General Information of Drug (ID: DMBK9AM)

Drug Name
PLX-4720
Synonyms PLX 4720; PLX4720 (BRAF inhibitor)
Indication
Disease Entry ICD 11 Status REF
Cutaneous melanoma 2C30 Phase 1 [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 413.8
Logarithm of the Partition Coefficient (xlogp) 3.3
Rotatable Bond Count (rotbonds) 6
Hydrogen Bond Donor Count (hbonddonor) 2
Hydrogen Bond Acceptor Count (hbondacc) 7
Chemical Identifiers
Formula
C17H14ClF2N3O3S
IUPAC Name
N-[3-(5-chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonyl)-2,4-difluorophenyl]propane-1-sulfonamide
Canonical SMILES
CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=C2C=C(C=N3)Cl)F
InChI
InChI=1S/C17H14ClF2N3O3S/c1-2-5-27(25,26)23-13-4-3-12(19)14(15(13)20)16(24)11-8-22-17-10(11)6-9(18)7-21-17/h3-4,6-8,23H,2,5H2,1H3,(H,21,22)
InChIKey
YZDJQTHVDDOVHR-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
24180719
ChEBI ID
CHEBI:90295
CAS Number
918505-84-7
UNII
EQY31RO8HA
DrugBank ID
DB06999
TTD ID
D0F5JZ
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
B-Raf messenger RNA (BRAF mRNA) TT0EOB8 BRAF_HUMAN Inhibitor [2]
Vascular endothelial growth factor receptor 2 (KDR) TTUTJGQ VGFR2_HUMAN Inhibitor [3]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Heat shock factor protein 1 (HSF1) OTYNJ4KP HSF1_HUMAN Gene/Protein Processing [4]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Cutaneous melanoma
ICD Disease Classification 2C30
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
B-Raf messenger RNA (BRAF mRNA) DTT BRAF 1.56E-01 -0.23 -0.43
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1; GDSC2 6.1918 8.127 2.6947 0.3334
EW-12 GDSC2 3.2727 4.8901 2.4965 5.3709
NOS-1 [Human HNSCC] GDSC1; GDSC2 3.4016 6.4457 1.826 9.2327
CHSA8926 GDSC1; GDSC2 3.573 5.9465 2.2126 6.3263
ES1 GDSC1; GDSC2 3.8666 6.3805 2.2194 5.5467
CHSA0011 GDSC1; GDSC2 3.8779 6.3845 2.2256 5.481
ES5 GDSC1; GDSC2 4.0812 9.2874 0.9459 12.7194
CHSA0108 GDSC1; GDSC2 4.4095 7.0382 2.2731 4.0634
EW-24 GDSC1; GDSC2 4.4297 7.2517 2.1858 4.5361
TC-71 GDSC1; GDSC2; CCLE 4.4348 6.9565 2.3272 3.0836
ES4 GDSC1; GDSC2 4.5247 7.4493 2.1538 4.5397
EW-22 GDSC1; GDSC2 4.5273 6.6095 2.5408 2.3496
EW-1 GDSC1; GDSC2 4.5394 6.9443 2.3967 3.1217
EW-18 GDSC1; GDSC2 4.5582 10.0488 0.9249 11.6561
ES7 GDSC1; GDSC2 4.5899 7.0874 2.3615 3.2331
U-CH2 GDSC2 4.649 8.5659 1.7064 6.9211
ES6 GDSC1; GDSC2 4.696 7.3922 2.2859 3.4766
EW-11 GDSC1; GDSC2 4.7128 9.0244 1.53 7.822
SK-ES-1 GDSC1; GDSC2; CTRP2; CCLE 4.7382 8.6784 2.9663 9.3413
CAL-72 GDSC1; GDSC2 4.778 10.575 0.8256 11.6942
CADO-ES1 GDSC1; GDSC2 4.8502 10.0022 1.1537 9.6952
HuO9 GDSC1; GDSC2 4.8775 8.8285 1.732 6.3107
EW-3 GDSC1; GDSC2 4.9325 7.3766 2.4273 2.3562
EW-16 GDSC1; GDSC2 5.0205 8.8425 1.8161 5.5583
A-673 GDSC1; GDSC2; CTRP2; CCLE 5.1079 9.2518 2.9934 8.4951
EW-13 GDSC1; GDSC2 5.1173 7.817 2.3354 2.5713
SK-N-MC CTRP2 5.2046 6.9658 4.2137 3.1945
Hs 822.T CTRP2 5.3018 7.3526 4.0971 3.5119
SK-PN-DW GDSC1; GDSC2 5.3047 10.0185 1.4466 7.1133
EW-7 GDSC1; GDSC2 5.329 8.8009 2.0191 3.9159
NY GDSC1; GDSC2 5.4152 11.3733 0.8787 10.02
HuO-3N1 GDSC1; GDSC2 5.4583 10.188 1.4639 6.7328
Hs 888.T CTRP2 5.4767 7.8569 3.9801 3.7052
ES8 GDSC1; GDSC2 5.5212 7.2266 2.7614 0.4451
U2OS GDSC1; GDSC2; CCLE 5.5725 7.495 2.6827 0.5381
SaOS-2 GDSC1; GDSC2; CTRP2; CCLE 5.6045 8.8663 3.5778 5.1642
MG-63 GDSC1; GDSC2; CTRP2; CCLE 5.7674 8.0941 4.0719 2.8851
TC71 CTRP2 5.787 8.6272 3.8278 3.8458
SJSA-1 GDSC1; GDSC2; CTRP2; CCLE 5.7941 7.6649 4.2939 1.9672
MHH-ES-1 GDSC1; GDSC2; CTRP2; CCLE 5.8447 7.934 4.1997 2.2705
HOS GDSC1; GDSC2; CTRP2; CCLE 5.8609 7.6712 4.333 1.7329
SW1353 CTRP2; CCLE 6.0538 7.569 4.4909 0.9561
CAL-78 GDSC1; GDSC2; CTRP2; CCLE 6.0584 10.523 3.0973 6.4173
G-292 clone A141B1 GDSC1; GDSC2; CTRP2 6.3287 10.3965 3.3482 4.9968
H-EMC-SS GDSC1; GDSC2 6.4756 8.6604 2.6121 0.4099
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 223 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 4.4809 6.0236 4.0316 5.4863
MEC1 CTRP2 4.7585 6.3485 4.1411 4.3873
JM1 GDSC1; GDSC2; CTRP2 5.4222 6.8689 4.4246 1.96
SIG-M5 GDSC2; CTRP2; CCLE -1.0421 1.9825 -1.0748 40.6444
OCI-Ly7 GDSC1; GDSC2 1.772 3.9133 1.4387 17.3667
EoL-1 GDSC1; GDSC2; CTRP2 1.8698 3.731 1.8308 21.2812
BC-3 GDSC2 2.5256 4.7264 1.8811 11.7354
JVM-3 GDSC1; GDSC2; CCLE 2.5427 5.6102 1.4776 11.7877
MOLM-16 GDSC1; GDSC2; CTRP2 2.6639 4.972 2.4659 16.5498
JVM-2 GDSC1; GDSC2; CTRP2 3.0644 5.4752 2.4273 9.8709
NCO2 CTRP2; CCLE 3.2048 6.3447 2.5766 14.5753
Peer CTRP2 3.2475 4.6899 3.1676 12.2456
Pfeiffer CTRP2; CCLE 3.2722 5.0756 3.1017 12.4038
697 GDSC1; GDSC2; CTRP2; CCLE 3.3768 6.2082 2.8135 13.1892
BONNA-12 GDSC2 3.3938 7.1353 1.4748 11.4411
CMK-86 CCLE 3.4071 5.5064 2.0678 4.1241
Mono-Mac-1 CTRP2; CCLE 3.4315 5.4648 3.1537 11.7399
NU-DUL-1 GDSC1; GDSC2; CTRP2 3.5531 5.772 3.1731 11.3193
MEC-1 CCLE 3.574 7.1092 1.402 7.3246
DoHH2 GDSC1; GDSC2; CCLE 3.6301 6.171 2.1454 5.4964
P30/OHK GDSC1; GDSC2 3.6325 5.8766 2.2933 5.6636
MV4-11 GDSC1; GDSC2; CTRP2 3.6409 5.6828 3.3009 10.5858
KE-97 CTRP2; CCLE 3.6533 6.2094 3.1029 11.316
BE-13 GDSC1; GDSC2 3.6822 9.3173 0.6189 15.6395
MEG-01 GDSC1; GDSC2; CCLE 3.7089 5.3736 2.598 2.976
SUP-B8 GDSC1; GDSC2 3.7768 8.1229 1.2892 11.5046
BC-1 GDSC1; GDSC2 3.7992 6.0737 2.3207 5.0787
NU-DHL-1 CTRP2 3.8777 10.1603 1.4592 17.334
KYO-1 CTRP2 3.9004 6.2819 3.3277 9.7782
SKM-1 GDSC1; GDSC2; CTRP2 3.904 6.4188 3.2711 9.9935
JURL-MK1 GDSC1; GDSC2; CTRP2 3.9218 5.586 3.6381 8.5119
TALL-1 [Human adult T-ALL] GDSC2; CTRP2 3.9385 6.8051 3.131 10.467
CML-T1 GDSC1; GDSC2; CTRP2 3.952 5.9963 3.5041 8.9474
P32/ISH GDSC1; GDSC2 3.9669 5.6071 2.6618 2.6345
ALL-SIL GDSC1; GDSC2; CCLE 3.9774 6.1281 2.4204 3.3814
Ku812 GDSC1; GDSC2; CTRP2; CCLE 3.9849 5.869 3.5919 8.5162
NK-92MI GDSC2 3.994 8.1421 1.4465 9.9905
SU-DHL-5 GDSC1; GDSC2 3.9999 5.467 2.748 2.0715
CTB-1 GDSC1; GDSC2 4.0016 9.1997 0.9285 13.027
LAMA-84 GDSC1; GDSC2; CTRP2 4.003 6.6294 2.7455 6.2014
HC-1 GDSC1; GDSC2 4.0063 6.0451 2.4798 3.6397
SU-DHL-16 GDSC1; GDSC2 4.0151 5.7284 2.6357 2.6943
IM-9 GDSC1; GDSC2 4.0243 5.9807 2.5225 3.3466
CESS GDSC1; GDSC2 4.0289 6.8887 2.0878 5.9788
KG-1 GDSC1; GDSC2; CCLE 4.032 6.5984 2.2311 4.2428
MLMA GDSC1; GDSC2 4.0579 6.7381 2.1815 5.3387
EM-2 GDSC1; GDSC2; CTRP2; CCLE 4.0883 5.8115 3.7241 7.7225
Jurkat GDSC1; GDSC2; CTRP2; CCLE 4.0906 6.473 2.8973 5.3366
BV-173 GDSC1; GDSC2; CTRP2 4.0925 7.6771 2.8698 11.1587
DB GDSC1; GDSC2; CTRP2 4.1363 7.2171 3.1322 9.9808
Loucy GDSC1; GDSC2 4.1544 7.3903 1.9329 6.6396
WIL2 NS GDSC1; GDSC2 4.1773 5.7852 2.709 1.987
YT GDSC1; GDSC2 4.2261 6.4474 2.4331 3.4775
A4/Fukuda GDSC1; GDSC2; CTRP2 4.2403 6.0117 3.7948 7.0434
KMS-34 CTRP2; CCLE 4.2485 5.7103 3.9339 6.473
MOLT-16 GDSC1; GDSC2; CTRP2; CCLE 4.2529 6.7192 3.4816 8.2753
U-698-M GDSC1; GDSC2 4.2533 6.6694 2.3462 3.9362
MY-M12 GDSC1; GDSC2 4.293 7.5615 1.9467 6.2464
KOPN-8 GDSC1; GDSC2 4.2941 6.4012 2.4973 2.9792
QIMR-WIL GDSC1; GDSC2 4.3003 8.2725 1.607 8.2797
Sc-1 GDSC1 4.3151 5.7123 2.8177 1.5137
ATN-1 GDSC1; GDSC2 4.3263 9.4205 1.0638 11.4245
ALL-PO GDSC1; GDSC2 4.3335 9.7839 0.8903 12.3966
OCI-Ly19 GDSC1; GDSC2 4.3348 9.8108 0.8781 12.4622
EB2 GDSC1; GDSC2; CCLE 4.3351 6.5916 2.4345 2.7198
HDLM-2 GDSC1; GDSC2; CTRP2 4.3486 7.7282 3.0862 9.6795
Karpas-231 GDSC1; GDSC2 4.3816 5.8658 2.7868 1.2828
JSC-1 GDSC1; GDSC2 4.3821 6.4854 2.5121 2.7421
MHH-CALL-2 GDSC1; GDSC2 4.3849 6.6399 2.4429 3.1283
RPMI-8866 GDSC1; GDSC2 4.3991 11.8746 -0.0932 17.3819
SCC-3 GDSC2 4.4018 5.6391 2.8917 0.7749
MOLM-13 GDSC1; GDSC2; CTRP2 4.4152 6.2481 3.8621 6.3345
WSU-DLCL2 GDSC1; GDSC2; CTRP2 4.4202 7.3391 3.3428 8.4559
Ri-1 CTRP2 4.429 7.3892 3.3265 8.5034
Ki-JK CTRP2 4.4398 5.9413 4.0285 5.6013
WSU-NHL GDSC1; GDSC2 4.44 7.2417 2.1971 4.4498
SUP-T11 CTRP2 4.4409 5.9441 4.0283 5.5994
Mino CTRP2; CCLE 4.4471 7.3773 3.3492 8.3685
KMOE-2 GDSC1; GDSC2 4.4486 6.9402 2.3433 3.584
EB1 CCLE 4.4626 6.6714 2.1922 1.8112
CRO-AP2 GDSC1; GDSC2 4.4943 6.3288 2.6465 1.8399
Kasumi-1 GDSC1; GDSC2; CTRP2 4.4958 7.0396 3.5594 7.3885
LC4-1 GDSC1; GDSC2 4.5094 7.0362 2.3364 3.5147
BL-70 CTRP2; CCLE 4.5542 5.2894 4.4271 3.7292
GR-ST GDSC1; GDSC2 4.5687 11.5009 0.2193 15.41
Farage GDSC1; GDSC2 4.5754 8.4735 1.7011 7.1075
KM-H2 GDSC1; GDSC2; CTRP2 4.5799 5.9952 3.5062 1.7521
Mono-Mac-6 GDSC1; GDSC2; CTRP2 4.5822 8.544 2.8959 9.9608
Hs 445 GDSC1; GDSC2 4.5904 6.5862 2.5863 2.0155
HL-60 GDSC1; GDSC2 4.5927 6.0915 2.7981 0.9877
TUR GDSC1; GDSC2 4.6067 10.3717 0.802 12.226
HAL-01 GDSC1; GDSC2 4.6078 8.1096 1.8962 5.8877
DG-75 GDSC1; GDSC2 4.6235 8.1874 1.8696 6.0125
KE-37 GDSC1; GDSC2; CTRP2 4.6379 7.4327 3.4966 7.3352
L-428 GDSC1; GDSC2; CTRP2; CCLE 4.6392 7.1652 3.6299 6.7767
RC-K8 GDSC1; GDSC2 4.6429 7.9901 1.9755 5.353
VL51 GDSC1; GDSC2 4.6524 6.9959 2.4395 2.7025
KY821 GDSC1; GDSC2 4.6605 6.9594 2.4604 2.5771
KMS-12-BM GDSC2; CTRP2; CCLE 4.6634 7.7625 3.3561 7.8676
MOLT-4 GDSC1; GDSC2 4.6682 8.6138 1.6964 6.9402
Karpas-299 GDSC1; GDSC2; CTRP2; CCLE 4.6795 6.6719 3.9096 5.5243
