General Information of Drug (ID: DMIQAY4)

Drug Name
VER-155008
Synonyms Heat shock protein 70 inhibitor (cancer), Vernalis; Hsp 70 inhibitor (cancer), Vernalis
Indication
Disease Entry ICD 11 Status REF
Alzheimer disease 8A20 Preclinical [1]
Solid tumour/cancer 2A00-2F9Z Investigative [2]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
Chemical Identifiers
Formula
C25H23Cl2N7O4
Canonical SMILES
C1=CC(=CC=C1COCC2C(C(C(O2)N3C4=NC=NC(=C4N=C3NCC5=CC(=C(C=C5)Cl)Cl)N)O)O)C#N
InChI
1S/C25H23Cl2N7O4/c26-16-6-5-15(7-17(16)27)9-30-25-33-19-22(29)31-12-32-23(19)34(25)24-21(36)20(35)18(38-24)11-37-10-14-3-1-13(8-28)2-4-14/h1-7,12,18,20-21,24,35-36H,9-11H2,(H,30,33)(H2,29,31,32)/t18-,20-,21-,24-/m1/s1
InChIKey
ZXGGCBQORXDVTE-UMCMBGNQSA-N
Cross-matching ID
PubChem CID
25195348
ChEBI ID
CHEBI:95010
CAS Number
1134156-31-2
TTD ID
D0H0AU
Repurposed Drugs (RPD) Click to Jump to the Detailed RPD Information of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 150 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 1.2726 4.4247 1.099 26.7703
MEC1 CTRP2 4.7296 7.6425 3.5731 7.8498
JM1 CTRP2 4.7802 8.2208 3.3326 8.7417
SKM-1 CTRP2; CTRP1 1.0901 2.7354 1.084 27.4136
EM-2 CTRP2 1.0919 3.241 1.0633 27.477
THP-1 CTRP2; CTRP1 1.1082 3.6589 1.0422 27.4951
PL21 CTRP2; CTRP1 1.1348 4.2949 0.9748 27.6384
NCO2 CTRP2 1.3175 3.0279 1.3071 25.9159
OPM-2 CTRP2 1.373 2.9065 1.3673 25.5313
HH [Human lymphoma] CTRP2 1.4262 3.6744 1.3767 25.325
A4/Fukuda CTRP2 1.4515 3.715 1.3992 25.1661
Peer CTRP2 1.456 3.6706 1.4084 25.1203
EoL-1 CTRP2 1.5812 2.8848 1.5786 24.1362
Ku812 CTRP2; CTRP1 1.6517 3.5437 1.6245 23.7499
Pfeiffer CTRP2 1.6582 4.7953 1.4386 24.3706
MOLM-13 CTRP2 1.7281 3.4842 1.7079 23.2183
Ki-JK CTRP2 1.7343 4.7329 1.5356 23.7925
KMS-26 CTRP2 1.8281 4.0499 1.7591 22.7189
JURL-MK1 CTRP2 1.8297 3.5201 1.811 22.5377
SU-DHL-1 CTRP2 1.8397 3.3099 1.8311 22.4375
RPMI-8226 CTRP2; CTRP1 1.8423 3.3903 1.8305 22.4306
M-07e CTRP2 2.0439 5.6146 1.6362 22.4837
KMS-12-BM CTRP2 2.1169 3.2481 2.1144 20.5735
BL-70 CTRP2; CTRP1 2.1591 3.6166 2.1458 20.3291
KMS-11 CTRP2; CTRP1 2.2717 4.635 2.14 19.9869
MOLM-16 CTRP2; CTRP1 2.3033 3.8855 2.2783 19.4096
OCI-AML-3 CTRP2; CTRP1 2.3149 6.328 1.6874 21.4975
GA-10 CTRP2 2.4745 4.8472 2.3153 18.7362
ALL-SIL CTRP2 2.5025 6.6638 1.7613 20.6863
SU-DHL-5 CTRP1 2.5255 3.9923 2.5019 38.4971
OCI-AML-2 CTRP2 2.5458 4.7691 2.4098 18.1803
Mino CTRP2 2.5468 7.855 1.3162 22.2184
F-36P CTRP2 2.5556 5.0241 2.3617 18.3202
KE-97 CTRP2; CTRP1 2.5993 5.5135 2.2724 18.5105
LAMA-84 CTRP2 2.6035 5.2156 2.3638 18.1662
KCL-22 CTRP2 2.6307 5.2488 2.3844 18.0094
PF-382 CTRP2 2.6761 5.5644 2.3402 18.0342
JVM-3 CTRP2 2.6781 5.2224 2.4434 17.6528
CML-T1 CTRP2 2.7445 4.9482 2.5859 16.9398
SIG-M5 CTRP2 2.7502 4.613 2.6618 16.6553
MOLT-16 CTRP2 2.761 5.0045 2.5905 16.8727
KMS-34 CTRP2 2.823 4.8481 2.6941 16.3135
WSU-DLCL2 CTRP2; CTRP1 2.8856 6.6098 2.1897 17.9967
NB4 CTRP2 2.8996 4.5276 2.8367 15.5741
Daudi CTRP2 2.9706 5.2854 2.745 15.6785
NALM-6 CTRP2 2.9832 6.2919 2.4174 16.8594
OCI-Ly19 CTRP2 2.9986 7.8387 1.7873 19.2332
Reh CTRP2 3.0657 5.9876 2.6193 15.8635
Ri-1 CTRP2 3.1206 6.2761 2.5702 15.894
SR CTRP2 3.1684 4.5676 3.1188 13.741
697 CTRP2 3.1969 5.6039 2.894 14.4599
MV4-11 CTRP2 3.215 7.1714 2.3017 16.6723
Jurkat CTRP2 3.2205 5.685 2.8926 14.3958
P31/FUJ CTRP2 3.2281 6.7539 2.4922 15.8978
KE-37 CTRP2 3.255 6.414 2.659 15.1814
Namalwa CTRP2 3.3399 6.0412 2.894 14.0486
RPMI-8402 CTRP2 3.3675 6.3159 2.8173 14.264
SU-DHL-6 CTRP2 3.3871 5.699 3.0683 13.2588
MOLM-6 CTRP2 3.3892 6.7321 2.6698 14.7751
CA46 CTRP2 3.42 5.8301 3.0578 13.203
NU-DUL-1 CTRP2; CTRP1 3.4787 5.4992 3.2342 12.3761
DEL CTRP2 3.4804 5.3025 3.2963 12.1441
U-937 CTRP2; CTRP1 3.57 5.8419 3.215 12.1833
P12-Ichikawa CTRP2 3.5904 6.9529 2.7834 13.798
SUP-T1 CTRP2 3.5981 7.3509 2.6146 14.4453
Karpas-299 CTRP2 3.6029 6.9693 2.7891 13.7429
OCI-AML-5 CTRP2 3.6434 6.2625 3.1306 12.3013
EB1 CTRP2 3.6454 6.9354 2.8476 13.4016
L-540 CTRP2 3.6582 5.9123 3.2835 11.6745
TF-1 CTRP2 3.6617 5.9327 3.2795 11.6803
Kasumi-1 CTRP2 3.6937 6.1747 3.2191 11.822
SU-DHL-10 CTRP2 3.7466 5.6103 3.488 10.653
KYO-1 CTRP2 3.7595 6.0136 3.3527 11.1276
ST486 CTRP2 3.7837 6.522 3.1694 11.7728
HuNS1 CTRP2 3.8177 8.2727 2.4055 14.7362
KMS-21-BM CTRP2 3.8296 6.4905 3.2305 11.4115
JeKo-1 CTRP2 3.8602 6.4984 3.2589 11.2195
AMO1 CTRP2; CTRP1 3.9372 5.3951 3.7662 9.0658
SU-DHL-8 CTRP2 3.9746 6.5766 3.3427 10.5897
DB CTRP2 3.9871 6.3947 3.4348 10.1938
CMK CTRP2 4.0442 5.4299 3.8714 8.3625
BV-173 CTRP2 4.0554 6.1236 3.6208 9.2848
SU-DHL-4 CTRP2; CTRP1 4.085 6.9985 3.2646 10.6205
K-562 CTRP2 4.0899 6.3954 3.5405 9.5081
HT CTRP2; CTRP1 4.1318 7.8258 2.9221 11.8941
HEL 92.1.7 CTRP2 4.1395 6.1228 3.7089 8.7158
MOLP-8 CTRP2 4.1422 6.3956 3.5941 9.1605
MC116 CTRP2; CTRP1 4.2107 4.9096 4.1842 6.7316
L-363 CTRP2 4.2259 5.8646 3.9064 7.7157
ME1 CTRP2 4.3584 8.298 2.909 11.4227
MOTN-1 CTRP2 4.411 7.3828 3.4023 9.2748
GDM-1 CTRP2; CTRP1 4.415 8.1501 3.034 10.7804
RS4;11 CTRP2 4.4219 10.773 1.7469 15.9814
HL-60 CTRP2 4.425 8.1705 3.0334 10.7603
RL CTRP2 4.455 6.4638 3.8796 7.2264
MOLT-13 CTRP2 4.4552 9.7134 2.3017 13.6947
EJM CTRP2; CTRP1 4.4946 10.3556 2.0188 14.7488
Ci-1 CTRP2 4.5292 6.4882 3.9418 6.7925
