General Information of Drug (ID: DMFLCW4)

Drug Name
AZD8931
Synonyms
Sapitinib; AZD8931; 848942-61-0; AZD8931 (Sapitinib); AZD-8931; Sapitinib(AZD8931); UNII-3499328002; CHEMBL2408045; 2-(4-((4-((3-Chloro-2-fluorophenyl)amino)-7-methoxyquinazolin-6-yl)oxy)piperidin-1-yl)-n-methylacetamide; 2-[4-({4-[(3-chloro-2-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}oxy)piperidin-1-yl]-N-methylacetamide; Sapitinib [INN]; 4-(3-chloro-2-fluoroanilino)-7-methoxy-6-((1-(n-methylcarbamoylmethyl)piperidin-4-yl)oxy)quinazoline
Indication
Disease Entry ICD 11 Status REF
Breast cancer 2C60-2C65 Phase 2 [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 473.9
Logarithm of the Partition Coefficient (xlogp) 4
Rotatable Bond Count (rotbonds) 7
Hydrogen Bond Donor Count (hbonddonor) 2
Hydrogen Bond Acceptor Count (hbondacc) 8
Chemical Identifiers
Formula
C23H25ClFN5O3
IUPAC Name
2-[4-[4-(3-chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypiperidin-1-yl]-N-methylacetamide
Canonical SMILES
CNC(=O)CN1CCC(CC1)OC2=C(C=C3C(=C2)C(=NC=N3)NC4=C(C(=CC=C4)Cl)F)OC
InChI
InChI=1S/C23H25ClFN5O3/c1-26-21(31)12-30-8-6-14(7-9-30)33-20-10-15-18(11-19(20)32-2)27-13-28-23(15)29-17-5-3-4-16(24)22(17)25/h3-5,10-11,13-14H,6-9,12H2,1-2H3,(H,26,31)(H,27,28,29)
InChIKey
DFJSJLGUIXFDJP-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
11488320
ChEBI ID
CHEBI:132986
CAS Number
848942-61-0
UNII
3499328002
DrugBank ID
DB12183
TTD ID
D0BM7M

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Erbb2 tyrosine kinase receptor (HER2) TT6EO5L ERBB2_HUMAN Inhibitor [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Breast cancer
ICD Disease Classification 2C60-2C65
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Erbb2 tyrosine kinase receptor (HER2) DTT ERBB2 5.67E-03 -1.26 -2.05
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 77 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1 2.0279 4.2896 1.5643 19.377
RPMI-3460/CS1 GDSC2 4.3795 6.634 2.4423 2.8549
ES4 GDSC1 0.6274 9.3541 -2.1549 42.4666
ES8 GDSC1 0.9487 2.7137 0.8691 30.1659
ES7 GDSC1 1.0232 2.8644 0.9217 29.3761
HuO9 GDSC1 1.084 3.3063 0.8838 29.2449
EW-1 GDSC1 1.201 3.0581 1.0737 27.327
ES1 GDSC1 1.2759 2.9245 1.1837 26.166
SJSA-1 GDSC1 1.8556 4.9125 1.1197 23.3713
U2OS GDSC1 1.9387 5.9293 0.7409 25.4025
CHSA0011 GDSC1 2.0408 7.3336 0.169 28.134
EW-7 GDSC1 2.0578 4.8658 1.3472 20.7708
NY GDSC1 2.0858 3.6076 1.8854 16.7939
SaOS-2 GDSC1 2.1062 3.9499 1.7832 17.4052
H-EMC-SS GDSC1 2.1524 5.0461 1.3616 20.2004
A-673 GDSC1 2.1781 3.1062 2.1252 14.6387
MHH-ES-1 GDSC1 2.2447 5.8466 1.0787 21.7241
NOS-1 [Human HNSCC] GDSC1 2.3146 5.4594 1.3301 19.6478
ES5 GDSC1 2.3766 4.3043 1.921 15.0266
CAL-78 GDSC1 2.5002 4.939 1.7567 15.6613
HOS GDSC1 2.5206 3.5619 2.3718 11.0189
CHSA0108 GDSC1 2.6186 6.2576 1.2334 18.9574
EW-22 GDSC1 2.6414 3.9855 2.3323 10.68
G-292 clone A141B1 GDSC1 2.8161 5.0783 1.9933 12.4574
CAL-72 GDSC1 2.8219 4.4779 2.2882 10.1645
CHSA8926 GDSC1 2.8486 7.9361 0.6094 22.0709
MG-63 GDSC1 2.9265 3.9112 2.6563 6.8827
SK-ES-1 GDSC1 2.951 4.3827 2.4577 8.2898
CADO-ES1 GDSC1 3.0271 7.3051 1.0796 18.3214
HuO-3N1 GDSC1 3.0866 5.075 2.2423 9.4045
SK-PN-DW GDSC1 3.1586 4.7699 2.4577 7.4315
TC-71 GDSC1 3.3814 9.209 0.4278 21.0592
CHSA8926 GDSC2 3.5191 6.1145 2.0863 6.6047
ES6 GDSC1 3.7368 5.7653 2.4264 5.6939
EW-13 GDSC1 3.9548 6.0461 2.4444 4.9352
CHSA0011 GDSC2 4 7.8253 0.8113 5.6231
NOS-1 [Human HNSCC] GDSC2 4.0593 7.6469 1.7389 7.3243
MG-63 GDSC2 4.0767 11.9553 -0.383 18.1844
EW-11 GDSC1 4.1881 7.1063 2.0939 6.9405
ES8 GDSC2 4.1922 6.1212 2.5639 2.5272
CHSA0108 GDSC2 4.2592 13.3451 -1.6703 17.9012
EW-7 GDSC2 4.2966 11.5806 -0.0259 16.0237
HuO-3N1 GDSC2 4.4094 7.5139 2.0483 4.9018
EW-24 GDSC1 4.4843 6.4909 2.5692 2.8179
U-CH2 GDSC2 4.545 6.2883 1.7483 0.4691
EW-12 GDSC2 4.593 6.7744 1.5846 0.9632
SK-PN-DW GDSC2 4.6768 6.8196 2.5314 1.9793
ES6 GDSC2 4.8383 13.2295 -0.4319 16.6077
EW-18 GDSC1 4.8509 8.9636 1.6509 8.4175
EW-3 GDSC1 4.994 9.0133 1.7198 7.593
U2OS GDSC2 5.0215 7.6967 2.3359 2.4563
NY GDSC2 5.0469 8.6758 1.9095 4.5345
CAL-72 GDSC2 5.0954 6.9096 2.7028 0.8312
CAL-78 GDSC2 5.1571 6.5613 2.8611 0.3209
EW-18 GDSC2 5.2268 7.29 2.6113 1.0582
ES7 GDSC2 5.281 8.2773 2.2236 2.6514
G-292 clone A141B1 GDSC2 5.3215 10.9487 1.0186 8.6603
HOS GDSC2 5.3653 6.6652 2.9026 0.168
H-EMC-SS GDSC2 5.3689 8.0453 2.3691 1.8974
EW-11 GDSC2 5.4106 7.9715 2.4208 1.6379
CADO-ES1 GDSC2 5.4145 6.9412 2.8234 0.3044
TC-71 GDSC2 5.4224 6.8378 2.8632 0.2211
ES1 GDSC2 5.4735 7.3793 2.6852 0.6358
EW-1 GDSC2 5.4764 8.1375 2.3843 1.7228
EW-24 GDSC2 5.4961 7.3537 2.7042 0.5678
A-673 GDSC2 5.4972 6.9134 2.8642 0.1977
SJSA-1 GDSC2 5.5013 7.596 2.6138 0.8419
ES5 GDSC2 5.5571 8.0813 1.4917 0.67
HuO9 GDSC2 5.5891 8.2502 2.3927 1.5801
EW-13 GDSC2 5.6882 7.4252 2.7544 0.3526
EW-22 GDSC2 5.811 7.666 2.7149 0.3935
SaOS-2 GDSC2 5.9215 12.603 0.6278 9.5103
SK-ES-1 GDSC2 6.0445 7.6463 2.8079 0.1569
MHH-ES-1 GDSC2 6.1707 7.9069 2.7635 0.1933
ES4 GDSC2 6.5968 15.2419 -0.1796 12.011
EW-3 GDSC2 6.826 9.1475 2.5706 0.3433
EW-16 GDSC2 7.5059 19.1257 -1.4241 15.3569
⏷ Show the Full List of 77 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 320 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JM1 GDSC1 2.9776 4.0591 2.6381 6.7849
JM1 GDSC2 5.235 17.4388 -2.9677 20.6807
EoL-1 GDSC1 0.0314 1.0894 0.0304 41.1373
CTV-1 GDSC1 0.4523 1.7701 0.4424 35.9311
SU-DHL-16 GDSC2 0.4524 4.3329 -0.4784 23.8593
CTV-1 GDSC2 0.6906 2.6644 0.5994 24.4229
SUP-B8 GDSC2 0.7753 5.7364 -0.799 24.2314
MLMA GDSC1 0.8669 2.603 0.7992 31.1118
Jurkat GDSC1 1.0669 3.0814 0.9222 29.1057
697 GDSC1 1.2333 2.6219 1.1885 26.3921
SU-DHL-5 GDSC1 1.3908 3.3386 1.2099 25.3156
SUP-M2 GDSC1 1.4324 3.2165 1.2877 24.5585
JeKo-1 GDSC1 1.5466 3.0669 1.4477 22.8307
TK [Human B-cell lymphoma] GDSC1 1.559 3.8991 1.2144 24.3255
BE-13 GDSC1 1.6145 3.0707 1.5206 21.9501
SU-DHL-6 GDSC2 1.6466 3.6022 1.41 16.4289
WSU-NHL GDSC2 1.7084 4.6071 1.0977 17.8094
WSU-DLCL2 GDSC2 1.7211 12.8537 -2.8359 33.1431
Sc-1 GDSC1 1.7419 3.8859 1.4163 21.9377
SR GDSC1 1.7939 3.1386 1.7006 19.7059
BL-41 GDSC1 1.8028 3.7912 1.5157 20.9166
H9 GDSC1 1.8275 5.0716 1.0209 24.1783
RPMI-8402 GDSC1 1.8299 3.1617 1.7344 19.2705
OCI-Ly7 GDSC1 1.8852 2.9315 1.8407 18.2433
RCH-ACV GDSC1 1.8964 2.9319 1.8527 18.0989
Karpas-231 GDSC1 1.8971 3.318 1.7681 18.6567
WSU-NHL GDSC1 1.9104 2.8904 1.8742 17.8752
SU-DHL-16 GDSC1 1.9127 3.0098 1.8566 17.976
JVM-2 GDSC1 1.9262 8.4501 -0.4815 31.6541
NB4 GDSC1 1.9727 3.0515 1.9135 17.2462
EoL-1 GDSC2 1.9749 4.9736 1.2147 16.2171
AMO1 GDSC1 1.9753 3.1001 1.9064 17.2776
HC-1 GDSC1 2.0045 3.4318 1.8527 17.4715
BONNA-12 GDSC2 2.0808 5.7429 0.4065 12.7983
SU-DHL-6 GDSC1 2.1265 3.2355 2.0399 15.5071
KCL-22 GDSC1 2.1313 3.2574 2.0396 15.4812
A4/Fukuda GDSC1 2.1383 3.9456 1.8189 16.9816
DoHH2 GDSC2 2.143 3.4726 1.5914 5.1734
Karpas-1106P GDSC1 2.1579 4.1741 1.7484 17.3867
ALL-SIL GDSC1 2.1669 3.3315 2.0588 15.1481
Hs 445 GDSC1 2.2001 3.7195 1.9699 15.5804
Kasumi-1 GDSC1 2.2004 3.7247 1.9684 15.5895
RPMI-8866 GDSC1 2.2237 3.5576 2.0517 14.8784
KE-37 GDSC1 2.227 2.9418 2.2053 13.8244
Namalwa GDSC1 2.2367 3.5728 2.0607 14.7448
NU-DUL-1 GDSC2 2.2461 9.0621 -1.1116 20.7019
OCI-AML-3 GDSC1 2.2491 3.0299 2.216 13.622
SU-DHL-10 GDSC1 2.2496 2.888 2.2354 13.4941
BALL-1 GDSC1 2.2508 3.2139 2.1806 13.8454
GR-ST GDSC1 2.2662 5.6376 1.1987 20.7992
MV4-11 GDSC1 2.2828 6.5154 0.7938 23.4099
TUR GDSC1 2.2995 3.08 2.2617 13.0231
U-698-M GDSC1 2.3042 3.4768 2.1654 13.6458
KOPN-8 GDSC1 2.3051 3.1977 2.2435 13.1098
ATN-1 GDSC1 2.3392 3.366 2.2371 12.9568
K-562 GDSC1 2.41 3.4442 2.2908 12.1914
Kasumi-1 GDSC2 2.4178 5.1199 1.0021 8.0786
RS4;11 GDSC1 2.4343 4.2656 1.9972 14.1797
L-363 GDSC1 2.4408 3.5623 2.2854 12.0586
Farage GDSC2 2.4448 4.48 1.3435 5.8463
MOLM-13 GDSC1 2.4479 4.987 1.6829 16.4537
JURL-MK1 GDSC1 2.4761 3.9259 2.1848 12.5931
MOLM-16 GDSC1 2.483 3.437 2.3726 11.2206
Daudi GDSC1 2.4889 4.3272 2.026 13.6987
OCI-AML-5 GDSC1 2.5007 3.2914 2.4339 10.7021
VAL GDSC1 2.5111 6.2659 1.1295 20.154
SKM-1 GDSC1 2.5507 3.4597 2.439 10.3854
GDM-1 GDSC1 2.5613 4.2157 2.1494 12.4294
Karpas-45 GDSC1 2.5939 3.5476 2.4561 10.03
OCI-M1 GDSC1 2.5947 3.4723 2.4827 9.8395
JVM-3 GDSC2 2.6218 7.1666 0.7889 16.4053
ML-2 GDSC1 2.6583 3.7302 2.4562 9.6885
P12-Ichikawa GDSC1 2.6632 3.549 2.5303 9.1331
DG-75 GDSC1 2.672 4.5064 2.1282 12.0649
HDLM-2 GDSC1 2.7381 4.5721 2.1622 11.5047
SUP-HD1 GDSC1 2.7637 4.3421 2.2953 10.3738
DND-41 GDSC1 2.7782 4.132 2.4067 9.4628
PL-21 GDSC1 2.7813 4.319 2.3234 10.0798
JJN-3 GDSC1 2.7859 3.7511 2.5821 8.1205
KY821 GDSC1 2.7963 3.746 2.5951 7.9727
SU-DHL-4 GDSC1 2.7975 3.6994 2.6156 7.8169
KM-H2 GDSC1 2.818 4.0256 2.4952 8.6087
SIG-M5 GDSC2 2.8406 4.8134 1.4776 4.0132
OCI-Ly19 GDSC1 2.862 5.3315 1.9121 12.8881
P32/ISH GDSC1 2.8634 6.106 1.5315 15.763
RPMI-6666 GDSC2 2.8849 7.7173 0.7502 15.8279
JSC-1 GDSC1 2.8962 4.3401 2.4256 8.7779
GA-10 GDSC2 2.9297 7.534 0.8807 14.9964
LC4-1 GDSC1 2.9344 4.3287 2.4679 8.284
MN-60 GDSC1 2.9503 5.9025 1.7102 14.0666
Karpas-1106P GDSC2 2.9549 5.2337 2.0453 8.3765
NCI-H929 GDSC1 2.9561 5.5177 1.906 12.5459
SU-DHL-4 GDSC2 3.0035 4.5054 1.7324 2.154
WIL2 NS GDSC1 3.0212 4.3693 2.5305 7.4236
P30/OHK GDSC1 3.029 5.39 2.0346 11.2553
MC116 GDSC2 3.0663 12.1 -1.9615 22.0898
NB4 GDSC2 3.1283 4.8075 1.6696 2.2908
JURL-MK1 GDSC2 3.1291 4.9417 1.608 2.6419
SU-DHL-5 GDSC2 3.1412 5.6046 2.0267 7.9441
Jiyoye GDSC2 3.1448 7.3517 1.1576 12.8675
HL-60 GDSC1 3.1628 4.4456 2.6226 6.1202
H9 GDSC2 3.168 6.0442 1.8305 8.9943
Karpas-422 GDSC1 3.1762 7.6287 1.0459 17.9648
NU-DUL-1 GDSC1 3.1817 4.691 2.5173 6.8727
HEL GDSC1 3.2 4.8301 2.464 7.221
L-540 GDSC1 3.2324 4.7769 2.5185 6.6678
CTB-1 GDSC1 3.234 5.7326 2.0426 10.3994
BC-3 GDSC2 3.247 5.7294 1.3137 4.1407
THP-1 GDSC1 3.2755 4.7943 2.5467 6.2843
OPM-2 GDSC1 3.2911 4.8541 2.53 6.3582
NOMO-1 GDSC1 3.303 4.7064 2.6139 5.653
EJM GDSC1 3.3036 5.0724 2.4314 7.0898
MV4-11 GDSC2 3.3202 11.8142 -0.9256 22.4352
JVM-2 GDSC2 3.3302 7.0001 1.4897 10.4993
Granta-519 GDSC1 3.3342 5.4856 2.2503 8.4033
RCH-ACV GDSC2 3.3362 5.1972 1.6158 2.2427
RPMI-8866 GDSC2 3.3533 5.9267 1.2895 4.0751
U266B1 GDSC1 3.3789 4.9897 2.535 6.0031
VAL GDSC2 3.3926 7.6922 1.1954 11.9874
CA46 GDSC1 3.3992 7.6133 1.2403 15.7863
NALM-6 GDSC1 3.4046 4.9653 2.5681 5.6526
L-428 GDSC1 3.4312 5.4472 2.3489 7.2852
CRO-AP2 GDSC1 3.4363 5.3146 2.4192 6.7147
ALL-PO GDSC1 3.46 5.8156 2.1882 8.4472
HL-60 GDSC2 3.5212 5.8118 2.239 5.7242
VL51 GDSC1 3.534 5.6921 2.3086 7.2531
CESS GDSC2 3.5617 4.9127 2.7165 2.8991
MOLM-13 GDSC2 3.5628 5.6658 2.3442 5.0209
MEG-01 GDSC1 3.5807 8.0362 1.1768 15.576
EM-2 GDSC1 3.5934 6.904 1.7518 11.3568
