rh41 GDSC1; CTRP2 3.6704 5.1991 3.626 15.9663
SW982 GDSC1; CTRP2 3.8228 7.2839 3.1967 17.0891
Rh18 CTRP2 3.8814 7.8314 3.036 17.545
TE 441.T GDSC1; CTRP2 3.9543 8.381 2.875 17.9737
SK-LMS-1 GDSC1; CTRP2 4.0952 8.8356 2.8148 17.8411
BT-16 CTRP2 4.1169 6.2483 3.8818 13.6717
TTC-709 CTRP2 4.1619 7.322 3.5407 14.8314
G-402 GDSC1; CTRP2 4.3989 7.7537 3.6061 13.9411
TE 617.T CTRP2 4.638 8.1186 3.6867 13.0053
RD GDSC1; CTRP2 4.7823 9.9733 2.9495 15.6224
Rh30 GDSC1 4.8494 6.6842 3.5463 4.4503
Tm87-16 CTRP2 4.9308 10.7808 2.6944 16.2934
GCT GDSC1; CTRP2 5.0424 6.5048 4.798 7.5639
SW872 GDSC1 5.175 8.006 3.1332 6.6823
Hs 729.T CTRP2 5.1844 10.0837 3.2698 13.4097
MFH-ino GDSC1 5.1953 9.2221 2.5561 10.8842
KYM-1 GDSC1; CTRP2 5.4798 6.6907 5.1816 4.8873
VA-ES-BJ GDSC1 5.5469 8.6257 3.0852 6.0831
MES-SA GDSC1; CTRP2 5.5592 6.9616 5.1378 4.8635
SW684 GDSC1 5.9619 7.2113 3.9121 0.3867
HT-1080 GDSC1; CTRP2 6.1511 9.0782 4.6155 5.8032
BT-12 CTRP2 6.2629 7.6652 5.4081 2.2811
SK-UT-1 GDSC1; CTRP2 6.5497 13.479 2.7393 12.7945
RKN GDSC1; CTRP2 7.8527 14.333 3.2932 8.4398
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H GDSC1; CTRP2 2.866 5.7919 2.6413 21.9536
IST-Mes1 GDSC1; CTRP2 3.3853 6.633 2.9627 19.2209
NCI-H2052 GDSC1; CTRP2 4.7582 8.7194 3.5268 13.3519
NCI-H28 GDSC1; CTRP2 4.9906 8.6274 3.7959 11.7006
NCI-H2452 GDSC1; CTRP2 5.8558 9.7595 4.0275 8.8462
MPP 89 GDSC1; CTRP2 5.9553 8.9555 4.514 6.6068
ACC-MESO-1 CTRP2 6.4508 10.528 4.1316 7.2862
JL-1 CTRP2 7.439 17.8991 1.2354 16.682
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
VCaP GDSC1; CTRP2 3.1733 5.8389 2.9647 19.8518
PC-3 GDSC1 4.5829 9.5458 1.9242 17.267
22Rv1 GDSC1; CTRP2 4.8057 9.8191 3.0463 15.1798
DU145 GDSC1; CTRP2 6.0042 11.2963 3.3848 11.2249
LNCaP clone FGC GDSC1; CTRP2 6.1301 12.8369 2.7193 13.668
PaCa-3 CTRP2 7.1771 10.1377 4.8472 3.2197
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 2.1876 5.0407 2.0608 26.1255
A-253 GDSC1; CTRP2 5.83 8.3757 4.6956 6.0972
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1 3.1795 6.5651 2.1482 21.5617
Cancer Drug Sensitivity Data Curated from 43 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RF-48 GDSC1 0.0493 4.2383 -0.3183 52.661
NUGC-4 GDSC1; CTRP2 1.7236 5.9746 1.3479 30.0467
SNU-620 CTRP2 2.2052 3.5963 2.2023 25.5871
HGC-27 GDSC1; CTRP2 2.5855 4.5768 2.5464 23.1752
ECC10 GDSC1; CTRP2 2.6456 6.752 2.1204 24.4903
GSS CTRP2 2.9303 5.2467 2.8257 21.1035
RERF-GC-1B GDSC1 3.286 8.2238 1.4523 25.4463
SNU-16 GDSC1; CTRP2 3.4915 4.6045 3.485 17.0296
IM95 GDSC1; CTRP2 3.6915 7.8509 2.8291 18.8566
SNU-668 CTRP2 3.946 8.2559 2.9212 17.8161
Fu97 GDSC1; CTRP2 4.0046 7.7218 3.2106 16.5364