SUP-M2 GDSC1; GDSC2; CTRP2; CCLE 4.6819 5.8351 4.3175 3.8356
HD-MY-Z CTRP2; CCLE 4.6912 8.1725 3.1771 8.5575
GDM-1 GDSC1; GDSC2; CTRP2 4.6965 6.3535 4.0814 4.7735
L-540 GDSC1; GDSC2; CTRP2 4.7014 7.0782 3.7292 6.2282
HH [Human lymphoma] GDSC1; GDSC2; CTRP2; CCLE 4.7074 6.8247 3.8598 5.6702
ARH-77 GDSC1; GDSC2 4.7263 7.4839 2.2622 3.5581
H9 GDSC1; GDSC2 4.73 7.4413 2.2837 3.4318
K-562 GDSC1; GDSC2; CTRP2 4.731 6.1161 4.2293 4.0832
BALL-1 GDSC1; GDSC2 4.7429 7.0433 2.4695 2.4058
CCRF-CEM GDSC1; GDSC2 4.7812 8.076 2.023 4.8163
JM-1 CCLE 4.7899 6.4071 2.4582 0.5325
PL-21 GDSC1; GDSC2 4.8215 9.809 1.2271 9.3399
Karpas-45 GDSC1; GDSC2 4.8245 7.1085 2.4856 2.207
Daudi GDSC1; GDSC2; CTRP2 4.8276 6.1755 4.2893 3.6188
Kasumi-2 CTRP2; CCLE 4.844 7.943 3.4249 7.204
MHH-PREB-1 GDSC1; GDSC2 4.8445 6.7278 2.6582 1.345
Hs 611.T CTRP2 4.8652 7.4622 3.6831 6.0776
GA-10 GDSC1; GDSC2; CTRP2 4.8739 6.9795 3.9313 5.0188
RCH-ACV GDSC1; GDSC2; CTRP2 4.8809 7.2716 3.7918 5.5894
M-07e CTRP2 4.8817 11.376 1.742 14.0691
KMS-20 CTRP2 4.8957 15.9157 -0.5156 21.9765
KMM-1 CCLE 4.9477 7.33 2.1621 1.4291
Ramos.2G6.4C10 GDSC1; GDSC2 4.9525 9.5994 1.416 7.9805
VAL GDSC1; GDSC2 4.9601 6.9602 2.6187 1.3978
CTV-1 GDSC1; GDSC2 4.9665 6.6026 2.766 0.7787
MN-60 GDSC1; GDSC2 4.9883 7.4549 2.4233 2.301
BDCM CCLE 4.9934 7.4929 2.1169 1.5619
SU-DHL-6 GDSC1; GDSC2; CTRP2; CCLE 5.0282 7.1467 3.9797 4.5065
RPMI-8402 GDSC1; GDSC2; CTRP2; CCLE 5.0729 7.2697 3.9554 4.5228
MOTN-1 CTRP2 5.0739 6.8141 4.184 3.5599
THP-1 GDSC1; GDSC2 5.0768 6.9324 2.6853 0.9996
RPMI-6666 GDSC1; GDSC2; CTRP2 5.0797 7.1316 4.03 4.196
MOLM-6 CTRP2 5.086 6.8514 4.1753 3.5736
NALM-6 GDSC1; GDSC2; CTRP2 5.0897 7.4222 3.893 4.753
LP-1 GDSC1; GDSC2; CTRP2; CCLE 5.096 6.2778 4.4702 2.3158
AML-193 CTRP2 5.1008 6.7039 4.2612 3.1849
Toledo CTRP2; CCLE 5.1037 10.893 2.1694 11.9133
KCL-22 GDSC1; GDSC2; CTRP2; CCLE 5.1145 6.4971 4.3756 2.6786
SET-2 CTRP2 5.1323 6.3549 4.4609 2.2883
OCI-Ly3 CTRP2 5.1529 6.5388 4.3856 2.5669
EHEB GDSC1; CTRP2 5.1571 8.3783 3.4704 6.4015
ME1 GDSC1; GDSC2 5.1684 6.392 2.9259 0.1992
HT GDSC1; GDSC2; CTRP2; CCLE 5.1748 7.0909 4.1277 3.609
BL-41 GDSC1; GDSC2; CTRP2; CCLE 5.1786 7.6878 3.8328 4.8396
TK [Human B-cell lymphoma] GDSC1; GDSC2 5.1953 6.7358 2.8121 0.4702
ML-2 GDSC1; GDSC2 5.2033 7.2115 2.6319 1.1017
KMS-26 CTRP2; CCLE 5.207 6.2629 4.5648 1.723
MJ CCLE 5.2101 7.7099 2.1327 1.3087
P31/FUJ GDSC1; GDSC2; CTRP2; CCLE 5.2404 7.1505 4.1499 3.3984
TF-1 CTRP2 5.2487 7.2143 4.1247 3.489
Namalwa GDSC1; GDSC2; CTRP2 5.2741 8.73 3.3894 6.5252
KO52 CTRP2; CCLE 5.2789 6.4676 4.5175 1.8012
KMS-21-BM CTRP2 5.29 6.7044 4.4091 2.2321
NOMO-1 GDSC1; GDSC2; CTRP2 5.2965 6.3877 4.5695 1.5591
HEL 92.1.7 CTRP2; CCLE 5.3241 6.6907 4.4411 2.0444
PF-382 GDSC1; GDSC2; CTRP2 5.3251 7.376 4.1034 3.4455
Reh GDSC1; GDSC2; CTRP2; CCLE 5.3343 8.0525 3.7746 4.8037
SU-DHL-1 GDSC2; CTRP2 5.3396 7.5921 4.0075 3.821
SU-DHL-8 GDSC1; GDSC2; CTRP2; CCLE 5.3564 8.2251 3.706 5.0518
OCI-AML-2 GDSC1; GDSC2; CTRP2; CCLE 5.3615 8.561 3.5428 5.7254
SU-DHL-10 GDSC1; GDSC2; CTRP2; CCLE 5.3641 9.0656 3.2936 6.7634
PL21 CTRP2 5.3914 7.2798 4.201 2.929
Jiyoye GDSC1; GDSC2 5.3972 9.8638 1.5762 6.2221
Karpas-1106P GDSC1; GDSC2 5.4066 7.1793 2.7328 0.5891
U266B1 GDSC1; GDSC2; CTRP2 5.4114 8.096 3.8126 4.5111
P12-Ichikawa GDSC1; GDSC2; CTRP2; CCLE 5.4125 7.4073 4.1539 3.0898
ST486 GDSC1; GDSC2; CTRP2 5.4388 7.2289 4.2608 2.606
RS4;11 GDSC1; GDSC2; CTRP2 5.478 8.6935 3.5674 5.4198
OCI-AML-3 GDSC1; GDSC2; CTRP2 5.4839 6.6425 4.5752 1.2677
L-1236 GDSC1; GDSC2; CTRP2 5.4913 10.5062 2.6764 9.1063
KHM-1B CTRP2; CCLE 5.5028 6.966 4.4335 1.8061
OCI-M1 GDSC1; GDSC2; CTRP2 5.5031 7.5823 4.1344 3.0253
MOLT-3 CTRP2 5.504 6.7863 4.5202 1.4581
MHH-CALL-4 GDSC2; CTRP2 5.5259 8.5993 3.6506 4.9923
RPMI-8226 GDSC1; GDSC2; CTRP2 5.5297 8.1517 3.8743 4.057
F-36P CTRP2; CCLE 5.565 10.0516 2.9603 7.7986
OPM-2 GDSC1; GDSC2; CTRP2; CCLE 5.5802 6.9266 4.5035 1.4234
U-937 CTRP2; CCLE 5.5893 7.88 4.0511 3.2336
Raji GDSC1; GDSC2; CTRP2; CCLE 5.6075 6.9766 4.4976 1.4118
Karpas-620 GDSC1; GDSC2; CTRP2; CCLE 5.6304 7.3279 4.3463 1.9772
JeKo-1 GDSC1; GDSC2; CTRP2 5.6528 10.1472 2.9806 7.5625
SEM CTRP2 5.6635 7.8164 4.1342 2.7832
SU-DHL-4 GDSC1; GDSC2; CTRP2; CCLE 5.678 9.1398 3.4978 5.375
CMK GDSC1; CTRP2 5.7095 6.8652 4.6104 0.8715
REC-1 CTRP2 5.721 8.5294 3.8285 3.9436
MHH-CALL-3 CTRP2 5.7294 9.238 3.4875 5.3343
CA46 GDSC1; GDSC2; CTRP2 5.7581 9.4546 3.4022 5.6405
SUP-B15 GDSC1; GDSC2; CTRP2 5.7635 7.5439 4.3311 1.8612
KMS-11 GDSC1; GDSC2; CTRP2; CCLE 5.7651 8.3698 3.9373 3.4327
HuT 78 CTRP2; CCLE 5.7857 7.7171 4.2638 2.0958
MOLT-13 GDSC1; GDSC2; CTRP2 5.7886 7.3032 4.4584 1.3432
NB4 GDSC1; GDSC2; CTRP2 5.8241 8.571 3.881 3.5744
SR GDSC1; GDSC2; CTRP2 5.8447 10.7114 2.8471 7.7903
Ci-1 CTRP2; CCLE 5.8573 6.8712 4.6866 0.4872
KMS-18 CTRP2 5.9296 7.4325 4.4824 1.1041
SUP-T1 GDSC1; GDSC2; CTRP2; CCLE 5.9378 8.3431 4.067 2.6702
P3HR-1 CTRP2; CCLE 5.9745 8.3097 4.1065 2.4668
MC116 GDSC1; GDSC2; CTRP2; CCLE 5.9873 11.0636 2.7799 7.8309
SUP-HD1 GDSC1; GDSC2; CTRP2 6.0146 8.1915 4.1872 2.1047
RL GDSC1; GDSC2; CTRP2 6.0689 8.7384 3.9655 2.897
HEL GDSC1; GDSC2; CTRP2 6.0791 9.6587 3.5322 4.6143
ROS-50 GDSC1; GDSC2 6.0919 8.358 2.5725 0.6825
A3/Kawakami GDSC1; GDSC2; CTRP2 6.1611 9.5723 3.6299 4.1041
NCI-H929 GDSC1; GDSC2; CTRP2 6.1682 8.319 4.2218 1.7969
KMS-27 CTRP2 6.1862 7.6772 4.5137 0.7708
DEL GDSC1; GDSC2; CTRP2; CCLE 6.2275 10.8871 3.0407 6.3878
NKM-1 GDSC1; GDSC2 6.2304 8.2321 2.6719 0.368
HPB-ALL CTRP2 6.2466 8.0381 4.3909 1.1197
L-363 GDSC1; GDSC2; CTRP2; CCLE 6.2478 10.0135 3.4771 4.5944
Karpas-422 GDSC1; GDSC2; CTRP2; CCLE 6.4271 7.7683 4.5904 0.4017
JJN-3 GDSC1; GDSC2; CTRP2 6.5085 7.8145 4.6076 0.3236
EJM GDSC1; GDSC2; CTRP2 6.5929 8.1801 4.5025 0.5335
AMO1 GDSC1; GDSC2; CTRP2; CCLE 6.6123 8.3206 4.4554 0.6472
Granta-519 GDSC1; GDSC2; CTRP2; CCLE 6.9526 8.6885 4.4623 0.4504
OCI-AML-5 GDSC1; GDSC2; CTRP2; CCLE 6.9882 7.8882 4.7587 0.0236
SK-MM-2 GDSC1; GDSC2; CTRP2; CCLE 7.1229 8.9347 4.4403 0.4249
MOLP-2 CTRP2 7.2215 9.0245 4.4472 0.372
ME1 CTRP2 7.2612 8.6743 4.5885 0.1343
MOLP-8 GDSC1; GDSC2; CTRP2; CCLE 7.2792 8.6408 4.6065 0.1106
MM1.S GDSC1; GDSC2; CTRP2 7.3783 8.6306 4.6446 0.0628
DND-41 GDSC1; GDSC2; CTRP2 7.5934 9.0762 4.5689 0.1018
OCI-Ly10 CTRP2; CCLE 8.3137 9.9602 4.5202 0.0632
⏷ Show the Full List of 223 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 5.1936 6.9001 4.2377 3.1136
TE15 CTRP2 5.9849 9.83 3.3829 5.363
T.T GDSC1; GDSC2 3.8298 6.5384 2.1148 6.2845
TE-15 GDSC1; GDSC2; CCLE 4.0544 7.3896 1.8616 6.0947
KYSE-140 GDSC1; GDSC2; CTRP2; CCLE 4.4845 7.4988 3.3242 8.3887
KYSE-270 GDSC1; GDSC2 4.4971 6.5132 2.5666 2.2574
TE-8 GDSC1; GDSC2 4.862 7.744 2.2243 3.5429
KYSE-70 GDSC1; GDSC2; CTRP2; CCLE 5.0484 7.3073 3.9163 4.734
EC-GI-10 GDSC1; GDSC2; CTRP2 5.0881 7.1254 4.0401 4.1379
TE-10 GDSC1; GDSC2; CTRP2 5.1364 7.0998 4.0923 3.8278
TE-11 GDSC1; GDSC2; CTRP2 5.1734 8.82 3.263 7.2412
TE-6 GDSC1; GDSC2; CTRP2 5.1747 7.9102 3.7186 5.3263
KYSE-410 GDSC1; GDSC2; CTRP2; CCLE 5.221 7.1348 4.1425 3.4635
TE-5 GDSC1; GDSC2; CTRP2; CCLE 5.4801 7.8645 3.9789 3.7045
TE-14 CTRP2 5.5268 7.9496 3.9716 3.6594
TE-9 GDSC1; GDSC2; CTRP2; CCLE 5.5974 7.9094 4.0425 3.2561
COLO 680N GDSC1; GDSC2; CTRP2 5.6841 7.3192 4.3857 1.7498
KYSE-520 GDSC1; GDSC2; CTRP2; CCLE 5.7127 9.0466 3.5693 5.0233
TE-1 GDSC1; GDSC2; CTRP2; CCLE 5.7696 8.2636 3.9917 3.2055
OE33 GDSC1; GDSC2; CTRP2; CCLE 5.9501 7.9218 4.2722 1.8578
KYSE-450 GDSC1; GDSC2; CTRP2; CCLE 6.1157 7.7987 4.4243 1.1261
KYSE-180 GDSC1; GDSC2; CTRP2; CCLE 6.1621 8.8574 3.9694 2.7618
TE-4 GDSC1; GDSC2; CTRP2 6.3401 8.1608 4.3875 1.0494
OE19 GDSC1; GDSC2; CTRP2 6.8989 8.1872 4.6257 0.1618
OE21 GDSC1; GDSC2; CTRP2; CCLE 6.9614 11.3244 3.3219 4.2662
KYSE-30 CTRP2; CCLE 7.2757 12.0099 3.1988 4.3564
KYSE-150 GDSC1; GDSC2; CTRP2; CCLE 7.3572 10.8268 3.7771 2.1875
KYSE-510 GDSC1; GDSC2; CTRP2; CCLE 7.9478 15.0543 2.2027 7.281
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 5.9323 8.1963 4.1328 2.4187
PK-1 CCLE 3.7012 5.9315 2.0694 3.5414
KP-1NL CCLE 4.1708 7.4302 1.6682 4.7679
BxPC-3 GDSC1; GDSC2; CTRP2; CCLE 4.2491 7.5844 3.063 10.0014
HuP-T4 GDSC1; GDSC2; CTRP2; CCLE 4.471 6.3781 3.8552 6.2278
HPAC GDSC1; GDSC2; CTRP2; CCLE 4.4776 7.7757 3.1817 8.9962
MZ-PC-1 GDSC1; GDSC2 4.5582 9.077 1.3982 8.932
SW1990 GDSC1; GDSC2; CTRP2; CCLE 4.6042 7.6056 3.3807 7.8918
KCI-MOH1 CCLE 4.7516 7.606 1.9409 2.5753
KP-1N GDSC1; GDSC2; CCLE 4.8697 8.8039 1.7385 5.2531
Hs 766T GDSC1; GDSC2; CTRP2; CCLE 4.898 6.943 3.9705 4.8048
PL45 CCLE 5.0493 7.2262 2.2526 1.0126
SUIT-2 GDSC1; GDSC2; CTRP2; CCLE 5.1118 6.6039 4.3201 2.917
Panc 08.13 GDSC1; GDSC2; CTRP2 5.1311 7.4849 3.8956 4.6641
KP-3 GDSC1; GDSC2; CTRP2; CCLE 5.1489 8.1605 3.5725 5.9879
L3.3 CTRP2; CCLE 5.3352 7.6641 3.9683 3.9921
PSN1 GDSC1; GDSC2; CTRP2; CCLE 5.3569 7.3656 4.1328 3.2691
DAN-G GDSC1; GDSC2; CTRP2 5.4023 8.8044 3.4537 6.0259
PL4 GDSC1; GDSC2 5.4079 6.9304 2.8248 0.3344
