Details of the Drug

General Information of Drug (ID: DMJWE3I)

Drug Name
Gossypol
Synonyms
gossypol; 303-45-7; (-)-Gossypol; 90141-22-3; (+)-Gossypol; Pogosin; Tash 1; racemic-Gossypol; (R)-(-)-Gossypol; (R)-Gossypol; (+-)-Gossypol; (+/-)-Gossypol; CCRIS 2689; NSC56817; NSC 56817; NSC 624336; BRN 1917878; CHEMBL51483; AI3-22957; 20300-26-9; 1,1',6,6',7,7'-Hexahydroxy-5,5'-diisopropyl-3,3'-dimethyl-[2,2'-binaphthalene]-8,8'-dicarbaldehyde; 2,2'-bi[8-Formyl-1,6,7-trihydroxy-5-isopropyl-3-methylnaphthalene]; 2,2'-Bis(1,6,7-trihydroxy-3-methyl-5-isopropyl-8-aldehydonaphthalene); NSC624336; Gossypol acetate
Indication
Disease Entry ICD 11 Status REF
Prostate cancer 2C82.0 Phase 2 [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 3 Molecular Weight (mw) 518.6
Logarithm of the Partition Coefficient (xlogp) 6.9
Rotatable Bond Count (rotbonds) 5
Hydrogen Bond Donor Count (hbonddonor) 6
Hydrogen Bond Acceptor Count (hbondacc) 8
Chemical Identifiers
Formula
C30H30O8
IUPAC Name
7-(8-formyl-1,6,7-trihydroxy-3-methyl-5-propan-2-ylnaphthalen-2-yl)-2,3,8-trihydroxy-6-methyl-4-propan-2-ylnaphthalene-1-carbaldehyde
Canonical SMILES
CC1=CC2=C(C(=C(C(=C2C(C)C)O)O)C=O)C(=C1C3=C(C4=C(C=C3C)C(=C(C(=C4C=O)O)O)C(C)C)O)O
InChI
InChI=1S/C30H30O8/c1-11(2)19-15-7-13(5)21(27(35)23(15)17(9-31)25(33)29(19)37)22-14(6)8-16-20(12(3)4)30(38)26(34)18(10-32)24(16)28(22)36/h7-12,33-38H,1-6H3
InChIKey
QBKSWRVVCFFDOT-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
3503
CAS Number
20300-26-9
UNII
KAV15B369O
DrugBank ID
DB13044
TTD ID
D0Z0HH
VARIDT ID
DR00896

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Apoptosis regulator Bcl-2 (BCL-2) TTJGNVC BCL2_HUMAN Regulator [2]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Bcl-2-binding component 3, isoforms 3/4 (BBC3) OTUAXDAY BBC3B_HUMAN Gene/Protein Processing [3]
Bcl-2-like protein 1 (BCL2L1) OTRC5K9O B2CL1_HUMAN Gene/Protein Processing [3]
Bcl-2-like protein 11 (BCL2L11) OTNQQWFJ B2L11_HUMAN Gene/Protein Processing [3]
C-C motif chemokine 2 (CCL2) OTAD2HEL CCL2_HUMAN Gene/Protein Processing [4]
Caspase-3 (CASP3) OTIJRBE7 CASP3_HUMAN Gene/Protein Processing [4]
Caspase-7 (CASP7) OTAPJ040 CASP7_HUMAN Gene/Protein Processing [4]
Caspase-9 (CASP9) OTD4RFFG CASP9_HUMAN Protein Interaction/Cellular Processes [3]