NCI-H929 CTRP2 4.5357 8.7832 2.8341 11.3376
KM-H2 CTRP2 4.5366 8.8968 2.7789 11.5633
RCH-ACV CTRP2 4.5746 8.3444 3.0858 10.211
KMS-27 CTRP2 4.6026 7.9798 3.2909 9.2994
HuT 78 CTRP2 4.6335 8.0578 3.2808 9.2738
SEM CTRP2 4.663 7.0796 3.7874 7.1102
HEL CTRP2 4.6683 7.5196 3.5773 7.967
HD-MY-Z CTRP2 4.7217 7.7325 3.5215 8.081
Mono-Mac-1 CTRP2 4.7514 7.6829 3.5729 7.8027
KMS-20 CTRP2 4.8079 7.0644 3.9292 6.1988
TALL-1 [Human adult T-ALL] CTRP2 4.839 7.3118 3.8355 6.5203
Mono-Mac-6 CTRP2 4.875 18.9602 -1.9466 26.5771
KMS-18 CTRP2 4.9139 8.2248 3.4489 7.9757
OCI-Ly3 CTRP2 4.9173 6.2208 4.4436 3.8244
SUP-B15 CTRP2 4.9186 7.6458 3.7411 6.7448
KHM-1B CTRP2 4.9766 11.7772 1.7295 14.884
SET-2 CTRP2 5.0501 9.6011 2.8795 10.0768
OCI-M1 CTRP2 5.0743 7.7675 3.8161 6.1115
SK-MM-2 CTRP2 5.1115 7.6325 3.9154 5.6211
NU-DHL-1 CTRP2 5.2975 9.5219 3.1262 8.5677
AML-193 CTRP2 5.3327 9.9284 2.9518 9.2276
MHH-CALL-3 CTRP2 5.3751 7.6461 4.1263 4.2353
Raji CTRP2 5.3843 9.7375 3.0894 8.5576
SUP-M2 CTRP2 5.4011 7.0988 4.4194 2.9634
KO52 CTRP2 5.5445 7.2991 4.429 2.6829
EHEB CTRP2 5.5499 10.252 2.9659 8.7667
HPB-ALL CTRP2 5.5986 8.9033 3.676 5.7216
MM1.S CTRP2 5.5992 11.3562 2.4545 10.7814
NOMO-1 CTRP2; CTRP1 5.7045 10.6196 2.905 8.7416
KMM-1 CTRP2 5.8565 9.4644 3.5942 5.6269
Granta-519 CTRP2 5.8756 12.3102 2.1978 11.3185
SUP-T11 CTRP2 5.9013 10.1376 3.2955 6.7882
Hs 611.T CTRP2 5.9017 10.0422 3.3429 6.5918
U266B1 CTRP2 6.0236 10.0403 3.4344 6.0162
Karpas-620 CTRP2 6.0475 9.1541 3.8844 4.1376
REC-1 CTRP2 6.0684 11.2746 2.8596 8.3038
MHH-CALL-4 CTRP2 6.1047 11.1861 2.9304 7.9539
HDLM-2 CTRP2 6.1523 11.6483 2.738 8.6605
MOLP-2 CTRP2 6.2102 9.1041 4.0197 3.361
Karpas-422 CTRP2 6.2617 10.4887 3.3871 5.8384
Kasumi-2 CTRP2 6.3003 8.3728 4.4179 1.7156
RPMI-6666 CTRP2 6.3099 9.2296 4.0259 3.2029
A3/Kawakami CTRP2 6.4102 7.8211 4.7167 0.6122
JJN-3 CTRP2 6.4442 10.6143 3.454 5.2965
P3HR-1 CTRP2; CTRP1 6.5782 9.805 3.9276 3.2422
MOLT-3 CTRP2 6.6681 8.0551 4.7414 0.3969
OCI-Ly10 CTRP2; CTRP1 6.6819 15.2797 1.3426 13.2187
L-428 CTRP2 6.8699 9.9445 4.0408 2.4789
LP-1 CTRP2; CTRP1 6.9252 15.7014 1.3157 12.9164
Toledo CTRP2 7.2549 10.9884 3.7941 2.9646
L-1236 CTRP2 7.2852 9.5176 4.4414 0.8236
SUP-HD1 CTRP2 7.5662 12.4908 3.295 4.4599
⏷ Show the Full List of 150 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 4.7967 6.7403 4.0777 5.6085
TE8 CTRP2 4.8331 11.0743 1.9578 14.2779
TE-5 CTRP2 2.739 6.7142 1.9929 19.1516
OE21 CTRP2 3.0964 5.3964 2.8498 14.92
KYSE-410 CTRP2; CTRP1 3.1073 5.9171 2.6894 15.4813
TE-11 CTRP2 3.9295 5.708 3.6506 9.5184
OE33 CTRP2 3.9953 8.0578 2.6798 13.2033
KYSE-520 CTRP2 4.0313 6.8089 3.297 10.6257
KYSE-140 CTRP2; CTRP1 4.0801 7.7227 2.921 12.0219
TE-10 CTRP2 4.3555 8.7145 2.7028 12.2765
TE-4 CTRP2 4.5294 7.6885 3.3658 9.1531
KYSE-450 CTRP2; CTRP1 4.7005 6.8889 3.9154 6.4968
KYSE-150 CTRP2 4.9473 7.2353 3.9706 5.726
KYSE-30 CTRP2 5.0632 9 3.1909 8.7521
EC-GI-10 CTRP2 5.1257 8.2771 3.6053 6.8934
OE19 CTRP2 5.3605 7.1183 4.3778 3.2091
TE-6 CTRP2 5.3677 7.9631 3.9622 4.9361
TE-9 CTRP2 5.4492 11.5553 2.234 11.9539
TE-14 CTRP2 5.8074 8.6445 3.9612 4.1916
KYSE-70 CTRP2 5.8702 9.8889 3.3949 6.4288
COLO 680N CTRP2 5.9132 12.599 2.0836 11.7061
TE-1 CTRP2 6.1459 10.5973 3.2506 6.576
KYSE-180 CTRP2 6.2788 16.8428 0.2581 17.7011
KYSE-510 CTRP2 7.9677 16.1147 1.8488 9.3855
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 4.2299 7.5884 3.1299 10.8149
PK-45H CTRP2 3.5284 8.0259 2.2365 16.1214
Panc 03.27 CTRP2; CTRP1 3.8849 6.3287 3.3567 10.7709
KP-4 CTRP2 3.9543 6.2576 3.4591 10.186
HuP-T4 CTRP2; CTRP1 4.2029 7.5934 3.1015 10.9946
SU.86.86 CTRP2 4.2595 8.2545 2.8375 11.9418
AsPC-1 CTRP2 4.3115 8.1942 2.9156 11.5026
QGP-1 CTRP2; CTRP1 4.4632 8.2942 3.0083 10.778
PK-59 CTRP2 4.4822 9.8014 2.2824 13.7143
SNU-213 CTRP2 4.5609 8.3284 3.0812 10.2601
HPAC CTRP2; CTRP1 4.7024 7.6065 3.566 7.9387
Capan-2 CTRP2; CTRP1 4.7178 9.5289 2.6275 11.8
BxPC-3 CTRP2 4.7668 11.6015 1.6374 15.6734
Panc 08.13 CTRP2 4.7689 9.6314 2.6214 11.7179
Panc 04.03 CTRP2 4.7943 7.7982 3.5547 7.786
Panc 10.05 CTRP2; CTRP1 5.1585 8.6823 3.4304 7.5622
MIA PaCa-2 CTRP2 5.2789 6.5121 4.615 2.3634
DAN-G CTRP2 5.2912 8.811 3.4763 7.1151
Panc 02.03 CTRP2 5.359 8.1991 3.8374 8.224
Capan-1 CTRP2 5.5842 8.6899 3.7708 5.3512
PSN1 CTRP2 5.5934 7.459 4.3864 2.7801
PaTu 8988s CTRP2 5.6497 11.7314 2.3077 11.2845
KP-3 CTRP2; CTRP1 5.7549 10.2552 3.1255 7.7408
YAPC CTRP2 5.8621 9.6529 3.5054 5.985
KP-2 CTRP2 5.865 10.1456 3.2642 6.9785
SNU-410 CTRP2 5.9723 8.8446 3.9817 3.8541
Panc 05.04 CTRP2 6.1041 14.953 1.0617 15.2459
PaTu 8902 CTRP2; CTRP1 6.1109 9.5989 3.7131 4.7392
SUIT-2 CTRP2; CTRP1 6.2437 8.5422 4.3058 2.2007
TCC-Pan2 CTRP2 6.4339 11.1969 3.1647 6.4799
HuP-T3 CTRP2 6.5485 9.9 3.8641 3.5257
CFPAC-1 CTRP2; CTRP1 6.9306 10.2695 3.9292 2.8221
PaTu 8988t CTRP2 7.0025 11.7786 3.272 5.2475
L3.3 CTRP2 7.1248 12.9465 2.7972 6.942
Hs 766T CTRP2 7.3858 9.312 4.5659 0.4676
HPAF-II CTRP2 10.0965 23.3238 -0.1704 13.2743
SW1990 CTRP2 10.6739 31.4068 -3.6619 21.153
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 49 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 9.418 25.6727 -1.7624 18.5511
LOX-IMVI CTRP2 2.7934 5.1208 2.5964 16.7518