TCC-Pan2 CTRP2 5.4299 7.2062 4.2655 2.6008
HPAF-II GDSC1; GDSC2; CTRP2; CCLE 5.4375 7.5876 4.0837 3.3398
Capan-2 GDSC1; GDSC2; CTRP2; CCLE 5.4565 7.2601 4.2584 2.5883
AsPC-1 GDSC1; GDSC2; CTRP2; CCLE 5.4665 8.0628 3.871 4.1752
Capan-1 GDSC1; GDSC2; CTRP2 5.4679 7.1325 4.3288 2.2823
KP-2 GDSC1; GDSC2; CTRP2 5.4973 6.8805 4.4709 1.6639
SNU-213 CTRP2 5.5181 7.8871 3.9959 3.573
Panc 05.04 CTRP2 5.5255 7.8471 4.021 3.4574
PK-59 CTRP2; CCLE 5.5774 8.1574 3.9067 3.8466
CFPAC-1 GDSC1; GDSC2; CTRP2 5.6201 8.6821 3.6802 4.7141
MIA PaCa-2 GDSC1; GDSC2; CTRP2; CCLE 5.6385 7.1951 4.4147 1.6958
SNU-410 CTRP2 5.6764 8.7922 3.6676 4.6753
YAPC GDSC1; GDSC2; CTRP2 5.7196 8.4909 3.8463 3.8727
Panc 04.03 GDSC1; GDSC2; CTRP2; CCLE 5.7885 8.0542 4.1054 2.7207
SU.86.86 GDSC1; GDSC2; CTRP2; CCLE 5.8438 8.4952 3.9312 3.3428
PK-45H CTRP2; CCLE 5.915 8.0225 4.2033 2.1657
KP-4 GDSC1; GDSC2; CTRP2; CCLE 5.9958 8.1852 4.1783 2.1616
Panc 10.05 GDSC1; GDSC2; CTRP2; CCLE 6.0151 7.7378 4.3948 1.3298
Panc 03.27 GDSC1; GDSC2; CTRP2; CCLE 6.1066 9.8382 3.4646 4.8478
PaTu 8988s CTRP2 6.1593 8.1382 4.2981 1.528
Panc 02.03 GDSC1; GDSC2; CTRP2; CCLE 6.2347 8.0141 4.3949 1.1168
PaTu 8902 GDSC1; GDSC2; CTRP2; CCLE 6.3142 7.6394 4.5907 0.4618
PaTu 8988t GDSC1; GDSC2; CTRP2 6.7337 8.3117 4.5132 0.4349
QGP-1 GDSC1; GDSC2; CTRP2; CCLE 7.5102 9.1232 4.5229 0.1672
HuP-T3 GDSC1; GDSC2; CTRP2; CCLE 7.6238 9.2254 4.5286 0.1391
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 79 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 -0.3346 6.2888 -1.2074 38.1464
CP50-MEL-B GDSC1; GDSC2 -1.8942 4.6126 -2.7689 51.6087
WM88 CTRP2; CCLE -1.7933 1.6643 -1.8336 45.6308
G-mel GDSC1; GDSC2 -1.6725 1.4432 -1.7538 50.1122
451Lu GDSC1; GDSC2 -1.3718 3.6822 -1.9033 47.6995
Malme-3M CTRP2; CCLE -0.9924 3.3856 -1.1762 40.6984
M14 GDSC1; GDSC2 -0.678 4.7834 -1.5144 42.5218
MMAc-SF GDSC1; GDSC2 -0.6558 5.0707 -1.5966 42.5558
SH-4 GDSC1; GDSC2 -0.5908 3.784 -1.0828 40.9515
A-375 GDSC1; GDSC2; CTRP2; CCLE -0.4275 3.1728 -0.5398 36.8027
Mel Ho GDSC1; GDSC2; CTRP2; CCLE -0.3809 4.2751 -0.6855 37.0427
COLO 679 GDSC1; GDSC2; CCLE -0.2726 4.5903 -1.0081 32.9511
WM983B CTRP2; CCLE -0.1869 4.1291 -0.4433 35.6438
IGR-37 GDSC1; GDSC2; CTRP2; CCLE 0.0238 3.8926 -0.1687 34.0664
UACC-62 GDSC1; GDSC2; CTRP2; CCLE 0.3995 5.8717 -0.2726 33.0778
SK-MEL-1 GDSC1; GDSC2; CTRP2 0.625 4.5104 0.356 30.3432
HT-144 GDSC1; GDSC2; CTRP2; CCLE 0.8494 6.2434 0.0906 30.4715
WT2-iPS GDSC1; GDSC2; CTRP2; CCLE 0.8688 4.9621 0.5097 29.0351
SK-MEL-28 GDSC1; GDSC2; CTRP2 0.9006 14.3531 -3.3933 37.9812
COLO 829 GDSC1; GDSC2; CTRP2 1.0383 7.1669 -0.047 30.2976
WM1799 CTRP2; CCLE 1.0819 6.0601 0.4054 28.7049
UACC-257 GDSC1; GDSC2; CTRP2; CCLE 1.1791 6.422 0.3833 28.4738
COLO 800 GDSC1; GDSC2; CTRP2 1.2529 4.8503 0.958 26.2744
WM115 GDSC1; GDSC2; CTRP2; CCLE 1.2757 4.4462 1.078 25.7847
G-361 GDSC1; GDSC2; CTRP2; CCLE 1.2793 4.2348 1.1247 25.6113
Hs 938.T GDSC1; GDSC2; CCLE 1.2979 8.0419 -0.8817 26.6206
WM266-4 CTRP2; CCLE 1.4872 5.1418 1.1353 24.9212
RVH-421 GDSC1; GDSC2; CTRP2; CCLE 1.5011 8.124 0.0519 28.5657
WM278 GDSC1; GDSC2 1.6123 9.7221 -1.3947 31.4771
SK-MEL-24 GDSC1; GDSC2; CTRP2; CCLE 1.9491 8.4427 0.3779 26.1964
COLO 783 GDSC1; GDSC2 1.9879 5.6693 0.9107 19.5492
MZ-MEL-7 GDSC1; GDSC2 2.5002 8.3096 0.1141 22.0104
MZ-MEL-2 GDSC1; GDSC2 2.7052 6.6013 1.1436 15.6053
MDA-MB-435S CTRP2; CCLE 2.8543 7.1149 1.8874 18.1915
Hs 695T CCLE 2.9367 6.3153 1.2893 9.4213
K029AX CTRP2; CCLE 2.9491 9.8103 0.7498 22.2193
A-431 GDSC1; GDSC2 3.2625 8.8657 0.5004 17.5172
CP66-MEL GDSC1; GDSC2 3.344 6.6336 1.6844 10.2848
SF8657 CCLE 3.4117 5.4828 2.0828 4.0347
CHL-1 GDSC1; GDSC2; CCLE 3.639 5.3737 2.5468 3.3804
IST-MEL1 GDSC1; GDSC2 3.7089 8.8021 0.8972 13.9974
A101D GDSC1; GDSC2; CTRP2 3.8621 10.1257 1.4619 17.3595
Hs 940.T GDSC1; GDSC2; CTRP2 3.869 7.406 2.7827 12.0466
WM1552C GDSC1; GDSC2 3.8841 9.9802 0.4489 16.001
VMRC-MELG GDSC1; GDSC2 4.067 6.3703 2.365 4.2039
COLO 741 CTRP2; CCLE 4.1792 8.2385 2.6793 11.7416
SK-MEL-3 GDSC1; GDSC2; CTRP2 4.2233 12.5052 0.6094 19.7142
RPMI-7951 GDSC1; GDSC2; CCLE 4.2481 8.2854 1.5633 7.2429
LOX-IMVI GDSC1; GDSC2; CTRP2; CCLE 4.3165 10.0499 1.9119 14.5699
Hs 294T CTRP2; CCLE 4.354 10.6039 1.6702 15.4511
WM793 GDSC1; GDSC2; CTRP2; CCLE 4.3689 10.997 1.488 16.1331
GAK GDSC1; GDSC2 4.4239 6.549 2.508 2.6944
LB2518-MEL GDSC1; GDSC2 4.4903 6.0894 2.7478 1.3367
IGR-1 GDSC1; GDSC2; CTRP2 4.56 9.588 2.3573 12.2395
A-388 GDSC1; GDSC2 4.6303 8.6651 1.6463 7.3143
HMV-II GDSC1; GDSC2 4.655 7.4912 2.2157 3.943
Hs 852.T CTRP2; CCLE 4.7622 7.0923 3.7767 5.8993
WM35 GDSC1; GDSC2 4.861 15.3574 -1.4662 21.9952
LB373-MEL-D GDSC1; GDSC2 4.8954 6.0238 2.9541 0.2353
Hs 944.T CTRP2; CCLE 4.9491 7.4202 3.7762 5.5174
DJM-1 GDSC1; GDSC2 5.0436 9.9385 1.315 8.369
COLO 792 GDSC1; GDSC2; CTRP2 5.2042 6.6211 4.3849 2.4786
IGR-39 CTRP2; CCLE 5.2562 7.4453 4.0155 3.9328
Hs 895.T CTRP2; CCLE 5.2894 7.3183 4.1046 3.5022
CJM [Human melanoma] CTRP2 5.311 6.2234 4.6596 1.1697
Hs 839.T CTRP2 5.4265 7.3965 4.1696 3.0021
SK-MEL-5 GDSC1; GDSC2; CTRP2; CCLE 5.5169 14.6772 0.6159 17.0532
Hs 934.T CTRP2 5.5533 8.5594 3.6909 4.7794
Hs 688(A).T CTRP2 5.5707 10.928 2.5289 9.5729
HMCB CTRP2; CCLE 5.6168 7.1681 4.4133 1.73
MeWo GDSC1; GDSC2; CTRP2; CCLE 5.7568 7.6039 4.2985 1.9972
A2058 GDSC1; GDSC2; CTRP2; CCLE 5.9534 10.7158 2.926 7.2867
Mel JuSo GDSC1; GDSC2; CTRP2 6.0452 7.7542 4.4046 1.2637
Hs 936.T CTRP2; CCLE 6.1156 7.6719 4.4794 0.9398
SK-MEL-2 GDSC1; GDSC2; CTRP2; CCLE 6.2298 7.3688 4.6594 0.3342
IPC-298 GDSC1; GDSC2; CTRP2; CCLE 6.271 10.9068 3.0619 6.2361
SK-MEL-30 GDSC1; GDSC2; CTRP2; CCLE 6.8024 7.9561 4.6713 0.1209
SK-MEL-31 GDSC1; GDSC2; CTRP2; CCLE 7.1962 14.0492 2.1845 8.3628
EquiPSC Line K2 GDSC1; GDSC2 1.2285 7.6312 -0.7548 30.7211
⏷ Show the Full List of 79 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE-12 GDSC1; GDSC2 4.0196 8.4788 1.2993 10.8094
HCE-4 GDSC1; GDSC2 4.2987 6.7766 2.325 3.972
FLO-1 GDSC1; GDSC2 4.3096 8.6828 1.4134 9.4159
SK-GT-4 GDSC1; GDSC2 4.5962 8.1804 1.8549 6.1545
ESO-51 GDSC1; GDSC2 4.6745 7.5124 2.2179 3.8967
KYAE-1 GDSC1; GDSC2 5.0135 8.1838 2.1141 3.9012
ESO-26 GDSC1; GDSC2 5.1535 6.8887 2.7366 0.7434
KYSE-50 GDSC1; GDSC2 5.1774 6.9703 2.7154 0.8022
OACP4 C GDSC1; GDSC2 5.4262 7.6321 2.5662 1.1681
KYSE-220 GDSC1; GDSC2 5.4772 8.0577 2.4177 1.7448
OACM5.1 C GDSC1; GDSC2 5.6707 8.5179 2.322 1.9654
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1; GDSC2 5.1154 8.0836 2.2174 3.1854
Cancer Drug Sensitivity Data Curated from 36 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SJNB-13 GDSC1; GDSC2 2.3689 4.6878 1.7423 13.1656
SJNB-6 GDSC1; GDSC2 3.4273 4.794 2.6717 3.8205
KP-N-YS GDSC1; GDSC2 3.7915 8.1015 1.3113 11.3324
NB69 GDSC1; GDSC2 3.8321 5.4412 2.6514 2.9713
SJNB-5 GDSC1; GDSC2 4.0197 6.0918 2.4665 3.6917
SJNB-7 GDSC1; GDSC2 4.1505 6.6 2.3113 4.352
GI-ME-N GDSC1; GDSC2 4.2749 6.3668 2.5014 2.9905
SJNB-12 GDSC1; GDSC2 4.3199 6.4747 2.4793 3.0362
CHP-134 GDSC1; GDSC2 4.3749 8.2986 1.6471 7.8686
KP-N-SI9s CTRP2; CCLE 4.6012 7.2363 3.5603 7.1499
SK-N-MC-IXC GDSC1; GDSC2 4.6605 6.0607 2.8423 0.7385
IMR-5 GDSC1; GDSC2 4.7725 7.7403 2.1727 3.981
SK-N-BE(2) CTRP2; CCLE 4.8221 7.3935 3.6798 6.1798
SK-N-SH GDSC1; GDSC2; CTRP2; CCLE 5.0173 6.5221 4.2829 3.2535
SJNB-14 GDSC1; GDSC2 5.0416 6.5242 2.8283 0.5098
SK-N-BE(2)-M17 GDSC1; GDSC2 5.0953 6.8233 2.7366 0.7871
GOTO GDSC1; GDSC2 5.1475 11.5793 0.5979 12.0882
MHH-NB-11 GDSC1; GDSC2 5.3741 7.2015 2.7109 0.6793
NH-6 CTRP2 5.4923 7.1532 4.3359 2.2164
NB(TU)1 GDSC1; GDSC2 5.515 7.0432 2.8252 0.2919
NH-12 GDSC1; GDSC2 5.6163 7.4038 2.7341 0.4726
TGW GDSC1; GDSC2 5.652 7.1466 2.8394 0.2186
SK-N-AS GDSC1; GDSC2; CTRP2; CCLE 5.7399 7.4047 4.3813 1.6961
SJNB-17 GDSC1; GDSC2 5.7718 8.1691 2.5094 1.1018
CHP-212 GDSC1; GDSC2; CCLE 5.7719 7.3522 2.8116 0.1961
IMR-32 CTRP2; CCLE 5.8863 7.2132 4.5552 0.8916
LA-N-6 GDSC1; GDSC2 5.941 7.3867 2.8597 0.1222
SK-N-FI GDSC1; GDSC2; CTRP2; CCLE 5.954 7.3966 4.5119 0.9769
Kelly GDSC1; GDSC2; CTRP2; CCLE 5.9746 7.4195 4.5132 0.953
SJNB-10 GDSC1; GDSC2 6.0484 7.7648 2.7686 0.2354
KP-N-RT-BM-1 GDSC2 6.0612 7.9863 2.6956 0.3776
SiMa GDSC1; GDSC2; CCLE 6.1016 7.8534 2.7572 0.2009
SK-N-DZ GDSC1; GDSC2; CTRP2; CCLE 6.7149 8.1846 4.5538 0.3524
CHP-126 GDSC1; GDSC2; CTRP2 6.7978 8.5548 4.4467 0.5637
NB1 GDSC1; GDSC2; CTRP2 6.7994 8.2931 4.5479 0.3303
KP-N-YN GDSC1; GDSC2; CTRP2 7.1983 10.4665 3.8481 2.0917
⏷ Show the Full List of 36 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 2.5039 5.1112 2.2533 17.8035
HuH-28 CTRP2 5.0418 7.1425 3.9931 4.4238
SNU-478 CTRP2 5.0669 7.5704 3.8001 5.187
HuCC-T1 GDSC1; GDSC2; CTRP2; CCLE 5.1331 8.5358 3.372 6.8597
SNU-308 CTRP2 5.578 8.3191 3.8277 4.1719
SNU-1196 CTRP2 5.9369 8.4901 3.9965 2.9505
SNU-869 CTRP2 7.0789 8.7088 4.5067 0.3084
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 90 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 GDSC1; GDSC2; CTRP2 -1.1497 1.0764 -1.1541 41.2794
MDA-MB-157 GDSC1; GDSC2; CTRP2; CCLE 3.5297 5.5784 3.2199 11.2083