DNA-binding protein inhibitor ID-1 (ID1) OTKGNZN5 ID1_HUMAN Gene/Protein Processing [4]
Fibroblast growth factor 2 (FGF2) OT7YUJ9F FGF2_HUMAN Gene/Protein Processing [4]
Fibroblast growth factor receptor 3 (FGFR3) OTSAXDIL FGFR3_HUMAN Gene/Protein Processing [4]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Prostate cancer
ICD Disease Classification 2C82.0
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Apoptosis regulator Bcl-2 (BCL-2) DTT BCL2 2.52E-02 0.17 0.72
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 134 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 1.7464 2.4313 1.7464 23.029
JK1 CTRP2 3.7787 5.0172 3.3883 4.4262
JM1 CTRP2 1.8462 2.8164 1.8457 22.367
SKM-1 CTRP2; CTRP1 0.7564 2.2682 0.7542 29.6198
WSU-DLCL2 CTRP2; CTRP1 0.8779 1.2895 0.8779 30.9983
NU-DUL-1 CTRP2; CTRP1 0.9755 1.6803 0.9755 28.1554
SU-DHL-5 CTRP1 1.0184 1.6841 1.0184 59.8711
GA-10 CTRP2 1.0566 2.1463 1.0564 27.617
TF-1 CTRP2 1.0939 1.8943 1.0939 27.3679
EB1 CTRP2 1.1048 2.722 1.0992 27.3143
Daudi CTRP2 1.1807 2.0242 1.1807 26.7909
HT CTRP2; CTRP1 1.3229 2.2027 1.3229 25.8454
GDM-1 CTRP1 1.344 3.1122 1.3309 55.0829
ST486 CTRP2 1.3498 2.2108 1.3498 25.6663
Mino CTRP2 1.3856 2.0118 1.3856 25.4282
PL21 CTRP2; CTRP1 1.4102 2.525 1.4097 25.2665
THP-1 CTRP2; CTRP1 1.4831 2.1606 1.4831 24.7797
EoL-1 CTRP2 1.5565 2.4924 1.5564 24.2921
BL-70 CTRP2; CTRP1 1.5778 2.0086 1.5778 24.1504
OCI-AML-5 CTRP2 1.5944 2.0456 1.5944 24.04
Pfeiffer CTRP2 1.5967 2.6451 1.5962 24.0264
P12-Ichikawa CTRP2 1.5991 2.3509 1.5991 24.0085
A4/Fukuda CTRP2 1.615 2.5593 1.6148 23.9037
Kasumi-2 CTRP2 1.6151 2.1146 1.6151 23.9023
KE-37 CTRP2 1.622 2.4134 1.622 23.8566
AML-193 CTRP2 1.6471 2.4763 1.6471 23.6895
MV4-11 CTRP2 1.6603 2.9154 1.658 23.6093
F-36P CTRP2 1.6609 2.564 1.6607 23.5982
KMS-20 CTRP2 1.6685 2.2371 1.6685 23.547
OCI-Ly3 CTRP2 1.6699 2.8551 1.6683 23.5431
NALM-6 CTRP2 1.6744 2.4723 1.6744 23.508
DND-41 CTRP2 1.6767 2.6884 1.6763 23.494
OPM-2 CTRP2 1.6812 3.1319 1.6749 23.4838
HEL 92.1.7 CTRP2 1.6863 2.0837 1.6863 23.4288
MOLM-13 CTRP2 1.6959 2.4525 1.6959 23.365
RPMI-8226 CTRP2; CTRP1 1.7045 3.0425 1.7006 23.3207
M-07e CTRP2 1.7084 2.2049 1.7084 23.2818
DoHH2 CTRP2 1.7128 2.2466 1.7128 23.2528
JeKo-1 CTRP2 1.719 2.1541 1.719 23.2112
KMS-34 CTRP2 1.7339 2.6946 1.7306 17.4141
Ki-JK CTRP2 1.7396 2.6633 1.7394 23.075