CML-T1 GDSC1 3.6123 5.2738 2.5762 4.9095
RL GDSC2 3.6214 6.0655 1.3901 3.0219
MHH-PREB-1 GDSC1 3.6256 7.9275 1.2671 14.7895
SKM-1 GDSC2 3.6376 5.3502 1.7128 1.3269
BV-173 GDSC1 3.6475 7.0626 1.7155 11.4469
Jiyoye GDSC1 3.6813 9.0452 0.754 18.0102
CML-T1 GDSC2 3.7109 5.4701 2.5523 3.5006
CTB-1 GDSC2 3.7207 10.1361 -0.4896 13.5318
MOLT-4 GDSC1 3.7306 9.2098 0.7112 18.1051
PF-382 GDSC2 3.7424 5.2455 2.684 2.6971
SUP-T1 GDSC2 3.7475 5.8291 2.4029 4.264
JVM-3 GDSC1 3.7601 10.2017 0.24 20.7604
Ku812 GDSC1 3.8056 6.5207 2.1055 7.9619
SR GDSC2 3.8171 5.4018 2.6601 2.6813
HT GDSC2 3.8182 6.6675 1.2331 3.5661
MC116 GDSC1 3.8405 8.2425 1.2793 13.9729
MOLT-13 GDSC2 3.858 6.595 2.1078 5.6896
EB2 GDSC1 3.8586 5.6595 2.5645 4.2868
GR-ST GDSC2 3.8646 6.5043 2.1573 5.396
RPMI-8402 GDSC2 3.8764 6.5964 2.1207 5.5767
A3/Kawakami GDSC1 3.879 6.5208 2.1596 7.3237
MOLT-16 GDSC1 3.9021 6.7277 2.075 7.9015
CESS GDSC1 3.9515 7.2447 1.8573 9.4022
EB2 GDSC2 3.9556 8.6845 1.1487 10.8381
SUP-B8 GDSC1 3.9577 6.262 2.3421 5.7024
Raji GDSC1 3.9635 7.4041 1.7877 9.8871
SK-MM-2 GDSC1 3.9779 6.7245 2.1315 7.2475
Ramos.2G6.4C10 GDSC1 4.018 9.8936 0.5966 17.8325
MLMA GDSC2 4.0241 10.8221 0.1398 15.8946
KMS-11 GDSC1 4.0247 9.088 1.0016 15.2546
OCI-AML-5 GDSC2 4.03 5.727 1.7454 0.8055
Ku812 GDSC2 4.0313 5.9427 2.5451 2.9065
P12-Ichikawa GDSC2 4.0434 7.2835 1.9055 6.4254
QIMR-WIL GDSC2 4.0499 12.6988 -1.5063 17.6788
RPMI-6666 GDSC1 4.0535 11.5394 -0.1942 22.0296
MY-M12 GDSC2 4.0826 11.9989 -1.1392 15.9262
ST486 GDSC2 4.0856 7.3523 1.9023 6.353
JeKo-1 GDSC2 4.0962 7.9782 0.8001 5.511
A3/Kawakami GDSC2 4.1031 6.1178 2.5091 2.971
HAL-01 GDSC1 4.1097 9.8746 0.6767 17.0462
KMOE-2 GDSC2 4.1172 5.9658 2.5894 2.519
GDM-1 GDSC2 4.1309 9.4632 0.8967 11.786
SCC-3 GDSC2 4.1435 5.3264 2.8932 0.9657
KMS-11 GDSC2 4.152 9.6878 0.0299 9.7412
PF-382 GDSC1 4.1521 6.3618 2.4257 4.5645
HEL GDSC2 4.1615 5.5882 1.853 0.3725
GA-10 GDSC1 4.1746 12.0458 -0.3514 22.3942
CMK GDSC1 4.1815 5.8453 2.6842 2.6379
RC-K8 GDSC2 4.1874 6.271 2.4912 2.9189
Mono-Mac-6 GDSC1 4.1982 7.7034 1.8116 9.0119
KG-1 GDSC1 4.2018 6.2527 2.5088 3.838
MOLT-13 GDSC1 4.2467 7.9045 1.7481 9.3394
MEG-01 GDSC2 4.2601 6.8297 2.2748 3.9504
CCRF-CEM GDSC1 4.2701 9.7814 0.8443 15.4907
LAMA-84 GDSC2 4.2719 6.6776 2.3543 3.5009
MHH-PREB-1 GDSC2 4.277 6.392 2.491 2.7684
ALL-SIL GDSC2 4.289 6.2858 2.5474 2.4566
DEL GDSC1 4.2907 13.2564 -0.8629 24.2883
DEL GDSC2 4.3255 5.4592 2.9287 0.6288
ARH-77 GDSC1 4.3535 10.2506 0.6752 16.2826
IM-9 GDSC1 4.3724 7.1968 2.1744 5.8639
OCI-M1 GDSC2 4.3729 5.8564 2.7863 1.178
KY821 GDSC2 4.3732 6.4159 2.5384 2.3718
TALL-1 [Human adult T-ALL] GDSC2 4.3774 8.3056 0.8199 4.9149
OCI-Ly7 GDSC2 4.3774 5.718 1.8886 0.2073
P32/ISH GDSC2 4.3814 6.8389 2.3485 3.3425
NOMO-1 GDSC2 4.3828 6.1825 2.649 1.8082
EHEB GDSC1 4.3973 7.0137 2.2769 5.057
Karpas-299 GDSC1 4.4162 8.6676 1.497 10.661
DB GDSC2 4.4332 6.0451 2.7369 1.3297
QIMR-WIL GDSC1 4.4334 10.5946 0.5652 16.6988
Daudi GDSC2 4.4428 7.8694 1.9009 5.6404
HH [Human lymphoma] GDSC1 4.4473 6.8953 2.3633 4.3213
P30/OHK GDSC2 4.448 6.9383 2.3438 3.2558
MOLT-4 GDSC2 4.4637 6.304 2.6406 1.74
ALL-PO GDSC2 4.4677 7.9519 1.8781 5.7166
U266B1 GDSC2 4.4833 7.1654 2.2603 3.635
WSU-DLCL2 GDSC1 4.4876 5.8426 2.8496 1.0841
Jurkat GDSC2 4.4916 5.9316 2.8148 0.9274
HH [Human lymphoma] GDSC2 4.4934 6.4224 2.6048 1.8716
OCI-AML-3 GDSC2 4.5004 7.1981 2.2558 3.6297
HC-1 GDSC2 4.503 6.5603 2.5489 2.1294
THP-1 GDSC2 4.51 6.1462 1.7863 0.3856
BC-1 GDSC2 4.5107 8.669 1.5626 7.3522
KG-1 GDSC2 4.5114 6.474 2.592 1.9087
HT GDSC1 4.5278 11.0435 0.4142 17.2916
L-363 GDSC2 4.5583 6.583 2.57 1.9517
MOLP-8 GDSC1 4.5671 7.0552 2.3627 4.0642
Mono-Mac-6 GDSC2 4.5683 7.218 2.2886 3.347
Karpas-422 GDSC2 4.5947 9.1976 1.3653 8.2519
L-540 GDSC2 4.6054 6.6199 2.5798 1.8432
BC-1 GDSC1 4.6168 9.8865 1.0462 13.1506
CCRF-CEM GDSC2 4.6235 6.3477 2.7066 1.2473
BL-41 GDSC2 4.6268 5.8652 2.9041 0.4839
SUP-M2 GDSC2 4.6421 9.4724 1.2653 8.6928
LP-1 GDSC2 4.6467 6.5525 1.6915 0.5771
ROS-50 GDSC2 4.648 7.8272 1.1809 2.6487
ML-2 GDSC2 4.6581 6.3906 2.7061 1.2126
L-1236 GDSC2 4.6685 8.2282 1.8798 5.3342
U-698-M GDSC2 4.6747 8.8981 1.5648 7.0166
AMO1 GDSC2 4.6969 6.3429 2.7451 1.0115
Farage GDSC1 4.7264 7.2017 2.3898 3.5546
NK-92MI GDSC2 4.7264 6.2415 1.8335 0.2085
YT GDSC2 4.7296 6.1278 2.8469 0.6029
RC-K8 GDSC1 4.7344 6.9412 2.5097 2.7501
BE-13 GDSC2 4.7432 7.338 2.3382 2.8267
SUP-B15 GDSC2 4.7604 6.438 2.7368 0.9852
OCI-Ly19 GDSC2 4.7737 6.8515 1.6317 0.6847
ME1 GDSC1 4.8078 6.0984 2.8919 0.5629
LP-1 GDSC1 4.8156 7.0702 2.4975 2.6879
CA46 GDSC2 4.816 9.5136 1.3653 7.8116
NKM-1 GDSC1 4.8304 9.3928 1.433 9.9738
ROS-50 GDSC1 4.8332 7.5477 2.296 3.9762
Loucy GDSC2 4.834 7.184 2.4579 2.1233
KOPN-8 GDSC2 4.8693 11.1399 0.6154 11.6071
ME1 GDSC2 4.8762 6.2444 2.8652 0.4496
OCI-AML-2 GDSC1 4.8763 6.2546 2.8614 0.6318
WIL2 NS GDSC2 4.8926 6.6076 2.7304 0.8932
LAMA-84 GDSC1 4.8941 8.5363 1.8795 6.7196
HAL-01 GDSC2 4.9024 8.6245 1.8435 5.1158
Karpas-45 GDSC2 4.9497 7.5281 2.3704 2.386
KE-37 GDSC2 4.9544 6.4819 2.8076 0.5786
K-562 GDSC2 4.9578 6.6914 2.7269 0.8524
Raji GDSC2 4.9665 7.9233 2.2042 3.1681
A4/Fukuda GDSC2 4.9667 7.2137 2.5155 1.7022
MHH-CALL-2 GDSC1 4.9977 6.6373 2.7662 0.9386
Namalwa GDSC2 5.0215 10.2921 1.1313 8.6473
RL GDSC1 5.0295 12.5383 0.0478 17.8322
Karpas-620 GDSC1 5.048 6.9073 2.682 1.2934
Loucy GDSC1 5.0592 6.8311 2.7175 1.1061
MOLM-16 GDSC2 5.0614 6.9915 1.6939 0.3814
L-428 GDSC2 5.0783 6.8442 2.7209 0.7808
KMOE-2 GDSC1 5.0821 7.7221 2.3577 3.1179
L-1236 GDSC1 5.0831 7.4635 2.4693 2.431
SK-MM-2 GDSC2 5.1112 6.9062 2.7112 0.7902
TK [Human B-cell lymphoma] GDSC2 5.1183 6.4642 2.8813 0.2898
SU-DHL-8 GDSC1 5.1232 6.8072 2.755 0.8724
EJM GDSC2 5.1418 7.2684 2.58 1.253
P31/FUJ GDSC2 5.1486 6.0719 3.028 0.0493
SU-DHL-1 GDSC2 5.1586 19.9407 -4.2496 24.6669
MN-60 GDSC2 5.1611 7.0873 2.6621 0.9252
CRO-AP2 GDSC2 5.1673 7.0632 1.708 0.3144
Reh GDSC1 5.1695 6.8283 2.7666 0.7832
MHH-CALL-4 GDSC2 5.1901 18.8828 -3.7068 23.0906
P31/FUJ GDSC1 5.1907 6.2413 2.9857 0.1188
MHH-CALL-2 GDSC2 5.1909 6.5187 2.8895 0.2445
RPMI-8226 GDSC1 5.198 11.7877 0.5322 14.6971
OCI-AML-2 GDSC2 5.2154 6.8099 2.7927 0.47
Ramos.2G6.4C10 GDSC2 5.2195 6.9235 2.7515 0.5872
BALL-1 GDSC2 5.2307 7.2796 2.6172 1.0329
IM-9 GDSC2 5.259 6.5801 2.8933 0.2144
MM1.S GDSC2 5.2729 7.2009 2.6674 0.8226
ST486 GDSC1 5.2843 6.9874 2.7544 0.7414
Karpas-299 GDSC2 5.2857 6.8634 2.8013 0.4119
MOLP-8 GDSC2 5.318 6.9852 2.7691 0.4814
VL51 GDSC2 5.3394 7.3394 2.6427 0.8588
OPM-2 GDSC2 5.34 7.0804 2.7425 0.5443
MOLT-16 GDSC2 5.369 6.9997 2.7843 0.4161
Reh GDSC2 5.3807 7.1435 2.7355 0.5417
PL-21 GDSC2 5.3852 7.6637 1.5765 0.5287
JSC-1 GDSC2 5.3865 7.3299 2.667 0.7459
SU-DHL-10 GDSC2 5.4053 6.5236 2.9649 0.0768
ARH-77 GDSC2 5.4158 7.2193 2.7215 0.5624
Karpas-231 GDSC2 5.4388 6.5712 2.9605 0.0767
KMS-12-BM GDSC2 5.4946 7.1272 2.7872 0.3546
Hs 445 GDSC2 5.5167 7.0008 2.8408 0.2345
ATN-1 GDSC2 5.5311 7.0981 2.8117 0.2872
DND-41 GDSC2 5.5318 7.1659 2.7876 0.3388
SU-DHL-8 GDSC2 5.5353 6.8855 2.8877 0.1508
NCI-H929 GDSC2 5.5374 6.8776 2.8911 0.1453
697 GDSC2 5.5463 7.1263 2.8074 0.2909
SUP-HD1 GDSC2 5.5568 7.5763 2.6453 0.7062
YT GDSC1 5.5587 7.2775 2.7576 0.545
RS4;11 GDSC2 5.567 7.3861 2.721 0.4856
Granta-519 GDSC2 5.584 7.2696 2.7704 0.3573
LC4-1 GDSC2 5.6066 13.3179 0.0761 12.7081
DB GDSC1 5.6402 7.2392 2.8026 0.3685
DG-75 GDSC2 5.6634 7.7459 2.6257 0.7015
Karpas-620 GDSC2 5.6947 7.0686 2.8815 0.1268
EM-2 GDSC2 5.6955 7.1504 2.8538 0.1653
TUR GDSC2 5.7063 7.199 2.841 0.1826
RPMI-8226 GDSC2 5.7973 7.6157 2.7277 0.37
HDLM-2 GDSC2 5.8379 7.8152 2.6711 0.4865
KM-H2 GDSC2 5.8819 7.6658 2.742 0.3097
SUP-T1 GDSC1 5.897 7.4032 2.8388 0.1979
JJN-3 GDSC2 5.923 7.8272 2.7 0.3834
BV-173 GDSC2 5.9958 8.0482 2.6482 0.4732
KCL-22 GDSC2 6.2782 8.1622 2.714 0.245
NKM-1 GDSC2 6.329 8.1792 2.7265 0.213
NALM-6 GDSC2 6.9348 17.7226 -1.1356 15.2848
⏷ Show the Full List of 320 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KYAE-1 GDSC1 -3.4828 0.679 -3.5843 75.6016
KYSE-220 GDSC1 -3.4651 12.0799 -7.4899 59.481
SK-GT-4 GDSC1 -0.1015 9.4955 -2.9356 46.9166
ESO-26 GDSC1 0.0989 6.2298 -1.2644 44.0515
KYAE-1 GDSC2 0.1444 3.5578 -0.2129 30.6076
TE-12 GDSC1 0.4951 10.4685 -2.8137 43.9546
OACP4 C GDSC1 0.7874 10.3088 -2.4572 42.1593
FLO-1 GDSC1 1.8601 4.0413 1.4854 20.8172
TE-12 GDSC2 1.902 17.3245 -5.5321 34.8683
HCE-4 GDSC1 2.0118 3.6408 1.7939 17.8367
KYSE-50 GDSC1 2.3113 6.0402 1.0501 21.6049
OACM5.1 C GDSC2 3.5043 7.125 1.5702 9.5909
OACM5.1 C GDSC1 3.6132 7.1514 1.6441 12.0978
ESO-51 GDSC1 3.6552 6.8162 1.8442 10.4472
ESO-26 GDSC2 3.8779 12.7361 -0.9302 20.9849
FLO-1 GDSC2 4.1233 11.0643 0.0967 15.8593
OACP4 C GDSC2 4.2456 11.358 0.0453 15.8095
KYSE-50 GDSC2 4.4218 11.1943 0.2606 14.3585
KYSE-220 GDSC2 4.52 17.2582 -2.6746 25.3472
SK-GT-4 GDSC2 5.2035 18.0307 -2.5293 23.4206
HCE-4 GDSC2 5.5344 7.4339 1.7122 0.2086
ESO-51 GDSC2 6.1121 7.9675 2.7212 0.2778
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1 4.6997 7.865 2.0702 5.8288
COLO 684 GDSC2 5.6084 7.7195 2.6125 0.7756
Cancer Drug Sensitivity Data Curated from 60 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SJNB-12 GDSC1 -1.3 24.1423 -11.1529 51.3292
NB69 GDSC1 0.0212 6.2673 -1.3611 44.7141
Kelly GDSC1 0.1803 10.5712 -3.1663 45.7244
CHP-212 GDSC1 0.4287 2.7223 0.3056 36.8596
GI-ME-N GDSC1 0.6387 3.1944 0.4275 34.7709
SJNB-5 GDSC1 0.7559 19.4499 -6.969 45.8715
NB1 GDSC1 1.414 3.7325 1.1147 25.8106
NB69 GDSC2 1.5618 14.1486 -3.6202 35.3051
GOTO GDSC1 1.5639 3.7564 1.2693 23.9281
SK-N-AS GDSC1 1.8757 4.084 1.4855 20.7336
KP-N-RT-BM-1 GDSC2 1.9294 9.3703 -1.5345 23.6278
SJNB-10 GDSC1 2.0078 3.0772 1.9464 16.8221
SJNB-7 GDSC1 2.0508 17.9922 -5.0976 40.927
SK-N-SH GDSC1 2.2388 3.3124 2.1425 14.1702
SK-N-DZ GDSC1 2.309 4.2563 1.8718 15.7236
TGW GDSC1 2.542 3.4011 2.4479 10.372
NH-12 GDSC1 2.5847 5.2971 1.6684 15.9389
KP-N-YN GDSC1 2.5974 3.9904 2.2846 11.2498
SJNB-14 GDSC1 2.6599 3.6641 2.4839 9.48
SK-N-FI GDSC1 2.7951 4.0558 2.4583 8.9945
LA-N-6 GDSC1 2.953 6.1253 1.602 14.8714
SJNB-6 GDSC1 3.0174 6.1632 1.6401 14.3269
SJNB-17 GDSC1 3.1418 5.0747 2.2913 8.8033
SiMa GDSC1 3.1475 4.9616 2.3526 8.2999
SJNB-13 GDSC1 3.1839 4.7223 2.5036 6.9717
CHP-126 GDSC1 3.2814 5.1718 2.363 7.7102
NB(TU)1 GDSC1 3.4015 5.4133 2.3418 7.4453
SJNB-6 GDSC2 3.4303 12.1149 -1.6843 19.9827
CHP-212 GDSC2 3.6816 7.1731 1.6873 8.486
SK-N-BE(2)-M17 GDSC1 3.9108 7.0234 1.9361 8.9324
SK-N-MC-IXC GDSC2 3.9773 5.5225 1.8018 0.6405
NB1 GDSC2 4.033 6.5238 2.2679 4.8666
SJNB-17 GDSC2 4.0815 9.4883 0.0779 9.6239
SiMa GDSC2 4.1365 6.8291 2.192 4.6375
GI-ME-N GDSC2 4.3046 7.079 2.1857 4.3511
SK-N-DZ GDSC2 4.5109 6.3894 2.629 1.7331