SNU-719 CTRP2 4.0163 9.0739 2.627 18.7729
ECC12 CTRP2 4.2577 8.0073 3.3502 15.3187
KATO III CTRP2 4.3413 8.8493 3.0549 16.2714
HuG1-N CTRP2 4.5121 10.4318 2.4719 18.1414
SNU-1 GDSC1; CTRP2 4.5865 8.9705 3.2407 14.9229
OCUM-1 GDSC1; CTRP2 4.5903 6.7975 4.2031 11.1007
TMK-1 GDSC1 4.701 9.7809 1.9016 16.9985
GCIY GDSC1 4.7765 7.7252 2.9827 8.9953
NCI-N87 GDSC1; CTRP2 4.8268 7.4311 4.1868 10.5278
23132/87 GDSC1; CTRP2 4.9994 8.7641 3.739 11.9122
KE-39 CTRP2 5.0234 11.8167 2.2687 17.736
NCC-StC-K140 CTRP2 5.2394 18.7555 -0.9939 27.2944
Hs 746.T GDSC1; CTRP2 5.2547 7.3916 4.6366 7.6416
MKN28 GDSC1 5.2606 10.6144 1.9196 15.0396
SNU-5 GDSC1; CTRP2 5.3343 6.4916 5.114 5.5407
MKN74 CTRP2 5.406 9.6943 3.6634 11.3042
TGBC11TKB GDSC1 5.4818 7.6401 3.5008 3.2866
LMSU CTRP2 5.5095 8.5369 4.3284 8.3161
NUGC-3 GDSC1; CTRP2 5.9342 10.7225 2.9085 7.9115
HSC-39 GDSC1 5.9734 7.6485 3.751 1.034
GSU CTRP2 6.0104 6.573 5.7513 1.2992
SH-10-TC CTRP2 6.1499 7.3377 5.4834 2.162
SCH GDSC1 6.1791 7.434 3.9151 0.2711
SNU-216 CTRP2 6.5193 11.0146 3.9432 7.9501
SNU-601 CTRP2 6.5332 7.9043 5.4835 1.5645
MKN45 GDSC1; CTRP2 6.6091 8.9881 5.0125 3.3615
MKN7 GDSC1; CTRP2 7.5121 13.1078 3.6485 7.5401
AGS GDSC1; CTRP2 7.8939 14.0822 3.4429 7.7917
MKN1 GDSC1; CTRP2 8.4577 16.873 2.4855 10.6247
SNG-M GDSC1; CTRP2 3.8674 7.9776 2.9596 17.8776
SNU-1077 CTRP2 4.7836 7.3932 4.1592 10.7498
SNU-685 CTRP2 6.4035 8.8153 4.9457 3.9699
⏷ Show the Full List of 43 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 18 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HTC-C3 GDSC1 0.4222 6.1923 -0.559 49.1956
CGTH-W-1 GDSC1; CTRP2 3.0567 5.2052 2.9687 20.2042
IHH-4 GDSC1 3.0648 5.0453 2.7019 18.2026
B-CPAP GDSC1; CTRP2 3.2086 7.4297 2.4855 21.504
ML-1 [Human leukemia] GDSC1; CTRP2 3.2479 7.1184 2.6441 20.8022
SW579 CTRP2 3.3463 7.2131 2.7147 20.2562
8305C GDSC1; CTRP2 3.9659 6.5781 3.6107 15.1184
BHT-101 GDSC1; CTRP2 4.2681 6.2922 4.0329 12.6674
KMH-2 GDSC1 4.5735 5.9109 3.7261 3.8624
K5 GDSC1 4.6444 8.6736 2.4086 13.7182
FTC-238 CTRP2 5.0317 7.986 4.1394 10.2031
8505C GDSC1; CTRP2 5.0515 9.9045 3.2351 13.85
TT GDSC1; CTRP2 5.0715 7.0917 4.5868 8.3065
ASH-3 GDSC1 5.54 6.9457 3.8325 1.1109
CAL-62 GDSC1; CTRP2 5.7222 8.655 4.4617 7.3014
WRO GDSC1 6.1523 8.621 3.438 2.5129
TT2609-C02 GDSC1; CTRP2 7.7136 16.1225 2.3198 12.3897
FTC-133 GDSC1; CTRP2 7.7668 9.4336 5.4804 0.4967
⏷ Show the Full List of 18 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 54 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 1.4763 4.5928 1.3673 30.7975
SCC-25 GDSC1; CTRP2 2.5813 5.146 2.4669 23.4615
PCI-06A GDSC1 2.6676 8.266 0.845 31.5301