LAMA-84 CTRP2 1.7481 2.6361 1.7479 23.0186
NCI-H929 CTRP2 1.7512 2.5398 1.7512 22.9973
NU-DHL-1 CTRP2 1.7519 2.515 1.7519 22.9925
U-937 CTRP2; CTRP1 1.7589 3.3417 1.747 22.9858
KCL-22 CTRP2 1.7612 3.0811 1.7573 22.9435
P31/FUJ CTRP2 1.7694 2.2591 1.7694 22.8762
SEM CTRP2 1.7711 2.2779 1.7711 22.865
SU-DHL-10 CTRP2 1.7825 2.5267 1.7819 17.0574
EM-2 CTRP2 1.7947 2.4148 1.7947 22.7077
SU-DHL-1 CTRP2 1.7993 2.2519 1.7993 22.6773
CML-T1 CTRP2 1.803 2.9163 1.8018 22.6568
HEL CTRP2 1.808 2.2926 1.808 22.6194
RL CTRP2 1.8083 3.3252 1.7984 22.6505
SET-2 CTRP2 1.8241 2.2644 1.8241 22.5124
MOLM-16 CTRP2; CTRP1 1.8254 2.9503 1.824 22.5083
CMK CTRP2 1.8305 2.197 1.8305 22.4696
DB CTRP2 1.8405 2.7145 1.8403 22.4038
Peer CTRP2 1.8427 2.7208 1.8425 22.3894
Jurkat CTRP2 1.8497 3.4268 1.8365 22.3862
SU-DHL-8 CTRP2 1.8572 2.5645 1.8567 16.5231
PF-382 CTRP2 1.8693 3.0985 1.8665 22.2211
KM-H2 CTRP2 1.8931 3.3874 1.8828 22.088
K-562 CTRP2 1.9165 3.8285 1.8778 22.0282
Karpas-422 CTRP2 1.9327 2.6837 1.9326 21.7905
KMS-26 CTRP2 1.9634 3.1688 1.9605 21.5958
Kasumi-1 CTRP2 1.9838 3.1026 1.982 21.4566
LP-1 CTRP2; CTRP1 2.0125 4.2165 1.933 21.529
SUP-HD1 CTRP2 2.016 3.7772 1.9867 21.3348
KMS-11 CTRP2; CTRP1 2.0393 3.8626 2.0037 21.2012
KO52 CTRP2 2.0519 2.7602 2.0519 20.9976
NCO2 CTRP2 2.0824 3.6215 2.0664 20.8482
RPMI-6666 CTRP2 2.0926 3.3309 2.0881 20.7417
DEL CTRP2 2.1103 3.3359 2.106 20.6238
RPMI-8402 CTRP2 2.1143 3.3993 2.1085 20.6018
Ri-1 CTRP2 2.1206 4.2721 1.9047 15.4536
KE-97 CTRP2; CTRP1 2.1893 3.0042 2.1891 20.0846
Ku812 CTRP2; CTRP1 2.2083 2.9885 2.2082 19.9577
KMS-21-BM CTRP2 2.2178 3.5518 2.209 19.9237
SUP-B15 CTRP2 2.2484 3.2649 2.2469 19.6957
MOLT-16 CTRP2 2.2574 3.7243 2.1853 13.9272
NOMO-1 CTRP1 2.3001 3.0454 2.3 41.5629
JURL-MK1 CTRP2 2.3243 3.9577 2.2942 19.2871
EHEB CTRP2 2.3253 3.9948 2.2919 19.292
MOTN-1 CTRP2 2.3605 4.074 2.3211 19.0781
KMS-12-BM CTRP2 2.4272 4.314 2.2269 13.2066
HL-60 CTRP2 2.5266 3.5631 2.5234 17.8512
MOLP-8 CTRP2 2.5425 3.8403 2.5297 17.7778
L-428 CTRP2 2.573 4.5556 2.4808 17.8466
SU-DHL-6 CTRP2 2.6339 4.4195 2.4194 11.7895
Hs 611.T CTRP2 2.646 4.4655 2.5742 17.2907
Granta-519 CTRP2 2.6535 5.4809 2.3414 18.0968
L-540 CTRP2 2.708 4.0802 2.5981 10.8537
MC116 CTRP2; CTRP1 2.7408 3.052 2.7408 16.4164
Mono-Mac-1 CTRP2 2.7442 5.2128 2.243 12.1732