CHP-126 GDSC2 4.5286 6.1584 1.7891 0.3707
SK-N-BE(2)-M17 GDSC2 4.5376 6.2014 2.7246 1.2637
SK-N-FI GDSC2 4.6213 6.7965 2.5107 2.1518
MHH-NB-11 GDSC2 4.6251 8.1437 1.0324 3.4146
SK-N-MC-IXC GDSC1 4.7014 5.8041 2.9583 0.3891
NH-12 GDSC2 4.7616 6.8445 2.5663 1.7121
LA-N-6 GDSC2 4.8564 6.523 1.7829 0.2646
SK-N-SH GDSC2 4.8615 10.1406 1.0947 9.1534
IMR-5 GDSC1 4.9313 12.5144 -0.0118 18.4206
NB(TU)1 GDSC2 5.0048 16.3251 -1.836 21.6478
Kelly GDSC2 5.0977 6.4775 2.8683 0.3291
TGW GDSC2 5.1895 7.0764 2.6792 0.8431
SJNB-5 GDSC2 5.2429 15.2694 -1.9088 16.7501
SJNB-7 GDSC2 5.3248 7.1389 2.7139 0.6379
KP-N-YS GDSC2 5.3382 7.3262 1.6788 0.3181
SJNB-14 GDSC2 5.3882 7.4003 2.6404 0.8318
SJNB-13 GDSC2 5.405 7.2097 2.7207 0.5708
CHP-134 GDSC2 5.4329 7.0374 2.7957 0.36
IMR-5 GDSC2 5.7054 7.4972 2.735 0.3896
SK-N-AS GDSC2 5.8772 8.1013 2.5806 0.7113
GOTO GDSC2 5.9173 7.9094 2.6679 0.4594
SJNB-12 GDSC2 5.9188 8.4602 2.4605 1.0617
SJNB-10 GDSC2 6.0328 13.5199 0.2666 11.0189
KP-N-YN GDSC2 6.4208 8.8756 2.5132 0.617
⏷ Show the Full List of 60 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuCC-T1 GDSC1 2.5031 6.2806 1.1149 20.2897
HuCC-T1 GDSC2 5.136 16.65 -1.8973 21.5671
Cancer Drug Sensitivity Data Curated from 100 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-175-VII GDSC2 -2.8198 1.2293 -2.9468 55.2622
HCC1599 GDSC1 -2.5368 11.4193 -6.253 57.0378
MDA-MB-175-VII GDSC1 -2.3685 2.1161 -2.6054 65.5223
AU565 GDSC1 -0.8333 2.4112 -1.0005 51.6972
UACC-893 GDSC2 -0.345 4.3163 -1.3006 31.322
MDA-MB-468 GDSC1 0.3164 7.9424 -1.8023 43.5686
BT-474 GDSC1 0.4081 5.3212 -0.5622 40.4044
OCUB-M GDSC1 0.4251 2.1948 0.3821 36.4649
HDQ-P1 GDSC2 0.5062 10.1597 -2.6555 36.7365
UACC-893 GDSC1 0.5299 3.7929 0.1344 36.9883
AU565 GDSC2 0.6192 6.8198 -0.9882 31.582
EFM-192A GDSC1 0.6235 4.426 0.0159 36.8716
HCC1954 GDSC1 0.7075 5.0462 -0.135 36.9397
HCC1806 GDSC1 0.8088 2.9102 0.6798 32.209
BT-20 GDSC1 0.8524 6.1135 -0.4364 37.1621
CAL-85-1 GDSC1 0.9274 6.4072 -0.4906 36.906
ZR-75-30 GDSC1 0.946 5.5496 -0.095 35.2754
HCC1419 GDSC1 0.9716 4.9152 0.1968 33.7969
BT-474 GDSC2 1.0986 6.7846 -0.4892 27.7408
Evsa-T GDSC1 1.1457 3.3907 0.9278 28.595
HCC2157 GDSC1 1.2028 5.7754 0.0713 33.0134
MDA-MB-330 GDSC1 1.2068 40.7242 -17.1698 47.393
HCC202 GDSC1 1.2938 4.937 0.5263 30.1407
HCC1187 GDSC1 1.3625 3.088 1.2426 25.2665
MDA-MB-330 GDSC2 1.4552 8.05 -1.293 24.0516
HCC70 GDSC1 1.4718 7.2413 -0.3333 33.2977
JIMT-1 GDSC1 1.5117 5.8153 0.3673 29.7932
ZR-75-30 GDSC2 1.5123 7.346 -0.3434 25.585
HCC1143 GDSC1 1.5574 10.4655 -1.8093 37.4852
MDA-MB-361 GDSC1 1.5843 6.0812 0.319 29.6591
MDA-MB-453 GDSC1 1.6098 4.2484 1.1384 24.5552
OCUB-M GDSC2 1.6486 5.0215 0.8592 19.2248
COLO 824 GDSC1 1.6679 3.8078 1.3642 22.7029
HCC1395 GDSC1 1.8076 4.5751 1.2148 22.9744
HCC2218 GDSC2 1.84 6.3975 -0.1302 16.7169
HCC2218 GDSC1 1.9288 6.407 0.5063 26.8488
UACC-812 GDSC2 1.9378 7.0223 0.2212 21.4733
HCC38 GDSC1 2.1878 4.7942 1.5113 18.9542
CAL-120 GDSC1 2.1924 4.3539 1.7091 17.4954
HCC2157 GDSC2 2.3337 10.5798 -1.1602 26.1456
EFM-192A GDSC2 2.4227 8.3501 0.0241 20.852
CAL-51 GDSC1 2.502 3.3705 2.4134 10.8343
MCF-7 GDSC1 2.5546 4.603 1.967 13.829
BT-549 GDSC1 2.685 4.4187 2.1818 11.5994
MDA-MB-157 GDSC1 2.7557 5.2871 1.8351 13.9287
Hs 578T GDSC1 2.7623 4.2755 2.3249 10.1556
HCC1569 GDSC1 2.8122 7.421 0.8335 20.8253
CAMA-1 GDSC1 2.8216 3.9771 2.5206 8.4013
MDA-MB-415 GDSC1 2.9647 5.6216 1.8623 12.8467
DU4475 GDSC1 2.9917 4.3677 2.5036 7.7585
MRK-nu-1 GDSC1 2.9999 4.1241 2.6287 6.7571
MFM-223 GDSC1 3.0208 4.8479 2.2955 9.255
EFM-19 GDSC1 3.0384 5.2125 2.131 10.4672
MDA-MB-468 GDSC2 3.0795 14.4279 -2.4343 28.1478
HCC1419 GDSC2 3.0867 9.7317 -0.081 19.3757
MDA-MB-231 GDSC1 3.1764 5.4088 2.1549 9.7392
HCC1806 GDSC2 3.1814 15.478 -2.8736 29.0791
MDA-MB-436 GDSC1 3.2064 4.7067 2.531 6.669
HCC1937 GDSC1 3.3091 7.3769 1.2838 15.8129
HDQ-P1 GDSC1 3.6158 14.6635 -2.1059 30.7088
Hs 578T GDSC2 3.644 6.6042 1.9408 7.1103
HCC1569 GDSC2 3.7703 10.7755 -0.7669 14.8054
Evsa-T GDSC2 3.9609 6.1856 2.3813 3.9265
HCC1428 GDSC1 4.0725 8.8644 1.1487 14.1175
HCC38 GDSC2 4.2582 7.3694 2.0153 5.3549
MDA-MB-453 GDSC2 4.2722 10.6579 0.4126 13.9164
HCC1428 GDSC2 4.2764 6.1315 2.6104 2.1476
HCC1954 GDSC2 4.3493 9.5779 1.0033 10.6879
DU4475 GDSC2 4.3924 6.6054 2.4633 2.7169
T-47D GDSC1 4.4145 8.4251 1.6136 9.837
HCC1500 GDSC1 4.5113 6.8283 2.4328 3.6945
MDA-MB-361 GDSC2 4.624 17.3915 -2.6594 25.0236
MRK-nu-1 GDSC2 4.7086 6.3368 2.7534 0.9644
MDA-MB-415 GDSC2 4.7567 6.4861 2.7152 1.0717
HCC1143 GDSC2 4.7929 15.6836 -1.6799 21.5407
HCC1599 GDSC2 4.7996 6.8257 1.6519 0.6074
CAMA-1 GDSC2 4.8904 7.5388 2.3326 2.6378
MDA-MB-231 GDSC2 4.9098 8.8763 1.7303 5.681
MDA-MB-436 GDSC2 4.9174 7.4564 2.3841 2.356
BT-483 GDSC1 4.957 20.4087 -3.8999 31.4023
CAL-120 GDSC2 5.0097 6.8237 2.6979 0.9138
BT-20 GDSC2 5.0836 14.1091 -0.6832 17.0938
EFM-19 GDSC2 5.1204 10.4913 1.1026 8.5814
CAL-51 GDSC2 5.2871 10.1376 1.3796 6.8469
JIMT-1 GDSC2 5.4191 14.3981 -0.5805 15.9506
CAL-148 GDSC2 5.4444 7.177 2.7491 0.4699
BT-549 GDSC2 5.4865 8.6445 2.1745 2.616
YMB-1-E GDSC2 5.5204 7.8875 1.5478 0.5415
MCF-7 GDSC2 5.5447 7.2601 2.7584 0.4003
HCC1187 GDSC2 5.6197 7.2209 2.8014 0.2771
MFM-223 GDSC2 5.696 8.937 2.1589 2.4432
HCC1500 GDSC2 5.8562 7.429 2.8155 0.1866
HCC1395 GDSC2 5.9458 10.4106 1.6517 4.4641
HCC70 GDSC2 5.9859 8.2902 2.5544 0.7236
COLO 824 GDSC2 6.019 8.8477 2.3527 1.3581
T-47D GDSC2 6.1058 13.005 0.5573 9.4973
BT-483 GDSC2 6.268 13.348 0.4998 9.4894
HCC1937 GDSC2 6.7519 16.1177 -0.4929 13.0336
CAL-85-1 GDSC2 6.8326 15.8496 -0.3135 12.1441
MDA-MB-157 GDSC2 7.1069 18.4691 -1.3768 15.8408
⏷ Show the Full List of 100 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 109 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNB-75 GDSC1 0.4924 11.3089 -3.2198 44.3853
D-542MG GDSC1 0.5791 26.3492 -10.5504 47.3484
PFSK-1 GDSC1 0.7561 1.9052 0.7484 32.1209
Becker GDSC1 0.7607 2.0502 0.746 32.1073
KALS-1 GDSC1 0.8314 3.8769 0.4344 33.4681
YH-13 GDSC1 0.8827 2.4586 0.8364 30.7808
Daoy GDSC1 1.094 2.2451 1.0793 27.9421
U-251MG GDSC1 1.3524 3.7791 1.0324 26.7048
H4 GDSC1 1.5239 2.9203 1.453 22.9302
SK-MG-1 GDSC1 1.5247 3.7511 1.2286 24.4234
SF539 GDSC1 1.6321 3.1157 1.5297 21.7863
SF268 GDSC1 1.7062 5.4733 0.7182 26.7378
KS-1 [Human Krukenberg tumour] GDSC1 1.8547 6.4398 0.4187 27.7146
SF126 GDSC1 1.8595 3.8487 1.5564 20.3242
U-87MG ATCC GDSC1 1.8768 11.5222 -2.0371 36.6866
MOG-G-UVW GDSC1 2.0008 3.4697 1.8373 17.5982
GI-1 GDSC1 2.0548 3.3029 1.9443 16.5632
T98G GDSC1 2.2077 3.752 1.9663 15.5649
M059J GDSC1 2.2251 4.8986 1.5019 18.8405
NMC-G1 GDSC1 2.2369 4.4691 1.7054 17.3007
D-247MG GDSC1 2.3341 4.3671 1.8498 15.7603
D-336MG GDSC1 2.4032 5.1968 1.5405 17.7136
MOG-G-CCM GDSC1 2.4741 4.1984 2.0675 13.4633
KNS-42 GDSC1 2.4954 4.0347 2.1597 12.6786
SF295 GDSC1 2.5424 4.7074 1.9065 14.3405
LN-229 GDSC1 2.6012 3.5602 2.4595 9.9658
YKG-1 GDSC1 2.6053 4.172 2.2136 11.7377
Hs 683 GDSC1 2.6336 3.4798 2.5224 9.349
D-423MG GDSC1 2.654 4.3623 2.1769 11.7807
DBTRG-05MG GDSC1 2.6786 4.3628 2.2013 11.4813
GaMG GDSC1 2.7017 5.306 1.7751 14.6189
Onda 10 GDSC1 2.7043 8.938 -0.0161 26.1157
SW1783 GDSC1 2.7342 11.2275 -1.1307 30.6792
KINGS-1 GDSC1 2.7823 5.6864 1.6645 15.1083
A-172 GDSC1 2.8161 4.4236 2.3083 10.0361
YKG-1 GDSC2 2.8792 5.9084 0.9693 7.0671
ONS-76 GDSC1 2.8889 4.3756 2.4017 8.9943
LN-18 GDSC1 2.9297 3.8136 2.7036 6.5119
D-263MG GDSC1 3.0094 6.3649 1.5327 15.161
D-566MG GDSC1 3.1275 4.5063 2.5608 6.7462
8-MG-BA GDSC1 3.1569 5.7131 1.9862 11.1307
SW1088 GDSC1 3.2562 5.3609 2.2472 8.714
D-502MG GDSC2 3.2788 8.1853 0.1445 11.074
D-502MG GDSC1 3.3189 7.9755 0.9926 17.7796
D-392MG GDSC1 3.3248 7.5044 1.2331 16.1118
U-118MG GDSC1 3.3269 5.196 2.389 7.3387
LN-405 GDSC1 3.3793 5.2788 2.3909 7.1365
D283 Med GDSC1 3.4416 4.9644 2.5982 5.289
D-247MG GDSC2 3.457 8.2342 0.25 10.0314
42-MG-BA GDSC1 3.4733 5.4343 2.3891 6.8254
Onda 11 GDSC1 3.6818 5.7822 2.3773 6.2416
SF126 GDSC2 3.7076 5.6073 1.6397 1.5915
GB-1 GDSC1 3.7462 6.6262 2.0087 8.8921
SF295 GDSC2 3.7685 5.1492 1.8557 0.6013
SW1088 GDSC2 3.8476 8.6512 1.0817 11.4631
CAS-1 GDSC1 3.8482 8.4049 1.2046 14.4659
GB-1 GDSC2 3.9466 7.0217 1.9634 6.3102
GaMG GDSC2 4.0461 9.0346 1.0444 11.1918
T98G GDSC2 4.0761 6.1252 2.488 3.1333
CAS-1 GDSC2 4.0819 6.7929 2.1717 4.859
PFSK-1 GDSC2 4.1092 6.3233 2.4157 3.4642
KNS-81-FD GDSC2 4.1499 6.3741 1.5404 1.5454
D-245MG GDSC2 4.1602 11.7647 -0.969 14.9325
D-542MG GDSC2 4.1699 13.0448 -1.5883 17.7553
DK-MG GDSC1 4.1784 8.6901 1.3139 12.6506
DBTRG-05MG GDSC2 4.2291 5.921 2.6779 1.885
NMC-G1 GDSC2 4.3101 5.9641 1.7738 0.5202
Onda 10 GDSC2 4.3228 10.0487 -0.0281 9.7048
YH-13 GDSC2 4.3453 7.2055 2.1525 4.4556
KNS-42 GDSC2 4.3795 5.948 1.8074 0.3904
SF268 GDSC2 4.383 7.3174 2.1242 4.5392
SNB-75 GDSC2 4.3923 6.6203 1.5553 1.2417
Hs 683 GDSC2 4.448 5.8803 1.8577 0.246
M059J GDSC2 4.5573 7.1324 2.3213 3.1958
42-MG-BA GDSC2 4.6398 7.173 2.3523 2.9096
D-336MG GDSC2 4.6594 7.5523 1.3023 2.0666
D-566MG GDSC2 4.7011 6.2233 1.8307 0.2206
LN-18 GDSC2 4.7627 9.3379 1.4134 7.6586
LNZTA3WT4 GDSC2 4.8525 6.6225 1.7463 0.342
Daoy GDSC2 4.8888 7.4099 2.3888 2.3784
SW1783 GDSC2 4.9397 7.3953 2.423 2.1525
8-MG-BA GDSC2 4.9903 10.3951 1.0606 9.0766
GI-1 GDSC2 5.0239 7.6305 2.3662 2.3112
MOG-G-CCM GDSC2 5.0451 7.132 2.5892 1.3077
D-263MG GDSC2 5.058 6.5112 2.8399 0.4219
D-392MG GDSC2 5.0663 7.4746 2.4559 1.8526
D-423MG GDSC2 5.0871 7.5554 1.4963 0.9228
KNS-81-FD GDSC1 5.1163 7.0715 2.6478 1.39
LN-405 GDSC2 5.1906 6.7062 2.8212 0.4056
AM-38 GDSC2 5.231 7.2055 2.6469 0.9252
KS-1 [Human Krukenberg tumour] GDSC2 5.2671 10.179 1.3473 7.07
MOG-G-UVW GDSC2 5.2727 7.2862 2.6338 0.9396
U-118MG GDSC2 5.3109 6.8425 2.8189 0.3563
Onda 11 GDSC2 5.3151 7.321 1.6721 0.3388
SF539 GDSC2 5.3169 9.7784 1.5661 5.8573
D283 Med GDSC2 5.3305 7.1887 2.6973 0.6859
DK-MG GDSC2 5.3335 12.6839 0.1929 12.7087
A-172 GDSC2 5.4404 10.4174 1.346 6.7757
H4 GDSC2 5.5115 12.9372 0.1941 12.3469
LNZTA3WT4 GDSC1 5.5141 7.3493 2.7132 0.7304
Becker GDSC2 5.6254 7.1073 2.8434 0.1989
U-251MG GDSC2 5.6632 7.0479 2.8775 0.1383
AM-38 GDSC1 5.7297 7.5384 2.7295 0.5379
KINGS-1 GDSC2 5.7675 7.9937 2.5753 0.7918
ONS-76 GDSC2 5.8168 7.4382 2.798 0.2251
SK-MG-1 GDSC2 5.9142 7.8066 2.704 0.378
LN-229 GDSC2 6.2639 15.9585 -0.7444 14.987
U-87MG ATCC GDSC2 6.2818 13.1899 0.5825 9.1038
KALS-1 GDSC2 8.6819 22.0327 -2.0327 15.5419
⏷ Show the Full List of 109 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TGBC24TKB GDSC1 -0.9397 6.1903 -2.3364 51.7935
ETK-1 GDSC1 0.437 6.2704 -0.932 41.1966
TGBC24TKB GDSC2 0.7516 8.7684 -1.7568 33.6311
TGBC1TKB GDSC1 2.6293 5.8063 1.464 17.2552
ETK-1 GDSC2 3.5848 10.7208 -0.1608 18.4368