MDA-MB-435S CTRP2 3.2981 6.521 2.6616 15.0534
K029AX CTRP2 3.626 7.9443 2.3713 15.3428
Mel JuSo CTRP2 3.6526 6.5516 3.0205 12.704
COLO 792 CTRP2 3.7968 5.9359 3.4226 10.7569
WM793 CTRP2 4.0577 7.6389 2.9389 12.003
Mel Ho CTRP2 4.3739 8.3291 2.9083 11.3906
SK-MEL-3 CTRP2 4.3963 7.1181 3.5147 8.8495
COLO 741 CTRP1 4.5035 6.3195 3.9945 14.2654
HMCB CTRP2 4.5331 7.0571 3.6754 7.8697
IPC-298 CTRP2 4.5679 8.5608 2.9731 10.6925
WM983B CTRP2 4.6847 7.3364 3.6822 7.496
SK-MEL-5 CTRP2; CTRP1 4.7479 7.8481 3.4882 8.163
IGR-37 CTRP2 4.7819 8.314 3.2879 8.9246
WM266-4 CTRP2 4.8164 7.938 3.5052 7.9452
COLO 800 CTRP2 4.8762 9.4143 2.8233 10.6617
Hs 895.T CTRP2 5.0602 25.8207 -5.2208 32.2366
RVH-421 CTRP2 5.0902 8.4299 3.4988 7.4098
COLO 829 CTRP2 5.1746 8.4012 3.5844 6.8851
MeWo CTRP2 5.1979 7.8778 3.8656 5.6605
WT2-iPS CTRP2 5.5262 7.1854 4.4714 2.5374
CJM [Human melanoma] CTRP2 5.561 15.2051 0.5015 18.2231
WM88 CTRP2 5.6457 8.4826 3.9207 4.6227
UACC-257 CTRP2 5.6675 8.4631 3.9468 4.4778
SK-MEL-30 CTRP2 5.7415 11.042 2.7238 9.4227
UACC-62 CTRP2 5.8675 9.5463 3.562 5.7424
WM115 CTRP2 6.0152 9.4664 3.7094 4.9004
WM1799 CTRP2 6.0339 12.2831 2.334 10.4952
Hs 944.T CTRP2; CTRP1 6.0862 10.5128 3.2483 6.6806
Hs 936.T CTRP2; CTRP1 6.1282 9.4293 3.8075 4.3301
SK-MEL-28 CTRP2; CTRP1 6.1542 11.7356 2.6964 8.8267
HT-144 CTRP2 6.1643 9.7499 3.6774 4.8043
Hs 294T CTRP2 6.33 9.803 3.7661 4.2067
SK-MEL-1 CTRP2; CTRP1 6.4166 10.034 3.7139 4.2944
Hs 852.T CTRP2; CTRP1 6.54 8.3172 4.5743 0.9492
Hs 839.T CTRP2 6.6635 7.8018 4.835 0.202
IGR-39 CTRP2 6.7231 14.1912 1.9091 11.0169
G-361 CTRP2; CTRP1 6.7235 11.3023 3.3137 5.4613
SK-MEL-2 CTRP2 6.825 19.2004 -0.4895 19.0756
SK-MEL-31 CTRP2 6.8282 8.7424 4.5401 0.8399
Hs 940.T CTRP2 6.8321 8.6052 4.5978 0.6743
A2058 CTRP2 6.8647 8.2376 4.7547 0.2838
Hs 688(A).T CTRP2 6.8963 8.3169 4.7379 0.3053
RPMI-7951 CTRP2 6.9055 8.7061 4.5913 0.6478
A-375 CTRP2; CTRP1 6.9384 12.5323 2.8695 6.9208
SK-MEL-24 CTRP2 7.1999 13.2182 2.7178 7.1476
A101D CTRP2 7.4251 8.675 4.8094 0.0762
IGR-1 CTRP2 7.7942 16.4858 1.5529 10.7151
⏷ Show the Full List of 49 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 2.7239 8.4689 1.2265 22.0684
Cancer Drug Sensitivity Data Curated from 13 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Kelly CTRP2 3.4191 5.7584 3.0822 13.114
CHP-212 CTRP2 3.9364 6.3637 3.3955 10.4821
SK-N-BE(2) CTRP2 4.3557 10.4917 1.827 15.8116
CHP-126 CTRP2 5.2213 11.5991 2.0245 13.2325
SK-N-AS CTRP2 5.3231 7.9909 3.9122 5.2278
SK-N-FI CTRP2 5.4617 11.236 2.4038 11.2428
KP-N-SI9s CTRP2 5.471 10.7908 2.6336 10.2848
NH-6 CTRP2 5.7187 9.6053 3.4202 6.5796
IMR-32 CTRP2 5.7925 7.6787 4.4205 2.3413
SK-N-DZ CTRP2 5.9798 7.6152 4.5719 1.5045
SK-N-SH CTRP2 6.3599 11.4675 2.9797 7.3434
KP-N-YN CTRP2 6.3842 11.3144 3.072 6.9313
NB1 CTRP2 6.5146 12.2941 2.6872 8.2828
⏷ Show the Full List of 13 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 3.4189 10.5337 0.9395 21.3347
SNU-478 CTRP2 3.7333 7.37 2.7423 13.5943
SNU-869 CTRP2 4.7373 10.0141 2.4032 12.6795
SNU-1196 CTRP2 5.2688 8.3505 3.6881 6.2693
HuH-28 CTRP2 5.3903 8.8752 3.525 6.7258
SNU-308 CTRP2 5.4828 8.4215 3.8252 5.3021
HuCC-T1 CTRP2 6.2776 9.5814 3.8368 3.997
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 16 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RD-ES CTRP2 0.177 42.5259 -17.7925 46.8195
MHH-ES-1 CTRP2 3.1404 7.2176 2.2046 17.2474
SJSA-1 CTRP2 3.7823 7.676 2.6506 13.8386
SK-ES-1 CTRP2 3.8744 7.7133 2.7242 13.316
SK-N-MC CTRP2 3.8919 6.1552 3.4361 10.4436
TC71 CTRP2 4.6753 6.6273 4.0178 6.1338
HOS CTRP2 5.2306 6.1477 4.7578 1.8545
A-673 CTRP2 5.7914 10.7616 2.9022 8.6005
SaOS-2 CTRP2 5.8697 10.6389 3.0234 7.9657
CAL-78 CTRP2 5.9067 8.7686 3.9722 3.992
Hs 888.T CTRP2 6.2852 11.6213 2.8499 7.9891
Hs 822.T CTRP2 6.3978 7.3974 4.8777 0.2142
SW1353 CTRP2 6.4828 14.1952 1.7286 12.1047
G-292 clone A141B1 CTRP2 6.8938 9.4593 4.2697 1.6471
U2OS CTRP2; CTRP1 8.2157 10.4191 4.4897 0.3247
MG-63 CTRP2 11.9282 23.4474 0.8942 7.9954
⏷ Show the Full List of 16 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 72 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HCC1954 CTRP2 2.3663 8.7912 0.7193 24.8461
HMC-1-8 CTRP2 2.6704 4.6524 2.5683 17.2336
HCC1569 CTRP2 2.7044 8.5105 1.1881 22.2612
DU4475 CTRP2 3.3739 7.714 2.2242 16.5611
BT-549 CTRP2 3.7192 7.1946 2.8076 13.3699
MDA-MB-157 CTRP2 3.8834 21.2933 -3.9626 32.5203
HCC1428 CTRP2 4.2569 6.8047 3.5251 9.1451
ZR-75-1 CTRP2 4.3972 7.7469 3.2134 10.0824
HCC1806 CTRP2 4.4066 8.1033 3.049 10.7376
HCC1500 CTRP2 4.7659 8.6578 3.103 9.7283
AU565 CTRP2 5.0172 9.3987 2.9526 9.8382
CAL-85-1 CTRP2 5.2692 7.947 3.8902 5.4212
MDA-MB-231 CTRP2 5.2809 14.2058 0.7707 17.8393
HCC1419 CTRP2 5.3553 10.3967 2.7363 10.0784
KPL-1 CTRP2 5.4635 8.3496 3.8457 5.2506
BT-20 CTRP2 5.472 9.0504 3.5032 6.6682
HCC38 CTRP2 5.6767 9.4178 3.4809 6.3996
MDA-MB-453 CTRP2 5.6973 9.3425 3.5341 6.1426
HCC1143 CTRP2 5.7367 11.3888 2.5474 10.1535
HCC202 CTRP2 5.7581 13.9233 1.3009 15.0021
ZR-75-30 CTRP2 5.7968 9.9908 3.2889 6.9914
SK-BR-3 CTRP2 5.9937 11.2715 2.8047 8.6539
MDA-MB-361 CTRP2 6.1083 10.5768 3.2331 6.7075
HDQ-P1 CTRP2 6.1182 12.0152 2.5311 9.5568
BT-474 CTRP2 6.2634 9.2582 3.9817 3.4394