Ci-1 CTRP2 2.7828 4.3252 2.7399 16.2817
SIG-M5 CTRP2 2.8781 3.3166 2.8781 15.5035
KYO-1 CTRP2 2.8917 4.4592 2.6865 9.9167
HPB-ALL CTRP2 2.8994 4.5208 2.6739 9.9432
P3HR-1 CTRP2; CTRP1 2.9037 3.6796 2.9026 15.3367
HDLM-2 CTRP2 2.9163 4.9382 2.7753 15.7361
OCI-AML-3 CTRP2; CTRP1 2.9273 3.6608 2.9266 15.1785
SU-DHL-4 CTRP2; CTRP1 2.9674 4.0767 2.9557 14.9486
Mono-Mac-6 CTRP2 3.0336 5.2388 2.5342 10.121
HD-MY-Z CTRP2 3.1382 4.8793 3.0299 14.1463
RS4;11 CTRP2 3.148 4.7779 2.8451 8.4919
OCI-M1 CTRP2 3.1594 3.9406 3.1572 13.6401
JJN-3 CTRP2 3.1737 5.1278 3.0095 14.1088
SUP-T1 CTRP2 3.2529 4.7519 2.9666 7.6803
KMS-18 CTRP2 3.2534 5.0572 2.8398 8.2091
KMS-27 CTRP2 3.2833 4.889 3.1854 13.1454
OCI-Ly19 CTRP2 3.3828 5.6284 3.0877 13.199
RCH-ACV CTRP2 3.4333 4.8757 3.1041 6.5837
SR CTRP2 3.4409 4.7308 3.1733 6.2719
REC-1 CTRP2 3.5898 6.6963 2.3958 9.2832
MM1.S CTRP2 3.6119 5.13 3.1714 5.8063
BV-173 CTRP2 3.6207 4.6919 3.3771 4.9012
EJM CTRP2; CTRP1 3.6269 6.2951 3.0999 12.4645
MOLM-6 CTRP2 3.7224 4.5079 3.5607 3.8396
L-1236 CTRP2 3.7276 5.5967 3.0611 5.9952
MHH-CALL-4 CTRP2 3.7385 5.3796 3.1764 5.4588
TALL-1 [Human adult T-ALL] CTRP2 3.7666 5.8454 2.9762 6.2781
L-363 CTRP2 3.831 4.3841 3.7255 2.8374
KHM-1B CTRP2 3.8378 5.5023 3.6235 9.8843
SUP-T11 CTRP2 3.8434 4.6397 3.6279 3.2153
AMO1 CTRP2; CTRP1 3.8668 4.2571 3.8666 8.9294
HuT 78 CTRP2 4.0343 5.9565 3.6668 9.164
ME1 CTRP2 4.1098 4.8875 3.7599 1.9763
MHH-CALL-3 CTRP2 4.3309 5.9108 3.4297 3.0178
MOLP-2 CTRP2 4.5221 6.034 3.5126 2.3085
Karpas-620 CTRP2 4.5727 5.9613 3.5836 1.9161
KMM-1 CTRP2 4.6544 11.5684 1.5564 16.2223
OCI-Ly10 CTRP1 6.4739 9.0959 4.1916 5.0562
SK-MM-2 CTRP2 6.9014 30.4561 -6.7719 29.3471
⏷ Show the Full List of 134 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 1.9646 3.489 1.9518 21.6211
TE8 CTRP2 4.4669 8.2545 2.3695 7.5177
TE-11 CTRP2 2.6975 4.7699 2.5743 17.1274
TE-5 CTRP2 2.6994 4.6275 2.6043 17.0164
KYSE-140 CTRP2; CTRP1 2.9546 4.9025 2.8252 15.4405
KYSE-30 CTRP2 2.9939 4.9597 2.8549 15.2135
OE21 CTRP2 2.9953 4.9928 2.8486 15.2312
KYSE-450 CTRP2; CTRP1 3.1403 4.8101 3.0465 14.0814
KYSE-520 CTRP2 3.1594 5.6977 2.822 14.8361
EC-GI-10 CTRP2 3.362 5.3753 3.1457 13.047
KYSE-410 CTRP2; CTRP1 3.4002 5.3476 3.1956 12.7508
TE-9 CTRP2 3.4412 5.2567 3.2666 12.37
OE33 CTRP2 3.5126 6.5004 2.8955 13.5662