TGBC1TKB GDSC2 4.084 10.6092 0.2923 15.0034
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 16 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
EN GDSC1 -1.144 193.6662 -95.597 50.1314
MFE-319 GDSC1 0.4267 8.4373 -1.921 43.1424
MFE-296 GDSC1 1.3124 3.4364 1.0966 26.5186
ESS-1 GDSC1 1.5537 3.1491 1.4365 22.8636
RL95-2 GDSC1 1.5872 4.1673 1.1457 24.6307
KLE GDSC1 2.0715 7.6747 0.0322 28.6763
AN3-CA GDSC1 2.7477 3.7219 2.5541 8.5191
MFE-280 GDSC1 3.2622 5.4222 2.2216 8.8932
ESS-1 GDSC2 3.9721 6.9972 1.9939 6.0827
KLE GDSC2 4.2351 13.7484 -1.1512 20.9623
AN3-CA GDSC2 4.4915 12.8151 -0.4887 17.6479
MFE-280 GDSC2 4.6616 11.7968 0.1425 14.3826
RL95-2 GDSC2 5.0479 13.5869 -0.4528 16.2354
MFE-296 GDSC2 5.5016 7.312 2.7221 0.5153
EN GDSC2 5.5418 7.6424 2.6135 0.8157
MFE-319 GDSC2 6.0473 16.194 -1.0085 16.4538
⏷ Show the Full List of 16 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 65 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LB2241-RCC GDSC1 -5.1769 6.2866 -6.9034 69.5187
SW13 GDSC1 -3.2909 2.709 -3.7372 69.4846
ACHN GDSC1 -3.2124 17.7287 -9.8545 56.5152
TK-10 GDSC1 -3.0645 17.0118 -9.3714 56.3926
LB1047-RCC GDSC1 -2.6447 11.7648 -6.5183 57.2235
SW13 GDSC2 -0.984 4.1798 -1.6367 41.2269
769-P GDSC1 -0.7833 5.1576 -1.7658 50.8276
LB996-RCC GDSC1 -0.7152 7.7627 -2.7682 50.221
CAL-54 GDSC2 -0.5061 15.4791 -6.1815 44.5895
KTCTL-1M GDSC1 -0.0351 12.3759 -4.2363 47.2699
UO-31 GDSC1 0.4232 6.7089 -1.1383 41.7528
KTCTL-21 GDSC1 0.89 11.1655 -2.7739 42.1551
CAL-54 GDSC1 0.8987 10.8276 -2.6019 41.873
KTCTL-140 GDSC1 1.0285 8.2811 -1.2567 38.633
RXF 393L GDSC1 1.1019 5.4796 0.0966 33.4855
KTCTL-195 GDSC1 1.3359 8.8532 -1.2337 37.0297
786-O GDSC1 1.3502 3.978 0.961 27.1794
NCC010 GDSC1 1.507 5.5723 0.4717 29.2481
LB996-RCC GDSC2 1.5833 12.8637 -2.9654 33.8682
SN12C GDSC1 1.6221 7.9633 -0.5326 33.3192
SW156 GDSC1 1.8127 9.6503 -1.1739 34.6316
KTCTL-26A GDSC1 1.9756 7.5326 0.0111 29.2357
RCC10RGB GDSC1 2.0606 14.9819 -3.5899 38.9642
Caki-1 GDSC1 2.1221 17.3694 -4.7251 40.3032
KTCTL-13 GDSC1 2.4122 4.4467 1.8947 15.0472
BB65-RCC GDSC1 2.5971 7.0952 0.8017 21.9443
A-704 GDSC1 2.6031 5.1267 1.7677 15.1102
KMRC-1 GDSC1 2.6512 11.3683 -1.273 31.4834
HA7-RCC GDSC1 2.6878 6.9651 0.9482 20.6047
BFTC-909 GDSC1 2.7939 4.0849 2.4439 9.1085
VMRC-RCZ GDSC1 2.9329 7.0729 1.1132 18.4705
NCC010 GDSC2 3.0945 9.9205 -0.8543 17.0048
NCC021 GDSC2 3.1559 5.4528 1.385 3.9
Caki-1 GDSC2 3.2115 19.1336 -5.3545 31.404
ACHN GDSC2 3.2206 16.0477 -3.1256 29.6711
NCC021 GDSC1 3.2406 5.1624 2.3331 8.0966
LB1047-RCC GDSC2 3.3086 20.2832 -5.8503 32.1244
KMRC-20 GDSC1 3.3447 5.6262 2.1887 8.8494
OS-RC-2 GDSC1 3.3523 6.2225 1.8968 11.0949
A-498 GDSC1 3.3818 12.833 -1.3838 29.2159
LB2241-RCC GDSC2 3.8066 8.5055 0.3628 8.5929
BB65-RCC GDSC2 3.9078 7.1071 1.0862 4.2332
KTCTL-1M GDSC2 3.9237 12.1374 -1.3233 17.1575
KMRC-1 GDSC2 3.9252 7.3482 1.7868 7.353
KTCTL-13 GDSC2 3.9405 6.6422 1.3149 2.93
769-P GDSC2 3.9601 16.7535 -2.8697 27.1906
BFTC-909 GDSC2 4.0693 5.9098 2.5852 2.6232
SN12C GDSC2 4.1731 6.6058 2.3237 3.8456
A-498 GDSC2 4.1874 6.8562 2.2136 4.4199
KTCTL-195 GDSC2 4.1901 10.0673 0.6426 12.9793
KTCTL-21 GDSC2 4.2027 18.2357 -4.1271 26.3619
786-O GDSC2 4.3114 7.4865 1.9954 5.3773
UO-31 GDSC2 4.353 6.7264 1.4938 1.5387
OS-RC-2 GDSC2 4.3859 8.6891 1.465 8.1416
VMRC-RCW GDSC2 4.5745 6.4608 1.6963 0.6031
KTCTL-140 GDSC2 4.6074 16.3824 -2.9064 21.8148
KTCTL-26A GDSC2 4.6885 6.6936 1.6559 0.6602
VMRC-RCZ GDSC2 4.8706 7.6822 2.2572 3.0442
SW156 GDSC2 4.8741 17.7846 -3.3993 22.8258
RXF 393L GDSC2 4.9067 8.1776 1.1644 2.4207
A-704 GDSC2 5.1196 13.6643 -0.4383 16.0173
HA7-RCC GDSC2 5.1488 8.0963 1.3129 1.5436
TK-10 GDSC2 5.9113 21.3045 -3.6132 24.9427
KMRC-20 GDSC2 5.9314 12.4972 0.684 9.2215
RCC10RGB GDSC2 7.988 28.1673 -5.4593 25.4253
⏷ Show the Full List of 65 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 94 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DiFi GDSC2 -7.093 9.7729 -10.2816 64.9085
DiFi GDSC1 -5.9671 2.2828 -6.5518 78.6328
SNU-407 GDSC1 -5.1056 2.7648 -5.7293 75.6246
NCI-H508 GDSC2 -1.4733 27.2035 -13.4078 47.7216
SW48 GDSC1 -1.4399 8.1415 -3.679 54.0766
CCK-81 GDSC2 -0.5064 8.292 -2.7901 41.0285
HT115 GDSC1 -0.4793 3.6169 -0.9106 48.0361
SW1463 GDSC1 0.2367 11.7723 -3.6866 45.8522
GP5d GDSC1 0.2733 2.0066 0.2409 38.2938
LoVo GDSC1 0.2937 4.5024 -0.3665 40.6104
HCT 116 GDSC1 0.5647 2.1714 0.5318 34.6665
LS513 GDSC1 0.6615 3.5404 0.3561 34.9992
HT-55 GDSC1 0.9232 6.9872 -0.7576 37.8056
NCI-H747 GDSC1 1.0182 21.3478 -7.6762 45.4989
CCK-81 GDSC1 1.1503 11.1853 -2.5394 40.6888
SW48 GDSC2 1.2997 17.448 -5.4899 38.8735
SW1116 GDSC1 1.3387 10.3257 -1.9444 38.7504
SK-CO-1 GDSC1 1.5179 3.3487 1.3458 23.6751
MDST8 GDSC1 1.7302 2.9652 1.6676 20.2983
CW-2 GDSC2 1.8397 10.3217 -1.4788 28.8438
SNU-81 GDSC1 1.8774 7.1604 0.0972 29.2918
LoVo GDSC2 1.8845 10.9213 -1.7334 29.5302
SNU-C2B GDSC1 1.9282 6.6551 0.3877 27.5184
NCI-H508 GDSC1 2.2575 23.0014 -7.4183 42.3992
LS180 GDSC1 2.3043 5.4876 1.3067 19.8625
HCC2998 GDSC1 2.3615 3.7766 2.1221 13.6392
HCT 15 GDSC1 2.4795 3.964 2.1727 12.6632
CaR-1 GDSC1 2.5161 4.6369 1.913 14.4146
C2BBe1 GDSC1 2.5714 6.9186 0.8653 21.6499
SW620 GDSC1 2.6216 5.0272 1.8331 14.5338
SNU-C5 GDSC1 2.639 4.4037 2.1429 12.1075
HT-29 GDSC1 2.6453 4.3279 2.1839 11.7685
SW626 GDSC1 2.747 5.2897 1.8257 14.0382
COLO 320HSR GDSC1 2.7559 4.0564 2.4184 9.4813
SK-CO-1 GDSC2 2.7915 10.1158 -0.5266 22.229
CW-2 GDSC1 2.8446 8.933 0.1093 24.8995
RKO GDSC1 3.0901 4.2654 2.6454 6.2393
SW1463 GDSC2 3.2143 12.8806 -1.5474 24.9849
RCM-1 [Human ESC] GDSC1 3.2915 9.6408 0.1371 23.007
NCI-H716 GDSC1 3.3385 5.2229 2.3852 7.3265
SW948 GDSC1 3.3918 5.1373 2.4718 6.4559
CL-11 GDSC1 3.3983 5.4719 2.3099 7.7068
LS1034 GDSC1 3.4081 9.8841 0.1124 22.7048
LS513 GDSC2 3.4205 13.7285 -2.4937 23.1365
T84 GDSC1 3.4336 8.2503 0.9502 17.6355
LS411N GDSC1 3.4836 6.9549 1.6383 12.5919
SW837 GDSC1 3.5399 11.7854 -0.7296 26.1952
KM12 GDSC1 3.6248 5.2919 2.5766 4.8682
SNU-283 GDSC2 3.6733 18.8794 -4.8594 29.3211
HT115 GDSC2 3.7903 9.2191 0.0071 10.6225
SW1417 GDSC1 4.0903 11.3747 -0.0834 21.3571
SW1116 GDSC2 4.2891 12.1352 -0.307 17.2844
COLO 320HSR GDSC2 4.2986 5.9012 2.7265 1.5435
LS411N GDSC2 4.3104 5.7091 2.8166 1.1111
COLO205 GDSC1 4.42 9.173 1.2533 12.3415
SNU-81 GDSC2 4.4438 6.3158 1.6968 0.6782
SNU-175 GDSC2 4.4495 20.2565 -4.225 29.2898
SW837 GDSC2 4.4891 8.4499 1.6534 6.8787
SNU-C5 GDSC2 4.548 7.2616 2.2559 3.5386
RKO GDSC2 4.6111 7.4776 2.195 3.7522
COLO205 GDSC2 4.7119 6.0966 2.8513 0.5989
HT-29 GDSC2 4.7333 8.5183 1.7848 5.7068
LS123 GDSC1 4.8607 14.0864 -0.8379 22.4875
SW626 GDSC2 4.8916 7.5556 2.3259 2.6772
C2BBe1 GDSC2 4.9085 17.0091 -2.2486 23.1584
COLO 678 GDSC1 4.9404 15.3464 -1.4005 24.48
HCT 116 GDSC2 4.9778 7.5433 2.3792 2.3015
SNU-1040 GDSC2 5.0928 14.305 -1.5472 15.508
SW948 GDSC2 5.0972 6.7666 2.7594 0.6373
SNU-C1 GDSC1 5.1224 12.7501 0.0111 17.7635
SNU-61 GDSC1 5.1489 13.9053 -0.5351 20.3469
NCI-H716 GDSC2 5.2648 7.3796 2.5929 1.0914
HT-55 GDSC2 5.3239 16.0611 -1.4659 19.6168
SNU-C2B GDSC2 5.4223 14.2782 -0.5197 15.6867
CL-11 GDSC2 5.4601 7.5508 2.6133 0.8693
LS1034 GDSC2 5.4794 7.0773 2.7994 0.3318
NCI-H747 GDSC2 5.559 20.6543 -3.5578 25.4562
HCT 15 GDSC2 5.5731 11.3929 0.973 8.4083
MDST8 GDSC2 5.574 6.722 2.9563 0.0634
KM12 GDSC2 5.6594 7.329 2.7779 0.3116
RCM-1 [Human ESC] GDSC2 5.8288 15.1558 -0.6584 15.443
LS180 GDSC2 5.8442 12.4527 0.6486 9.5204
LS123 GDSC2 5.8664 14.4997 -0.3148 13.9144
SNU-1040 GDSC1 5.9181 14.5837 -0.3197 17.3205
SNU-C1 GDSC2 5.9824 7.5292 2.826 0.1445
SNU-61 GDSC2 6.0226 15.3996 -0.6412 15.0274
SW620 GDSC2 6.0325 9.2148 2.2107 1.8836
HCC2998 GDSC2 6.1435 7.7334 2.8131 0.1319
CaR-1 GDSC2 6.2949 16.9706 -1.2116 16.7165
T84 GDSC2 6.5206 15.1335 -0.1781 12.1086
GP5d GDSC2 6.6295 15.5619 -0.3097 12.4809
SNU-407 GDSC2 6.882 18.1764 -1.3887 16.2834
SW1417 GDSC2 7.0222 17.2254 -0.8406 13.9632
COLO 678 GDSC2 7.7556 22.1004 -2.6786 19.0092
⏷ Show the Full List of 94 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1 3.5395 5.286 2.5148 5.6198
MO-T GDSC2 4.4934 6.5232 2.56 2.089
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHH-1 GDSC1 -4.8714 3.6076 -5.6994 73.2095
SNU-387 GDSC1 1.7966 3.9675 1.4452 21.4391
HuH-1 GDSC1 1.925 4.5088 1.3652 21.3194
JHH-6 GDSC1 1.9277 4.091 1.5381 20.087
JHH-4 GDSC1 2.1492 5.1116 1.3285 20.4513
Huh-7 GDSC1 2.4814 3.9995 2.1599 12.7478
HLE GDSC1 2.5401 4.3927 2.0486 13.2839
JHH-7 GDSC1 3.3228 4.7136 2.6268 5.4787
Hep 3B2.1-7 GDSC2 3.5112 5.3291 1.6556 1.7695
Hep-G2/C3A GDSC2 3.671 5.0694 2.7193 2.647
JHH-2 GDSC1 3.8562 7.1444 1.8356 9.8617
SNU-449 GDSC1 3.8931 15.3321 -2.214 30.165
SK-HEP-1 GDSC1 4.2464 5.944 2.6777 2.5499
HLE GDSC2 4.467 11.3611 0.2121 14.49
JHH-6 GDSC2 4.4741 7.7367 1.9851 5.1235
Huh-7 GDSC2 4.878 7.8252 2.1969 3.3343
Hep 3B2.1-7 GDSC1 4.9344 6.5359 2.7779 0.9462
HuH-1 GDSC2 5.0579 8.0245 2.2112 3.0045
SNU-423 GDSC1 5.1457 7.5042 2.484 2.2519
SNU-398 GDSC1 5.2389 12.5898 0.1721 16.5952
JHH-7 GDSC2 5.249 6.7845 2.8157 0.3922
SNU-449 GDSC2 5.2652 12.5951 0.1881 12.8711
Hep-G2/C3A GDSC1 5.3436 6.7078 2.8797 0.2934
SK-HEP-1 GDSC2 5.3947 6.6517 2.9178 0.1375
SNU-387 GDSC2 5.5757 7.291 2.7593 0.3863
SNU-398 GDSC2 5.7743 8.2057 2.4962 1.0442
JHH-2 GDSC2 5.82 11.8458 0.9185 8.2703
JHH-4 GDSC2 6.1093 12.3064 0.8856 7.9437
SNU-423 GDSC2 7.0112 15.3922 0.0143 10.4693
JHH-1 GDSC2 7.1961 20.3903 -2.2391 18.6532
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 357 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PC-14 GDSC2 -5.955 30.1118 -18.4168 55.7011
NCI-H292 GDSC1 -5.7535 4.5832 -6.9535 73.554
HCC827 GDSC1 -5.6193 6.5426 -7.4724 70.2213
NCI-H3255 GDSC1 -5.4899 5.5116 -6.9707 71.4229
EMC-BAC-1 GDSC1 -4.3707 3.7062 -5.1813 71.5337
PC-14 GDSC1 -4.2361 5.2049 -5.5078 68.4722
NCI-H1568 GDSC1 -3.9615 4.9829 -5.1352 67.9164
COR-L105 GDSC2 -3.8927 3.9341 -4.7269 60.0989
NCI-H1666 GDSC1 -3.8402 13.019 -8.2921 59.9444
NCI-H322M GDSC2 -3.4252 11.8769 -7.3585 54.3088
PaCa-3 GDSC2 -2.9308 24.8921 -13.0329 51.4968
PaCa-3 GDSC1 -2.8381 12.25 -6.9333 57.5913
HCC827 GDSC2 -2.5105 15.3191 -8.0319 51.0386
RERF-LC-Sq1 GDSC1 -2.4698 9.2257 -5.2113 57.9748
Calu-3 GDSC1 -2.2575 3.5133 -2.8204 62.4524
NCI-H3255 GDSC2 -2.0106 32.7295 -16.628 48.9809
COR-L105 GDSC1 -1.7428 9.2751 -4.4868 55.0274
NCI-H1623 GDSC1 -1.5864 7.3544 -3.4954 55.1536
NCI-H1623 GDSC2 -1.197 5.5252 -2.3477 43.7478
NCI-H2030 GDSC1 -1.046 6.7012 -2.6576 52.359
NCI-H1648 GDSC2 -0.9915 10.1961 -4.1438 44.7743
NCI-H1437 GDSC1 -0.9602 29.4217 -13.4484 50.5066
LOU-NH91 GDSC1 -0.7789 34.3328 -15.7209 50.1569
NCI-H2170 GDSC1 -0.7022 4.1296 -1.3141 50.2171
NCI-H2170 GDSC2 -0.673 3.5518 -1.1027 38.0408