NCI-H3118 GDSC1 3.2094 9.3903 0.8099 29.0941
SNU-1076 CTRP2 3.2788 6.4046 2.9206 19.6911
SNU-1214 CTRP2 3.3558 8.5339 2.1912 22.1817
SCC-9 GDSC1; CTRP2 3.4296 8.2687 2.3806 21.274
BB30-HNC GDSC1 3.4405 7.2579 2.0674 20.8954
JHU-011 GDSC1 3.4466 9.009 1.2141 26.0339
SNU-899 CTRP2 3.4927 6.7203 3.0496 18.5849
SNU-46 CTRP2 3.5598 9.4291 2.0061 22.3078
LB771-HNC GDSC1 3.6732 7.1332 2.3448 17.9287
SNU-1041 CTRP2 3.6837 9.7472 1.9857 22.0533
BICR 18 CTRP2 3.7105 6.6431 3.3119 16.9746
BHY GDSC1; CTRP2 3.7279 7.0838 3.1722 17.449
SAS GDSC1 3.7326 11.0006 0.4797 28.3252
YD-8 CTRP2 3.7585 7.0033 3.235 17.1247
PE/CA-PJ34 (clone C12) CTRP2 3.8207 7.6483 3.0482 17.6633
Ca9-22 GDSC1 3.8689 9.1944 1.4985 22.6469
PCI-38 GDSC1 3.882 8.1914 2.0094 19.3824
CAL-27 GDSC1; CTRP2 4.2426 8.019 3.3296 15.4392
BB49-HNC GDSC1 4.2972 5.9467 3.4889 6.6597
SCC-4 GDSC1; CTRP2 4.3541 7.3807 3.7185 13.6197
BICR 31 GDSC1; CTRP2 4.3756 8.0472 3.4532 14.6055
PCI-04B GDSC1 4.4112 10.1687 1.4726 20.6889
OSC-20 GDSC1 4.4642 10.6021 1.2996 21.4818
KOSC-2 GDSC1 4.5164 7.1834 3.0498 9.3325
PE/CA-PJ49 CTRP2 4.5491 7.0707 4.051 11.7994
SCC-15 GDSC1 4.5554 9.3029 2.0233 16.7094
SKN-3 GDSC1 4.7181 8.7203 2.4436 13.2146
CAL-33 GDSC1; CTRP2 4.8128 9.4195 3.2458 14.359
HSC-3 GDSC1; CTRP2 4.8416 7.6999 4.0818 10.9082
OSC-19 GDSC1 4.9795 11.4413 1.2943 19.7138
SAT [Human HNSCC] GDSC1 5.0264 7.8979 3.0816 7.486
Detroit 562 GDSC1; CTRP2 5.0689 7.4784 4.4112 9.0134
HO-1-N-1 GDSC1 5.0879 10.1737 2.0073 15.0136
HO-1-u-1 GDSC1 5.1537 8.8 2.7326 9.7232
BICR 22 GDSC1; CTRP2 5.3055 6.6386 5.0235 5.97
BICR 16 CTRP2 5.4211 9.1135 3.9638 10.0258
PE/CA-PJ15 GDSC1; CTRP2 5.4367 8.7073 4.1779 9.1024
BICR 78 GDSC1 5.6131 9.9226 2.5109 10.015
BICR 6 CTRP2 5.6188 12.2392 2.5856 15.2236
BICR 56 CTRP2 5.6584 12.6327 2.4233 15.7728
HSC-4 GDSC1; CTRP2 5.8063 9.2267 4.2507 8.0111
HSC-2 GDSC1; CTRP2 6.0219 9.057 4.5193 6.4539
PCI-15A GDSC1 6.2066 8.8767 3.3571 2.917
FaDu GDSC1; CTRP2 6.2388 12.1274 3.1633 11.679
BICR 10 GDSC1 6.281 8.1326 3.6976 0.9828
PE/CA-PJ41 (clone D2) CTRP2 6.327 9.3166 4.6374 5.3903
PCI-30 GDSC1 6.4085 9.7723 3.0764 4.334
KON GDSC1 6.5604 8.2353 3.7736 0.4925
SNU-1066 CTRP2 6.9314 11.4575 4.0368 6.8674
DOK GDSC1 6.9481 11.4752 2.6242 6.2008
JHU-022 GDSC1 6.958 13.1757 1.8517 10.9333
⏷ Show the Full List of 54 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 25 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RT-4 GDSC1; CTRP2 0.8697 6.4902 0.2693 36.2311
JMSU-1 CTRP2 1.6824 4.7878 1.5588 29.4759
U-BLC1 CTRP2 1.9709 6.5525 1.4504 28.9071
253J CTRP2 2.5765 5.1175 2.4666 23.4781
UM-UC-1 CTRP2 2.7414 6.6302 2.2643 23.6855
5637 GDSC1; CTRP2 2.7453 6.1648 2.4104 23.1492