KYSE-150 CTRP2 3.5334 5.0705 3.4163 11.5511
KYSE-180 CTRP2 3.5625 5.525 3.317 11.8243
TE-14 CTRP2 3.6498 5.7313 3.3409 11.482
TE-10 CTRP2 3.7046 5.6971 3.4122 11.0576
TE-6 CTRP2 3.8905 6.4086 2.81 6.7337
KYSE-510 CTRP2 4.0968 7.385 3.0967 11.2692
TE-4 CTRP2 4.2255 6.6754 2.9632 5.3249
TE-1 CTRP2 4.2831 5.7615 3.4664 2.9445
COLO 680N CTRP2 4.3759 6.0084 4.0033 7.464
OE19 CTRP2 4.5866 6.3234 4.0753 6.1122
KYSE-70 CTRP2 5.2782 7.0198 2.6239 0.4276
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 36 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 3.5406 5.5835 3.2738 12.0482
KP-4 CTRP2 1.9238 3.3283 1.9164 21.8741
PSN1 CTRP2 2.2852 3.3814 2.2824 19.4555
Capan-2 CTRP2; CTRP1 2.4604 4.4255 2.3813 18.55
KP-3 CTRP2; CTRP1 2.4672 5.3944 2.1642 19.2996
BxPC-3 CTRP2 2.7464 8.4497 1.258 21.8929
AsPC-1 CTRP2 2.9641 5.4168 2.6994 15.8633
DAN-G CTRP2 3.0654 5.0629 2.9079 14.8041
MIA PaCa-2 CTRP2 3.0807 4.5223 3.0314 14.3229
HPAF-II CTRP2 3.1635 4.9695 3.0373 14.0409
Panc 04.03 CTRP2 3.1809 5.3972 2.9417 14.3322
SUIT-2 CTRP2; CTRP1 3.2271 4.9422 3.1127 13.5766
SW1990 CTRP2 3.2339 5.9141 2.8269 14.6027
HuP-T4 CTRP2; CTRP1 3.434 4.897 3.3473 12.1043
HPAC CTRP2; CTRP1 3.5656 4.9367 3.4819 11.2191
Panc 03.27 CTRP2; CTRP1 3.7158 5.1633 3.5918 10.3646
QGP-1 CTRP2; CTRP1 3.7386 5.6985 3.4484 10.824
HuP-T3 CTRP2 3.888 6.2417 3.3963 10.6083
Panc 08.13 CTRP2 3.9206 5.889 3.5727 9.8391
PK-59 CTRP2 4.0438 5.2789 3.5071 3.2592
PK-45H CTRP2 4.071 6.3093 3.5583 9.4877
YAPC CTRP2 4.0713 4.668 3.8346 1.7287
PaTu 8988s CTRP2 4.0722 6.038 3.6737 9.0341
SU.86.86 CTRP2 4.1514 5.3626 3.5581 2.7964
Hs 766T CTRP2 4.2599 5.4747 4.0902 6.9218
KP-2 CTRP2 4.2603 6.8627 3.5017 9.2312
PaTu 8988t CTRP2 4.2842 5.4711 4.1178 6.7487
L3.3 CTRP2 4.3583 5.3364 3.7353 1.6019
Panc 02.03 CTRP2 4.3806 6.9975 3.5567 8.7157
CFPAC-1 CTRP2; CTRP1 4.562 7.1551 3.6556 7.8841
SNU-410 CTRP2 4.7566 6.9007 3.2572 3.0465
TCC-Pan2 CTRP2 4.7834 6.7465 2.5093 1.0782
Panc 10.05 CTRP2; CTRP1 4.8023 6.002 4.4381 4.1169
SNU-213 CTRP2 4.8735 5.7104 4.6438 3.1112
PaTu 8902 CTRP2; CTRP1 4.9845 5.7768 4.7219 2.5246
Panc 05.04 CTRP2 5.0323 7.6946 3.0642 3.4562
⏷ Show the Full List of 36 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 4.127 16.4563 -1.3397 26.6563
WM266-4 CTRP2 1.7371 2.122 1.7371 23.0906
CJM [Human melanoma] CTRP2 1.8864 2.5125 1.8864 22.0983