SK-BR-3 CCLE 3.95 7.1498 1.6535 5.2414
Hs 578Bst CTRP2 4.4408 8.8887 2.5986 11.4974
OCUB-M GDSC1; GDSC2 4.524 6.8291 2.44 2.9062
MFM-223 GDSC1; GDSC2 4.5783 6.3893 2.6654 1.6298
HCC1599 GDSC2 4.6618 8.4527 1.7689 6.5273
HCC2218 GDSC1; GDSC2; CTRP2 4.7104 7.7058 3.426 7.476
Hs 739.T CCLE 4.7173 7.4074 2.0094 2.3119
MDA-MB-175-VII GDSC1; GDSC2; CCLE 4.8053 6.4989 2.7334 0.8776
Evsa-T GDSC1; GDSC2 4.8671 6.5293 2.75 0.9257
HCC1569 GDSC1; GDSC2; CCLE 4.8823 8.6103 1.8375 4.7523
HCC2157 GDSC1; GDSC2 4.95 8.0192 2.1514 3.8003
COLO 824 GDSC1; GDSC2 4.9769 7.3164 2.477 2.0483
CAL-85-1 GDSC1; GDSC2; CTRP2; CCLE 5.067 7.7122 3.7293 5.4845
MDA-MB-436 GDSC1; GDSC2; CCLE 5.1002 7.0349 2.655 1.0665
MDA-MB-453 GDSC1; GDSC2; CTRP2; CCLE 5.1051 7.8388 3.6975 5.5455
BT-474 GDSC1; GDSC2; CCLE 5.1496 6.6399 2.8292 0.3706
MDA-MB-415 GDSC1; GDSC2; CCLE 5.1504 6.7816 2.7764 0.5072
Hs 578T GDSC1; GDSC2; CTRP2; CCLE 5.1759 7.3811 3.9837 4.211
MRK-nu-1 GDSC1; GDSC2 5.1905 6.6035 2.8588 0.3438
MDA-MB-330 GDSC1; GDSC2 5.2324 9.0948 1.8295 5.1063
BT-20 GDSC1; GDSC2; CTRP2; CCLE 5.3045 7.3185 4.1162 3.4275
HMC-1-8 CTRP2; CCLE 5.3143 6.2617 4.6434 1.2303
T-47D GDSC1; GDSC2; CTRP2; CCLE 5.3315 7.7303 3.9326 4.1475
HCC70 GDSC1; GDSC2; CCLE 5.4015 9.0321 1.9572 3.4499
HCC1954 GDSC1; GDSC2; CTRP2; CCLE 5.4132 7.1056 4.3027 2.4739
MDA-MB-231 GDSC1; GDSC2; CTRP2 5.42 7.4873 4.1201 3.2176
UACC-893 GDSC1; GDSC2 5.4433 8.714 2.1211 3.2149
UACC-812 GDSC2; CCLE 5.4648 7.2473 2.7312 0.4667
CAL-51 GDSC1; GDSC2; CTRP2 5.4908 7.1364 4.343 2.1901
HCC1428 GDSC1; GDSC2; CTRP2 5.5898 7.6169 4.1795 2.7081
HCC1395 GDSC1; GDSC2; CTRP2; CCLE 5.5909 7.8741 4.0551 3.2147
MDA-MB-468 GDSC1; GDSC2; CTRP2; CCLE 5.6269 7.3466 4.3351 2.0268
ZR-75-1 CTRP2; CCLE 5.6621 7.1955 4.4298 1.6061
ZR-75-30 GDSC1; GDSC2; CTRP2; CCLE 5.7122 7.8612 4.1462 2.6647
EFM-19 GDSC1; GDSC2; CCLE 5.7389 7.6765 2.6827 0.4607
HCC1143 GDSC1; GDSC2; CTRP2 5.7701 7.7823 4.2227 2.2787
HCC1500 GDSC1; GDSC2; CTRP2 5.7826 7.9499 4.1512 2.5457
YMB-1-E GDSC2 5.8095 7.5853 2.7434 0.3651
HCC1419 GDSC1; GDSC2; CTRP2 5.8156 8.313 3.9996 3.1073
CAMA-1 GDSC1; GDSC2; CTRP2; CCLE 5.8444 7.3248 4.4817 1.195
BT-549 GDSC1; GDSC2; CTRP2; CCLE 5.925 9.0684 3.7106 4.1173
HCC1187 GDSC1; GDSC2; CCLE 5.9253 7.5509 2.7982 0.1806
EFM-192A GDSC1; GDSC2; CTRP2 5.9667 7.4776 4.4833 1.0642
HCC1937 GDSC1; GDSC2; CTRP2 5.9687 8.7888 3.8752 3.3907
MDA-MB-361 GDSC1; GDSC2; CTRP2 6.0477 8.6204 4.0074 2.7599
JIMT-1 GDSC1; GDSC2; CTRP2 6.0484 8.5165 4.0567 2.5666
KPL-1 CTRP2 6.0583 6.7339 4.8256 0.0744
AU565 GDSC1; GDSC2; CTRP2; CCLE 6.0773 8.5936 4.0391 2.5985
BT-483 GDSC1; GDSC2 6.1174 7.7347 2.8035 0.1638
CAL-120 GDSC1; GDSC2; CTRP2 6.1287 8.974 3.8931 3.103
HCC1806 GDSC1; GDSC2; CTRP2; CCLE 6.1534 8.5464 4.1086 2.2376
HDQ-P1 GDSC1; GDSC2; CTRP2; CCLE 6.3997 9.9307 3.6173 3.8311
CAL-148 GDSC2; CTRP2 6.5285 7.9915 4.548 0.4535
HCC38 GDSC1; GDSC2; CTRP2 6.6856 8.5263 4.4067 0.7361
MCF-7 GDSC1; GDSC2; CTRP2; CCLE 6.8211 8.9456 4.3001 0.9517
HCC202 GDSC1; CTRP2 6.8377 16.0196 0.9701 13.465
BT 416 CTRP2 4.5905 6.3021 4.0064 5.3262
BT 498 CTRP2 5.3987 6.969 4.359 2.2649
BT164 CTRP2 5.434 6.7235 4.5032 1.6239
BT 179 CTRP2 5.5321 6.6123 4.62 1.033
BT 239 CTRP2 5.589 7.1521 4.4026 1.81
BT 224 CTRP2 5.5904 6.8231 4.5584 1.198
BT 440 CTRP2 5.6958 7.9738 4.0806 2.9531
BT 422 CTRP2 5.7141 8.1838 3.9917 3.2874
BT 172 CTRP2 5.7143 7.2827 4.4221 1.5702
BT 320 CTRP2 5.7396 7.4993 4.3367 1.87
BT 112 CTRP2 5.7614 8.4012 3.9195 3.5106
BT 340 CTRP2 5.7706 8.8194 3.7225 4.3016
BT 231 CTRP2 5.7709 7.9768 4.1306 2.6445
BT 145 CTRP2 5.7901 7.2612 4.4785 1.2664
BT147 CTRP2 5.8459 7.5023 4.4018 1.4899
BT 330 CTRP2 5.8465 7.5062 4.4003 1.4948
BT 482 CTRP2 5.8681 7.7939 4.2805 1.9258
BT 444 CTRP2 5.8768 7.8487 4.2604 1.9927
BT 187 CTRP2 5.8901 9.7471 3.3552 5.6238
BT 328 CTRP2 5.9158 8.8204 3.824 3.6716
BT 139 CTRP2 6.0669 9.7561 3.4767 4.8573
BT 333 CTRP2 6.098 7.6462 4.4811 0.9497
BT 248 CTRP2 6.1033 11.5424 2.6301 8.2535
BT 245 CTRP2 6.2037 8.6076 4.1112 2.1689
BT 504 CTRP2 6.428 8.3183 4.366 1.046
BT 232 CTRP2 6.4387 8.2797 4.3878 0.9679
BT 286 CTRP2 6.8029 7.8454 4.7097 0.0767
BT 216 CTRP2 6.8966 8.7678 4.407 0.6105
BT 228 CTRP2 7.0962 16.5942 0.8774 13.3796
BT 131 CTRP2 7.1483 8.4274 4.6331 0.1031
BT 359 CTRP2 7.4729 8.8889 4.5903 0.098
BT 159 CTRP2 11.8489 26.5265 -0.6946 12.0525
⏷ Show the Full List of 90 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 5.8112 8.1022 4.0977 2.72
Cancer Drug Sensitivity Data Curated from 70 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DBTRG-05MG GDSC1; GDSC2; CTRP2; CCLE 2.5626 7.9324 1.2309 21.4705
MOG-G-UVW GDSC1; GDSC2 2.9863 8.9234 0.2368 19.774
D-245MG GDSC2 3.1361 7.901 0.8757 15.7989
H4 GDSC1; GDSC2; CCLE 3.24 5.2767 2.2754 5.7195
KG-1-C CTRP2 3.2655 13.8739 -0.9283 26.7523
D-566MG GDSC1; GDSC2 3.6595 7.3474 1.5831 10.03
D-423MG GDSC1; GDSC2 3.6978 7.3441 1.6148 9.7311
GI-1 GDSC1; GDSC2; CCLE 3.7699 5.673 2.4956 3.3849
D-247MG GDSC1; GDSC2 3.9659 5.9603 2.4932 3.6436
SF539 GDSC1; GDSC2; CTRP2 4.2959 7.1876 3.2993 8.9201
Onda 10 GDSC1; GDSC2 4.4346 7.6122 2.0182 5.518
D-263MG GDSC1; GDSC2 4.4502 6.2457 2.6588 1.839
D-502MG GDSC1; GDSC2 4.4595 8.1181 1.7928 6.8099
PFSK-1 GDSC1; GDSC2 4.5211 6.6632 2.5132 2.5086
KNS-81-FD GDSC1; GDSC2 4.5994 9.9367 1.0093 11.0826
D-542MG GDSC1; GDSC2 4.7381 6.4691 2.7131 1.2122
NMC-G1 GDSC1; GDSC2; CTRP2 4.7649 8.8788 2.8896 9.6069
1321N1 CCLE 4.8142 8.5519 1.5507 4.3164
LN-405 GDSC1; GDSC2 4.8262 6.9365 2.5608 1.8277
MOG-G-CCM GDSC1; GDSC2; CCLE 4.8417 8.6351 1.8 4.9991
SNU-466 CTRP2 4.8704 7.5178 3.6599 6.1642
Onda 11 GDSC1; GDSC2 4.8871 7.9802 2.1318 4.0139
D-392MG GDSC1; GDSC2 4.8927 7.5071 2.348 2.8261
D-336MG GDSC1; GDSC2 4.9054 7.3563 2.4214 2.4241
AM-38 GDSC1; GDSC2 4.9587 10.5269 0.9755 10.4584
SF268 GDSC1; GDSC2; CTRP2 5.0043 7.3232 3.8713 5.0087
DK-MG GDSC1; GDSC2; CTRP2; CCLE 5.1198 6.8124 4.2224 3.3123
42-MG-BA GDSC1; GDSC2; CTRP2; CCLE 5.1443 7.016 4.1406 3.6106
SNB-75 GDSC1; GDSC2; CTRP2 5.1603 8.278 3.5232 6.1737
M059J GDSC1; GDSC2; CCLE 5.1692 7.4389 2.5229 1.3351
D283 Med GDSC1; GDSC2; CTRP2 5.1843 7.7056 3.8285 4.8471
GB-1 GDSC1; GDSC2; CTRP2; CCLE 5.2113 9.3821 3.013 8.2177
LNZTA3WT4 GDSC1 5.2376 6.7089 2.8389 0.4657
Hs 683 GDSC1; GDSC2; CTRP2; CCLE 5.2397 8.0432 3.7045 5.2664
ONS-76 GDSC1; GDSC2; CTRP2; CCLE 5.2823 8.6329 3.4443 6.2798
T98G GDSC1; GDSC2; CTRP2; CCLE 5.3294 7.6946 3.9487 4.084
KNS-60 CTRP2; CCLE 5.3731 7.1773 4.2379 2.8058
Becker GDSC1; GDSC2; CTRP2 5.3875 6.7804 4.443 1.9374
YH-13 GDSC1; GDSC2; CTRP2 5.4243 7.3842 4.174 2.9875
SW1783 GDSC1; GDSC2; CTRP2 5.429 8.4769 3.6372 5.2128
SW1088 GDSC1; GDSC2; CTRP2; CCLE 5.4445 8.5676 3.6041 5.3244
CCF-STTG1 CTRP2 5.5225 7.2672 4.3018 2.3103
GMS-10 CTRP2; CCLE 5.579 7.2771 4.336 2.0901
Daoy GDSC1; GDSC2; CTRP2; CCLE 5.6064 8.9284 3.5486 5.2823
U-118MG GDSC1; GDSC2; CTRP2; CCLE 5.6122 7.4378 4.2814 2.2626
GOS-3 CTRP2 5.6199 6.9904 4.499 1.3906
YKG-1 GDSC1; GDSC2; CTRP2; CCLE 5.6312 8.2832 3.8841 3.8544
CAS-1 GDSC1; GDSC2; CTRP2; CCLE 5.6336 7.9141 4.066 3.105
SF126 GDSC1; GDSC2; CTRP2; CCLE 5.6354 7.7317 4.1557 2.7371
SNU-1105 CTRP2 5.66 8.4764 3.8105 4.1125
KALS-1 GDSC1; GDSC2; CTRP2; CCLE 5.6807 9.1537 3.4929 5.3911
LN-229 GDSC1; GDSC2; CTRP2; CCLE 5.6949 7.7943 4.1665 2.6072
LN-18 GDSC1; GDSC2; CTRP2 5.7431 7.5993 4.2917 2.0419
KINGS-1 GDSC1; GDSC2 5.7849 7.9599 2.5955 0.7925
8-MG-BA GDSC1; GDSC2; CTRP2; CCLE 5.7899 10.1157 3.1001 6.8372
TM-31 CTRP2 5.7962 8.0959 4.0906 2.7692
SNU-201 CTRP2 5.8 7.7633 4.2513 2.1263
SK-MG-1 GDSC1; GDSC2 5.8552 7.4886 2.7944 0.2431
SNU-738 CTRP2 5.865 7.2137 4.5432 0.9538
A-172 GDSC1; GDSC2; CTRP2; CCLE 5.9025 7.2699 4.5392 0.9314
M059K CTRP2 5.9539 7.2784 4.5633 0.8025
GaMG GDSC1; GDSC2; CTRP2; CCLE 6.0484 8.4007 4.1109 2.3564
SNU-626 CTRP2 6.1687 7.554 4.5565 0.6526
U-87MG ATCC GDSC1; GDSC2; CTRP2; CCLE 6.259 8.9936 3.9669 2.6514
KS-1 [Human Krukenberg tumour] GDSC1; GDSC2 6.2931 8.2225 2.6985 0.294
KNS-81 CTRP2; CCLE 6.3655 7.8013 4.5495 0.5415
SNU-489 CTRP2 6.5745 8.0552 4.5433 0.4412
KNS-42 GDSC1; GDSC2; CTRP2; CCLE 6.6006 8.0502 4.5566 0.397
U-251MG GDSC1; GDSC2; CTRP2 7.0663 8.6479 4.5241 0.2806
SF295 GDSC1; GDSC2; CTRP2; CCLE 7.6614 14.1686 2.4353 6.7738
⏷ Show the Full List of 70 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TGBC1TKB GDSC1; GDSC2 4.4776 6.71 2.4666 2.8353
ETK-1 GDSC1; GDSC2 4.8608 7.5328 2.3185 3.0319
TGBC24TKB GDSC1; GDSC2 6.1775 8.2157 2.6578 0.4189
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-2 CTRP2; CCLE 3.7916 5.4192 3.1614 4.8108
JHUEM-3 CTRP2 4.1175 7.2018 3.1212 10.0702
JHUEM-7 CTRP2 4.5801 6.37 3.9637 5.5262
MFE-280 GDSC1; GDSC2; CCLE 4.5981 7.1757 2.3261 2.8469
RL95-2 GDSC1; GDSC2; CTRP2; CCLE 4.7753 7.4387 3.6161 6.544
TEN CCLE 4.8629 7.2333 2.1603 1.5165
KLE GDSC1; GDSC2; CTRP2; CCLE 5.1231 8.2169 3.5233 6.2434
JHUEM-1 CTRP2 5.194 6.3864 4.4936 2.0421
AN3-CA GDSC1; GDSC2; CTRP2; CCLE 5.321 7.9459 3.8172 4.6486