CAL-148 CTRP2 6.3337 11.9806 2.709 8.482
MDA-MB-415 CTRP2 6.4001 14.6927 1.4199 13.4103
MCF-7 CTRP2; CTRP1 6.4668 11.1144 3.2279 6.1751
HCC1937 CTRP2 6.6479 13.3794 2.2524 9.8011
CAMA-1 CTRP2 6.6511 10.0543 3.8572 3.423
Hs 578Bst CTRP2 6.7098 13.9124 2.0362 10.5472
CAL-120 CTRP2 6.7885 8.2032 4.736 0.3536
CAL-51 CTRP2 6.8119 11.06 3.4876 4.6551
T-47D CTRP2 6.9079 12.5692 2.8308 7.1177
JIMT-1 CTRP2 7.1368 13.0227 2.7689 7.0361
MDA-MB-468 CTRP2 7.2154 11.6319 3.4762 4.1916
Hs 578T CTRP2 7.3635 11.1464 3.7858 2.8809
HCC1395 CTRP2 8.2027 19.7392 0.2628 14.5402
BT 271 CTRP2 4.9594 5.9756 4.6022 3.0744
BT 172 CTRP2 5.0026 5.9298 4.6651 2.7164
BT 145 CTRP2 5.0415 7.3883 3.9771 5.5037
BT 330 CTRP2 5.1443 6.3655 4.5763 2.7848
BT 416 CTRP2 5.1591 6.1104 4.7164 2.1679
BT147 CTRP2 5.1788 6.5236 4.5266 2.9244
BT164 CTRP2 5.2 5.8856 4.8634 1.4702
BT 112 CTRP2 5.2287 6.1578 4.7512 1.8857
BT 179 CTRP2 5.3164 6.365 4.7182 1.864
BT 504 CTRP2 5.3438 6.2676 4.7878 1.5266
BT 245 CTRP2 5.482 7.0597 4.5005 2.489
BT 286 CTRP2 5.6258 6.9818 4.6417 1.6895
BT 340 CTRP2 5.6391 6.9903 4.6467 1.6505
BT 328 CTRP2 5.6694 7.1175 4.6062 1.7703
BT 359 CTRP2 5.6706 7.109 4.6111 1.7488
BT 232 CTRP2 5.6757 7.4579 4.4461 2.4083
BT 440 CTRP2 5.7792 7.7749 4.3649 2.5846
BT 482 CTRP2 5.7928 7.7849 4.3695 2.5464
BT 320 CTRP2 5.8087 8.7253 3.9225 4.3487
BT 422 CTRP2 5.8138 7.5735 4.4853 2.0523
BT 248 CTRP2 5.8289 9.7556 3.4298 6.3533
BT 131 CTRP2 5.8343 7.4292 4.5671 1.7022
BT 216 CTRP2 5.847 7.449 4.566 1.6901
BT 428 CTRP2 5.9576 7.4656 4.6271 1.3227
BT 333 CTRP2 6.0181 7.6911 4.5603 1.5036
BT 224 CTRP2 6.2824 8.9308 4.1489 2.7575
BT 159 CTRP2 6.4074 9.6067 3.9111 3.5253
BT 498 CTRP2 6.5252 7.633 4.8418 0.2379
BT 139 CTRP2 6.9227 11.865 3.1784 5.7223
BT 444 CTRP2 7.0724 8.2418 4.8326 0.1053
BT 239 CTRP2 7.3218 8.6233 4.7906 0.1098
BT 231 CTRP2 7.5472 14.4387 2.3676 8.0184
BT 228 CTRP2 7.7063 14.7411 2.3294 7.9461
BT 187 CTRP2 7.7345 11.2128 3.9592 1.9446
⏷ Show the Full List of 72 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 4.287 8.1412 2.9183 11.5476
Cancer Drug Sensitivity Data Curated from 46 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
AM-38 CTRP2 -11.1105 10.0674 -14.1297 70.5159
SF539 CTRP2 2.5637 4.608 2.4612 17.9444
D283 Med CTRP2 3.9204 6.5558 3.2961 10.9149
SF268 CTRP2 4.3961 8.4493 2.8702 11.4976
Becker CTRP2 4.8953 7.8344 3.6268 7.2713
DK-MG CTRP2 5.136 9.8874 2.809 10.1999
ONS-76 CTRP2 5.2433 7.6888 3.9978 5.0188
SF295 CTRP2; CTRP1 5.3414 9.152 3.347 7.562
U-87MG ATCC CTRP2 5.723 10.3358 3.0607 8.0648
SW1783 CTRP2 5.7818 11.3848 2.5849 9.9202
42-MG-BA CTRP2 5.8032 9.4906 3.5413 5.9339
Hs 683 CTRP2 5.8038 7.9733 4.2861 2.8679
SF126 CTRP2 5.9537 9.4313 3.6821 5.1085
YKG-1 CTRP2 6.2382 8.3526 4.39 1.8887
SW1088 CTRP2 6.239 11.6103 2.8213 8.1798
KNS-81 CTRP2 6.2895 7.4966 4.7915 0.4788
SNU-489 CTRP2 6.3006 10.6221 3.3497 5.9311
U-118MG CTRP2 6.3127 7.9071 4.6312 0.9543
CCF-STTG1 CTRP2 6.3738 10.0387 3.6828 4.4785
LN-229 CTRP2; CTRP1 6.4342 8.6972 4.3496 1.8206
KNS-60 CTRP2 6.4397 7.7596 4.7555 0.4847
KALS-1 CTRP2 6.4546 10.2622 3.6303 4.5749
NMC-G1 CTRP2 6.4738 7.6712 4.8056 0.3397
TM-31 CTRP2 6.501 9.4089 4.0636 2.8145
Daoy CTRP2 6.552 9.9696 3.8336 3.6402
DBTRG-05MG CTRP2 6.5526 11.4255 3.1372 6.4134
SNU-626 CTRP2 6.5784 8.3905 4.5629 0.9548
SNU-738 CTRP2 6.6149 12.4153 2.7001 8.0753
CAS-1 CTRP2 6.6624 7.942 4.7822 0.307
LN-18 CTRP2 6.677 7.9716 4.7771 0.3119
GaMG CTRP2; CTRP1 6.7225 9.2257 4.278 1.7809
GB-1 CTRP2 6.8902 12.1138 3.0376 6.3237
8-MG-BA CTRP2 6.9028 12.5266 2.8479 7.0574
SNB-75 CTRP2 6.9075 17.0239 0.6508 15.2966
SNU-1105 CTRP2 6.9551 13.71 2.3115 9.0928
U-251MG CTRP2 7.3639 12.6593 3.0905 5.4829
A-172 CTRP2 7.6769 13.6483 2.8264 6.0956
KNS-42 CTRP2 8.0896 15.3893 2.273 7.6504
KG-1-C CTRP2 8.1343 14.8506 2.5537 6.5503
SNU-466 CTRP2 8.1558 18.3044 0.9251 12.4107
M059K CTRP2 9.2637 19.0241 1.3178 9.5709
T98G CTRP2 9.8031 18.0578 2.0895 6.3131
SNU-201 CTRP2 10.4874 24.8478 -0.6363 14.128
GMS-10 CTRP2 10.8047 21.9958 0.8938 9.16
GOS-3 CTRP2 10.9635 21.3568 1.2773 7.7772
YH-13 CTRP2 11.4424 24.2855 0.2295 10.4914
⏷ Show the Full List of 46 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-2 CTRP2; CTRP1 3.281 6.9305 2.4732 15.8293
RL95-2 CTRP2 3.8573 7.8888 2.6253 13.7561
HEC-151 CTRP2; CTRP1 4.2242 6.984 3.4096 9.6918
JHUEM-7 CTRP2 4.3512 7.3619 3.3549 9.6091
HEC-1-A CTRP2 4.367 9.1093 2.5196 13.0011
ESS-1 CTRP2 4.7854 8.6997 3.0994 9.7022
JHUEM-3 CTRP2 4.8264 7.4638 3.7491 6.9074
MFE-319 CTRP2; CTRP1 5.0367 9.4171 2.96 9.7687
KLE CTRP2; CTRP1 5.115 7.9899 3.7397 6.3508
JHUEM-1 CTRP2 5.2785 9.2589 3.2419 8.1201
AN3-CA CTRP2 5.4244 10.9498 2.5164 10.853
HEC-108 CTRP2; CTRP1 5.587 9.1578 3.5404 6.3075
HEC-265 CTRP2; CTRP1 5.6039 7.2774 4.4829 2.3672
HEC-50B CTRP2 5.6158 8.3477 3.9648 4.4897
HEC-6 CTRP2; CTRP1 5.7952 10.3194 3.1247 7.6747
EFE-184 CTRP2 5.8338 9.0108 3.8007 4.8111
HEC-251 CTRP2; CTRP1 6.3017 10.096 3.6057 4.8919
HEC-59 CTRP2; CTRP1 6.9953 10.6074 3.8136 3.1784
MFE-296 CTRP2 7.2398 13.5169 2.6017 7.5443
EN CTRP2 7.5518 12.8008 3.1429 5.0493
HEC-1-B CTRP2 7.5641 9.4421 4.5902 0.3506
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 6.181 9.6901 3.7181 4.6144