NCI-H1648 GDSC1 -0.4902 10.1089 -3.6053 49.0785
NCI-H1666 GDSC2 -0.0861 15.7153 -5.9024 43.1598
NCI-H2122 GDSC1 -0.0376 3.3554 -0.3536 43.137
NCI-H1944 GDSC1 0.0172 9.1954 -2.6785 46.1371
CAL-12T GDSC1 0.0554 8.6129 -2.371 45.6761
SK-MES-1 GDSC1 0.2331 12.6751 -4.1254 46.1437
EPLC-272H GDSC1 0.2656 8.9804 -2.333 44.5297
NCI-H290 GDSC1 0.3629 7.6318 -1.6139 43.0105
NCI-H1781 GDSC1 0.4104 4.5201 -0.2477 39.3767
Calu-3 GDSC2 0.4529 4.2166 -0.0921 28.7096
NCI-H2110 GDSC1 0.5667 6.6492 -0.9653 40.4764
LC-1/sq GDSC1 0.5879 11.3115 -3.1302 43.8842
EMC-BAC-1 GDSC2 0.6113 13.1395 -4.5711 36.8026
NCI-H1703 GDSC1 0.6653 1.8158 0.6588 33.2483
LC-2/ad GDSC1 0.7607 3.2333 0.5505 33.2791
RERF-LC-Sq1 GDSC2 0.8116 17.9947 -6.1989 40.9659
NCI-H647 GDSC1 0.8272 2.3946 0.7853 31.446
NCI-H524 GDSC1 0.9403 2.949 0.8143 30.5609
NCI-H1869 GDSC1 1.0268 15.1613 -4.6046 43.6137
NCI-H2595 GDSC1 1.0342 13.2668 -3.6656 42.6764
NCI-H1792 GDSC1 1.0817 6.7945 -0.5106 36.0895
NCI-H1355 GDSC1 1.1877 8.0027 -0.97 37.0142
HARA [Human squamous cell lung carcinoma] GDSC1 1.2033 8.1544 -1.0269 37.1023
RERF-LC-KJ GDSC1 1.2161 5.9513 0.0067 33.2349
NCI-H358 GDSC2 1.2752 9.9576 -1.825 31.9199
Lu-99A GDSC1 1.2938 4.129 0.8455 28.2387
NCI-H1975 GDSC1 1.3379 3.5841 1.0798 26.4793
DMS 273 GDSC1 1.3442 3.246 1.1838 25.7605
A-549 GDSC1 1.4158 8.4517 -0.9643 35.8417
NCI-H1975 GDSC2 1.4299 4.9037 0.6826 21.0154
CAL-12T GDSC2 1.4503 14.8792 -4.6971 34.5519
LCLC-97TM1 GDSC1 1.5036 3.3266 1.3363 23.8211
NCI-H513 GDSC1 1.5172 5.7745 0.3913 29.634
NCI-H292 GDSC2 1.6245 14.202 -4.2089 33.0408
NCI-H358 GDSC1 1.6594 9.6635 -1.3223 35.7633
SHP-77 GDSC1 1.6708 3.2315 1.5439 21.4661
VMRC-LCD GDSC1 1.705 3.435 1.5252 21.3965
NCI-H2110 GDSC2 1.7256 17.2823 -5.6609 35.53
NCI-H446 GDSC1 1.7386 3.8175 1.4372 21.8112
EMC-BAC-2 GDSC1 1.8275 7.3632 -0.0479 30.2391
NCI-H1568 GDSC2 1.8279 16.6975 -4.6484 36.358
LK-2 GDSC1 1.8284 3.0423 1.7589 19.1168
NCI-H196 GDSC1 1.9074 39.3997 -15.9089 46.2364
NCI-H2342 GDSC1 1.9143 10.1344 -1.3184 34.6256
HCC44 GDSC1 1.9216 3.2116 1.8224 18.1503
LXF 289 GDSC1 1.9641 3.6485 1.7396 18.4768
NCI-H661 GDSC1 1.9672 8.2642 -0.3526 30.9278
NCI-H1915 GDSC1 1.9841 3.5892 1.7811 18.0784
NCI-H841 GDSC1 2.0092 3.6642 1.7831 17.927
HOP-62 GDSC1 2.0897 5.7541 0.9714 23.1854
NCI-H1573 GDSC1 2.1167 6.4997 0.6433 25.1239
NCI-H1781 GDSC2 2.1489 7.4849 0.197 20.9511
NCI-H522 GDSC1 2.2195 4.8397 1.5229 18.715
LC-2/ad GDSC2 2.269 5.47 0.7035 10.3856
NCI-H2369 GDSC1 2.3472 3.4943 2.2066 13.1219
LB647-SCLC GDSC1 2.3593 6.5865 0.8314 22.8181
RERF-LC-MS GDSC2 2.3793 3.7514 1.6544 4.0625
NCI-H1436 GDSC1 2.3801 5.6648 1.296 19.5854
HOP-92 GDSC1 2.4043 6.2003 1.0612 21.1018
NCI-H2795 GDSC1 2.4462 5.1345 1.6119 16.9883
HCC366 GDSC1 2.4561 4.8585 1.7508 15.9099
NCI-H2373 GDSC1 2.4682 6.1922 1.1253 20.3755
A-427 GDSC1 2.4893 3.6479 2.3072 11.6438
SBC-3 GDSC1 2.4983 3.8995 2.2189 12.2313
NCI-H838 GDSC2 2.5135 6.9886 0.1462 13.0893
NCI-H23 GDSC1 2.5291 3.5694 2.3784 10.9264
RERF-LC-MS GDSC1 2.5347 3.4079 2.4378 10.4828
NCI-H1793 GDSC1 2.5425 9.8799 -0.6273 29.5422
NCI-H1299 GDSC1 2.5561 4.4768 2.0265 13.3739
NCI-H847 GDSC1 2.606 3.5901 2.4539 9.9797
NCI-H441 GDSC1 2.6153 6.6943 1.0159 20.4667
SBC-5 GDSC1 2.6495 3.3913 2.568 8.9452
NCI-H1755 GDSC1 2.652 5.2328 1.7636 14.9241
EBC-1 GDSC1 2.6572 3.7845 2.4331 9.8614
NCI-H1048 GDSC1 2.6577 3.7171 2.4608 9.6584
ABC-1 GDSC1 2.666 6.0961 1.3563 17.8775
NCI-H2009 GDSC1 2.6717 3.9825 2.3649 10.2896
ChaGo-K-1 GDSC1 2.6936 3.9573 2.3984 9.9336
NCI-H460 GDSC1 2.696 3.706 2.5058 9.1353
NCI-H513 GDSC2 2.7032 10.685 -0.8872 24.0388
NCI-H2722 GDSC1 2.726 6.7984 1.0651 19.659
UMC-11 GDSC1 2.7746 4.0107 2.4579 9.0958
NCI-H2444 GDSC2 2.7971 4.2911 1.6997 2.7535
NCI-H810 GDSC1 2.802 3.798 2.579 8.0624
NCI-H3122 GDSC1 2.8178 4.1284 2.448 8.966
NCI-H1650 GDSC1 2.8224 6.127 1.4841 16.2832
NCI-H1876 GDSC1 2.8289 5.3213 1.8866 13.2232
HCC15 GDSC1 2.831 4.5558 2.2598 10.341
NCI-H1155 GDSC1 2.8614 3.9788 2.5601 7.9148
NCI-H2087 GDSC1 2.8642 5.1279 2.0139 12.0941
COR-L23 GDSC1 2.8723 4.404 2.3721 9.295
NCI-H2804 GDSC1 2.8902 5.8992 1.6578 14.7082
NCI-H520 GDSC1 2.9214 5.1187 2.0713 11.4102
NCI-H1993 GDSC1 2.9371 4.4813 2.3969 8.8194
NCI-H650 GDSC1 2.9643 4.5814 2.3739 8.881
Ms-1 GDSC1 2.9696 4.2536 2.5375 7.5929
NCI-H2023 GDSC1 3.0107 7.089 1.1731 17.7435
Lu-135 GDSC1 3.0171 5.0739 2.1805 10.167
NCI-H1581 GDSC1 3.0299 4.1476 2.6461 6.4912
NCI-H2818 GDSC1 3.0512 4.3739 2.5563 7.0962
SW1271 GDSC1 3.0563 4.7212 2.3902 8.3701
SK-LU-1 GDSC1 3.1079 5.8871 1.8568 12.3204
DMS 114 GDSC1 3.1133 4.7306 2.437 7.773
NCI-H2731 GDSC1 3.1456 4.9237 2.3698 8.1725
DMS 53 GDSC1 3.1802 5.9715 1.8772 11.885
NCI-H345 GDSC2 3.1865 4.3391 1.9101 0.9265
HCC78 GDSC1 3.1913 5.6243 2.0601 10.4233
NCI-H1688 GDSC1 3.2174 5.8539 1.9678 11.0436
NCI-H2228 GDSC1 3.2216 5.9159 1.9405 11.2395
COR-L321 GDSC1 3.2291 4.4635 2.6721 5.4715
SW1573 GDSC1 3.2345 5.3223 2.2479 8.7893
NCI-H1770 GDSC2 3.2484 6.0547 1.1598 5.0582
NCI-H2810 GDSC1 3.267 5.4798 2.1968 9.0694
NCI-H2227 GDSC1 3.2796 5.7274 2.0838 9.9084
NCI-H2066 GDSC1 3.2846 6.555 1.6742 13.043
NCI-H2461 GDSC1 3.2863 6.3693 1.7685 12.3213
NCI-H720 GDSC1 3.292 6.0824 1.9167 11.1616
NCI-H838 GDSC1 3.3026 6.5241 1.7047 12.7452
NCI-H596 GDSC1 3.3169 4.8448 2.5563 6.0566
NCI-H1105 GDSC2 3.3182 8.415 0.0606 11.4632
NCI-H226 GDSC1 3.3421 6.5652 1.7171 12.5064
NCI-H2122 GDSC2 3.3547 9.745 0.1376 17.6385
NCI-H2405 GDSC1 3.3714 5.5578 2.2449 8.3124
NCI-H1755 GDSC2 3.411 5.9564 2.0782 6.9238
KNS-62 GDSC1 3.4525 4.8473 2.6652 4.7259
BEN GDSC2 3.4787 4.5897 1.9464 0.4905
SBC-1 GDSC1 3.4838 7.278 1.4771 13.7832
LCLC-103H GDSC1 3.4962 5.1546 2.5464 5.5133
IST-SL1 GDSC2 3.5065 5.9858 1.3578 3.3977
NCI-H2171 GDSC2 3.5552 8.7781 0.055 10.9261
EPLC-272H GDSC2 3.568 21.2987 -5.4622 33.5201
NCI-H1694 GDSC1 3.5957 5.5902 2.4071 6.2806
NCI-H2172 GDSC1 3.601 5.9574 2.2289 7.6553
BEN GDSC1 3.6022 6.545 1.9376 9.9095
NCI-H526 GDSC1 3.6102 5.4339 2.4955 5.5448
IA-LM GDSC1 3.6169 6.6862 1.8788 10.3111
NCI-H1770 GDSC1 3.6336 5.6273 2.4176 6.079
NCI-H2803 GDSC1 3.6567 6.0035 2.2489 7.3195
NCI-H2085 GDSC1 3.6672 10.1315 0.2004 21.3013
NCI-H1651 GDSC1 3.6909 6.2741 2.1409 8.0484
NCI-H1793 GDSC2 3.7053 11.1758 -0.2903 18.712
NCI-H1563 GDSC1 3.7065 9.7645 0.4153 19.9599
NCI-H2347 GDSC1 3.7075 6.1878 2.1962 7.5677
NCI-H2030 GDSC2 3.7103 14.1662 -2.4866 22.4369
COLO 668 GDSC1 3.7156 9.4665 0.5713 19.0108
NCI-H1563 GDSC2 3.7156 7.2828 1.6593 8.5627
NCI-H1915 GDSC2 3.722 6.1642 2.2188 5.3651
NCI-H1838 GDSC1 3.7239 9.4437 0.5892 18.874
NCI-H1435 GDSC1 3.7876 5.9385 2.3785 5.9124
NCI-H2141 GDSC1 3.789 6.0314 2.334 6.2516
COR-L32 GDSC1 3.8103 6.5178 2.1105 7.9089
NCI-H2869 GDSC2 3.8161 6.3959 1.3542 2.9089
EMC-BAC-2 GDSC2 3.8182 12.5649 -0.8927 20.9872
EKVX GDSC1 3.8614 19.4661 -4.3051 34.9029
UMC-11 GDSC2 3.8662 5.6794 2.5602 3.1365
NCI-H2591 GDSC1 3.9028 6.1586 2.3537 5.7681
NCI-H460 GDSC2 3.9196 5.4052 1.8222 0.6103
NCI-H1105 GDSC1 3.9295 6.2061 2.3495 5.7254
NCI-H650 GDSC2 3.9303 5.5519 2.6641 2.4473
COR-L303 GDSC2 3.9523 5.4174 1.8314 0.5565
NCI-H2869 GDSC1 3.9691 6.9292 2.0251 8.0813
EKVX GDSC2 4.0093 17.1886 -3.7563 25.7871
NCI-H647 GDSC2 4.012 6.5225 1.4067 2.353
NCI-H2444 GDSC1 4.0166 5.9898 2.5131 4.258
NCI-H250 GDSC2 4.0224 6.7122 1.3296 2.7335
NCI-H82 GDSC2 4.0306 6.2841 2.3817 3.7994
NCI-H1341 GDSC1 4.0396 8.4288 1.3391 12.9074
NCI-H2347 GDSC2 4.0437 6.571 2.2525 4.4873
HOP-62 GDSC2 4.0568 5.8461 2.6071 2.5284
NCI-H2172 GDSC2 4.0629 5.4021 1.8822 0.3418
NCI-H1963 GDSC2 4.0633 5.9534 2.5608 2.7642
NCI-H1836 GDSC2 4.0757 8.6551 0.4705 7.421
SHP-77 GDSC2 4.0796 8.1402 1.5114 8.5495
COR-L279 GDSC2 4.1145 5.8279 2.6517 2.1967
HCC44 GDSC2 4.1592 7.1063 2.0739 5.2456
NCI-H1436 GDSC2 4.1595 5.7091 1.8075 0.5044
NCI-H2291 GDSC2 4.172 12.6204 -1.3786 16.8222
NCI-H69 GDSC2 4.1896 7.0945 2.1006 5.0373
SBC-5 GDSC2 4.1961 5.4993 2.8465 1.1156
NCI-H146 GDSC1 4.2 7.3063 2.0056 7.5666
LC-1/sq GDSC2 4.2208 23.3425 -5.9496 32.9409
LCLC-103H GDSC2 4.2278 5.5383 2.8466 1.077
NCI-H82 GDSC1 4.2283 8.8482 1.2729 12.7814
COR-L23 GDSC2 4.2315 6.471 2.4255 3.1917
NCI-H2291 GDSC1 4.235 13.6544 -1.1045 25.4265
NCI-H2461 GDSC2 4.256 8.6304 1.4002 8.775
IST-SL2 GDSC1 4.2768 6.9767 2.216 5.7994
Calu-6 GDSC2 4.2789 7.0283 2.1928 4.3603
NCI-H226 GDSC2 4.2962 7.5382 1.9601 5.601
NCI-H345 GDSC1 4.3029 5.341 2.9657 0.6976
NCI-H69 GDSC1 4.3054 6.7558 2.3391 4.8246
NCI-H1092 GDSC2 4.3235 7.6035 1.9474 5.6175
NCI-H1573 GDSC2 4.3245 7.7016 1.9008 5.8714
NCI-H1304 GDSC1 4.3246 9.8742 0.8392 15.3536
NCI-H1838 GDSC2 4.3355 8.688 1.4295 8.4427
NCI-H2196 GDSC2 4.3435 6.0396 1.7592 0.545
CPC-N GDSC2 4.3528 6.3672 2.5485 2.3519
HCC33 GDSC2 4.3675 11.9356 -0.9053 14.1552
KNS-62 GDSC2 4.3727 7.0386 2.2494 3.884
NCI-H2081 GDSC2 4.3827 7.5345 1.1665 3.0667
NCI-H1734 GDSC2 4.3964 6.3466 1.6648 0.8213
Lu-139 GDSC1 4.4017 7.1186 2.2304 5.3835
NCI-H1836 GDSC1 4.4035 6.816 2.3729 4.3513
NCI-H841 GDSC2 4.4036 10.5859 0.5473 12.9729
HCC366 GDSC2 4.4043 14.3531 -2.0588 19.1674
NCI-H835 GDSC1 4.4067 7.5862 2.012 6.9654
COR-L95 GDSC1 4.4217 6.9954 2.3008 4.8264
NCI-H2135 GDSC2 4.4254 6.0045 1.8048 0.3763
COR-L95 GDSC2 4.4348 6.099 1.774 0.4532
IST-SL1 GDSC1 4.446 7.6954 1.9862 7.0528
Lu-134-A GDSC2 4.4517 18.5786 -4.1069 25.764
EBC-1 GDSC2 4.4602 7.8767 1.9091 5.5624
NCI-H2795 GDSC2 4.4611 11.2978 0.239 14.3732
COR-L88 GDSC1 4.473 8.4431 1.6456 9.4458
DMS 79 GDSC2 4.4777 6.1104 1.7867 0.399
Calu-6 GDSC1 4.4949 6.409 2.6115 2.5179
SBC-3 GDSC2 4.499 8.5934 1.591 7.221
NCI-H446 GDSC2 4.5009 6.4502 2.5967 1.9003
NCI-H2009 GDSC2 4.5031 9.1563 1.3209 8.6805
NCI-H727 GDSC2 4.5061 7.5248 2.1064 4.4126
NCI-H2029 GDSC2 4.5086 6.2632 1.743 0.5023
NCI-H1703 GDSC2 4.5107 12.1311 -0.1354 16.0285
COR-L311 GDSC2 4.5166 6.544 2.5639 2.0375
COR-L279 GDSC1 4.5194 6.5179 2.577 2.6999
NCI-H510A GDSC2 4.5217 6.2212 1.7636 0.4389
NCI-H209 GDSC1 4.5398 8.5134 1.6576 9.1778
NCI-H835 GDSC2 4.554 8.5424 1.6534 6.7721
NCI-H1155 GDSC2 4.5586 6.586 2.5688 1.9568
SW1271 GDSC2 4.5795 7.196 2.3055 3.2415
NCI-H2227 GDSC2 4.5844 6.1813 1.8022 0.3173
IST-SL2 GDSC2 4.6092 9.4295 1.2631 8.772
NCI-H1869 GDSC2 4.6269 16.0396 -1.9848 22.9918
NCI-H748 GDSC2 4.6287 6.671 1.6396 0.7488
NCI-H2405 GDSC2 4.6458 9.3086 1.3472 8.2456
NCI-H146 GDSC2 4.6483 6.2763 1.7925 0.315
NCI-H2369 GDSC2 4.6638 6.3904 2.7091 1.194
COR-L321 GDSC2 4.6741 6.3777 1.7661 0.3658
Lu-65 GDSC1 4.6775 11.5429 0.2791 17.6038
NCI-H2085 GDSC2 4.6827 10.9976 0.5506 12.3337
NCI-H1651 GDSC2 4.6898 7.4485 2.2564 3.32
NCI-H727 GDSC1 4.7221 13.9131 -0.8568 22.9672
COR-L88 GDSC2 4.7246 6.7236 2.5988 1.6092
NCI-H526 GDSC2 4.7319 6.3597 2.7552 0.9389
NCI-H1581 GDSC2 4.744 6.2338 2.8115 0.7163