HEC-1-A CTRP2; CCLE 5.4526 7.3849 4.1945 2.8575
HEC-151 CTRP2; CCLE 5.5382 7.2363 4.3277 2.1823
HEC-59 CTRP2; CCLE 5.8147 8.8557 3.7363 4.1778
HEC-108 CTRP2 5.8179 7.7206 4.2829 1.9793
EN GDSC1; GDSC2; CTRP2; CCLE 5.8292 7.2451 4.5088 1.1126
MFE-296 GDSC1; GDSC2; CTRP2; CCLE 5.8583 8.184 4.0901 2.6857
HEC-1-B CTRP2; CCLE 5.8832 8.7394 3.8406 3.6517
ESS-1 GDSC1; GDSC2; CTRP2; CCLE 5.9561 7.514 4.4611 1.1529
HEC-251 CTRP2; CCLE 5.9725 7.7131 4.3812 1.4245
HEC-265 CTRP2; CCLE 6.2162 7.5824 4.5679 0.5858
HEC-6 CTRP2; CCLE 6.411 8.1284 4.4374 0.8355
EFE-184 CTRP2; CCLE 6.5672 9.4072 3.9634 2.3111
MFE-319 GDSC1; GDSC2; CTRP2; CCLE 6.6183 8.2471 4.4875 0.5581
HEC-50B CTRP2 9.2945 23.3985 -0.8776 15.7096
Ishikawa (Heraklio) 02 ER- CTRP2; CCLE 5.8599 8.9949 3.7006 4.2551
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
BB65-RCC GDSC1; GDSC2 3.1971 5.9552 1.8999 9.368
LB2241-RCC GDSC1; GDSC2 3.2614 6.4635 1.7004 10.4278
LB1047-RCC GDSC1; GDSC2 3.3924 5.8897 2.0963 7.556
UO-31 GDSC1; GDSC2; CTRP2 3.4962 6.9308 2.6279 13.6016
LB996-RCC GDSC1; GDSC2 3.5283 5.5355 2.3821 5.3766
KTCTL-26A GDSC1; GDSC2 3.8924 7.4802 1.697 8.7183
KTCTL-13 GDSC1; GDSC2 3.9936 5.8105 2.583 3.0482
A-704 GDSC1; GDSC2 4.0615 7.0465 2.0342 6.2324
KTCTL-1M GDSC1; GDSC2 4.098 6.3789 2.3818 4.038
RXF 393L GDSC1; GDSC2 4.1512 7.2171 2.0147 6.1481
NCC021 GDSC1; GDSC2 4.2092 7.1866 2.0697 5.6854
KTCTL-140 GDSC1; GDSC2 4.2703 9.7932 0.8387 12.8453
SW156 GDSC1; GDSC2 4.3273 6.971 2.2518 4.3481
KTCTL-21 GDSC1; GDSC2 4.3277 7.9921 1.7626 7.2804
SW13 GDSC1; GDSC2 4.3305 6.0802 2.665 1.984
A-498 GDSC1; GDSC2 4.3445 6.7436 2.3697 3.6236
CAL-54 GDSC1; GDSC2; CTRP2 4.3878 6.4181 3.7553 6.8347
HA7-RCC GDSC1; GDSC2 4.5711 6.6364 2.5536 2.2153
KTCTL-195 GDSC1; GDSC2 4.6017 6.7768 2.5085 2.4092
NCC010 GDSC1; GDSC2 5.1128 7.7055 2.3813 2.3464
KMRC-3 CTRP2 5.1248 8.5867 3.3398 7.0106
VMRC-RCZ GDSC1; GDSC2; CTRP2; CCLE 5.3006 7.5224 4.0119 3.8702
TUHR4TKB CTRP2 5.3347 7.4937 4.0525 3.6415
ACHN GDSC1; GDSC2; CTRP2; CCLE 5.3662 8.8128 3.4212 6.2261
SN12C GDSC1; GDSC2 5.3796 6.9671 2.8005 0.4085
KMRC-1 GDSC1; GDSC2; CTRP2; CCLE 5.4316 6.9646 4.3847 2.109
TK-10 GDSC1; GDSC2 5.4864 8.6741 2.1617 2.9503
Caki-2 CTRP2; CCLE 5.9374 9.4042 3.5564 4.7266
KMRC-20 GDSC1; GDSC2; CTRP2 5.9863 7.7994 4.3502 1.5235
769-P GDSC1; GDSC2; CTRP2; CCLE 5.9992 8.3887 4.0853 2.5181
KMRC-2 CTRP2; CCLE 6.0302 8.4606 4.0714 2.5328
VMRC-RCW GDSC1; GDSC2; CTRP2; CCLE 6.0572 8.5433 4.0498 2.5823
TUHR14TKB CTRP2 6.0831 10.222 3.2619 5.707
OS-RC-2 GDSC1; GDSC2; CTRP2 6.1475 9.4375 3.6852 3.9018
Caki-1 GDSC1; GDSC2; CTRP2 6.2598 8.8184 4.0483 2.3407
786-O GDSC1; GDSC2; CTRP2 6.3713 9.6939 3.7106 3.5029
RCC10RGB GDSC1; GDSC2; CTRP2 6.3745 8.4139 4.2964 1.3231
TUHR10TKB CTRP2 6.3881 7.75 4.5803 0.4474
BFTC-909 GDSC1; GDSC2; CTRP2; CCLE 6.5135 8.1265 4.4875 0.6201
SNU-1272 CTRP2 7.0506 8.5798 4.5428 0.2526
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 61 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO201 CTRP2; CCLE 1.206 4.7977 0.9201 26.554
COLO205 GDSC1; GDSC2; CTRP2; CCLE 1.7701 8.2582 0.2738 27.0566
HT-29 GDSC1; GDSC2; CTRP2; CCLE 2.6509 8.4853 1.0724 21.822
MDST8 GDSC1; GDSC2; CTRP2 3.4818 6.1839 2.9339 12.437
LS411N GDSC1; GDSC2; CTRP2; CCLE 3.5406 8.8629 1.7725 16.899
LoVo GDSC1; GDSC2; CTRP2 3.7398 5.9579 3.2978 10.3235
SNU-81 GDSC1; GDSC2 4.399 6.585 2.4767 2.9122
COLO 320HSR GDSC1; GDSC2 4.415 6.347 2.5939 2.2368
SNU-C5 GDSC1; GDSC2; CTRP2 4.434 9.8227 2.1293 13.4386
GP2d CTRP2 4.7658 6.3055 4.1688 4.2559
SNU-C1 GDSC1; GDSC2; CTRP2 4.8129 6.4184 4.1561 4.2059
SNU-1040 GDSC1; GDSC2 4.9593 6.5141 2.7973 0.6695
SW626 GDSC1; GDSC2 5.0023 7.5285 2.3989 2.4058
T84 GDSC1; GDSC2; CTRP2; CCLE 5.0726 7.0672 4.0564 4.0985
SW620 GDSC1; GDSC2; CTRP2; CCLE 5.0752 6.6194 4.2824 3.1442
SNU-283 GDSC2 5.1488 6.8455 2.7513 0.6952
CCK-81 GDSC1; GDSC2; CTRP2; CCLE 5.1789 6.4464 4.4521 2.2421
SNU-175 GDSC2 5.2217 6.8537 2.7789 0.5562
NCI-H716 GDSC1; GDSC2; CTRP2 5.2283 7.2523 4.0897 3.6717
SW1116 GDSC1; GDSC2 5.23 6.9146 2.7593 0.6135
SNU-1033 CTRP2 5.2324 8.135 3.6528 5.4961
SK-CO-1 GDSC1; GDSC2; CTRP2; CCLE 5.2712 6.8108 4.3424 2.5409
HCT 15 GDSC1; GDSC2; CTRP2; CCLE 5.2755 7.6989 3.9045 4.3635
COLO 678 GDSC1; GDSC2; CTRP2; CCLE 5.2771 7.0667 4.22 3.041
SW1417 GDSC1; GDSC2; CTRP2; CCLE 5.3199 11.8348 1.8759 12.6824
HT-55 GDSC1; GDSC2; CTRP2 5.3504 7.1842 4.2176 2.9277
DiFi GDSC1; GDSC2 5.3639 7.9433 2.4094 1.9056
CL-11 GDSC1; GDSC2; CTRP2 5.374 6.8559 4.3965 2.1495
SW1463 GDSC1; GDSC2 5.4522 7.1656 2.7564 0.4936
LS123 GDSC1; GDSC2; CTRP2; CCLE 5.4788 7.3419 4.2345 2.6517
SW948 GDSC1; GDSC2; CTRP2 5.489 6.8803 4.4653 1.6978
NCI-H747 GDSC1; GDSC2; CTRP2; CCLE 5.4944 7.2471 4.2918 2.3934
OUMS-23 CTRP2 5.5249 7.7929 4.0471 3.3504
SNU-61 GDSC1; GDSC2; CTRP2 5.5314 7.5949 4.1487 2.9223
SW48 GDSC1; GDSC2; CTRP2; CCLE 5.6091 7.2127 4.387 1.8444
CaR-1 GDSC1; GDSC2 5.6192 8.0028 2.5066 1.2366
HT115 GDSC1; GDSC2; CTRP2 5.6573 6.9321 4.5493 1.1532
SNU-C2A CTRP2; CCLE 5.6694 8.1229 3.9898 3.3619
COLO 320 CTRP2; CCLE 5.7107 11.9536 2.1282 10.955
RCM-1 [Human ESC] GDSC1; GDSC2; CTRP2 5.7167 7.4944 4.3241 1.9492
SNU-407 GDSC1; GDSC2; CTRP2 5.732 7.4474 4.3562 1.8036
SNU-C4 CTRP2 5.7514 8.0419 4.0861 2.8505
HCC2998 GDSC1; GDSC2 5.7519 7.6876 2.6838 0.5435
GP5d GDSC1; GDSC2 5.8333 7.7242 2.7025 0.4544
C2BBe1 GDSC1; GDSC2; CTRP2; CCLE 5.8927 7.6654 4.3553 1.6107
SW837 GDSC1; GDSC2 5.9565 7.7394 2.7439 0.3107
SW403 CCLE 5.9788 7.6774 2.456 0.1393
LS180 GDSC1; GDSC2; CTRP2 5.9925 7.7846 4.3606 1.4784
HCT 8 CTRP2 6.1754 11.0145 2.9414 6.8715
SW480 CCLE 6.1786 8.437 2.2645 0.3918
KM12 GDSC1; GDSC2; CTRP2 6.2838 7.7863 4.5167 0.6889
DLD-1 CTRP2 6.4658 7.6791 4.641 0.2702
SNU-C2B GDSC1; GDSC2; CCLE 6.5169 9.2075 2.4289 0.7268
LS1034 GDSC1; GDSC2; CTRP2 6.5684 8.1804 4.4913 0.5768
HCC-56 CTRP2; CCLE 6.5757 7.6602 4.6913 0.1445
RKO GDSC1; GDSC2; CTRP2; CCLE 6.6839 13.9899 1.8535 10.4125
NCI-H508 GDSC1; GDSC2; CTRP2 6.7172 16.9153 0.4388 15.5222
LS513 GDSC1; GDSC2; CTRP2; CCLE 7.1306 8.5382 4.5881 0.1613
CW-2 GDSC1; GDSC2; CTRP2 7.1374 8.8422 4.4809 0.337
SNU-503 CTRP2 7.3434 9.1011 4.4676 0.2928
HCT 116 GDSC1; GDSC2; CTRP2; CCLE 7.5921 8.8971 4.6287 0.0539
⏷ Show the Full List of 61 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1; GDSC2 5.4842 7.0009 2.8285 0.2958
Cancer Drug Sensitivity Data Curated from 26 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Li-7 CTRP2 3.9294 6.5797 3.2248 10.1132
Hep-G2/C3A GDSC1; GDSC2; CCLE 3.9646 5.4572 2.7305 1.8625
SNU-182 CCLE 4.4809 7.4686 1.846 3.3866
Huh-7 GDSC1; GDSC2 4.5724 7.7612 2.0379 5.1257
JHH-7 GDSC1; GDSC2; CCLE 4.719 8.8737 1.6063 6.1567
HLE GDSC1; GDSC2; CCLE 4.9331 7.5574 2.3484 2.3027
SNU-475 CTRP2; CCLE 5.0709 7.9634 3.6069 5.9911
SNU-449 GDSC1; GDSC2; CTRP2; CCLE 5.1005 8.5902 3.318 7.1484
JHH-2 GDSC1; GDSC2; CTRP2; CCLE 5.1225 7.4572 3.9025 4.6511
JHH-1 GDSC1; GDSC2; CTRP2 5.167 5.9612 4.6838 1.295
SNU-423 GDSC1; GDSC2; CTRP2; CCLE 5.4453 7.7009 4.0336 3.5347
SNU-761 CTRP2 5.54 7.7312 4.0883 3.1575
PLC/PRF/5 CTRP2; CCLE 5.6407 7.3955 4.3209 2.0643
SNU-398 GDSC1; GDSC2; CTRP2; CCLE 5.6709 7.3956 4.341 1.9437
JHH-4 GDSC1; GDSC2; CTRP2; CCLE 5.6742 9.1887 3.4709 5.4928
HuH-1 GDSC1; GDSC2; CTRP2; CCLE 5.6927 8.436 3.8538 3.8831
SNU-886 CTRP2 5.698 8.5497 3.8021 4.0873
HuH-6 CTRP2 5.8618 9.0959 3.6528 4.4472
JHH-6 GDSC1; GDSC2; CTRP2; CCLE 5.9897 7.2579 4.5908 0.6831
SNU-387 GDSC1; GDSC2; CTRP2; CCLE 6.1751 8.5553 4.1178 2.1773
Hep-G2 CTRP2; CCLE 6.2875 13.5318 1.7869 11.3141
HLF CTRP2; CCLE 6.3099 10.5353 3.2686 5.3437
JHH-5 CTRP2; CCLE 6.4502 7.977 4.5182 0.575
Hep 3B2.1-7 GDSC1; GDSC2; CTRP2; CCLE 6.5431 10.9068 3.2485 5.0958
SK-HEP-1 GDSC1; GDSC2; CTRP2; CCLE 6.7457 12.5634 2.5909 7.4229
SNU-878 CTRP2 7.0776 8.6619 4.5234 0.2782
⏷ Show the Full List of 26 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 227 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1648 GDSC1; GDSC2; CCLE 2.5244 3.8251 2.2766 7.8082
NCI-H2795 GDSC1; GDSC2 2.6317 5.4351 1.6466 12.792
NCI-H1755 GDSC1; GDSC2; CTRP2 2.8769 5.5251 2.5321 15.6705
NCI-H209 GDSC1; GDSC2 3.331 8.736 0.6224 16.6409
NCI-H1734 GDSC2; CTRP2 3.715 5.4237 3.4748 9.7184
NCI-H358 GDSC1; GDSC2; CTRP2; CCLE 3.8563 6.4791 3.1956 10.4167
EMC-BAC-2 GDSC1; GDSC2 3.8708 7.7801 1.5321 9.7849
IA-LM GDSC1; GDSC2; CCLE 3.918 5.8375 2.5196 2.9865
NCI-H82 GDSC1; GDSC2 4.0104 9.3418 0.8648 13.3672
NCI-H1781 GDSC1; GDSC2 4.0152 5.8327 2.5866 2.9838
NCI-H1563 GDSC1; GDSC2; CTRP2; CCLE 4.0297 5.6405 3.7319 7.852
COR-L23 GDSC1; GDSC2; CCLE 4.0597 6.8321 2.1372 4.6704
NCI-H1876 GDSC1; GDSC2 4.061 11.9588 -0.3971 19.6936
HCC33 GDSC2 4.0639 6.3998 2.3488 4.308
NCI-H2286 CTRP2; CCLE 4.0901 6.197 3.5593 8.3673
LXF 289 GDSC1; GDSC2; CTRP2 4.1405 6.4059 3.5162 8.4116
COLO 677 CCLE 4.1542 6.6905 2.005 3.1055
Hs 229.T CCLE 4.2031 6.8791 1.9479 3.3106
NCI-H2369 GDSC1; GDSC2 4.2043 5.7189 2.7544 1.6967
LC-2/ad GDSC1; GDSC2 4.2351 6.7355 2.303 4.2284