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
786-O CTRP2 4.3649 7.6677 3.2211 10.1254
UO-31 CTRP2 4.8393 8.8313 3.0815 9.6639
CAL-54 CTRP2 5.081 8.5368 3.4376 7.6846
769-P CTRP2 5.0957 9.1351 3.1511 8.8542
TUHR10TKB CTRP2 5.3965 15.0709 0.4337 18.7717
OS-RC-2 CTRP2 5.5198 9.2325 3.4503 6.8028
VMRC-RCZ CTRP2 5.7786 7.3587 4.5641 1.7875
Caki-1 CTRP2 6.0964 13.1405 1.9567 11.8834
KMRC-20 CTRP2 6.1108 9.9404 3.5466 5.419
KMRC-2 CTRP2 6.1259 10.4929 3.2871 6.4578
SNU-1272 CTRP2 6.3834 8.6646 4.3345 1.9313
RCC10RGB CTRP2; CTRP1 6.4401 8.6133 4.3908 1.6654
KMRC-1 CTRP2 6.59 12.6203 2.5821 8.5852
TUHR4TKB CTRP2 6.5958 8.5038 4.5238 1.0653
VMRC-RCW CTRP2; CTRP1 6.705 11.2849 3.3096 5.5036
TUHR14TKB CTRP2 6.772 17.6723 0.2275 16.9371
A-498 CTRP2 6.9442 8.3131 4.7587 0.2482
ACHN CTRP2 6.9708 13.0154 2.659 7.7053
BFTC-909 CTRP2 7.013 8.597 4.6808 0.3775
KMRC-3 CTRP2 7.8855 9.7033 4.6199 0.2125
Caki-2 CTRP2 8.5734 16.5306 2.0465 7.8678
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 52 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KM12 CTRP2; CTRP1 3.1434 5.5257 2.861 14.7392
SW1417 CTRP2 3.1912 7.6468 2.0689 17.6409
SNU-175 CTRP1 3.2951 5.3825 3.0706 28.9821
SW48 CTRP2; CTRP1 3.6092 7.465 2.5743 14.5771
COLO201 CTRP2 3.618 5.6802 3.3246 11.6348
SW620 CTRP2; CTRP1 3.7389 7.4564 2.7086 13.7148
NCI-H747 CTRP2 3.9314 7.4183 2.9179 12.396
SW403 CTRP1 4.1376 7.2894 3.1816 22.9315
NCI-H508 CTRP2; CTRP1 4.256 8.758 2.5892 12.9658
HT-55 CTRP2; CTRP1 4.3118 7.5585 3.223 10.2412
SNU-C5 CTRP2; CTRP1 4.3457 7.4766 3.2947 9.8685
SNU-81 CTRP1 4.376 6.6151 3.7312 17.194
SNU-61 CTRP2; CTRP1 4.4233 6.7021 3.7375 7.8785
SNU-1040 CTRP1 4.4283 6.2145 3.9664 14.9154
COLO 678 CTRP2; CTRP1 4.4369 8.6694 2.7999 11.6959
SNU-C2A CTRP2; CTRP1 4.5792 10.4528 2.0456 14.4597
SNU-407 CTRP2 4.5972 7.6827 3.4317 8.7283
SNU-C1 CTRP2 4.6101 6.4974 4.0167 6.2928
COLO205 CTRP2; CTRP1 4.6239 7.0942 3.7435 7.38
GP2d CTRP2; CTRP1 4.7827 6.3321 4.2622 4.8808
RKO CTRP2; CTRP1 4.8982 6.8799 4.1025 5.2812
LS513 CTRP2; CTRP1 5.0755 8.8863 3.2583 8.446
LS411N CTRP2; CTRP1 5.0832 6.5015 4.4554 3.4156
SW948 CTRP2; CTRP1 5.1196 6.6142 4.4309 3.4439
HT115 CTRP2; CTRP1 5.1693 9.2389 3.1612 8.6674
HCT 116 CTRP2; CTRP1 5.1953 8.9358 3.3345 7.8925
RCM-1 [Human ESC] CTRP2; CTRP1 5.2489 8.9357 3.3791 7.6024
HCC-56 CTRP2 5.2497 5.9964 4.849 1.4366
LS1034 CTRP2 5.2585 6.4432 4.633 2.3256
COLO 320 CTRP2; CTRP1 5.2597 7.9389 3.8864 5.455
LoVo CTRP2; CTRP1 5.2684 11.865 1.9307 13.513
HCT 15 CTRP2 5.2694 6.2347 4.7458 1.8328
C2BBe1 CTRP2; CTRP1 5.4348 7.0057 4.4915 2.6052
SK-CO-1 CTRP2; CTRP1 5.4541 7.6164 4.2033 3.7729
SNU-C4 CTRP2; CTRP1 5.5105 7.4354 4.3363 3.1227
DLD-1 CTRP2; CTRP1 5.5249 6.8867 4.617 1.9402
SNU-503 CTRP2 5.6011 9.6525 3.3053 7.263
CL-40 CTRP1 5.6521 8.253 4.039 8.8214
HT-29 CTRP2; CTRP1 5.6671 11.2099 2.5816 10.1392
SW1116 CTRP2 5.716 10.6653 2.8913 8.7781
LS123 CTRP2; CTRP1 5.8212 10.0624 3.272 7.02
CCK-81 CTRP2 5.8361 9.0731 3.7718 4.9265
OUMS-23 CTRP2 5.8406 7.0236 4.7587 0.9661
NCI-H716 CTRP2 5.8487 10.7944 2.9302 8.3859
CW-2 CTRP2; CTRP1 5.9026 8.0781 4.3036 2.6546
SW480 CTRP1 6.0222 11.3556 2.7846 17.3539
MDST8 CTRP2; CTRP1 6.2198 9.5703 3.8028 4.2158
CL-11 CTRP2 6.2699 8.6962 4.2507 2.3799
HCT 8 CTRP2; CTRP1 6.397 9.5411 3.9354 3.4436
SNU-1033 CTRP2 6.5861 12.1398 2.8138 7.6635
LS180 CTRP2; CTRP1 6.6846 13.6596 2.1418 10.1763
CL-34 CTRP1 7.0383 14.8744 1.8034 19.7934
⏷ Show the Full List of 52 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 20 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHH-5 CTRP2 3.7472 6.5203 3.1322 12.0151
SNU-398 CTRP2; CTRP1 4.2797 7.4307 3.2532 10.1935
Hep 3B2.1-7 CTRP2 4.4003 7.1485 3.5041 8.8831
SNU-878 CTRP2 4.4426 5.6402 4.2253 5.8934
PLC/PRF/5 CTRP2 4.6604 7.5681 3.5462 8.1135
Hep-G2 CTRP2; CTRP1 4.7334 7.9951 3.4024 8.5513
SNU-182 CTRP2 4.8344 12.1892 1.4023 16.4341
Li-7 CTRP2 5.0789 6.3894 4.5074 3.2069
SNU-761 CTRP2 5.1167 7.6778 3.8972 5.6871
SNU-423 CTRP2 5.2104 8.6873 3.4713 7.29
JHH-1 CTRP2 5.3594 6.3203 4.7735 2.3441
HLF CTRP2 5.4725 8.9019 3.5776 6.3559
HuH-1 CTRP2 5.6509 7.5542 4.3815 2.7101
SNU-387 CTRP2 5.6924 11.812 2.3015 11.2313
SNU-449 CTRP2; CTRP1 6.0336 10.0292 3.4472 5.9476
JHH-6 CTRP2; CTRP1 6.6049 7.6198 4.8781 0.1463
SNU-886 CTRP2 6.7633 8.6919 3.5389 0.3185
JHH-2 CTRP2 7.187 14.1254 2.2726 8.8975
SK-HEP-1 CTRP2 7.5944 11.7477 3.6489 3.1328
JHH-4 CTRP2 7.8083 10.2659 4.3807 0.695
⏷ Show the Full List of 20 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 160 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H146 CTRP2 -0.5052 11.6568 -3.4822 42.9501
NCI-H3255 CTRP1 1.2744 3.6844 1.2153 55.7125
NCI-H82 CTRP1 2.0797 3.5981 2.0649 44.7787
HCC2935 CTRP2; CTRP1 2.1645 5.5729 1.7804 21.6001
HCC827 CTRP2; CTRP1 2.2161 4.8717 2.0283 20.5539
HCC44 CTRP2; CTRP1 2.4477 5.2383 2.1876 19.2739
NCI-H596 CTRP1 2.5057 5.9252 2.0364 40.8651
PC-14 CTRP2 2.6305 4.366 2.5724 17.3466
NCI-H1048 CTRP1 2.7476 5.7879 2.3451 37.5204
NCI-H1703 CTRP2 2.8387 6.3172 2.2534 17.8869
NCI-H520 CTRP2 2.8771 5.8781 2.4546 17.0223
NCI-H1734 CTRP2 2.9902 8.0396 1.6892 19.6301
NCI-H1666 CTRP2; CTRP1 3.0317 7.0903 2.1461 17.7643
COR-L51 CTRP2; CTRP1 3.2138 9.1218 1.4151 20.0943