Lu-165 GDSC2 4.7636 6.2486 2.8146 0.69
SBC-1 GDSC2 4.778 6.1662 1.8775 0.1287
NCI-H2804 GDSC2 4.7996 10.0324 0.2837 7.1029
NCI-H2818 GDSC2 4.8059 8.5872 1.7995 5.5163
NCI-H2141 GDSC2 4.8115 6.9155 2.5621 1.6723
Lu-139 GDSC2 4.8116 6.3608 1.823 0.2041
IA-LM GDSC2 4.8137 6.9388 2.5532 1.7097
NCI-H290 GDSC2 4.8191 6.8231 1.6607 0.5739
NCI-H187 GDSC1 4.8214 6.6188 2.692 1.517
NCI-H847 GDSC2 4.8301 6.2885 2.8285 0.5938
NCI-H2066 GDSC2 4.8535 8.7355 1.7603 5.6393
NCI-H1092 GDSC1 4.8632 6.8156 2.6309 1.8048
DMS 273 GDSC2 4.866 9.3665 1.4694 7.1622
NCI-H211 GDSC1 4.8725 11.0597 0.6568 14.8597
HARA [Human squamous cell lung carcinoma] GDSC2 4.8733 17.9182 -2.727 24.7104
NCI-H2731 GDSC2 4.9042 7.8544 2.199 3.2847
NCI-H1437 GDSC2 4.9044 7.0375 1.6156 0.6586
NCI-H2228 GDSC2 4.9134 12.1926 0.1329 13.8734
NCI-H211 GDSC2 4.9167 7.6257 2.3088 2.7254
NCI-H810 GDSC2 4.9536 6.2701 2.8873 0.3475
NCI-H720 GDSC2 4.9645 6.2501 2.8989 0.3128
NCI-H441 GDSC2 4.9724 9.1653 1.6346 6.0928
SK-MES-1 GDSC2 4.9896 17.1114 -2.2371 22.9885
NCI-H596 GDSC2 5.019 7.4833 2.4274 2.0356
NCI-H209 GDSC2 5.0386 8.4308 2.0167 4.0001
NCI-H2810 GDSC2 5.0616 7.1049 1.6532 0.4779
DMS 79 GDSC1 5.1193 7.2392 2.5811 1.7397
NCI-H1694 GDSC2 5.1244 6.5348 2.8579 0.3429
LB647-SCLC GDSC2 5.1298 6.6727 1.8288 0.1281
ChaGo-K-1 GDSC2 5.1424 7.8438 1.4092 1.1853
NCI-H322M GDSC1 5.1641 16.7299 -1.9155 25.6627
Lu-99A GDSC2 5.1989 7.8682 2.3567 2.1421
Lu-65 GDSC2 5.2694 12.068 0.4463 11.6225
CPC-N GDSC1 5.2835 7.5154 2.5468 1.7183
ABC-1 GDSC2 5.287 7.4914 1.6007 0.5109
LCLC-97TM1 GDSC2 5.3102 8.3135 2.2236 2.6149
NCI-H2029 GDSC1 5.3185 6.9702 2.7749 0.6377
NCI-H1299 GDSC2 5.3732 10.6037 1.2157 7.5588
Lu-165 GDSC1 5.3735 7.1166 2.7427 0.72
DMS 53 GDSC2 5.3887 7.1553 2.7345 0.5404
LXF 289 GDSC2 5.3934 7.4506 2.6231 0.8867
NCI-H64 GDSC2 5.396 6.5354 2.9577 0.0859
Lu-134-A GDSC1 5.4025 8.8918 2.0202 4.7066
NCI-H2087 GDSC2 5.4185 7.8496 2.4748 1.4131
COR-L32 GDSC2 5.4234 9.8951 1.5778 5.6235
NCI-H661 GDSC2 5.4317 9.6806 1.6814 5.0865
NCI-H2803 GDSC2 5.4352 7.1802 1.7636 0.1566
NCI-H2373 GDSC2 5.4375 7.1204 2.7672 0.4278
NCI-H2722 GDSC2 5.486 7.6064 2.6031 0.8882
HOP-92 GDSC2 5.4913 10.8198 1.19 7.482
COLO 668 GDSC2 5.5261 7.5794 2.631 0.7699
NCI-H524 GDSC2 5.5319 7.1557 2.7913 0.3305
Lu-135 GDSC2 5.5467 7.6179 2.6251 0.7755
VMRC-LCD GDSC2 5.6105 7.6046 2.6571 0.6394
NCI-H2135 GDSC1 5.618 7.1192 2.8366 0.2915
NCI-H740 GDSC2 5.6239 7.8346 1.6058 0.3722
LK-2 GDSC2 5.634 7.226 2.805 0.2664
NCI-H1688 GDSC2 5.6537 7.4402 2.7356 0.4098
NCI-H1792 GDSC2 5.6649 10.0569 1.6486 4.8953
SW1573 GDSC2 5.6656 7.8877 2.5723 0.8668
NCI-H196 GDSC2 5.6852 7.0377 2.8887 0.1195
A-427 GDSC2 5.7273 18.2177 -2.998 19.7899
NCI-H1341 GDSC2 5.7858 7.2366 2.8564 0.1426
NCI-H1435 GDSC2 5.8103 13.3541 0.1974 11.753
NCI-H2081 GDSC1 5.8205 7.7218 2.6983 0.5865
NCI-H1876 GDSC2 5.905 7.5563 2.789 0.2169
HCC15 GDSC2 5.9246 7.7528 2.7272 0.3253
NCI-H520 GDSC2 5.9322 7.9081 2.6743 0.4382
NCI-H23 GDSC2 5.9862 7.9826 2.6682 0.4301
SK-LU-1 GDSC2 6.0117 11.8124 1.0539 7.2851
NCI-H1048 GDSC2 6.0164 7.2719 2.9233 0.0465
NCI-H1993 GDSC2 6.0448 7.8103 2.7516 0.2432
NCI-H3122 GDSC2 6.075 7.956 2.7115 0.3071
Ms-1 GDSC2 6.0942 7.6162 2.8355 0.1144
NCI-H2023 GDSC2 6.1112 13.7931 0.1886 11.2365
NCI-H2595 GDSC2 6.1203 8.6354 2.4799 0.8685
DMS 114 GDSC2 6.1738 7.516 2.8957 0.052
NCI-H2591 GDSC2 6.1753 8.2959 2.6282 0.4463
HCC78 GDSC2 6.2971 17.178 -1.3106 17.118
A-549 GDSC2 6.3788 17.2334 -1.2804 16.85
NCI-H1355 GDSC2 6.4707 15.0703 -0.1809 12.2396
NCI-H2342 GDSC2 6.5933 15.1318 -0.1299 11.8017
NCI-H1693 GDSC2 6.8108 20.4367 -2.531 20.2539
NCI-H522 GDSC2 6.9591 16.0677 -0.3347 12.047
LOU-NH91 GDSC2 7.5477 30.5178 -6.935 28.7154
RERF-LC-KJ GDSC2 7.8152 17.2196 -0.3351 10.6744
NCI-H1944 GDSC2 7.8198 20.543 -1.8903 16.4465
NCI-H1650 GDSC2 8.4806 32.2251 -7.0884 27.5768
⏷ Show the Full List of 357 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1 3.7836 11.6079 -0.4429 24.1072
CBTCi002-A GDSC2 5.2447 7.8582 2.3849 1.9648
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KYSE-450 GDSC1 -5.6966 4.7732 -6.9517 73.0999
EC-GI-10 GDSC1 -4.5034 2.4977 -5.008 74.5641
TE-4 GDSC1 -3.5892 -1.2043 -3.5929 82.1733
OE21 GDSC1 -3.2954 4.6584 -4.3045 65.9184
KYSE-140 GDSC1 -1.7694 8.0878 -3.9967 55.6851
TE-15 GDSC2 -1.6647 6.504 -3.6032 44.1758
OE19 GDSC1 -1.2964 1.2762 -1.3409 57.2172
KYSE-180 GDSC1 -1.1793 4.6778 -2.0177 53.9738
T.T GDSC1 -1.0061 11.3508 -4.6934 51.3994
TE-4 GDSC2 -0.7536 0.969 -0.7623 37.2071
KYSE-410 GDSC1 -0.7374 3.432 -1.1387 50.5807
EC-GI-10 GDSC2 -0.5753 9.9297 -3.6065 42.5635
OE19 GDSC2 -0.5005 4.5885 -1.253 37.6237
TE-15 GDSC1 0.1416 9.5715 -2.7317 45.5542
KYSE-140 GDSC2 0.5291 10.5767 -2.8328 37.1005
KYSE-270 GDSC1 0.5487 5.566 -0.5156 39.3291
TE-5 GDSC1 0.7498 5.5099 -0.2821 37.2364
KYSE-450 GDSC2 0.8523 19.2562 -6.7866 41.3985
TE-10 GDSC1 1.0114 3.6761 0.6955 30.8458
KYSE-510 GDSC1 1.025 2.9604 0.9039 29.4772
TE-8 GDSC1 1.3582 5.5913 0.3115 30.9391
OE21 GDSC2 1.4936 21.4524 -7.3086 40.3561
TE-1 GDSC1 1.6178 3.72 1.34 23.1466
TE-9 GDSC1 1.6535 3.108 1.5548 21.4945
KYSE-520 GDSC1 1.759 10.4771 -1.6291 36.1654
TE-11 GDSC1 1.8134 8.8774 -0.7951 33.3696
TE-6 GDSC2 1.9996 10.4637 -1.403 28.1326
KYSE-520 GDSC2 2.1081 16.8817 -4.4943 35.3698
KYSE-270 GDSC2 2.2975 13.5409 -2.6645 31.0012
KYSE-410 GDSC2 2.3283 9.4831 -0.6214 24.102
KYSE-150 GDSC1 2.4657 4.1416 2.0833 13.3886
OE33 GDSC1 2.6063 4.8442 1.9051 14.0577
KYSE-180 GDSC2 2.7476 12.4771 -1.7427 27.0049
TE-11 GDSC2 2.884 16.0508 -4.0799 29.3529
TE-6 GDSC1 2.9593 6.6127 1.3653 16.5873
KYSE-70 GDSC1 3.1709 4.6574 2.5245 6.8587
T.T GDSC2 3.188 13.2183 -1.7383 25.7613
TE-1 GDSC2 3.2614 10.0464 -0.0909 18.9857
COLO 680N GDSC1 3.8007 7.618 1.5587 12.102
TE-9 GDSC2 4.9211 9.7143 1.3402 7.7426
TE-8 GDSC2 5.2791 15.2261 -1.0883 18.3384
KYSE-510 GDSC2 5.8092 16.7854 -2.2505 16.9607
KYSE-70 GDSC2 5.8134 9.2649 2.08 2.6656
OE33 GDSC2 6.1446 19.0377 -2.3257 20.8792
TE-10 GDSC2 6.1876 18.1987 -2.6717 17.7833
TE-5 GDSC2 6.3509 16.5729 -0.9807 15.7612
COLO 680N GDSC2 6.941 17.655 -1.0991 15.1359
KYSE-150 GDSC2 7.4553 23.2779 -3.4565 21.7315
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 59 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RMG-I GDSC1 -2.27 12.911 -6.6693 55.5817
JHOS-2 GDSC1 -2.0525 9.2698 -4.8014 56.3199
TOV-112D GDSC1 -0.8376 3.7157 -1.3309 51.4887
OVTOKO GDSC1 -0.3523 10.1946 -3.509 48.3955
IGROV-1 GDSC2 0.004 8.7878 -2.5028 38.4325
TOV-21G GDSC1 0.0332 4.1148 -0.5112 42.9912
OAW42 GDSC1 0.7182 5.4665 -0.2968 37.4917
OC 314 GDSC1 0.9632 3.3192 0.7485 30.8237
A2780 GDSC1 0.9724 2.6029 0.9123 29.7476
SK-OV-3 GDSC1 1.3294 6.391 -0.0779 32.9778
JHOS-4 GDSC1 1.4761 8.4618 -0.9116 35.3765
OVCAR-8 GDSC1 1.501 3.6749 1.2282 24.5601
DOV13 GDSC1 1.6337 8.3968 -0.7305 33.9927
OVCAR-4 GDSC1 1.8514 4.9712 1.0897 23.5956
JHOS-4 GDSC2 2.0833 10.2752 -1.8553 24.4919
OVCAR-3 GDSC1 2.2162 4.9593 1.4653 19.1481
OVCAR-5 GDSC1 2.3373 4.3839 1.8458 15.7742
OVISE GDSC1 2.5311 10.6968 -1.0436 31.1663
OVTOKO GDSC2 2.662 12.6237 -1.8897 27.7248
Kuramochi GDSC1 2.8417 7.0471 1.0454 19.3067
OVK18 GDSC1 2.8803 4.5362 2.3165 9.6878
OAW28 GDSC1 2.949 5.1265 2.0927 11.1294
EFO-21 GDSC1 3.002 6.3158 1.5507 15.0569
ES-2 GDSC1 3.1268 4.3738 2.6257 6.2412
IGROV-1 GDSC1 3.2109 6.4155 1.6817 13.2622
OVKATE GDSC1 3.2335 7.65 1.0838 17.4884
EFO-27 GDSC2 3.268 14.831 -3.1627 25.8155
Caov-4 GDSC1 3.2752 6.1494 1.8691 11.5909
A2780 GDSC2 3.2869 9.0544 0.4265 16.384
EFO-27 GDSC1 3.3135 4.9268 2.5125 6.4138
TOV-21G GDSC2 3.3204 6.8407 1.5613 10.1194
OV56 GDSC1 3.3255 5.0017 2.485 6.5875
TYK-nu GDSC1 3.3533 5.7762 2.1208 9.3508
DOV13 GDSC2 3.4141 5.8325 2.1426 6.5457
OAW42 GDSC2 3.7741 4.9846 2.8305 1.8322
OV-90 GDSC1 3.9945 6.146 2.4234 4.987
OVK18 GDSC2 4.4224 6.1728 1.7417 0.5528
RMG-I GDSC2 4.4323 24.448 -6.3306 33.1044
FU-OV-1 GDSC1 4.6004 13.0307 -0.5125 21.823
SK-OV-3 GDSC2 4.6227 14.5005 -1.2238 20.3203
OV-90 GDSC2 4.7182 6.8625 2.5352 1.9084
Caov-3 GDSC2 4.7704 6.3921 1.7971 0.2636
OAW28 GDSC2 5.0207 8.1931 2.1141 3.537
ES-2 GDSC2 5.1149 6.5696 2.8413 0.3897
TOV-112D GDSC2 5.1565 7.8235 2.3536 2.2065
Caov-4 GDSC2 5.1947 12.2922 0.2855 12.5523
FU-OV-1 GDSC2 5.198 15.5625 -1.3139 19.3704
OVCAR-5 GDSC2 5.3635 14.211 -0.5291 15.8879
OV56 GDSC2 5.6039 6.6701 2.9834 0.04
OVCAR-3 GDSC2 5.6639 12.0977 0.6987 9.6294
TYK-nu GDSC2 5.8893 7.6539 2.749 0.2935
JHOS-2 GDSC2 5.9447 20.4427 -3.9255 22.2351
OVISE GDSC2 6.8098 21.6244 -3.1105 21.9349
Kuramochi GDSC2 6.8187 15.0149 0.0692 10.5454
OC 314 GDSC2 6.8676 15.5913 -0.1695 11.5013
OVCAR-8 GDSC2 7.6655 16.4065 -0.0526 9.7334
OVCAR-4 GDSC2 8.054 18.0607 -0.5767 11.279
OVKATE GDSC2 8.5852 20.8355 -1.5337 14.0145
EFO-21 GDSC2 9.4578 22.1373 -1.5971 12.9612
⏷ Show the Full List of 59 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 60 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DAN-G GDSC1 0.2373 1.5616 0.2302 38.6003
HuP-T4 GDSC1 0.2407 7.8993 -1.8585 44.0743
Panc 02.03 GDSC1 0.4973 6.6181 -1.0224 41.0376
Panc 03.27 GDSC1 0.8859 4.8464 0.1338 34.6319
HuP-T3 GDSC1 0.9638 8.247 -1.3037 39.0872
CFPAC-1 GDSC1 1.1333 4.9716 0.3438 32.0747
KP-1N GDSC1 1.2709 3.4433 1.0493 27.0704
MIA PaCa-2 GDSC1 1.6424 4.2121 1.1873 24.0481
KP-3 GDSC1 1.9045 5.1426 1.0677 23.4703
PaTu 8902 GDSC1 2.0813 5.3286 1.161 21.9511
SW1990 GDSC1 2.1908 7.589 0.1853 27.3427
HPAF-II GDSC1 2.3031 6.0835 1.0214 21.8357
SUIT-2 GDSC1 2.4582 4.9984 1.6876 16.3711
PaTu 8988t GDSC1 2.4809 3.8699 2.2126 12.3664
Capan-1 GDSC1 2.5271 10.9587 -1.1776 31.6462
MZ-PC-1 GDSC1 2.5304 6.4178 1.0733 20.4523
SU.86.86 GDSC1 2.6424 8.3068 0.2428 25.032
KP-4 GDSC1 2.6456 3.5862 2.498 9.456
PL4 GDSC1 2.7383 5.2768 1.8238 14.09
PSN1 GDSC1 2.8406 3.9681 2.5439 8.1357
Panc 10.05 GDSC1 2.8573 7.7347 0.7173 21.3732
Panc 04.03 GDSC1 3.1321 14.9828 -2.6675 33.6968
KP-2 GDSC1 3.2109 4.5221 2.627 5.8962
Panc 08.13 GDSC1 3.2875 7.8663 1.021 17.7084
QGP-1 GDSC1 3.4785 6.6963 1.7634 11.6664
HPAC GDSC1 3.6295 8.2274 1.1205 15.7903
MIA PaCa-2 GDSC2 3.9033 11.2914 -0.1893 17.7453
PaTu 8902 GDSC2 3.9363 5.6965 2.5993 2.7874
Panc 02.03 GDSC2 4.1428 10.6682 0.3085 14.7813
HuP-T3 GDSC2 4.1905 8.6557 1.3398 9.2508
SUIT-2 GDSC2 4.2129 5.4223 2.8884 0.9074
KP-1N GDSC2 4.2252 7.0117 2.1647 4.6154
KP-3 GDSC2 4.2299 6.5234 2.3999 3.3314
SU.86.86 GDSC2 4.2321 8.7556 1.3213 9.2599
PL4 GDSC2 4.3283 8.6678 1.4343 8.4319
HPAC GDSC2 4.3606 8.7382 1.4231 8.4246
Capan-2 GDSC2 4.5128 12.7515 -0.4409 17.3906
QGP-1 GDSC2 4.6045 6.4221 1.7228 0.5097
BxPC-3 GDSC1 4.6758 8.6065 1.705 8.4828
HPAF-II GDSC2 4.7837 11.7927 0.2344 13.6708
Hs 766T GDSC1 4.7869 11.6961 0.2841 17.2547
KP-4 GDSC2 4.9321 6.4016 2.8289 0.5258