NCI-H3255 GDSC1; GDSC2; CCLE 4.2412 6.7474 2.3014 3.5198
GLC-82 CCLE 4.2457 7.0959 1.8737 3.61
NCI-H2461 GDSC1; GDSC2 4.32 6.426 2.5018 2.9077
NCI-H1568 GDSC1; GDSC2; CTRP2; CCLE 4.3373 6.3568 3.7345 7.0421
Calu-6 GDSC1; GDSC2; CTRP2; CCLE 4.3416 6.3113 3.76 6.9284
NCI-H1581 GDSC1; GDSC2; CTRP2; CCLE 4.3651 6.3475 3.7663 6.8453
NCI-H290 GDSC1; GDSC2 4.3664 6.1977 2.633 2.101
NCI-H1975 GDSC1; GDSC2; CCLE 4.375 7.0092 2.2646 3.4811
NCI-H1341 GDSC1; GDSC2; CTRP2; CCLE 4.3753 5.3085 4.2282 4.9898
NCI-H2405 GDSC1; GDSC2; CTRP2 4.3819 6.8987 3.5203 7.8109
SBC-3 GDSC1; GDSC2 4.3905 6.3708 2.5691 2.4116
NCI-H345 GDSC1; GDSC2 4.3992 5.5535 2.925 0.6381
COR-L279 GDSC1; GDSC2 4.4246 6.4895 2.5354 2.5416
NCI-H2171 GDSC2 4.4351 6.8418 2.3805 3.3952
CPC-N GDSC1; GDSC2 4.4705 9.7319 1.0164 11.3472
Lu-99A GDSC1; GDSC2 4.4887 6.5833 2.5304 2.4659
SBC-1 GDSC1; GDSC2 4.4981 7.3736 2.1723 4.4826
NCI-H1436 GDSC1; GDSC2 4.4983 6.922 2.3822 3.2742
NCI-H1048 GDSC1; GDSC2; CCLE 4.5122 6.6204 2.5273 2.0371
NCI-H847 GDSC1; GDSC2 4.5165 7.4321 2.1567 4.5389
NCI-H524 GDSC1; GDSC2 4.5273 7.4677 2.1469 4.5754
SW900 CCLE 4.5336 6.7114 2.2128 1.6423
LCLC-97TM1 GDSC1; GDSC2; CTRP2 4.5353 8.432 2.9097 10.0032
IST-SL1 GDSC1; GDSC2 4.5671 6.7279 2.5106 2.4508
NCI-H1993 GDSC1; GDSC2 4.5855 6.5316 2.6076 1.9125
SK-LU-1 GDSC1; GDSC2; CTRP2; CCLE 4.5979 8.0885 3.1359 8.9265
NCI-H1666 GDSC1; GDSC2; CTRP2; CCLE 4.6039 10.4779 1.9524 13.7963
HCC2108 CTRP2 4.6105 8.2928 3.0458 9.276
NCI-H2087 GDSC1; GDSC2; CTRP2; CCLE 4.6333 6.4555 3.9726 5.367
NCI-H2731 GDSC1; GDSC2 4.654 6.7062 2.5686 2.0178
A-427 GDSC1; GDSC2 4.6594 7.1548 2.3721 3.0594
RERF-LC-Sq1 GDSC1; GDSC2 4.6771 8.5079 1.7528 6.5901
NCI-H1573 GDSC1; GDSC2; CTRP2; CCLE 4.6906 5.971 4.2611 4.0457
HCC44 GDSC1; GDSC2; CTRP2; CCLE 4.6962 7.1729 3.6776 6.4544
NCI-H1355 GDSC1; GDSC2; CTRP2; CCLE 4.7011 7.5193 3.5104 7.1428
NCI-H2810 GDSC1; GDSC2 4.7055 7.0143 2.4614 2.5038
EPLC-272H GDSC1; GDSC2; CTRP2 4.709 8.7865 2.887 9.7328
NCI-H1703 GDSC1; GDSC2; CTRP2; CCLE 4.713 6.6545 3.9488 5.2875
HCC1171 CTRP2 4.7199 8.0764 3.2501 8.192
NCI-H64 GDSC1; GDSC2 4.7204 6.7735 2.5751 1.8944
EKVX GDSC1; GDSC2; CTRP2 4.7369 6.9807 3.8094 5.8169
CAL-12T GDSC1; GDSC2; CTRP2; CCLE 4.7701 9.0571 2.8051 9.9488
Ms-1 GDSC1; GDSC2 4.8157 7.6289 2.2492 3.4812
NCI-H2085 GDSC1; GDSC2; CTRP2; CCLE 4.8431 8.1239 3.3338 7.5878
NCI-H1915 GDSC1; GDSC2; CTRP2; CCLE 4.8447 7.6205 3.5864 6.5252
COR-L321 GDSC1; GDSC2 4.859 7.2459 2.4444 2.3705
NCI-H146 GDSC1; GDSC2 4.8628 9.1305 1.5796 7.2213
NCI-H596 GDSC1; GDSC2 4.8686 6.8349 2.6255 1.468
NCI-H187 GDSC1 4.8742 6.4528 2.7837 0.9795
NCI-H2030 GDSC1; GDSC2; CTRP2; CCLE 4.887 7.2826 3.0971 3.043
NCI-H2804 GDSC1; GDSC2 4.8932 9.8717 1.2459 9.0775
IST-SL2 GDSC1; GDSC2 4.9173 8.4573 1.9307 5.0952
LB647-SCLC GDSC1; GDSC2 4.9299 9.1924 1.5942 7.0022
NCI-H2818 GDSC1; GDSC2 4.9348 7.0203 2.581 1.5991
NCI-H1435 GDSC1; GDSC2; CTRP2 4.9895 8.5277 3.2568 7.6196
Lu-165 GDSC1; GDSC2 5.036 10.203 1.1838 9.1266
HOP-62 GDSC1; GDSC2; CTRP2 5.0581 7.2575 3.9492 4.577
NCI-H446 GDSC1; GDSC2; CTRP2 5.0627 7.361 3.9013 4.7696
NCI-H1688 GDSC1; GDSC2 5.0713 8.8583 1.8402 5.3297
NCI-H2591 GDSC1; GDSC2 5.0782 7.9309 2.2642 2.9942
PaCa-3 GDSC1; GDSC2 5.0848 7.6244 2.4014 2.2829
Lu-135 GDSC1; GDSC2 5.094 7.1774 2.5942 1.3654
DMS 454 CTRP2 5.0998 10.2757 2.4747 10.6686
RERF-LC-MS GDSC1; GDSC2; CTRP2; CCLE 5.1241 6.5759 4.344 2.7936
NCI-H2009 GDSC1; GDSC2; CTRP2; CCLE 5.1302 7.8316 3.7216 5.3967
NCI-H748 GDSC2 5.155 7.4132 2.5266 1.6018
NCI-H661 GDSC1; GDSC2; CTRP2; CCLE 5.1566 7.1317 4.0927 3.789
NCI-H2227 GDSC1; GDSC2 5.1627 7.3353 2.5625 1.4334
NCI-H2228 GDSC1; GDSC2; CTRP2; CCLE 5.1737 7.7187 3.8135 4.9298
NCI-H2595 GDSC1; GDSC2 5.1746 7.7656 2.388 2.2337
NCI-H1385 CTRP2 5.1811 6.5293 4.4125 2.4036
NCI-H720 GDSC1; GDSC2 5.1873 6.8725 2.7573 0.6481
Lu-139 GDSC1; GDSC2 5.1904 7.0342 2.6962 0.8627
DV-90 CTRP2; CCLE 5.2104 6.3447 4.5268 1.8754
COR-L303 GDSC2 5.2151 7.014 2.7149 0.7757
NCI-H810 GDSC1; GDSC2; CTRP2; CCLE 5.2188 6.5174 4.4477 2.1913
NCI-H1651 GDSC1; GDSC2; CTRP2; CCLE 5.2209 7.6962 3.8626 4.6372
NCI-H647 GDSC1; GDSC2; CTRP2; CCLE 5.2217 9.008 3.2083 7.3806
NCI-H2373 GDSC1; GDSC2 5.2294 7.05 2.7071 0.7929
DMS 79 GDSC1; GDSC2 5.2314 7.7421 2.4272 1.9753
NCI-H1963 GDSC2 5.2322 6.9983 2.7283 0.7164
NCI-H1694 GDSC1; GDSC2; CTRP2; CCLE 5.2499 6.6046 4.4282 2.2194
NCI-H1838 GDSC1; GDSC2; CTRP2 5.2742 7.559 3.9731 4.0787
HCC827 GDSC1; GDSC2; CTRP2; CCLE 5.2946 9.4904 2.3139 5.7869
NCI-H838 GDSC1; GDSC2; CTRP2 5.2946 6.6258 4.4513 2.0495
COR-L311 GDSC2 5.3016 7.7933 2.441 1.8302
NCI-H1304 GDSC1 5.3136 13.4035 -0.1708 18.1621
LK2 CTRP2 5.3143 6.1578 4.6934 1.0284
NCI-H2803 GDSC1; GDSC2 5.3163 7.2664 2.661 0.8949
NCI-H2029 GDSC1; GDSC2; CTRP2 5.3232 6.5137 4.5271 1.6916
NCI-H2126 CTRP2 5.3434 6.9865 4.3099 2.556
NCI-H211 GDSC1; GDSC2; CTRP2; CCLE 5.3452 7.318 4.1475 3.2277
NCI-H513 GDSC1; GDSC2 5.348 7.0689 2.7501 0.5703
NCI-H2291 GDSC1; GDSC2; CTRP2 5.3481 6.8226 4.3939 2.2008
NCI-H3122 GDSC1; GDSC2 5.3497 7.5031 2.5826 1.1697
NCI-H1105 GDSC1; GDSC2; CTRP2 5.3783 7.1461 4.2572 2.7175
HOP-92 GDSC1; GDSC2; CTRP2 5.3827 9.4439 3.1198 7.4569
NCI-H2066 GDSC1; GDSC2 5.3839 6.9789 2.7979 0.4134
SK-MES-1 GDSC1; GDSC2; CTRP2; CCLE 5.3841 9.1638 3.2605 6.8662
SHP-77 GDSC1; GDSC2; CTRP2; CCLE 5.3845 6.7464 4.4575 1.8828
NCI-H526 GDSC1; GDSC2; CTRP2 5.3989 7.3525 4.1708 3.0419
NCI-H841 GDSC1; GDSC2; CTRP2 5.4006 7.3161 4.19 2.9595
NCI-H441 GDSC1; GDSC2; CTRP2; CCLE 5.4026 8.2901 3.7095 4.9566
Calu-3 GDSC1; GDSC2; CTRP2; CCLE 5.4222 7.6925 4.0205 3.6274
Lu-65 GDSC1; GDSC2; CTRP2 5.4275 7.5245 4.1073 3.2583
COR-L105 GDSC1; GDSC2; CTRP2; CCLE 5.4283 7.8489 3.9479 3.9191
DMS 273 GDSC1; GDSC2; CTRP2 5.4442 7.6472 4.0593 3.4301
NCI-H1092 GDSC1; GDSC2; CCLE 5.4481 7.1688 2.7536 0.4196
NCI-H1693 GDSC1; GDSC2; CTRP2; CCLE 5.4535 7.7314 4.0247 3.5583
NCI-H1944 GDSC1; GDSC2; CTRP2; CCLE 5.454 7.328 4.2234 2.7364
HCC15 GDSC1; GDSC2; CTRP2; CCLE 5.4558 8.245 3.7727 4.6023
HCC2279 CTRP2 5.4769 7.7269 4.0443 3.4389
COLO 699 CTRP2; CCLE 5.4806 7.8035 4.0094 3.5776
NCI-H835 GDSC1; GDSC2 5.4883 8.5279 2.2256 2.6314
NCI-H1155 GDSC1; GDSC2; CTRP2; CCLE 5.4965 8.4498 3.7022 4.827
NCI-H2196 GDSC2; CTRP2 5.4974 7.0095 4.4089 1.9129
LC-1/sq GDSC1; GDSC2 5.4976 7.7248 2.5617 1.1247
NCI-H2444 GDSC1; GDSC2; CTRP2; CCLE 5.4982 7.1505 4.3414 2.1856
NCI-H322M GDSC1; GDSC2 5.5006 12.4853 0.4042 12.3254
Lu-99 CTRP2; CCLE 5.5027 8.0622 3.8983 4.002
NCI-H1770 GDSC1; GDSC2 5.5116 11.2505 1.0002 9.1708
ChaGo-K-1 GDSC1; GDSC2; CTRP2 5.5179 8.2999 3.7925 4.416
NCI-H1373 CTRP2; CCLE 5.5201 8.2512 3.8181 4.3058
HCC1833 CTRP2 5.5347 7.6087 4.1443 2.9356
Sq-1 CTRP2; CCLE 5.5353 8.6336 3.6407 5.018
UMC-11 GDSC1; GDSC2 5.541 7.205 2.7771 0.3953
NCI-H740 GDSC2 5.5451 8.119 2.4253 1.6415
COLO 668 GDSC1; GDSC2; CTRP2 5.5635 7.6762 4.132 2.9416
NCI-H2110 GDSC1; GDSC2; CTRP2 5.5691 7.5717 4.1869 2.7089
NCI-H250 GDSC2 5.5736 7.4405 2.7035 0.582
NCI-H2023 GDSC1; GDSC2; CTRP2; CCLE 5.5741 7.3929 4.2769 2.3358
PC-14 GDSC1; GDSC2; CTRP2; CCLE 5.5778 8.4364 3.7698 4.4118
T3M-10 CTRP2; CCLE 5.5835 7.1955 4.3782 1.9146
NCI-H1836 GDSC1; GDSC2 5.5905 7.1025 2.8323 0.251
SW1573 GDSC1; GDSC2; CTRP2; CCLE 5.5964 9.7732 3.1228 7.0688
DMS 114 GDSC1; GDSC2; CTRP2; CCLE 5.5987 7.2536 4.3606 1.9641
NCI-H1184 CTRP2; CCLE 5.6113 7.8669 4.0732 3.1095
LOU-NH91 GDSC1; GDSC2; CTRP2; CCLE 5.6335 8.3639 3.8463 4.0065
NCI-H2347 GDSC1; GDSC2 5.6346 7.5365 2.6925 0.5807
VMRC-LCD GDSC1; GDSC2; CTRP2; CCLE 5.6481 7.363 4.3414 1.9725
NCI-H23 GDSC1; GDSC2; CTRP2; CCLE 5.6637 7.2423 4.4088 1.6861
NCI-H226 GDSC1; GDSC2; CTRP2; CCLE 5.6827 7.1306 4.4731 1.4127
RERF-LC-KJ GDSC1; GDSC2 5.6893 7.1612 2.8479 0.1934
RERF-LC-Ad2 CTRP2 5.6953 8.8492 3.6534 4.7038
NCI-H2081 GDSC1; GDSC2; CTRP2 5.7153 7.7422 4.2053 2.423
NCI-H650 GDSC1; GDSC2; CTRP2; CCLE 5.7225 9.8546 3.1784 6.6249
NCI-H1623 GDSC1; GDSC2; CTRP2 5.7267 7.2231 4.4575 1.4191
NCI-H292 GDSC1; GDSC2; CTRP2 5.7285 7.1868 4.4754 1.349
SW1271 GDSC1; GDSC2; CTRP2; CCLE 5.7414 8.9135 3.6555 4.6222
EMC-BAC-1 GDSC1; GDSC2 5.7424 12.4895 0.5644 11.0074
HARA [Human squamous cell lung carcinoma] GDSC1; GDSC2; CTRP2; CCLE 5.746 8.2389 3.9873 3.2579
NCI-H522 GDSC1; GDSC2; CTRP2; CCLE 5.7481 7.9325 4.1363 2.6533
NCI-H510A GDSC1; GDSC2 5.7516 7.5154 2.7463 0.3814
NCI-H2869 GDSC1; GDSC2 5.7583 7.7046 2.6801 0.5507
NCI-H727 GDSC1; GDSC2; CTRP2; CCLE 5.7641 7.6467 4.283 2.0485
NCI-H520 GDSC1; GDSC2; CTRP2; CCLE 5.7925 7.4826 4.3781 1.6434
HCC2935 CTRP2; CCLE 5.8038 8.319 3.9886 3.1685
A-549 GDSC1; GDSC2; CTRP2; CCLE 5.814 8.1996 4.0529 2.8954
LCLC-103H GDSC1; GDSC2; CTRP2; CCLE 5.8424 7.8633 4.2315 2.1486
NCI-H2135 GDSC1; GDSC2 5.8691 7.4202 2.8231 0.1894
NCI-H1339 CTRP2; CCLE 5.8809 8.1387 4.1265 2.5107
HCC366 GDSC1; GDSC2; CTRP2 5.888 8.1069 4.1462 2.4239
LK-2 GDSC1; GDSC2 5.8888 7.3105 2.8673 0.1218
NCI-H1299 GDSC1; GDSC2; CTRP2; CCLE 5.8924 8.0577 4.1722 2.316
HCC95 CTRP2 5.8927 7.6619 4.3568 1.6049
NCI-H1650 GDSC1; GDSC2; CTRP2; CCLE 5.897 8.0581 4.175 2.299