WM115 CTRP2 1.9412 3.0147 1.94 21.7375
HMCB CTRP2 2.0984 3.1073 2.0974 20.6915
WT2-iPS CTRP2 2.1417 2.9102 2.1416 20.4006
MeWo CTRP2 2.4412 4.0814 2.4054 18.5292
Malme-3M CTRP2 2.5975 5.4894 2.2779 18.4956
SK-MEL-2 CTRP2 2.6568 4.4483 2.5886 17.2065
WM88 CTRP2 2.7447 4.6106 2.6562 16.6923
Hs 944.T CTRP2; CTRP1 2.7861 3.6484 2.7845 16.1203
COLO 741 CTRP1 2.8309 4.6398 2.7441 33.8497
G-361 CTRP2; CTRP1 2.8958 4.284 2.8641 15.4925
UACC-62 CTRP2 2.8977 3.3766 2.8977 15.3733
K029AX CTRP2 3.062 4.9165 2.9389 14.7045
SK-MEL-3 CTRP2 3.0855 4.0253 3.0796 14.1439
SK-MEL-28 CTRP2; CTRP1 3.3017 3.9987 3.3001 12.6918
SK-MEL-5 CTRP2; CTRP1 3.3175 4.2213 3.3094 12.6085
WM983B CTRP2 3.3719 4.9568 3.267 12.581
COLO 792 CTRP2 3.4245 5.4775 3.1822 12.7277
LOX-IMVI CTRP2 3.6289 4.8822 3.5617 10.7406
RVH-421 CTRP2 3.7193 5.2072 3.5838 10.3823
Mel Ho CTRP2 3.8123 5.7405 3.5126 10.3723
COLO 800 CTRP2 3.8433 5.8543 3.5035 10.3189
WM793 CTRP2 3.8483 4.3966 3.7388 2.7314
UACC-257 CTRP2 3.8609 5.0882 3.7689 9.2862
HT-144 CTRP2 4.0137 5.5448 3.7997 8.7175
SK-MEL-31 CTRP2 4.0808 5.2043 3.5767 2.8642
A-375 CTRP2; CTRP1 4.0959 5.3869 3.9415 7.952
MDA-MB-435S CTRP2 4.1657 5.8906 3.3061 3.9021
Hs 294T CTRP2 4.2371 5.4835 4.0626 7.0909
SK-MEL-1 CTRP2; CTRP1 4.2494 5.3082 4.1332 6.7941
IGR-37 CTRP2 4.3841 5.3752 4.2585 5.935
Hs 895.T CTRP2 4.3987 5.619 4.1868 6.1626
IPC-298 CTRP2 4.4357 6.0098 3.461 2.6858
Hs 936.T CTRP2; CTRP1 4.4729 5.5716 4.2842 5.584
COLO 829 CTRP2 4.4803 5.6703 4.2534 5.6815
WM1799 CTRP2 4.4934 5.6242 3.6916 1.5714
Mel JuSo CTRP2 4.507 5.9126 3.561 2.1204
A2058 CTRP2 4.5335 5.1584 4.485 4.663
Hs 852.T CTRP2; CTRP1 4.6382 5.8568 4.3393 4.9248
SK-MEL-30 CTRP2 4.66 6.5874 3.3412 2.8347
RPMI-7951 CTRP2 4.769 5.9619 4.4238 4.2565
A101D CTRP2 4.8328 5.2753 4.7787 2.6966
IGR-39 CTRP2 4.9598 8.7069 3.2485 8.7194
Hs 839.T CTRP2 5.0069 6.2715 4.5015 3.3851
Hs 688(A).T CTRP2 5.231 6.058 4.803 1.6644
IGR-1 CTRP2 8.1988 24.38 -2.013 20.946
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 1.364 3.6523 1.3133 25.7425
Cancer Drug Sensitivity Data Curated from 9 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IMR-32 CTRP2 1.0689 2.3386 1.068 27.5374
Kelly CTRP2 1.734 2.2365 1.734 17.4016
SK-N-BE(2) CTRP2 1.8076 2.8571 1.8068 22.6247
SK-N-SH CTRP2 2.0039 2.9844 2.0032 21.3189