NCI-H838 CTRP2 3.3013 5.5803 3.0151 13.7061
EPLC-272H CTRP2; CTRP1 3.3294 7.5566 2.2498 16.5753
NCI-H1568 CTRP2; CTRP1 3.5635 7.2346 2.6316 14.4672
NCI-H2171 CTRP2 3.5987 6.5972 2.9451 13.1421
NCI-H358 CTRP2; CTRP1 3.6451 5.9956 3.2378 11.8851
NCI-H1373 CTRP2; CTRP1 3.654 6.6894 2.9633 12.924
NCI-H1975 CTRP2; CTRP1 3.6587 7.0484 2.8114 13.5099
RERF-LC-MS CTRP2 3.6819 5.3729 3.4951 10.817
SW1271 CTRP2 3.7041 8.0521 2.3982 15.0422
NCI-H23 CTRP2; CTRP1 3.7107 6.6111 3.0557 12.4117
NCI-H2085 CTRP2 3.8325 7.7121 2.6835 13.5828
RERF-LC-Ad2 CTRP2 3.8481 7.9253 2.599 13.8844
Lu-65 CTRP2; CTRP1 3.8568 8.1659 2.4941 14.2856
NCI-H1623 CTRP2 3.8718 6.2109 3.3921 10.6687
NCI-H1437 CTRP1 3.9073 5.9165 3.5479 21.394
HOP-92 CTRP2 3.9414 11.2618 1.0709 19.6196
EBC-1 CTRP2; CTRP1 3.9688 7.6446 2.8493 12.5811
NCI-H2291 CTRP2 4.0718 9.0482 2.2755 14.6596
NCI-H1341 CTRP2 4.0951 7.4409 3.0687 11.3864
LCLC-97TM1 CTRP2; CTRP1 4.1103 7.414 3.0963 11.2377
COR-L23 CTRP1 4.1454 5.8521 3.8262 17.7074
HCC78 CTRP2; CTRP1 4.1832 7.2181 3.2598 10.3982
NCI-H1944 CTRP2; CTRP1 4.1862 6.3895 3.6419 8.8568
NCI-H2110 CTRP2; CTRP1 4.1884 8.742 2.5338 13.3459
NCI-H2009 CTRP2; CTRP1 4.1967 8.4152 2.7004 12.6471
NCI-H526 CTRP2 4.2559 9.9249 2.0165 15.2816
SW1573 CTRP2 4.2687 8.665 2.6463 12.7035
NCI-H2073 CTRP1 4.2721 5.8298 3.9691 15.7825
NCI-H441 CTRP2; CTRP1 4.2823 8.8294 2.5787 12.9492
HCC4006 CTRP2; CTRP1 4.2863 6.1181 3.8634 7.7216
NCI-H1573 CTRP2; CTRP1 4.2984 7.706 3.1393 10.6151
NCI-H1838 CTRP2 4.3051 7.863 3.0701 10.8833
NCI-H2087 CTRP2 4.3332 8.1306 2.967 11.2418
COR-L105 CTRP2 4.335 6.6748 3.6628 8.3971
NCI-H1793 CTRP2; CTRP1 4.3558 8.2886 2.9112 11.4196
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 4.3762 8.0146 3.0637 10.7459
LXF 289 CTRP2; CTRP1 4.3936 7.8926 3.1393 10.3953
Lu-99 CTRP2; CTRP1 4.4081 7.2541 3.4612 9.0403
NCI-H1792 CTRP2; CTRP1 4.4243 7.3887 3.4121 9.2035
EKVX CTRP2 4.4323 22.1255 -3.9046 31.3482
NCI-H292 CTRP2 4.4532 8.8286 2.7366 11.9205
RERF-LC-A1 CTRP2 4.4584 8.3498 2.9765 10.9198
NCI-H1355 CTRP2; CTRP1 4.4807 7.4885 3.4173 9.0515
Calu-6 CTRP2; CTRP1 4.4953 7.4345 3.4573 8.8535
NCI-H647 CTRP2 4.5063 8.407 2.9926 10.7471
NCI-H1693 CTRP2 4.5475 7.1327 3.6526 7.9301
HCC15 CTRP2; CTRP1 4.5831 7.6808 3.4196 8.81
NCI-H2170 CTRP2 4.5831 7.1358 3.6849 7.715
NCI-H1930 CTRP1 4.5878 6.7327 3.8833 14.7813
NCI-H661 CTRP2; CTRP1 4.5917 7.8076 3.3655 9.0148
NCI-H727 CTRP2; CTRP1 4.5974 8.4666 3.0464 10.3247
NCI-H1339 CTRP2 4.5988 5.3602 4.4965 4.4261
NCI-H1435 CTRP2; CTRP1 4.6254 8.4431 3.0834 10.1103
RERF-LC-KJ CTRP1 4.6448 7.2892 3.6683 16.337
SK-MES-1 CTRP2 4.7032 6.813 3.9547 6.3283
LUDLU-1 CTRP2 4.7203 6.3798 4.1794 5.3665
NCI-H1650 CTRP2 4.7262 8.168 3.3104 8.9497
HCC95 CTRP2 4.7452 8.0149 3.4032 8.5224
NCI-H2122 CTRP2; CTRP1 4.7497 7.1966 3.8108 6.8186
MOR/CPR CTRP2 4.7516 5.6538 4.5445 3.819
NCI-H1869 CTRP2 4.7547 8.344 3.2488 9.1451
NCI-H1755 CTRP2; CTRP1 4.7902 8.1841 3.3597 8.6075
NCI-H1963 CTRP1 4.8037 14.6575 0.1432 34.1171
NCI-H2405 CTRP2; CTRP1 4.829 9.5989 2.6901 11.3098
NCI-H322 CTRP2 4.8326 6.8239 4.0701 5.5595
HCC366 CTRP2 4.8391 9.3808 2.8077 10.8025
ChaGo-K-1 CTRP2; CTRP1 4.8472 8.4078 3.2992 8.7397
Sq-1 CTRP2; CTRP1 4.8699 7.8174 3.6127 7.3834
COLO 699 CTRP2; CTRP1 4.8796 11.5324 1.769 14.9273
NCI-H810 CTRP2; CTRP1 4.8851 7.7843 3.6426 7.2266
LK2 CTRP2 4.9057 5.4766 4.7801 2.4876
NCI-H2286 CTRP2; CTRP1 4.9173 7.8924 3.6173 7.265
HCC33 CTRP1 4.9231 7.5946 3.7706 14.1345
NCI-H522 CTRP2; CTRP1 4.931 8.2987 3.4271 8.0316
LOU-NH91 CTRP2 4.9397 8.499 3.3348 8.4
NCI-H2444 CTRP2 4.9969 8.0399 3.6134 7.1175
CAL-12T CTRP2; CTRP1 4.9977 8.2968 3.486 7.6493
HCC1195 CTRP2; CTRP1 5.0006 9.1657 3.0547 9.4464
COR-L279 CTRP1 5.0151 8.7349 3.2823 17.7603
A-549 CTRP2; CTRP1 5.0164 7.2143 4.0419 5.2839
COR-L88 CTRP2; CTRP1 5.0325 9.5498 2.8901 10.0678
NCI-H1299 CTRP2; CTRP1 5.0499 8.221 3.5688 7.1971
T3M-10 CTRP2; CTRP1 5.0862 8.3532 3.5338 7.2712
SCLC-21H CTRP1 5.1246 11.5531 1.9667 25.8232
Calu-3 CTRP2; CTRP1 5.1689 8.5535 3.5035 7.2357
NCI-H1395 CTRP2 5.1715 11.9212 1.8219 14.1323
VMRC-LCD CTRP2; CTRP1 5.2122 7.5803 4.0264 4.9585
NCI-H446 CTRP2 5.2442 8.1507 3.7677 5.9825
DMS 273 CTRP2; CTRP1 5.2746 6.7882 4.4737 2.9637
DMS 454 CTRP2 5.2998 7.8454 3.966 5.0457
DMS 53 CTRP2 5.3101 8.7064 3.5442 6.7948
NCI-H2030 CTRP2; CTRP1 5.3104 9.504 3.1457 8.4617
LC-1/sq-SF CTRP2; CTRP1 5.3297 8.5569 3.6348 6.3781
NCI-H841 CTRP2; CTRP1 5.3359 9.4471 3.1951 8.2074
NCI-H1155 CTRP2 5.3534 8.5087 3.6782 6.1522
HCC1359 CTRP1 5.3631 6.9069 4.4851 5.9192
NCI-H2342 CTRP2; CTRP1 5.4709 9.7317 3.1624 8.0934
NCI-H211 CTRP2 5.4974 11.9265 2.0878 12.4501
HCC1588 CTRP2 5.5029 9.956 3.0761 8.3944
COLO 668 CTRP2; CTRP1 5.536 8.332 3.9113 4.8491
DV-90 CTRP2; CTRP1 5.5448 10.0601 3.0576 8.395
IA-LM CTRP2 5.5659 8.0121 4.093 4.0409
NCI-H1581 CTRP2 5.5837 9.8133 3.2115 7.6845
HCC2108 CTRP2; CTRP1 5.5869 11.4015 2.4221 10.9355
NCI-H889 CTRP2 5.5992 9.6998 3.2803 7.3707
NCI-H2029 CTRP2; CTRP1 5.6098 7.4745 4.3908 2.7362
NCI-H69 CTRP2 5.6428 10.6864 2.8232 9.1894
NCI-H1836 CTRP1 5.6603 8.6008 3.8733 10.2281
NCI-H1092 CTRP2 5.6742 15.6594 0.3666 18.4601
NCI-H1105 CTRP2; CTRP1 5.6744 9.878 3.2504 7.3626
RERF-LC-Ad1 CTRP2 5.7619 9.4304 3.5398 6.0096