RT-112 GDSC1; CTRP2 2.9828 5.8714 2.7488 21.2098
BC-3C CTRP2 4.0953 12.4145 1.1181 24.015
BFTC-905 GDSC1 4.4566 6.8838 3.1514 8.7462
SCaBER CTRP2 4.4804 10.2149 2.546 17.9306
KMBC-2 CTRP2 4.5077 9.3431 2.9879 16.1254
647V GDSC1; CTRP2 4.8046 9.4669 3.2151 14.5022
VM-CUB-1 CTRP2 4.8216 11.2409 2.3679 17.8149
253J-BV CTRP2 4.8834 9.5866 3.2323 14.2477
SW1710 GDSC1; CTRP2 5.0423 8.9177 3.7061 11.9463
SW780 GDSC1 5.1158 8.1655 3.0148 7.7334
UM-UC-3 GDSC1; CTRP2 5.1332 8.614 3.939 10.7797
TCCSUP GDSC1; CTRP2 5.1711 9.6906 3.4507 12.6997
639V GDSC1; CTRP2 5.3433 7.6271 4.6131 7.5219
J82 GDSC1; CTRP2 5.6566 7.9952 4.7295 6.324
HT-1197 GDSC1; CTRP2 5.7385 6.8196 5.3795 3.4472
HT-1376 GDSC1; CTRP2 5.848 9.8403 3.9804 9.0587
T24 GDSC1; CTRP2 5.9475 12.3755 2.7977 13.7163
KU-19-19 GDSC1; CTRP2 6.005 9.0794 4.494 6.5931
CAL-29 GDSC1; CTRP2 6.5796 11.0555 3.9697 7.7344
⏷ Show the Full List of 25 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PA-1 GDSC1 -0.7052 1.8765 -0.7373 61.9153
C-33 A GDSC1 0.9574 8.4609 -0.9472 45.8241
Ca Ski GDSC1 1.814 7.0065 0.5711 37.3682
ME-180 GDSC1 1.865 5.4248 1.2753 34.0796
LB831-BLC GDSC1 2.017 5.4401 1.4322 32.3105
KGN GDSC1 2.4256 6.5508 1.3983 30.1008
SW954 GDSC1 2.4507 5.4155 1.9038 26.9736
NEC8 GDSC1 2.4558 4.9466 2.0862 25.7609
BPH-1 GDSC1 2.5439 4.8397 2.2189 24.3799
OVMIU GDSC1 3.4059 10.1598 0.6083 29.1282
CAL-39 GDSC1 3.6838 6.3669 2.7288 15.0476
SW962 GDSC1 4.0518 7.6886 2.4086 15.9047
DSH1 GDSC1 4.1881 5.8463 3.4455 7.4119
OVCA420 GDSC1 4.2639 5.4821 3.6928 5.1755
ACC-OV7 GDSC1 4.2943 7.9174 2.5011 14.297
UWB1.289 GDSC1 4.3804 11.2948 0.8841 23.9752
OMC-1 [Human cervical carcinoma] GDSC1 4.4028 9.0237 2.0381 17.1636
SiSo GDSC1 4.4598 11.0745 1.0598 22.792
JAR GDSC1 4.559 8.7934 2.2806 14.9279
HEY GDSC1 4.5631 9.4481 1.957 17.1221
PEO1 GDSC1 4.6006 8.0598 2.6798 11.874
HT-3 GDSC1 4.8033 11.4329 1.1592 21.0508
C-4-I GDSC1 4.906 9.0995 2.4007 12.9001
HeLa GDSC1; CTRP2 4.9973 7.2195 4.4545 9.0236
DoTc2 4510 GDSC1 5.128 10.1106 2.0689 14.4774
MS751 GDSC1 5.4167 8.8654 2.8851 7.8667
NCC-IT GDSC1 5.6846 7.7913 3.5481 2.5909
OVCA433 GDSC1 5.7501 10.1759 2.4826 9.8441
SW756 GDSC1 5.9053 8.1681 3.503 2.5051
SKG-IIIa GDSC1 6.0823 7.9599 3.6768 1.2813
JHOS-3 GDSC1 6.0974 13.6195 1.0569 17.5945
NT2-D1 GDSC1 6.1978 19.393 -1.7131 27.9664
HEC-1 GDSC1 6.2905 7.6417 3.8833 0.3068
SiHa GDSC1 6.3636 7.6837 3.8955 0.247
JEG-3 GDSC1 6.7195 8.4231 3.7671 0.4303
SKN GDSC1 7.1362 9.3228 3.6031 0.7144
OV17R GDSC1 7.6872 21.6299 -1.713 24.4685
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug

References

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