MZ-PC-1 GDSC2 5.0504 7.2532 1.5946 0.6408
DAN-G GDSC2 5.0782 12.84 -0.0646 14.4401
KP-2 GDSC2 5.318 8.9159 1.9612 3.8612
Hs 766T GDSC2 5.3758 13.1078 0.017 13.4429
CFPAC-1 GDSC2 5.3911 14.1831 -0.4957 15.6877
AsPC-1 GDSC2 5.4616 14.3787 -0.5406 15.7321
Panc 08.13 GDSC2 5.5239 10.5554 1.3341 6.6946
HuP-T4 GDSC2 5.5485 14.5956 -0.5843 15.7369
PSN1 GDSC2 5.9199 7.8405 2.694 0.398
Panc 03.27 GDSC2 5.9259 16.1111 -1.0539 16.8697
YAPC GDSC2 6.0313 13.5217 0.2648 11.0301
SW1990 GDSC2 6.1758 13.7901 0.2324 10.919
BxPC-3 GDSC2 6.2212 20.4161 -2.9457 22.573
Capan-1 GDSC2 6.2405 14.2332 0.0648 11.5654
PaTu 8988t GDSC2 6.6214 13.1102 0.8275 7.4091
Panc 04.03 GDSC2 6.7326 17.717 -1.2697 16.1515
YAPC GDSC1 6.7608 22.7883 -3.7153 26.9565
Panc 10.05 GDSC2 6.8302 16.7176 -0.7262 13.8773
⏷ Show the Full List of 60 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H28 GDSC1 -1.1344 14.8992 -6.4995 51.5248
MSTO-211H GDSC1 1.414 3.8079 1.0893 25.9782
NCI-H2452 GDSC1 1.9083 3.7686 1.6377 19.4921
IST-Mes1 GDSC1 2.5228 5.1005 1.7025 15.9627
MPP 89 GDSC1 3.1657 5.3498 2.175 9.623
MSTO-211H GDSC2 3.8811 8.0473 1.4075 9.584
NCI-H2452 GDSC2 4.0431 7.3038 1.8953 6.4834
MPP 89 GDSC2 4.5508 10.1248 0.8824 10.9164
IST-Mes1 GDSC2 4.974 8.6596 1.8721 4.8465
NCI-H2052 GDSC2 6.0836 8.5178 2.5092 0.8025
NCI-H28 GDSC2 7.8955 23.3627 -3.1905 20.2744
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LNCaP clone FGC GDSC1 1.2498 3.7433 0.9329 27.9441
22Rv1 GDSC1 2.5871 5.7776 1.4384 17.6279
PC-3 GDSC1 2.6306 5.131 1.792 14.8043
VCaP GDSC1 2.7229 3.8595 2.4707 9.2545
DU145 GDSC1 3.0926 12.8552 -1.6372 31.0411
NCI-H660 GDSC2 4.3186 5.8539 1.8178 0.3914
LNCaP clone FGC GDSC2 4.4143 6.75 2.4101 2.9656
22Rv1 GDSC2 4.877 6.8247 2.6339 1.2901
VCaP GDSC2 5.4688 6.8342 2.8814 0.1763
DU145 GDSC2 6.0098 7.7959 2.7437 0.2668
PC-3 GDSC2 6.1548 8.7399 2.4546 0.9246
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 GDSC1 0.6619 6.6895 -0.8864 39.699
A-253 GDSC2 5.6727 13.5529 0.0083 12.8891
Cancer Drug Sensitivity Data Curated from 113 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CHL-1 GDSC1 -3.3774 6.4986 -5.0492 63.7549
A-431 GDSC2 -1.0634 10.2364 -4.7186 42.837
A-388 GDSC1 0.0079 7.467 -1.8986 45.473
A-388 GDSC2 0.4421 9.6138 -2.9887 33.8798
WM278 GDSC1 0.6359 19.5409 -7.122 46.2563
WM115 GDSC1 0.9971 2.2551 0.9777 29.1824
COLO 800 GDSC1 1.1124 2.3337 1.0919 27.7486
WM1552C GDSC1 1.1779 2.6313 1.1281 27.1163
M14 GDSC1 1.1785 2.9666 1.0693 27.4901
COLO 792 GDSC1 1.2184 3.3119 1.029 27.5126
A-431 GDSC1 1.299 5.8921 0.1174 32.2456
CP50-MEL-B GDSC1 1.4845 3.0935 1.3741 23.6818
RVH-421 GDSC1 1.6148 3.9448 1.2582 23.7192
DJM-1 GDSC1 1.6818 5.2327 0.8007 26.3589
WM793 GDSC1 1.6851 3.9369 1.3367 22.7967
IGR-1 GDSC1 1.7365 3.3748 1.577 20.866
CHL-1 GDSC2 1.7555 10.008 -1.402 28.9284
HT-144 GDSC1 1.7979 3.5651 1.5865 20.4552
SK-MEL-2 GDSC1 1.8282 5.01 1.0489 23.9886
CP66-MEL GDSC1 1.892 4.0715 1.5078 20.4902
IGR-37 GDSC1 1.9717 3.5686 1.7743 18.1947
G-mel GDSC1 1.9769 3.7398 1.722 18.5297
WM35 GDSC1 1.9927 3.6691 1.7636 18.1529
A-375 GDSC1 2.2085 3.76 1.9643 15.5752
RPMI-7951 GDSC1 2.3659 5.0285 1.5826 17.5786
LOX-IMVI GDSC1 2.4128 3.7489 2.1875 12.9023
UACC-62 GDSC1 2.4255 4.0186 2.0935 13.5154
SK-MEL-24 GDSC1 2.5686 4.2479 2.1425 12.4459
IST-MEL1 GDSC1 2.5897 5.0507 1.7911 14.9944
Hs 938.T GDSC1 2.6116 4.7749 1.9429 13.7472
MZ-MEL-2 GDSC1 2.6603 5.9241 1.4353 17.3299
COLO 829 GDSC1 2.7323 5.3028 1.8055 14.2553
WT2-iPS GDSC1 2.7656 5.2789 1.8484 13.785
SK-MEL-30 GDSC1 2.8482 4.9722 2.075 11.6909
GAK GDSC1 2.9025 5.8684 1.6842 14.4585
MMAc-SF GDSC1 2.964 4.3572 2.4824 8.0421
G-361 GDSC1 2.975 4.0994 2.6164 6.9626
A101D GDSC1 2.9916 3.9593 2.6986 6.2591
Mel JuSo GDSC1 2.9972 4.1607 2.6086 6.9243
Hs 940.T GDSC2 3.0375 5.1211 1.4644 3.6674
LB2518-MEL GDSC1 3.251 5.4584 2.1941 9.1503
COLO 783 GDSC1 3.2693 5.1996 2.3388 7.9449
Hs 940.T GDSC1 3.2985 5.5197 2.2034 8.9018
COLO 783 GDSC2 3.3154 6.6841 0.903 6.4615
Mel Ho GDSC1 3.3318 4.9162 2.533 6.1865
MZ-MEL-7 GDSC1 3.3664 5.0072 2.5161 6.1963
SK-MEL-5 GDSC1 3.3702 6.342 1.8519 11.3761
SK-MEL-28 GDSC1 3.4085 5.1247 2.4917 6.2405
DJM-1 GDSC2 3.4318 6.1575 1.2314 4.2647
451Lu GDSC1 3.4736 6.0979 2.0582 9.4146
UACC-257 GDSC1 3.5293 5.0421 2.628 4.7665
MeWo GDSC1 3.5708 6.9515 1.7102 11.7483
SK-MEL-28 GDSC2 3.5993 5.2659 1.7288 1.2961
VMRC-MELG GDSC1 3.6473 6.0264 2.2304 7.4939
COLO 679 GDSC1 3.7352 5.8606 2.3784 6.0696
SH-4 GDSC1 3.7449 5.7897 2.4203 5.7163
HT-144 GDSC2 3.8522 5.4425 2.6644 2.5907
Mel Ho GDSC2 3.9004 7.6139 0.8473 5.6031
LB373-MEL-D GDSC2 3.9327 5.2586 1.8831 0.4057
SK-MEL-31 GDSC2 3.9795 15.4052 -2.8948 23.2097
CP66-MEL GDSC2 4.0304 5.2682 1.918 0.266
UACC-257 GDSC2 4.0736 6.1853 2.4578 3.3014
SK-MEL-3 GDSC2 4.08 5.7664 1.752 0.7425
SK-MEL-3 GDSC1 4.1162 6.0316 2.558 3.6819
RVH-421 GDSC2 4.1427 5.6457 1.8243 0.4633
A2058 GDSC2 4.2224 5.583 2.8243 1.1854
IPC-298 GDSC2 4.2331 15.1347 -2.5699 21.4902
CP50-MEL-B GDSC2 4.2913 13.9119 -1.925 18.889
SK-MEL-30 GDSC2 4.3342 5.5316 1.9375 0.1345
WM793 GDSC2 4.369 6.9563 2.2857 3.6968
VMRC-MELG GDSC2 4.3757 6.1551 1.7291 0.6193
MZ-MEL-7 GDSC2 4.3945 6.4995 1.6044 1.0458
SK-MEL-1 GDSC1 4.4192 5.9359 2.7764 1.6018
IST-MEL1 GDSC2 4.4376 7.0713 2.2755 3.6325
451Lu GDSC2 4.4822 18.148 -3.8708 25.0536
MeWo GDSC2 4.523 6.782 2.4607 2.5383
SK-MEL-31 GDSC1 4.5876 6.396 2.6674 2.0023
G-mel GDSC2 4.6174 6.4407 1.7211 0.5079
LB2518-MEL GDSC2 4.6305 6.0184 1.876 0.1619
SK-MEL-24 GDSC2 4.6362 7.5819 2.1622 3.894
LOX-IMVI GDSC2 4.7141 8.7933 1.6414 6.529
UACC-62 GDSC2 4.7306 6.015 2.8911 0.4585
MZ-MEL-2 GDSC2 4.7395 7.1191 1.5147 1.1074
WM278 GDSC2 4.7452 9.9346 1.1135 9.2901
RPMI-7951 GDSC2 4.8211 8.7319 1.741 5.7996
COLO 800 GDSC2 4.8694 19.5159 -4.2554 25.2732
COLO 792 GDSC2 4.8724 7.7586 2.2238 3.2078
SK-MEL-2 GDSC2 4.894 5.9632 2.9751 0.172
Hs 938.T GDSC2 4.9163 6.3946 1.8485 0.1413
WM115 GDSC2 4.9365 6.409 2.8279 0.526
A-375 GDSC2 4.9573 7.2881 2.4788 1.8762
Mel JuSo GDSC2 4.9915 6.767 2.7122 0.879
A101D GDSC2 5.0084 6.364 2.8746 0.3543
SK-MEL-5 GDSC2 5.0307 6.3028 1.918 0.0537
COLO 829 GDSC2 5.0536 8.1319 2.1608 3.2573
GAK GDSC2 5.0906 6.8121 2.7389 0.7111
COLO 679 GDSC2 5.1461 6.5028 2.878 0.2861
IGR-37 GDSC2 5.2179 6.4004 2.941 0.1428
WM1552C GDSC2 5.2209 6.8883 2.7655 0.5447
HMV-II GDSC2 5.2283 10.4853 1.1773 8.0185
LB373-MEL-D GDSC1 5.2735 22.0432 -4.4661 31.7947
MMAc-SF GDSC2 5.2991 18.4629 -3.4219 22.0112
SK-MEL-1 GDSC2 5.3219 6.4644 2.956 0.1002
WT2-iPS GDSC2 5.4158 6.6323 2.9319 0.1137
G-361 GDSC2 5.5425 6.8065 2.9172 0.1094
IGR-1 GDSC2 5.5545 7.1942 2.7861 0.3334
M14 GDSC2 5.7107 7.6811 2.6696 0.5509
SH-4 GDSC2 5.7368 8.0323 2.5472 0.9005
IPC-298 GDSC1 5.8379 7.0932 2.9224 0.0868
HMV-II GDSC1 5.8837 8.3159 2.5012 1.3033
WM35 GDSC2 6.3591 8.2884 2.6996 0.2481
EquiPSC Line K2 GDSC1 1.8097 4.292 1.3334 22.1458
EquiPSC Line K2 GDSC2 5.8316 20.4623 -4.0157 22.7056
⏷ Show the Full List of 113 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1 2.0557 3.1033 1.9931 16.232
HuTu 80 GDSC2 2.2736 9.2815 -1.1982 21.0306
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Rh30 GDSC1 -0.9961 6.9871 -2.7251 51.9903
G-401 GDSC1 0.3369 1.4808 0.3335 37.3339
SK-UT-1 GDSC1 1.3159 2.9457 1.2227 25.673
A-204 GDSC1 1.4353 3.8405 1.1012 25.7788
SW982 GDSC1 1.5687 3.2799 1.4199 22.8866
HT-1080 GDSC1 1.6976 3.1945 1.5824 21.0536
STS-0421 GDSC1 1.8092 4.0509 1.4273 21.4954
EW-8 GDSC1 1.8447 3.1068 1.7631 18.9934
SW872 GDSC1 1.997 3.4239 1.8469 17.5536
KYM-1 GDSC1 2.3538 3.2693 2.2793 12.5885
Rh41 GDSC1 2.3765 3.7373 2.153 13.3399
GCT GDSC1 2.5185 4.5702 1.9461 14.1545
MES-SA GDSC1 2.5297 3.5773 2.3763 10.938
SK-LMS-1 GDSC1 2.6819 3.7873 2.458 9.5543
RD GDSC1 2.7403 4.0831 2.3907 9.7638
G-402 GDSC1 2.9497 4.6495 2.3272 9.3056
RKN GDSC1 2.9797 4.0155 2.6606 6.6036
VA-ES-BJ GDSC1 3.2656 5.515 2.1781 9.2215
SW684 GDSC1 3.3495 10.7674 -0.3779 25.336
MFH-ino GDSC1 3.3546 4.9659 2.527 6.1522
Hs 633.T GDSC1 3.4524 5.9709 2.1046 9.1268
TE 441.T GDSC2 3.7489 5.0347 1.8913 0.4915
Rh41 GDSC2 3.7922 6.2354 2.2361 5.1098
Hs 633.T GDSC2 3.8694 5.2384 2.7725 1.9738
G-402 GDSC2 3.9879 6.3538 2.3187 4.2321
Rh30 GDSC2 4.1353 6.3412 2.4244 3.369
SK-LMS-1 GDSC2 4.3703 6.2619 2.6064 2.0349
RKN GDSC2 4.4155 6.1317 2.6897 1.57
Rh18 GDSC1 4.5274 8.4775 1.6664 9.1487
G-401 GDSC2 4.7742 10.6557 0.7836 10.9514
GCT GDSC2 4.8068 9.4217 1.4032 7.6277
SW982 GDSC2 4.8718 10.6504 0.8552 10.3794
SW684 GDSC2 4.9213 5.9493 2.99 0.1375
MES-SA GDSC2 4.9882 6.1864 2.9312 0.2289
A-204 GDSC2 5.0156 8.4163 2.0096 4.072
VA-ES-BJ GDSC2 5.2044 7.1708 2.6486 0.9398
EW-8 GDSC2 5.2958 6.6013 2.8995 0.192
STS-0421 GDSC2 5.4115 8.5181 1.2646 1.5107
HT-1080 GDSC2 5.5347 6.9175 2.8764 0.1681
KYM-1 GDSC2 5.5442 7.4079 2.7037 0.5437
SK-UT-1 GDSC2 5.7414 7.4015 2.783 0.2746
MFH-ino GDSC2 5.8436 7.5104 2.7826 0.2447
RD GDSC2 6.0586 12.2936 0.8599 8.152
SW872 GDSC2 6.8752 15.073 0.0777 10.4148
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 55 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NUGC-4 GDSC1 -5.0085 5.4218 -6.4186 70.364
NCI-N87 GDSC2 -2.5352 2.0418 -2.7716 52.9559
SK-GT-2 GDSC1 -2.4421 -0.3422 -2.4467 70.9802
SK-GT-2 GDSC2 -2.2542 -0.4654 -2.2559 50.8514
NCI-N87 GDSC1 -1.5904 1.6667 -1.6945 59.8912
IM95 GDSC1 -0.5502 11.8441 -4.4791 49.4559
TMK-1 GDSC1 -0.4253 4.2718 -1.0614 47.685
NUGC-3 GDSC1 -0.1459 15.6607 -5.9316 48.1975
AGS GDSC1 0.3852 2.1146 0.3484 36.9259
MKN28 GDSC1 1.1557 3.9058 0.7761 29.4826
23132/87 GDSC1 1.6551 3.4111 1.4777 22.0018
MKN1 GDSC1 1.7225 6.3567 0.3283 28.8832
RERF-GC-1B GDSC1 1.9301 4.2304 1.4854 20.4467
SNU-16 GDSC1 1.9554 3.3194 1.8313 17.8959
NUGC-3 GDSC2 2.2522 14.7658 -3.3142 32.6899
HSC-39 GDSC1 2.4924 3.4252 2.3864 11.0728
SCH GDSC1 2.5838 4.4123 2.0837 12.8136
SNU-5 GDSC1 2.9759 5.5263 1.9196 12.3603
Hs 746.T GDSC1 3.0091 4.0438 2.6759 6.3536
Fu97 GDSC1 3.1367 4.3835 2.6298 6.1682
KATO III GDSC1 3.1859 5.0868 2.3237 8.3784
OCUM-1 GDSC1 3.1987 5.3292 2.2139 9.1918
RERF-GC-1B GDSC2 3.2589 9.2629 0.2987 17.1059
GCIY GDSC2 3.2595 11.4743 -0.8064 22.1218
RF-48 GDSC1 3.3927 5.6226 2.2301 8.3538
MKN45 GDSC1 3.3986 5.9788 2.0568 9.6886
HSC-39 GDSC2 3.443 5.7395 2.2125 6.0704
TMK-1 GDSC2 3.6097 10.9257 -0.9596 16.2006
ECC12 GDSC2 3.8981 4.9275 1.9891 0.1599
KATO III GDSC2 3.9114 7.2026 1.8483 7.0374
MKN7 GDSC1 3.9676 16.9858 -2.9797 31.9323
23132/87 GDSC2 4.0431 10.0417 0.5425 13.8438
ECC10 GDSC1 4.1311 7.9767 1.6296 10.5441
SCH GDSC2 4.329 12.3787 -1.1478 15.4005
TGBC11TKB GDSC1 4.407 9.5401 1.0642 13.6488
HGC-27 GDSC2 4.5028 6.6154 2.5241 2.252
MKN45 GDSC2 4.631 5.6154 2.9995 0.2142
MKN1 GDSC2 4.7543 15.0891 -1.4147 20.728
RF-48 GDSC2 4.8914 7.0117 2.5625 1.5798