Lu-134-A GDSC1; GDSC2 5.9001 13.3714 0.2494 12.2688
KNS-62 GDSC1; GDSC2; CTRP2; CCLE 5.9225 7.996 4.2204 2.09
NCI-H2342 GDSC1; GDSC2; CTRP2 5.9338 9.6652 3.4267 5.2621
NCI-H2722 GDSC1; GDSC2 5.9501 7.3881 2.8624 0.1174
NCI-H196 GDSC1; GDSC2; CTRP2 5.9514 7.9315 4.2685 1.8702
Calu-1 CTRP2; CCLE 5.9698 8.4564 4.0343 2.7567
HCC1588 CTRP2 5.981 7.4413 4.5072 0.9677
NCI-H1395 CTRP2 5.9842 10.5251 3.0424 6.7594
LUDLU-1 CTRP2; CCLE 5.9874 8.0216 4.249 1.9014
NCI-H1437 GDSC1; GDSC2 5.9941 8.7276 2.389 1.3778
HCC1195 CTRP2 6.0248 9.1 3.764 3.7579
NCI-H1869 GDSC1; GDSC2; CTRP2; CCLE 6.0647 10.5842 3.0719 6.5114
RERF-LC-A1 CTRP2; CCLE 6.0758 8.9115 3.8881 3.193
COR-L88 GDSC1; GDSC2; CTRP2 6.0898 8.2713 4.1965 1.9799
COR-L47 CTRP2 6.1399 9.6445 3.5809 4.3306
RERF-LC-Ad1 CTRP2 6.1581 7.1632 4.7077 0.2559
ABC-1 GDSC1; GDSC2 6.1669 8.1786 2.667 0.402
HCC1438 CTRP2 6.2186 9.1146 3.8849 3.0188
DMS 53 GDSC1; GDSC2; CTRP2 6.2352 8.1371 4.3414 1.2991
NCI-H1793 GDSC1; GDSC2; CTRP2; CCLE 6.2469 10.0031 3.4815 4.5781
MOR/CPR CTRP2; CCLE 6.2672 7.0811 4.7809 0.0893
HCC78 GDSC1; GDSC2; CTRP2; CCLE 6.3466 8.2678 4.3449 1.1848
COR-L32 GDSC1; GDSC2 6.3505 8.0547 2.7765 0.1553
COR-L51 CTRP2 6.368 8.4462 4.2787 1.3898
NCI-H69 GDSC1; GDSC2; CTRP2 6.4018 11.9175 2.6629 7.6499
NCI-H460 GDSC1; GDSC2; CTRP2; CCLE 6.4075 8.4456 4.3005 1.2794
HCC4006 CTRP2; CCLE 6.4203 10.6528 3.2874 5.1111
NCI-H2106 CTRP2 6.4349 8.3338 4.3629 1.0503
EBC-1 GDSC1; GDSC2; CTRP2; CCLE 6.4792 9.5359 3.8519 2.8258
NCI-H2122 GDSC1; GDSC2; CTRP2; CCLE 6.4884 9.3758 3.931 2.5181
COR-L95 GDSC1; CTRP2 6.4905 7.9196 4.5593 0.4452
NCI-H1792 GDSC1; GDSC2; CTRP2; CCLE 6.5033 9.3007 3.9741 2.3417
NCI-H2141 GDSC1; GDSC2; CTRP2 6.508 8.4029 4.371 0.9667
NCI-H889 CTRP2 6.5569 8.1499 4.4982 0.5654
SBC-5 GDSC1; GDSC2; CTRP2; CCLE 6.5704 7.5857 4.7157 0.1112
BEN GDSC1; GDSC2; CTRP2 6.5731 7.4672 4.7576 0.0626
LC-1/sq-SF CTRP2; CCLE 6.5764 10.6334 3.4003 4.4513
NCI-H2172 GDSC1; GDSC2; CTRP2; CCLE 6.8552 8.2685 4.5796 0.2492
NCI-H322 CTRP2; CCLE 6.9282 8.4885 4.5276 0.3222
NCI-H2170 GDSC1; GDSC2; CTRP2; CCLE 7.5796 12.7448 3.0457 4.576
Hs 888.Lu CTRP2 4.7885 7.2877 3.7029 6.1529
⏷ Show the Full List of 227 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1; GDSC2 4.9342 7.0459 2.57 1.6517
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 4.6664 6.9782 3.7468 6.2304
ES-2 GDSC1; GDSC2; CCLE 2.9499 6.7162 1.3056 11.5518
TOV-21G GDSC1; GDSC2; CTRP2; CCLE 3.4169 6.0232 2.9302 12.6289
JHOS-4 GDSC1; GDSC2; CCLE 3.9498 6.0947 2.4175 3.4459
COV318 CCLE 3.952 5.8239 2.2804 2.0707
OVMANA CCLE 4.122 10.6725 0.0539 13.0288
OC 315 CCLE 4.278 5.9808 2.3917 1.1703
Caov-3 GDSC2; CTRP2 4.3649 6.6671 3.615 7.4628
OC 316 CCLE 4.3915 6.6881 2.1459 2.1039
OVTOKO GDSC1; GDSC2; CTRP2 4.4691 8.4245 2.8539 10.3776
A2780 GDSC1; GDSC2; CTRP2; CCLE 4.4713 6.1104 3.9817 5.7116
SK-OV-3 GDSC1; GDSC2; CTRP2; CCLE 4.555 6.5852 3.8359 6.1105
OVCAR-3 GDSC1; GDSC2; CCLE 4.6424 7.1789 2.3511 2.668
OVCAR-5 GDSC1; GDSC2; CTRP2 4.976 8.0415 3.4885 6.6731
HEY A8 CTRP2 4.9841 7.1686 3.9316 4.7951
OV-90 GDSC1; GDSC2; CTRP2; CCLE 4.9851 6.8718 4.0808 4.1661
TYK-nu GDSC1; GDSC2; CTRP2; CCLE 4.9985 8.8238 3.1163 8.1911
IGROV-1 GDSC1; GDSC2; CTRP2 5.086 7.6458 3.7782 5.2425
RMG-I GDSC1; GDSC2; CTRP2 5.2463 8.7645 3.3498 6.7418
COV434 CTRP2 5.2566 7.7308 3.8737 4.5265
ONCO-DG-1 CTRP2; CCLE 5.272 8.0004 3.7515 5.0107
JHOM-1 CTRP2 5.3035 8.5385 3.5083 5.9732
MCAS CTRP2; CCLE 5.4149 7.7469 3.9881 3.7741
SNU-119 CTRP2 5.4236 8.3296 3.7061 4.9343
OC 314 GDSC1; GDSC2; CTRP2; CCLE 5.4785 8.5135 3.657 5.0454
OAW28 GDSC1; GDSC2; CTRP2 5.5407 8.6541 3.6346 5.034
EFO-21 GDSC1; GDSC2; CTRP2; CCLE 5.6146 7.6152 4.1976 2.598
TOV-112D GDSC1; GDSC2; CTRP2; CCLE 5.6539 8.2275 3.9278 3.6396
OV56 GDSC1; GDSC2; CTRP2 5.6871 7.5879 4.2602 2.2426
EFO-27 GDSC1; GDSC2; CTRP2 5.7147 7.9286 4.1154 2.7848
Kuramochi GDSC1; GDSC2; CTRP2; CCLE 5.7407 7.51 4.3324 1.8856
Caov-4 GDSC1; GDSC2 5.7479 8.0391 2.5495 0.9747
SNU-8 CTRP2 5.8396 8.2913 4.0263 2.9658
DOV13 GDSC1; GDSC2; CTRP2; CCLE 5.845 9.6005 3.3942 5.5345
OVCAR-8 GDSC1; GDSC2; CTRP2; CCLE 5.8987 8.1145 4.1496 2.3965
ES2 CTRP2 5.9132 10.9245 2.7933 7.8976
OVKATE GDSC1; GDSC2 5.9973 7.4206 2.8677 0.1037
OVSAHO CTRP2; CCLE 5.9978 8.3307 4.1116 2.4173
JHOS-2 GDSC1; GDSC2; CTRP2; CCLE 6.0355 9.1637 3.7407 3.8363
OVCAR-4 GDSC1; GDSC2; CTRP2; CCLE 6.1226 8.315 4.1964 1.9423
OVISE GDSC1; GDSC2; CTRP2 6.2208 8.6639 4.0957 2.2073
COV362 CTRP2 6.3439 11.2327 2.9549 6.5595
OAW42 GDSC1; GDSC2; CTRP2 6.368 7.8612 4.5266 0.6035
JHOC-5 CTRP2 6.4969 8.294 4.411 0.8524
COV504 CCLE 6.5173 8.9097 2.224 0.3626
SNU-840 CTRP2 6.5703 9.7944 3.7885 2.9589
COV644 CTRP2 6.618 8.1872 4.511 0.4984
OVK18 GDSC1; GDSC2; CTRP2 6.6927 8.2857 4.5055 0.4732
OV7 CTRP2 6.9819 18.8252 -0.3055 17.4982
FU-OV-1 GDSC1; GDSC2; CTRP2; CCLE 7.063 8.6761 4.5124 0.3032
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 5.106 7.1003 4.0674 3.9894
Cancer Drug Sensitivity Data Curated from 31 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 5.8442 7.0896 4.5863 0.8242
Aska-SS CTRP2 6.1591 7.8539 4.4238 1.0877
SW872 GDSC1; GDSC2 3.2456 7.0824 1.3778 12.4723
Hs 633.T GDSC1; GDSC2 3.4492 5.1268 2.5233 4.6986
GCT GDSC1; GDSC2; CTRP2; CCLE 4.2418 7.7886 2.957 10.4552
VA-ES-BJ GDSC1; GDSC2 4.2963 9.209 1.1457 11.0241
A-204 GDSC1; GDSC2; CTRP2; CCLE 4.4002 7.228 3.3782 8.355
EW-8 GDSC1; GDSC2 4.4761 6.4078 2.6016 2.1022
Rh18 GDSC1; CTRP2 4.6986 7.8673 3.3353 7.8801
Rh41 GDSC1; GDSC2; CTRP2 4.7343 6.9988 3.7981 5.8697
G-402 GDSC1; GDSC2; CTRP2; CCLE 4.7644 6.4665 4.0884 4.5937
G-401 GDSC1; GDSC2; CTRP2; CCLE 4.9646 6.6603 4.169 3.8364
SW684 GDSC1; GDSC2 4.9757 6.3303 2.8739 0.4092
MFH-ino GDSC1; GDSC2 5.1944 7.1303 2.6601 0.9972
Rh30 GDSC1; GDSC2; CCLE 5.2667 7.0356 2.7287 0.5755
SW982 GDSC1; GDSC2; CTRP2 5.3226 14.1914 0.7006 17.1265
TE 441.T GDSC2; CTRP2 5.3243 8.3877 3.5999 5.5523
SK-LMS-1 GDSC1; GDSC2; CTRP2; CCLE 5.3681 8.1549 3.75 4.8471
TTC-709 CTRP2 5.4967 7.4549 4.1921 2.7981
HT-1080 GDSC1; GDSC2; CTRP2; CCLE 5.5589 8.3648 3.7911 4.3545
KYM-1 GDSC1; GDSC2; CTRP2; CCLE 5.5659 9.0258 3.4699 5.6769
STS-0421 GDSC1; GDSC2 6.0664 8.1788 2.6283 0.54
RKN GDSC1; GDSC2; CTRP2; CCLE 6.138 8.9032 3.9325 2.9364
BT-12 CTRP2 6.2081 7.0824 4.758 0.1387
TE 617.T CTRP2; CCLE 6.219 7.8393 4.4618 0.9095
MES-SA GDSC1; GDSC2; CTRP2; CCLE 6.2717 8.1749 4.3449 1.2528
Tm87-16 CTRP2 6.2735 8.0548 4.398 1.072
SK-UT-1 GDSC1; GDSC2; CTRP2 6.2939 8.2598 4.3199 1.3178
RD GDSC1; GDSC2; CTRP2; CCLE 6.3599 9.588 3.753 3.3519
Hs 729.T CTRP2; CCLE 6.5408 10.4159 3.4799 4.1856
BT-16 CTRP2 7.0671 8.431 4.6023 0.156
⏷ Show the Full List of 31 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 6.2936 8.3534 4.2784 1.4623
H-STS CTRP2 6.4261 7.3731 4.737 0.1141
Cancer Drug Sensitivity Data Curated from 9 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IST-Mes2 CCLE 2.1659 3.691 1.839 8.7308
MSTO-211H GDSC1; GDSC2; CTRP2; CCLE 3.2092 6.1364 2.6652 14.2218
NCI-H2452 GDSC1; GDSC2; CTRP2; CCLE 4.2192 7.0603 3.2869 9.151
NCI-H2052 GDSC1; GDSC2; CTRP2; CCLE 5.089 6.5999 4.3035 3.0294
IST-Mes1 GDSC1; GDSC2; CTRP2; CCLE 5.4513 7.7249 4.0263 3.5553
ACC-MESO-1 CTRP2 5.7437 7.4588 4.3584 1.7802
JL-1 CTRP2 5.8945 8.2254 4.0943 2.6198
NCI-H28 GDSC1; GDSC2; CTRP2; CCLE 5.9566 9.0299 3.7511 3.9073
MPP 89 GDSC1; GDSC2; CTRP2; CCLE 6.004 7.8155 4.3533 1.4925
⏷ Show the Full List of 9 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PC-3 GDSC1; GDSC2; CCLE 4.4678 7.1229 2.2704 3.3067
NCI-H660 GDSC2 4.9197 6.5849 2.752 0.8717
LNCaP clone FGC GDSC1; GDSC2; CTRP2 4.9539 6.6509 4.1646 3.8766
PaCa-3 CTRP2 5.3958 6.8279 4.4258 1.9954
22Rv1 GDSC1; GDSC2; CTRP2; CCLE 5.7708 9.2966 3.4891 5.2613
DU145 GDSC1; GDSC2; CTRP2; CCLE 6.0886 9.4357 3.6462 4.1406
VCaP GDSC1; GDSC2; CTRP2 7.3075 8.8014 4.5611 0.1595
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 4.4469 7.1799 3.4454 7.9708
A-253 GDSC1; GDSC2; CCLE 4.9412 6.9051 2.6322 1.1305
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1; GDSC2 4.083 6.1966 2.4586 3.6088
Cancer Drug Sensitivity Data Curated from 46 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-39 GDSC1; GDSC2 2.9871 6.9934 1.2002 14.3469
SCH GDSC1; GDSC2 3.6749 6.7496 1.8927 8.0649
ECC10 GDSC1; GDSC2; CTRP2 3.8065 6.8287 2.988 11.373
GSS CTRP2 4.043 5.6683 3.7349 7.8037
BGC-823 CCLE 4.0995 6.7232 1.9555 3.4373
SNU-16 GDSC1; GDSC2; CTRP2; CCLE 4.1959 6.7026 3.4337 8.6082
SNU-216 CTRP2 4.3263 7.7697 3.0452 9.8993
HGC-27 GDSC1; GDSC2; CTRP2; CCLE 4.3292 6.7522 3.54 7.8542
RF-48 GDSC1; GDSC2 4.3739 7.9287 1.8254 6.8003
SK-GT-2 GDSC1; GDSC2 4.4769 7.0951 2.2891 3.8445
Fu97 GDSC1; GDSC2; CTRP2; CCLE 4.5732 6.5326 3.8786 5.8924
OCUM-1 GDSC1; GDSC2; CCLE 4.7084 7.6777 2.1624 3.4594
NCC-StC-K140 CTRP2 4.7229 7.9364 3.3224 7.8831
TGBC11TKB GDSC1; GDSC2 4.7914 7.1076 2.468 2.3441
SNU-1 GDSC1; GDSC2; CTRP2; CCLE 4.8173 6.4442 4.1473 4.2335
MKN28 GDSC1; GDSC2 4.9541 7.3182 2.4641 2.1414