HCC1438 CTRP2 5.7736 11.2204 2.6602 9.6267
DMS 79 CTRP2 5.7929 9.9033 3.3293 6.8307
COR-L95 CTRP2 5.8267 7.3194 4.6138 1.53
SHP-77 CTRP2; CTRP1 5.8814 11.0565 2.8253 8.7614
SBC-5 CTRP2 5.8916 7.4946 4.573 1.6066
NCI-H1651 CTRP2 5.9171 10.6655 3.0464 7.7904
NCI-H650 CTRP2; CTRP1 5.9295 11.8293 2.4788 10.0921
NCI-H2126 CTRP2; CTRP1 5.9441 8.4921 4.1328 3.2829
NCI-H1915 CTRP2; CTRP1 6.0099 9.3051 3.7843 4.602
NCI-H226 CTRP2 6.023 9.8662 3.5194 5.6677
NCI-H2196 CTRP2 6.0276 7.431 4.6837 1.0412
NCI-H1563 CTRP2 6.0551 9.933 3.51 5.6555
NCI-H2081 CTRP2; CTRP1 6.1708 14.4415 1.3681 14.003
NCI-H196 CTRP2 6.2147 9.5426 3.8126 4.1834
HCC2279 CTRP2 6.2937 14.3411 1.5128 13.2461
NCI-H1184 CTRP2 6.33 10.5764 3.3928 5.7121
NCI-H1781 CTRP1 6.3459 15.5915 0.9324 25.9759
NCI-H2106 CTRP2 6.3554 13.5826 1.9353 11.5222
BEN CTRP2; CTRP1 6.4117 7.6699 4.7785 0.4401
HOP-62 CTRP2 6.4509 10.5245 3.5019 5.0945
NCI-H460 CTRP2; CTRP1 6.5068 10.8751 3.3713 5.5385
KNS-62 CTRP2; CTRP1 6.5451 10.0301 3.8007 3.778
NCI-H2228 CTRP2 6.7225 12.3588 2.8038 7.4975
SK-LU-1 CTRP2; CTRP1 6.9265 12.7855 2.7393 7.4526
NCI-H1876 CTRP1 6.9509 11.8627 3.1982 11.4267
NCI-H1694 CTRP2; CTRP1 7.1063 16.8181 0.9001 14.1079
NCI-H2141 CTRP2; CTRP1 7.1409 15.2176 1.7094 11.115
LCLC-103H CTRP2; CTRP1 7.2221 12.1573 3.2355 5.1049
DMS 114 CTRP2 7.4291 12.2003 3.3451 4.4328
HCC1171 CTRP2 7.4437 15.7028 1.688 10.7342
HCC1833 CTRP2; CTRP1 7.6096 15.9432 1.6873 10.4912
Calu-1 CTRP2 7.9557 16.5078 1.6527 10.1208
NCI-H2023 CTRP2; CTRP1 8.2738 14.2155 2.9314 4.9976
NCI-H2172 CTRP2; CTRP1 9.2188 17.032 2.211 6.5226
Hs 888.Lu CTRP2 6.6712 11.5611 3.1538 6.1731
⏷ Show the Full List of 160 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 4.7634 7.2355 3.8043 6.8151
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 5.499 9.465 3.3179 7.3934
P-STS CTRP2 6.2039 10.3285 3.4239 5.7768
SYO-1 CTRP2 6.2481 8.437 4.3572 2.0004
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 5.9254 11.2735 2.7514 8.9884
Aska-SS CTRP2 6.7162 8.582 4.5518 0.8846
Rh41 CTRP2 3.3006 7.415 2.2833 16.5188
GCT CTRP2 3.715 6.3136 3.1851 11.8957
G-402 CTRP2 3.8556 8.4602 2.3531 14.8555
TTC-709 CTRP2 4.0723 8.3132 2.6315 13.2172
HT-1080 CTRP2; CTRP1 4.1111 7.4045 3.1015 11.2149
TE 617.T CTRP2 4.2899 6.7918 3.5639 8.9072
MES-SA CTRP2 5.0522 6.1761 4.5896 2.9206
SK-LMS-1 CTRP2 5.0853 8.6944 3.3625 7.9904
KYM-1 CTRP2 5.2127 8.9317 3.3511 7.7893
Rh18 CTRP2 5.3 7.5061 4.1357 4.3338
A-204 CTRP2 5.4766 10.4793 2.7937 9.6145
G-401 CTRP2; CTRP1 5.7838 10.5921 2.9806 8.2904
BT-12 CTRP2 5.8343 7.6605 4.4574 2.1352
Hs 729.T CTRP2 6.1163 9.059 3.978 3.6588
RKN CTRP2; CTRP1 6.2434 10.5376 3.3502 6.0163
TE 441.T CTRP2 6.4255 8.4768 4.4433 1.493
SW982 CTRP2 6.7731 7.9613 4.8198 0.1942
BT-16 CTRP2 6.8068 8.2982 4.7075 0.4098
Tm87-16 CTRP2 7.4992 9.0235 4.7159 0.167
RD CTRP2 8.7552 19.3348 0.8385 11.8598
SK-UT-1 CTRP2 11.3311 22.4973 0.977 8.3404
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 6.437 11.5562 2.9919 7.1746
TYK-nu CTRP2; CTRP1 3.1435 7.2622 2.1886 17.3012
A2780 CTRP2; CTRP1 3.8322 6.3165 3.3068 11.1068
OVKATE CTRP1 4.0044 7.4031 2.9973 25.0437
IGROV-1 CTRP2; CTRP1 4.1851 7.1658 3.2862 10.2869
SNU-840 CTRP2; CTRP1 4.3355 8.4231 2.8266 11.8132
MCAS CTRP2 4.3551 6.4028 3.8074 7.7663
ES2 CTRP2 4.4496 7.6018 3.3332 9.4692
RMUG-S CTRP1 4.5182 11.2295 1.6055 30.2542
SNU-119 CTRP2 4.5907 8.1494 3.1966 9.7165
Kuramochi CTRP2 4.652 12.994 0.8434 18.8708
FU-OV-1 CTRP2 4.7278 8.5699 3.1128 9.7683
HEY A8 CTRP2; CTRP1 4.8606 8.6676 3.1817 9.202
EFO-27 CTRP2; CTRP1 4.9167 8.5559 3.2865 8.649
EFO-21 CTRP2; CTRP1 4.9264 7.0587 4.0396 5.4824
SNU-8 CTRP2 5.2091 8.1049 3.7614 6.0759
OC 314 CTRP2 5.21 10.8441 2.3926 11.7692
OVCAR-8 CTRP2; CTRP1 5.3767 9.6186 3.1426 8.3499
DOV13 CTRP2 5.3785 8.5559 3.6749 6.1197
RMG-I CTRP2; CTRP1 5.457 10.7648 2.6353 10.3041
JHOM-1 CTRP2; CTRP1 5.4719 8.814 3.6209 6.1759
OVSAHO CTRP2 5.5266 11.8398 2.1547 12.1277
JHOS-2 CTRP2 5.5759 9.1279 3.5466 6.3011
JHOS-4 CTRP1 5.6416 7.5051 4.3988 5.6983
COV434 CTRP2; CTRP1 5.6476 9.2886 3.5226 6.2762
OVCAR-5 CTRP2 5.7086 9.7165 3.3572 6.8592
OVK18 CTRP2; CTRP1 5.8535 12.5641 2.0541 11.9297
OV7 CTRP2; CTRP1 5.8712 11.44 2.627 9.5908
TOV-112D CTRP2 5.8978 8.0766 4.301 2.6717
COV362 CTRP2; CTRP1 5.9061 9.3556 3.6844 5.1747
ONCO-DG-1 CTRP2 5.922 10.7022 3.0319 7.8417
COV318 CTRP1 5.9402 7.1864 4.7431 1.9724
OVCAR-4 CTRP2; CTRP1 5.9969 9.8496 3.5084 5.7541
TOV-21G CTRP2 6.1032 9.0621 3.9675 3.7198
OAW28 CTRP2 6.1893 9.3583 3.8839 3.9331
OVMANA CTRP1 6.2896 9.7425 3.7677 9.0148
OAW42 CTRP2; CTRP1 6.3635 7.4551 4.8413 0.3088
OV56 CTRP2 6.4879 7.5486 4.8581 0.2195
OVTOKO CTRP2 6.7779 14.3647 1.8641 11.1013
OV-90 CTRP2; CTRP1 6.8051 11.9285 3.0687 6.3207
SK-OV-3 CTRP2; CTRP1 6.8979 9.8173 4.114 2.1853
COV644 CTRP2; CTRP1 7.1818 13.5835 2.5303 7.9047
JHOC-5 CTRP2; CTRP1 8.0152 13.8083 2.9624 5.1766
OVISE CTRP2 9.2633 19.2898 1.193 9.9958
Caov-3 CTRP2; CTRP1 9.2868 17.8599 1.8729 7.6265
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2; CTRP1 2.5721 5.2236 2.3273 18.393
NCI-H28 CTRP2; CTRP1 4.1789 7.1598 3.2829 10.3151
NCI-H2452 CTRP2 4.9027 8.2149 3.444 8.0199
NCI-H2052 CTRP2; CTRP1 5.012 8.5371 3.3783 8.0709