KP-N-YN CTRP2 2.9132 6.3656 2.3145 17.4462
NH-6 CTRP2 3.0998 4.8312 2.9982 14.3778
NB1 CTRP2 3.1464 5.1373 2.6946 9.1247
SK-N-FI CTRP2 3.5988 4.5951 3.5735 10.7963
SK-N-DZ CTRP2 4.4527 5.1567 4.3974 5.2239
⏷ Show the Full List of 9 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-478 CTRP2 1.8675 3.1774 1.8631 22.2385
SNU-869 CTRP2 2.5444 6.4412 1.8915 20.0809
SNU-1079 CTRP2 3.0721 4.666 2.9996 15.5616
HuH-28 CTRP2 3.9553 4.786 3.9288 8.4298
SNU-245 CTRP2 4.156 5.5462 3.9529 7.7346
SNU-308 CTRP2 4.2136 5.2151 4.1211 6.9454
HuCC-T1 CTRP2 4.3615 5.5849 4.16 6.369
SNU-1196 CTRP2 4.4595 7.4511 3.4154 9.8018
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-MC CTRP2 1.7046 2.1394 1.7046 23.307
HOS CTRP2 1.896 2.8079 1.8957 22.0352
MHH-ES-1 CTRP2 1.9067 3.104 1.9041 21.9718
TC71 CTRP2 2.0892 3.0272 2.0886 20.7516
A-673 CTRP2 2.2025 3.3372 2.1994 20.0063
MG-63 CTRP2 2.2852 3.2352 2.2842 19.4496
SK-ES-1 CTRP2 2.681 4.6305 2.5838 17.146
SaOS-2 CTRP2 2.8885 5.5121 2.5879 16.4963
CAL-78 CTRP2 4.1408 6.0296 3.2157 4.3613
G-292 clone A141B1 CTRP2 4.3368 6.2548 3.8554 7.6218
SW1353 CTRP2 4.4768 5.2299 4.4042 5.126
SJSA-1 CTRP2 4.594 7.9435 2.6239 6.1378
Hs 888.T CTRP2 4.7906 7.4533 3.7219 7.098
Hs 822.T CTRP2 4.8863 6.0425 4.5004 3.6623
U2OS CTRP1 5.0221 6.4567 4.4236 7.8987
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 71 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 CTRP2 1.0009 2.4219 0.999 27.993
MDA-MB-415 CTRP2 1.6907 3.3206 1.6779 23.4424
HCC2218 CTRP2 1.7004 2.463 1.7004 23.3348
MDA-MB-157 CTRP2 1.7474 2.8824 1.7461 23.0267
EFM-192A CTRP2 2.2139 4.3379 2.1304 20.2038
HCC1419 CTRP2 2.2502 4.8161 2.0782 20.2718
BT-549 CTRP2 2.2709 3.9283 2.2408 19.6421
SK-BR-3 CTRP2 2.9389 5.037 2.7764 15.6622
CAMA-1 CTRP2 2.9893 4.6197 2.9184 15.0053
ZR-75-30 CTRP2 3.0285 5.7301 2.6693 15.7842
HCC1500 CTRP2 3.0391 4.7587 2.947 14.748
MDA-MB-453 CTRP2 3.0606 4.9412 2.9318 14.7343
Hs 578T CTRP2 3.2297 18.64 -3.2195 32.6372
HCC202 CTRP2 3.3744 5.7562 3.0348 13.4204
HMC-1-8 CTRP2 3.4066 4.688 3.3559 12.1612
HCC1428 CTRP2 3.6096 6.343 3.0623 12.6571
HCC38 CTRP2 3.6112 5.4371 3.3981 11.3823
MDA-MB-468 CTRP2 3.6775 5.2312 3.5316 10.6977
HCC1937 CTRP2 3.7331 6.2842 3.2162 11.7258
MCF-7 CTRP2; CTRP1 3.8315 6.4315 3.2577 11.3002
BT-20 CTRP2 3.9628 5.5026 3.759 9.0169