NUGC-3 GDSC1; GDSC2; CTRP2; CCLE 5.0632 8.308 3.4282 6.7568
SNU-620 CTRP2 5.0953 6.3145 4.4513 2.3964
MKN7 GDSC1; GDSC2; CTRP2; CCLE 5.1138 7.6841 3.7819 5.1741
GCIY GDSC1; GDSC2; CCLE 5.1717 6.7409 2.8006 0.4317
SNU-5 GDSC1; GDSC2; CTRP2 5.1777 7.5997 3.876 4.6599
KATO III GDSC1; GDSC2; CTRP2 5.2091 6.7843 4.3076 2.7932
23132/87 GDSC1; GDSC2; CTRP2 5.2493 6.7852 4.3382 2.5956
NCI-N87 GDSC1; GDSC2; CTRP2; CCLE 5.3404 7.1063 4.2486 2.8154
SNU-668 CTRP2 5.4667 6.8091 4.4844 1.6528
AZ-521 CCLE 5.5313 8.2167 2.0782 1.2458
LMSU CTRP2 5.5492 8.2621 3.8344 4.191
SNU-601 CTRP2 5.6318 7.6731 4.1816 2.6375
TMK-1 GDSC1; GDSC2 5.7492 7.388 2.7907 0.2835
Hs 746.T GDSC1; GDSC2; CTRP2; CCLE 5.7652 7.3144 4.4391 1.4435
MKN74 CTRP2; CCLE 5.8146 8.448 3.9338 3.3743
ECC12 GDSC2; CTRP2 5.9126 7.2679 4.5457 0.8996
SH-10-TC CTRP2; CCLE 5.9686 8.6471 3.9429 3.1205
GSU CTRP2 5.9724 6.7792 4.7755 0.1879
NUGC-4 GDSC1; GDSC2; CTRP2; CCLE 6.2128 7.7626 4.4912 0.8205
SNU-719 CTRP2 6.3518 8.4964 4.2477 1.5132
RERF-GC-1B GDSC1; GDSC2; CCLE 6.3566 8.5499 2.6064 0.3898
KE-39 CTRP2; CCLE 6.3785 9.164 3.9617 2.5291
MKN45 GDSC1; GDSC2; CTRP2; CCLE 6.4484 9.3363 3.925 2.5862
AGS GDSC1; GDSC2; CTRP2 6.5927 9.02 4.1504 1.6199
MKN1 GDSC1; GDSC2; CTRP2 6.6792 8.2416 4.5167 0.453
HuG1-N CTRP2 6.7472 8.4107 4.4807 0.5059
IM95 GDSC1; GDSC2; CTRP2; CCLE 7.6819 9.3544 4.505 0.1562
SNU-1077 CTRP2 4.926 6.9337 3.9993 4.6267
SNG-M GDSC1; GDSC2; CTRP2; CCLE 4.9789 8.405 3.3092 7.4203
SNU-685 CTRP2 5.0546 8.613 3.2686 7.4438
⏷ Show the Full List of 46 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 18 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
K5 GDSC1; GDSC2 0.5527 4.5269 -0.0976 31.0077
HTC-C3 GDSC1; GDSC2 1.0402 5.631 -0.0326 28.4399
8305C GDSC1; GDSC2; CTRP2; CCLE 2.3149 9.2488 0.387 25.1475
IHH-4 GDSC1; GDSC2 3.1117 6.503 1.553 11.7988
B-CPAP GDSC1; GDSC2; CTRP2; CCLE 3.1664 8.3772 1.6368 18.3521
BHT-101 GDSC1; GDSC2; CTRP2 3.8507 10.438 1.298 18.0157
8505C GDSC1; GDSC2; CTRP2; CCLE 3.9042 9.4625 1.8256 15.8342
WRO GDSC1; GDSC2 4.0651 5.83 2.6199 2.6917
KMH-2 GDSC1; GDSC2 4.1396 5.6773 2.7357 1.9011
ML-1 [Human leukemia] GDSC1; GDSC2; CTRP2 4.3702 7.3393 3.2959 8.7632
CGTH-W-1 GDSC1; GDSC2; CTRP2 4.7453 6.5871 4.0115 4.9556
SW579 CTRP2; CCLE 4.9189 7.3843 3.7683 5.6109
FTC-238 CTRP2 5.3435 7.4414 4.0852 3.4903
TT GDSC1; GDSC2; CTRP2 5.645 7.9131 4.0745 3.0532
TT2609-C02 GDSC1; GDSC2; CTRP2; CCLE 5.7847 8.7376 3.7725 4.0751
ASH-3 GDSC1; GDSC2 5.8623 7.2784 2.869 0.1244
FTC-133 GDSC1; GDSC2; CTRP2 6.0355 8.9324 3.8514 3.3933
CAL-62 GDSC1; GDSC2; CTRP2 6.9665 8.3931 4.5777 0.2185
⏷ Show the Full List of 18 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 57 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
BB49-HNC GDSC1; GDSC2 3.7517 5.914 2.3643 4.9222
HO-1-N-1 GDSC1; GDSC2 3.8248 5.7251 2.5092 3.8546
KON GDSC1; GDSC2 3.8507 6.3878 2.2043 5.6781
KOSC-2 GDSC1; GDSC2 3.9924 15.3378 -2.1368 26.444
BICR 10 GDSC1; GDSC2 4.0578 6.3073 2.3891 4.0782
BB30-HNC GDSC1; GDSC2 4.1287 6.5673 2.3124 4.3912
YD-10B CTRP2 4.176 6.4337 3.5389 8.2317
PCI-04B GDSC1; GDSC2 4.1896 9.111 1.1148 11.4678
PCI-06A GDSC1; GDSC2 4.2057 6.5892 2.3531 3.9898
PCI-15A GDSC1; GDSC2 4.2552 6.2967 2.5217 2.9095
BICR 78 GDSC1; GDSC2 4.2716 6.7244 2.3321 3.9834
SNU-1214 CTRP2 4.3001 7.7901 3.0108 10.1006
JHU-029 GDSC1; GDSC2 4.3497 6.6958 2.3952 3.4658
DOK GDSC1; GDSC2 4.3513 7.4974 2.0172 5.697
JHU-011 GDSC1; GDSC2 4.362 9.7873 0.9098 12.216
SAS GDSC1; GDSC2 4.385 7.019 2.2665 4.1491
OSC-20 GDSC1; GDSC2 4.4651 7.6669 2.0123 5.4904
SCC-25 GDSC1; GDSC2; CTRP2; CCLE 4.6838 6.4906 4.0025 5.129
SNU-899 CTRP2 4.8076 7.7667 3.4812 7.0425
PCI-38 GDSC1 4.8101 9.9036 1.1736 11.7722
SKN-3 GDSC1; GDSC2 4.8186 9.9614 1.1516 9.7769
SCC-15 GDSC1; GDSC2 4.8423 9.6462 1.3196 8.765
HO-1-u-1 GDSC1; GDSC2 4.9639 6.7089 2.7227 0.9495
OSC-19 GDSC1; GDSC2 4.987 6.8828 2.6634 1.1738
JHU-022 GDSC1; GDSC2 5.2742 7.6397 2.4913 1.6321
PE/CA-PJ34 (clone C12) CTRP2 5.3673 8.2029 3.7255 4.9509
YD-8 CTRP2 5.3798 7.7491 3.9604 3.9486
BICR 18 CTRP2 5.3801 7.37 4.1481 3.1669
SNU-1076 CTRP2 5.3834 7.9783 3.8495 4.4052
Detroit 562 GDSC1; GDSC2; CTRP2; CCLE 5.4216 8.1654 3.786 4.6044
BHY GDSC1; GDSC2; CTRP2 5.4564 8.6036 3.5954 5.3401
PCI-30 GDSC1; GDSC2 5.5106 7.4176 2.6862 0.6729
CAL-27 GDSC1; GDSC2; CTRP2; CCLE 5.5391 7.3058 4.2947 2.3146
CAL-33 GDSC1; GDSC2; CTRP2 5.6117 8.2435 3.8895 3.8631
HSC-2 GDSC1; GDSC2; CTRP2; CCLE 5.629 7.9629 4.039 3.2223
Ca9-22 GDSC1; GDSC2 5.6446 7.3516 2.7641 0.3826
PE/CA-PJ15 GDSC1; GDSC2; CTRP2 5.6667 8.5841 3.7626 4.2991
FaDu GDSC1; GDSC2; CTRP2; CCLE 5.6769 7.8775 4.1141 2.8452
BICR 22 GDSC1; GDSC2; CTRP2 5.6785 8.0673 4.0233 3.2117
SNU-1066 CTRP2 5.6915 8.7098 3.719 4.4395
HSC-4 GDSC1; GDSC2; CTRP2 5.7105 8.6081 3.7826 4.1481
BICR 31 GDSC2; CTRP2 5.7269 7.9256 4.1252 2.728
SNU-1041 CTRP2 5.8452 8.215 4.0666 2.7972
PE/CA-PJ49 CTRP2 5.8488 7.4615 4.4222 1.4099
SNU-46 CTRP2 5.8626 9.4662 3.4728 5.1838
PE/CA-PJ41 (clone D2) CTRP2 5.8941 8.4395 3.9921 3.0272
BICR 16 CTRP2 5.9346 9.5482 3.4844 5.0248
SCC-9 GDSC1; GDSC2; CTRP2; CCLE 6.0306 9.3789 3.6338 4.274
SAT [Human HNSCC] GDSC1; GDSC2 6.0308 13.655 0.2011 12.2409
LB771-HNC GDSC1; GDSC2 6.0721 13.1342 0.4748 10.8117
BICR 6 CTRP2 6.1584 9.4164 3.7026 3.8173
HSC-3 GDSC1; GDSC2; CTRP2 6.1695 10.7962 3.0437 6.4642
NCI-H3118 GDSC1; GDSC2 6.1719 8.0702 2.7073 0.3144
UPCI-SCC-090 GDSC1; GDSC2 6.1896 8.0898 2.707 0.3094
Hs 840.T CCLE 7.1021 10.0851 2.0263 0.5546
BICR 56 CTRP2 7.4494 13.3 2.7074 6.0098
SCC-4 GDSC1; GDSC2; CTRP2 7.8345 19.2386 0.1168 14.8053
⏷ Show the Full List of 57 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
5637 GDSC1; GDSC2; CTRP2; CCLE 3.7543 6.3373 3.1532 10.8503
BFTC-905 GDSC1; GDSC2 3.8727 5.9022 2.457 4.0668
JMSU-1 CTRP2; CCLE 4.0688 6.7809 3.2718 9.5756
SW780 GDSC1; GDSC2; CCLE 4.5774 6.5152 2.6103 1.5905
U-BLC1 CTRP2 4.6896 9.0492 2.7391 10.3891
HT-1376 GDSC1; GDSC2; CTRP2; CCLE 5.038 8.8415 3.1405 8.0132
253J CTRP2 5.2048 7.2734 4.0606 3.8358
KMBC-2 CTRP2; CCLE 5.265 8.6161 3.4389 6.3341
T24 GDSC1; GDSC2; CTRP2; CCLE 5.3861 9.3748 3.157 7.2954
RT-112 GDSC1; GDSC2; CTRP2; CCLE 5.4297 6.8651 4.4317 1.9198
VM-CUB-1 CTRP2 5.4302 8.1717 3.7895 4.5754
SW1710 GDSC1; GDSC2; CTRP2 5.5802 7.8861 4.0416 3.2865
HT-1197 GDSC1; GDSC2; CTRP2; CCLE 5.6414 8.0556 4.0027 3.3521
BC-3C CTRP2 5.6499 10.3155 2.8949 7.9226
KU-19-19 GDSC1; GDSC2; CTRP2 5.7427 7.5737 4.3036 1.9957
SCaBER CTRP2; CCLE 5.807 7.9949 4.1461 2.5327
UM-UC-3 GDSC1; GDSC2; CTRP2; CCLE 5.8608 9.1861 3.6082 4.6314
UM-UC-1 CTRP2 6.0244 7.6725 4.4292 1.1974
TCCSUP GDSC1; GDSC2; CTRP2; CCLE 6.2155 9.4215 3.738 3.5993
J82 GDSC1; GDSC2; CTRP2; CCLE 6.4432 9.6271 3.7874 3.1153
639V GDSC1; GDSC2; CTRP2; CCLE 6.5012 7.4636 4.733 0.103
RT-4 GDSC1; GDSC2; CTRP2; CCLE 6.6505 8.6927 4.3211 1.0124
647V GDSC1; GDSC2; CTRP2 6.6777 8.1126 4.5655 0.3429
CAL-29 GDSC1; GDSC2; CTRP2 6.9556 8.7747 4.4304 0.5227
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PA-1 GDSC1; GDSC2 2.3274 4.3906 1.8328 12.7843
NT2-D1 GDSC1; GDSC2 3.3539 6.7604 1.6293 10.5997
SKN GDSC1; GDSC2 3.7195 6.7115 1.946 7.6151
KGN GDSC1; GDSC2 3.8573 7.0533 1.8815 7.6662
DoTc2 4510 GDSC1; GDSC2 4.0989 6.1397 2.496 3.3547
SiSo GDSC1; GDSC2 4.1984 6.709 2.2913 4.3729
SW954 GDSC1; GDSC2 4.2354 7.9318 1.7269 7.7064
HEY GDSC1; GDSC2 4.3325 6.7845 2.3429 3.802
JAR GDSC1; GDSC2 4.3405 6.1166 2.6544 2.0255
SKG-IIIa GDSC1; GDSC2 4.391 6.5943 2.4675 2.9777
UWB1.289 GDSC1; GDSC2 4.4365 6.978 2.3182 3.7504
OV17R GDSC1; GDSC2 4.4608 6.7003 2.461 2.895
LB831-BLC GDSC1; GDSC2 4.4842 6.6119 2.5149 2.5577
C-33 A GDSC1; GDSC2 4.5047 6.4982 2.5776 2.187
OMC-1 [Human cervical carcinoma] GDSC1; GDSC2 4.5312 6.4979 2.5925 2.0688
DSH1 GDSC1; GDSC2 4.5621 7.0664 2.3545 3.32
C-4-I GDSC1; GDSC2 4.588 6.3189 2.7006 1.4445
JEG-3 GDSC1; GDSC2 4.6307 6.2771 2.7399 1.2087
NCC-IT GDSC2 4.7032 10.202 0.954 11.1531
Ca Ski GDSC1; GDSC2 4.711 7.4059 2.2886 3.4366
HEC-1 GDSC1; GDSC2 4.7139 7.2461 2.3626 3.0236
SiHa GDSC1; GDSC2 4.7944 5.913 2.9551 0.2758
SW962 GDSC1; GDSC2 4.8493 6.6799 2.6804 1.2401
CAL-39 GDSC1; GDSC2 4.911 6.7969 2.6621 1.2562
NEC8 GDSC1; GDSC2 4.9789 6.7941 2.6955 1.0467
PWR-1E GDSC1; GDSC2 4.9958 7.2653 2.5086 1.8703
ME-180 GDSC1; GDSC2 5.0717 8.6782 1.9234 4.8614
ACC-OV7 GDSC1; GDSC2 5.0986 15.1787 -1.1988 20.4239
MS751 GDSC1; GDSC2 5.0999 6.6301 2.8126 0.524
JHOS-3 GDSC1; GDSC2 5.3029 7.1838 2.6873 0.8098
PEO1 GDSC1; GDSC2 5.3221 7.3433 2.6335 0.9939
TC-YIK GDSC1; GDSC2 5.5503 7.8319 2.5431 1.1525
OVCA420 GDSC1; GDSC2 5.5601 7.1404 2.8076 0.3143
SW756 GDSC1; GDSC2 5.5702 7.3725 2.7273 0.5146
BPH-1 GDSC1; GDSC2 5.6208 8.3678 2.3597 1.8507
OVMIU GDSC1; GDSC2 5.6832 9.3505 1.9737 3.6328
HT-3 GDSC1; GDSC2 5.8164 7.6289 2.7304 0.3929
OVCA433 GDSC1; GDSC2 5.986 7.8403 2.7192 0.353
HeLa GDSC1; GDSC2; CTRP2 6.4971 7.9245 4.5603 0.4395
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug

References

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