Fu97 GDSC2 4.9344 10.5273 0.9584 9.7182
IM95 GDSC2 5.1357 9.1963 1.7235 5.3477
Hs 746.T GDSC2 5.1648 6.7835 2.7817 0.5292
SNU-16 GDSC2 5.5262 6.8424 2.8992 0.1361
SNU-1 GDSC2 5.68 7.4242 2.7516 0.362
SNU-5 GDSC2 5.7127 7.1675 2.8541 0.1611
ECC10 GDSC2 5.7337 7.1877 2.8546 0.1557
SNU-1 GDSC1 5.8918 7.6194 2.7621 0.3672
TGBC11TKB GDSC2 5.9659 8.1873 2.5849 0.6509
NUGC-4 GDSC2 6.0785 25.0454 -5.3367 28.3814
AGS GDSC2 6.1778 12.7272 0.7327 8.5649
MKN28 GDSC2 6.2761 14.3459 0.0348 11.6362
OCUM-1 GDSC2 6.2815 9.2052 2.3296 1.2458
MKN7 GDSC2 6.9753 17.2329 -0.8752 14.2121
SNG-M GDSC1 -1.3261 2.4715 -1.5463 56.6175
SNG-M GDSC2 3.641 7.3532 1.5656 9.2744
⏷ Show the Full List of 55 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IHH-4 GDSC1 0.8183 1.7176 0.8165 31.3062
CAL-62 GDSC1 1.5159 3.1277 1.4004 23.323
KMH-2 GDSC1 1.8724 3.0859 1.7977 18.602
K5 GDSC1 1.9163 3.3967 1.7668 18.556
HTC-C3 GDSC1 2.2355 3.7222 2.0071 15.1273
BHT-101 GDSC1 2.4798 4.2585 2.047 13.5874
8505C GDSC1 2.531 4.3155 2.0741 13.1376
8305C GDSC1 2.7825 4.6625 2.1621 11.3063
WRO GDSC1 2.8925 5.562 1.8266 13.4169
B-CPAP GDSC1 2.9855 4.2643 2.5476 7.4449
FTC-133 GDSC1 3.0168 4.1287 2.6427 6.575
TT GDSC1 3.4423 6.7578 1.7033 12.2497
ASH-3 GDSC1 3.4441 5.4189 2.3735 7.0479
TT2609-C02 GDSC1 3.4495 5.2713 2.4514 6.4167
CAL-62 GDSC2 3.7869 5.448 2.617 2.9798
ML-1 [Human leukemia] GDSC2 4.1482 6.3237 1.5603 1.4582
BHT-101 GDSC2 4.2125 6.2688 2.5081 2.7866
FTC-133 GDSC2 4.2247 7.9586 1.7061 7.1518
IHH-4 GDSC2 4.2439 6.2102 2.5547 2.491
TT GDSC2 4.3004 11.033 0.2484 14.7014
K5 GDSC2 4.3631 8.7231 1.4322 8.3693
WRO GDSC2 4.4977 6.7857 2.4441 2.6601
CGTH-W-1 GDSC2 4.5592 6.1366 2.763 1.0751
KMH-2 GDSC2 4.8292 6.3913 1.8188 0.2067
B-CPAP GDSC2 4.8498 7.8889 2.1511 3.6086
TT2609-C02 GDSC2 5.0972 7.1227 2.6181 1.1439
8305C GDSC2 5.1911 8.9727 1.8606 4.556
ASH-3 GDSC2 5.2708 6.8391 2.8043 0.4111
HTC-C3 GDSC2 5.6726 8.5339 2.3164 1.8077
8505C GDSC2 6.306 8.1733 2.7203 0.228
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 80 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Ca9-22 GDSC1 -5.6439 4.2886 -6.7429 73.8327
JHU-029 GDSC1 -5.3496 1.4547 -5.705 79.4231
CAL-27 GDSC1 -5.154 7.2535 -7.2358 68.1895
SAT [Human HNSCC] GDSC1 -4.6457 6.7667 -6.5084 67.4745
HSC-4 GDSC1 -4.5124 9.5518 -7.4733 64.1245
DOK GDSC1 -4.2876 7.8984 -6.5628 65.1316
JHU-022 GDSC1 -4.1711 14.8066 -9.4376 59.8072
SCC-15 GDSC1 -3.7481 4.9283 -4.8854 67.2508
CAL-33 GDSC1 -3.3849 6.2309 -4.9563 64.1027
NCI-H3118 GDSC1 -3.1786 10.8923 -6.6693 59.3486
HSC-3 GDSC1 -3.0529 4.113 -3.8662 65.7318
DOK GDSC2 -2.9714 8.6595 -5.4895 53.515
JHU-022 GDSC2 -2.8934 10.163 -6.0559 52.8784
SCC-9 GDSC1 -2.732 12.4136 -6.9014 57.1981
FaDu GDSC1 -2.2778 9.7902 -5.2613 56.9328
PCI-04B GDSC1 -2.19 4.1194 -2.9287 61.2144
PCI-15A GDSC2 -1.8723 6.7328 -3.9165 45.5624
BB30-HNC GDSC1 -1.4898 6.9086 -3.2089 54.8582
BICR 78 GDSC1 -1.4236 8.9331 -4.0093 53.7264
UPCI-SCC-090 GDSC1 -1.1649 10.7778 -4.5846 52.1421
BB30-HNC GDSC2 -1.0752 6.7737 -3.1203 40.5104
BHY GDSC1 -1.0104 4.5482 -1.7898 52.7342
HSC-2 GDSC1 -0.9262 9.4686 -3.7457 51.238
Ca9-22 GDSC2 -0.8832 7.0045 -2.6148 42.5533
HO-1-N-1 GDSC1 -0.8455 7.1968 -2.6574 51.0418
PCI-15A GDSC1 -0.7748 4.8725 -1.651 50.7877
PCI-06A GDSC1 -0.7305 12.3302 -4.8847 50.2126
SAT [Human HNSCC] GDSC2 -0.6407 8.859 -3.1816 42.281
UPCI-SCC-090 GDSC2 -0.2131 12.1665 -4.3066 42.0447
PCI-38 GDSC1 -0.1592 3.4642 -0.517 44.5818
CAL-27 GDSC2 -0.064 11.0117 -3.6123 40.6207
JHU-029 GDSC2 0.0158 8.6644 -2.9293 35.3463
HO-1-u-1 GDSC2 0.0454 8.2022 -2.1928 37.5839
KOSC-2 GDSC1 0.4237 5.1291 -0.4684 40.0155
SCC-15 GDSC2 0.6551 9.073 -1.9948 34.6619
PE/CA-PJ15 GDSC1 0.6694 12.8306 -3.7906 44.1906
BICR 22 GDSC1 0.6884 13.4098 -4.0556 44.347
Detroit 562 GDSC1 0.8115 3.2354 0.6054 32.6336
SKN-3 GDSC1 0.8438 5.8017 -0.3092 36.7527
NCI-H3118 GDSC2 0.884 18.512 -6.3896 40.9621
LB771-HNC GDSC1 0.9748 5.4397 -0.0181 34.7697
KON GDSC1 0.9764 3.267 0.777 30.5674
FaDu GDSC2 1.0785 13.1527 -3.5689 36.6794
JHU-011 GDSC2 1.0872 17.151 -6.1451 37.8943
SCC-4 GDSC1 1.1389 7.6696 -0.8606 36.9384
SAS GDSC1 1.1723 10.3345 -2.1048 39.819
SCC-25 GDSC1 1.1996 11.0052 -2.4055 40.2513
KOSC-2 GDSC2 1.2525 9.9607 -2.4216 29.288
BB49-HNC GDSC1 1.3561 3.8087 1.0264 26.7224
PCI-04B GDSC2 1.3641 11.4686 -3.0722 30.9542
SCC-9 GDSC2 1.5547 11.0771 -2.1116 31.7999
BHY GDSC2 1.5988 7.23 -0.758 21.0209
HSC-2 GDSC2 1.7892 11.3184 -2.0159 30.7627
OSC-19 GDSC1 2.0236 6.165 0.713 25.1527
JHU-011 GDSC1 2.0818 6.0895 0.8054 24.2941
OSC-20 GDSC1 2.1128 6.8979 0.4479 26.2837
BICR 10 GDSC1 2.2128 3.9092 1.9125 15.9211
HSC-3 GDSC2 2.3695 10.4129 -1.0455 25.6666
PCI-06A GDSC2 2.4927 14.9005 -3.8256 29.7189
HO-1-u-1 GDSC1 2.6271 7.6302 0.5644 23.2738
CAL-33 GDSC2 2.7111 10.9665 -1.0206 24.5379
PCI-30 GDSC1 2.7138 6.5045 1.1992 18.7871
OSC-19 GDSC2 2.7963 13.4511 -2.8525 26.0605
Detroit 562 GDSC2 2.8409 12.4104 -1.6291 26.3599
HO-1-N-1 GDSC2 2.8741 10.8442 -0.8186 23.2621
PE/CA-PJ15 GDSC2 3.2572 6.2771 1.0591 5.6457
BB49-HNC GDSC2 3.2692 7.3072 1.2852 11.8151
SCC-25 GDSC2 3.8221 8.3099 0.467 7.9577
BICR 22 GDSC2 4.0526 6.7003 2.1961 4.7824
KON GDSC2 4.2603 15.4097 -2.6852 21.8364
SAS GDSC2 4.2991 15.2108 -1.8291 23.2409
BICR 10 GDSC2 4.3506 10.8129 0.3954 13.8585
PCI-30 GDSC2 4.5928 11.6526 0.1624 14.4424
BICR 31 GDSC2 4.8264 6.6334 1.7325 0.3837
BICR 78 GDSC2 4.9557 14.2676 -0.8562 18.1257
HSC-4 GDSC2 4.9967 15.208 -1.2896 19.721
SKN-3 GDSC2 5.0045 11.8394 0.371 12.5342
LB771-HNC GDSC2 5.5585 7.8091 2.5558 0.9971
SCC-4 GDSC2 6.2642 14.2564 0.0694 11.5023
OSC-20 GDSC2 6.4832 16.8528 -1.0246 15.6833
⏷ Show the Full List of 80 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 32 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
5637 GDSC1 -0.0259 4.6808 -0.7757 44.0516
CAL-29 GDSC1 0.4876 7.7492 -1.5425 42.1785
BFTC-905 GDSC1 1.6304 3.1845 1.5115 21.9173
HT-1376 GDSC1 1.6381 5.4682 0.6514 27.5017
RT-4 GDSC1 1.7364 3.7808 1.4477 21.7514
SW780 GDSC1 1.8322 6.7953 0.2282 28.8513
SW1710 GDSC1 1.9255 5.883 0.7495 25.4159
RT-112 GDSC1 1.9766 3.2231 1.8795 17.4492
647V GDSC1 2.0184 6.62 0.4914 26.4917
639V GDSC1 2.124 4.7492 1.4665 19.5915
TCCSUP GDSC1 2.4724 4.7566 1.8143 15.3591
UM-UC-3 GDSC1 2.6451 3.4958 2.5294 9.2369
KU-19-19 GDSC1 2.8764 3.887 2.6166 7.4192
T24 GDSC1 2.9207 3.9953 2.6118 7.2461
J82 GDSC1 3.0384 7.1135 1.185 17.5499
CAL-29 GDSC2 3.3904 13.9256 -1.923 25.8254
HT-1197 GDSC1 3.4019 4.9991 2.549 5.8123
SW1710 GDSC2 3.8233 5.7998 2.4719 3.7147
BFTC-905 GDSC2 4.069 7.1806 1.9742 5.9863
647V GDSC2 4.0732 6.2171 2.4424 3.3861
KU-19-19 GDSC2 4.1561 6.2224 2.494 2.9582
TCCSUP GDSC2 4.8082 7.1232 2.4704 2.0976
639V GDSC2 4.8204 7.0137 2.5246 1.8315
T24 GDSC2 5.0797 7.2559 1.6053 0.5956
HT-1197 GDSC2 5.1124 6.7472 2.7734 0.5855
RT-112 GDSC2 5.3517 9.4995 1.7161 5.0368
SW780 GDSC2 5.5029 6.9077 2.8683 0.1893
J82 GDSC2 6.0117 7.8332 2.7313 0.2891
5637 GDSC2 6.1498 19.7653 -2.6786 21.9408
HT-1376 GDSC2 6.3602 13.5989 0.441 9.633
RT-4 GDSC2 7.4202 20.0028 -1.8997 17.1533
UM-UC-3 GDSC2 8.934 18.9135 -0.4425 9.5056
⏷ Show the Full List of 32 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 76 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OVCA420 GDSC1 -5.7957 6.2524 -7.5587 71.0211
OVMIU GDSC1 -5.5953 3.4502 -6.4451 75.3292
DoTc2 4510 GDSC1 -3.2976 10.5907 -6.6583 59.9001
CAL-39 GDSC2 -2.8165 3.3608 -3.3878 54.483
CAL-39 GDSC1 -2.6361 3.1205 -3.1264 65.3189
BPH-1 GDSC1 -2.1718 9.3178 -4.9448 56.7724
OVCA420 GDSC2 -2.004 10.7074 -5.3934 49.37
C-33 A GDSC1 -1.0772 5.6177 -2.2554 52.8708
BPH-1 GDSC2 -0.8743 14.0696 -5.8525 45.5238
OVMIU GDSC2 -0.5938 11.5915 -4.4021 43.4955
DSH1 GDSC1 -0.1993 3.2405 -0.499 44.8888
SW954 GDSC1 -0.0064 7.4439 -1.9029 45.5627
DSH1 GDSC2 0.3136 8.2072 -1.9268 35.8242
UWB1.289 GDSC1 0.712 12.3532 -3.5182 43.7665
PEO1 GDSC1 0.7596 5.4525 -0.2476 37.0445
PWR-1E GDSC1 0.8848 2.1484 0.8684 30.5673
NEC8 GDSC1 1.6044 3.2387 1.4696 22.3481
ME-180 GDSC1 1.7354 17.813 -5.2848 42.0207
JAR GDSC1 1.7478 3.1667 1.6438 20.3525
C-4-I GDSC1 1.8318 3.8077 1.5412 20.581
KGN GDSC1 1.9324 4.3864 1.4241 20.8672
UWB1.289 GDSC2 1.9933 12.4779 -3.0324 28.9007
NT2-D1 GDSC1 2.1407 5.2221 1.2693 20.9097
SW962 GDSC1 2.1801 3.8187 1.912 16.0972
JEG-3 GDSC1 2.3042 3.4422 2.1763 13.5703
HEC-1 GDSC1 2.3559 8.4298 -0.0758 27.9017
OMC-1 [Human cervical carcinoma] GDSC2 2.6046 10.9934 -1.7805 22.6339
HEY GDSC1 2.6456 5.6825 1.5395 16.6288
DoTc2 4510 GDSC2 2.6996 9.631 -0.3652 21.8553
C-33 A GDSC2 2.7488 10.2661 -0.6386 22.8883
SKN GDSC1 2.8008 6.495 1.2826 17.8318
ACC-OV7 GDSC1 3.0191 5.7486 1.8479 12.7392
LB831-BLC GDSC1 3.2941 5.5041 2.2076 8.885
OV17R GDSC1 3.3661 9.488 0.2756 21.9768
JHOS-3 GDSC2 3.4838 7.2675 0.7377 7.0865
OMC-1 [Human cervical carcinoma] GDSC1 3.5071 8.6377 0.8168 18.2331
ME-180 GDSC2 3.5098 24.6594 -7.1906 36.0296
JEG-3 GDSC2 3.7504 6.4969 1.2706 3.4708
ACC-OV7 GDSC2 3.77 9.6276 -0.2057 11.8853
OVCA433 GDSC1 3.835 20.0909 -4.6389 35.5264
PA-1 GDSC2 3.8541 7.3038 1.7552 7.6934
HeLa GDSC2 3.8966 5.2485 2.7851 1.8597
SW954 GDSC2 3.9121 15.1745 -2.832 23.1581
JAR GDSC2 4.0143 5.9177 1.6622 1.1524
JHOS-3 GDSC1 4.0195 14.6555 -1.7745 28.4541
OV17R GDSC2 4.0274 7.1371 1.1433 3.719
Ca Ski GDSC2 4.0352 15.582 -2.2243 25.1472
SiHa GDSC1 4.0727 7.646 1.7492 9.8416
SKN GDSC2 4.2184 7.4134 1.9665 5.7209
HT-3 GDSC1 4.2271 13.838 -1.2022 25.8241
SiHa GDSC2 4.242 6.3694 2.4797 2.8865
NT2-D1 GDSC2 4.3081 7.0398 2.2066 4.2309
TC-YIK GDSC1 4.351 9.5756 1.0057 14.2019
SiSo GDSC1 4.4086 10.3612 0.6618 16.1945
SKG-IIIa GDSC1 4.4199 9.2099 1.2353 12.4646
HeLa GDSC1 4.571 5.8143 2.8994 0.738
MS751 GDSC1 4.5998 7.2155 2.3089 4.3696
HEC-1 GDSC2 4.6866 7.2649 2.3382 2.9104
LB831-BLC GDSC2 4.7945 8.157 1.9937 4.5116
SW962 GDSC2 4.9824 6.8254 1.7231 0.3457
NEC8 GDSC2 5.0911 6.5794 2.828 0.4375
HEY GDSC2 5.1277 8.3179 2.12 3.3527
SW756 GDSC1 5.1551 6.9271 2.7224 0.9882
OVCA433 GDSC2 5.2357 12.0875 -0.3988 9.8694
C-4-I GDSC2 5.3745 10.3951 1.3146 7.0498
TC-YIK GDSC2 5.3988 7.7276 2.5151 1.2743
PWR-1E GDSC2 5.4183 7.3098 2.6884 0.659
SW756 GDSC2 5.4785 11.666 0.7813 9.5642
SiSo GDSC2 5.5449 7.5865 2.6363 0.7412
Ca Ski GDSC1 5.6246 15.748 -1.0923 21.4602
NCC-IT GDSC2 5.6923 7.1675 2.8468 0.1768
HT-3 GDSC2 5.9005 13.6535 0.1149 11.9637
SKG-IIIa GDSC2 6.267 22.0353 -3.7082 24.5025
PEO1 GDSC2 6.9427 17.8749 -1.2031 15.5244
KGN GDSC2 8.5628 22.2517 -2.2128 16.3036
MS751 GDSC2 9.1283 25.9358 -3.5889 19.4034
⏷ Show the Full List of 76 Cancer Drug Sensitivity Data of This Drug

References

1 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 7717).
2 Clinical pipeline report, company report or official report of AstraZeneca (2009).