ACC-MESO-1 CTRP2 5.2366 10.1296 2.772 10.1574
MPP 89 CTRP2 6.9937 9.3463 4.3706 1.2321
JL-1 CTRP2 7.2276 11.8622 3.3768 4.5552
IST-Mes1 CTRP2 8.4041 16.4348 1.9835 8.3105
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
22Rv1 CTRP2 4.3291 10.5363 1.781 16.0511
LNCaP clone FGC CTRP2 4.9332 7.5934 3.7801 6.5512
VCaP CTRP2 5.4232 8.0104 3.9829 4.749
DU145 CTRP2 5.5238 9.521 3.3097 7.3829
PaCa-3 CTRP2; CTRP1 5.6063 6.902 4.6667 1.6165
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 CTRP2 5.3929 8.0866 3.9207 5.0638
YD-15 CTRP2 5.6811 11.6805 2.3581 11.0233
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-16 CTRP2 3.1351 5.076 2.9806 14.3305
SNU-1 CTRP2 3.4954 7.2598 2.551 14.961
SNU-5 CTRP2 3.6071 7.9457 2.3518 15.4675
SNU-620 CTRP2 3.883 5.4246 3.6979 9.4767
SNU-719 CTRP2 3.9558 7.1652 3.059 11.7684
NUGC-4 CTRP2; CTRP1 4.0341 7.2771 3.0852 11.4687
23132/87 CTRP2 4.2422 8.1188 2.8868 11.78
SNU-216 CTRP2 4.2861 9.2969 2.3531 13.8593
GSS CTRP2 4.4899 9.1521 2.6104 12.3584
ECC10 CTRP2 4.5803 7.9373 3.2912 9.3477
KE-39 CTRP2 4.6042 7.9195 3.322 9.1673
HGC-27 CTRP2 4.6621 7.2394 3.7087 7.4367
Fu97 CTRP2; CTRP1 4.7397 7.5495 3.6281 7.5991
HuG1-N CTRP2 4.779 7.4583 3.7089 7.1773
SNU-668 CTRP2 4.9609 9.8977 2.6551 11.185
IM95 CTRP2 4.9753 10.3987 2.4172 12.1337
GSU CTRP2 5.1933 5.8377 4.8817 1.4064
KATO III CTRP2 5.2223 7.0002 4.3248 3.687
SH-10-TC CTRP2; CTRP1 5.3311 8.773 3.528 6.8233
MKN74 CTRP2; CTRP1 5.3688 8.7539 3.5682 6.5848
MKN7 CTRP2; CTRP1 5.3742 10.4602 2.72 10.1101
NUGC-3 CTRP2 5.732 10.3908 3.0403 8.1338
LMSU CTRP2 5.7869 7.6608 4.4252 2.3303
AGS CTRP2; CTRP1 5.9083 11.1616 2.7938 8.8442
MKN45 CTRP2 5.9523 7.8489 4.4455 2.0247
ECC12 CTRP2 6.1799 10.4321 3.3561 6.0905
SNU-601 CTRP2 6.3936 9.7287 3.8442 3.8079
NCI-N87 CTRP2 6.4293 13.0969 2.2304 10.2415
MKN1 CTRP2 6.5544 10.3988 3.6319 4.4309
Hs 746.T CTRP2 6.5916 11.4495 3.1527 6.2936
SNU-685 CTRP2 4.9742 8.3928 3.4177 7.9826
SNG-M CTRP2; CTRP1 5.7525 9.6104 3.4436 6.4248
SNU-1077 CTRP2 8.0765 14.5072 2.6772 6.1618
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TT CTRP2 3.6675 8.8961 1.9637 16.8579
TT2609-C02 CTRP2 4.5844 7.9392 3.2942 9.3263
CGTH-W-1 CTRP2 5.5475 9.6919 3.2433 7.6169
SW579 CTRP2 5.6496 8.4929 3.9186 4.625
FTC-133 CTRP2 5.8292 7.8184 4.3784 2.4583
8305C CTRP2 6.0625 7.9304 4.4771 1.7656
B-CPAP CTRP2 6.0778 12.924 2.0498 11.5502
8505C CTRP2 6.0836 11.0148 2.9992 7.7072
CAL-62 CTRP2 6.7513 8.2523 4.7011 0.4522
ML-1 [Human leukemia] CTRP2 7.4778 9.4223 4.5626 0.4368
BHT-101 CTRP2 7.4787 11.7917 3.562 3.5697
FTC-238 CTRP2 8.1123 15.2652 2.3459 7.3503
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 1.9666 5.821 1.4863 23.2568
PE/CA-PJ49 CTRP2 3.4748 5.8703 3.1022 12.8797
HSC-2 CTRP2; CTRP1 3.9407 5.7103 3.6618 9.4445
SCC-25 CTRP2 4.2077 6.6195 3.5608 9.125
SNU-1214 CTRP2 4.2248 8.4975 2.6868 12.6381
Detroit 562 CTRP2 4.5191 8.0144 3.197 9.8737
PE/CA-PJ15 CTRP2 4.6967 9.2594 2.7427 11.3692
SNU-1076 CTRP2 4.7168 7.0603 3.8471 6.7417
PE/CA-PJ34 (clone C12) CTRP2 4.7991 6.258 4.3135 4.6324
BHY CTRP2 4.968 7.9118 3.6521 7.0146
SNU-46 CTRP2 5.1198 12.7005 1.3889 15.9037
SNU-1066 CTRP2 5.1321 9.6388 2.93 9.7045
FaDu CTRP2 5.1741 6.7006 4.4342 3.3212
SNU-899 CTRP2 5.2064 10.9383 2.3425 11.9802
HSC-4 CTRP2 5.2392 9.5747 3.0516 8.9901
PE/CA-PJ41 (clone D2) CTRP2 5.4091 9.7587 3.099 8.4717
SCC-9 CTRP2; CTRP1 5.4386 8.1144 3.9433 4.8872
BICR 6 CTRP2 5.4549 8.7778 3.6255 6.1875
BICR 22 CTRP2 5.5035 7.3789 4.359 3.0403
CAL-33 CTRP2 5.5647 8.0756 4.0606 4.1775
SNU-1041 CTRP2 5.6989 10.2872 3.066 8.0852
BICR 31 CTRP2 5.7085 8.9904 3.7171 5.363
BICR 18 CTRP2 6.4416 8.6176 4.3897 1.6677
HSC-3 CTRP2 6.8182 11.8231 3.1282 6.0657
SCC-4 CTRP2 7.0201 15.2263 1.6182 11.646
YD-8 CTRP2 7.1854 12.6695 2.9697 6.1842
BICR 16 CTRP2 7.6776 9.1512 4.7362 0.1111
BICR 56 CTRP2 9.1755 20.577 0.5265 12.3173
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HT-1197 CTRP2 1.1834 13.2621 -7.8323 20.9428
5637 CTRP2; CTRP1 3.3149 7.4734 2.272 16.5258
RT-4 CTRP2; CTRP1 4.1929 8.3763 2.7156 12.5938
UM-UC-3 CTRP2; CTRP1 4.3112 6.7419 3.6082 8.6759
SW1710 CTRP2 4.6684 8.2052 3.2398 9.3677
RT-112 CTRP2 4.6957 9.2196 2.7617 11.293
JMSU-1 CTRP2 4.7812 9.4383 2.7283 11.2513
VM-CUB-1 CTRP2 4.8226 10.102 2.4338 12.3774
253J CTRP2 4.8284 7.4316 3.7667 6.8297
HT-1376 CTRP2; CTRP1 4.9253 8.1833 3.4796 7.8243
BC-3C CTRP2 4.9655 8.8942 3.16 9.0775
KMBC-2 CTRP2; CTRP1 5.0008 8.4626 3.4059 7.9782
U-BLC1 CTRP2 5.0067 5.8508 4.7073 2.533
SCaBER CTRP2 5.1234 12.6738 1.4053 15.8347
253J-BV CTRP2 5.1433 7.6926 3.9123 5.5711
UM-UC-1 CTRP2 5.1676 9.3269 3.1157 8.8611
CAL-29 CTRP2 5.7563 7.4794 4.4915 2.1075
T24 CTRP2 5.9057 8.5448 4.0804 3.5523
KU-19-19 CTRP2 6.1311 10.8914 3.0952 7.2361
647V CTRP2 6.2603 13.9575 1.6774 12.6796
BFTC-905 CTRP2 6.8566 8.2955 4.7296 0.3386
639V CTRP2 6.9139 8.4713 4.6869 0.4074
TCCSUP CTRP2 7.9626 15.1562 2.3008 7.7121
J82 CTRP2 10.2452 18.3618 2.2043 5.4889
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 6.2291 9.0411 4.0623 3.1668

References

1 Lysosomes as a therapeutic target. Nat Rev Drug Discov. 2019 Dec;18(12):923-948.
2 The ChEMBL database in 2017. Nucleic Acids Res. 2017 Jan 4;45(D1):D945-D954.