T-47D CTRP2 4.0013 6.4812 3.4119 10.2467
AU565 CTRP2 4.0865 5.738 3.8077 8.48
HCC1954 CTRP2 4.1407 5.3937 3.988 7.6487
HCC1806 CTRP2 4.1817 5.7407 3.9084 7.8301
MDA-MB-361 CTRP2 4.2008 7.5242 3.1324 10.8738
HCC1143 CTRP2 4.3937 7.1282 2.8729 5.3991
ZR-75-1 CTRP2 4.4272 5.7302 3.5924 2.1164
MDA-MB-231 CTRP2 4.4694 6.4501 3.2688 3.4826
CAL-85-1 CTRP2 4.5965 5.9508 4.2551 5.3663
HCC1395 CTRP2 4.7353 6.289 4.2371 5.0955
CAL-51 CTRP2 4.804 5.4683 4.6768 3.1636
HDQ-P1 CTRP2 4.8165 6.1358 4.3886 4.2842
BT-474 CTRP2 5.2044 6.214 4.703 2.1348
CAL-148 CTRP2 5.2672 6.9109 4.4064 3.2596
JIMT-1 CTRP2 5.3432 7.5728 4.1374 4.5704
KPL-1 CTRP2 5.659 11.4191 2.4709 10.6054
CAL-120 CTRP2 5.727 7.2028 4.6041 1.6989
BT 239 CTRP2 1.116 1.9011 1.116 27.2214
BT 286 CTRP2 1.1351 2.0896 1.1351 27.0942
BT164 CTRP2 1.1882 1.9677 1.1882 26.741
BT 271 CTRP2 1.1948 2.4826 1.1936 26.7012
BT 145 CTRP2 1.1995 2.1221 1.1995 26.666
BT 112 CTRP2 1.2438 2.0083 1.2438 26.3716
BT 248 CTRP2 1.2884 2.2862 1.2882 26.0754
BT147 CTRP2 1.3722 2.8627 1.3675 25.5334
BT 428 CTRP2 1.4009 2.2478 1.4009 25.3267
BT 416 CTRP2 1.434 2.1481 1.434 25.1064
BT 228 CTRP2 1.5035 2.0431 1.5035 24.6445
BT 231 CTRP2 1.5155 2.5768 1.5151 24.5658
BT 330 CTRP2 1.5705 2.1559 1.5705 24.1985
BT 131 CTRP2 1.6053 2.1892 1.6053 23.9673
BT 139 CTRP2 1.6335 2.0339 1.6335 23.7796
BT 159 CTRP2 1.6494 2.2566 1.6494 23.6743
BT 232 CTRP2 1.685 2.6252 1.6848 23.4379
BT 172 CTRP2 1.7519 2.5734 1.7518 22.9929
BT 245 CTRP2 1.7718 3.1449 1.7667 22.877
BT 444 CTRP2 1.8175 3.4172 1.8038 22.602
BT 504 CTRP2 1.8287 2.2379 1.8287 22.4819
BT 482 CTRP2 1.8575 3.2929 1.8498 22.3162
BT 498 CTRP2 1.9105 3.5878 1.8904 22.0051
BT 422 CTRP2 2.0187 3.577 2.0031 21.2704
BT 216 CTRP2 2.1171 3.5837 2.1042 20.6072
BT 224 CTRP2 2.2137 3.4577 2.208 19.9404
BT 179 CTRP2 2.4787 3.7049 2.4704 18.1869
BT 333 CTRP2 2.8801 4.6435 2.7966 15.7749
BT 359 CTRP2 3.0739 4.7305 2.99 14.4879
BT 340 CTRP2 3.2507 5.482 2.9916 13.9419
BT 440 CTRP2 3.324 4.7125 3.263 12.7457
BT 320 CTRP2 4.3493 5.1607 4.2836 5.9484
BT 328 CTRP2 4.3871 5.2933 4.2878 5.8187
⏷ Show the Full List of 71 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 4.1118 5.0104 4.0594 7.4789
Cancer Drug Sensitivity Data Curated from 43 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW1783 CTRP2 0.3686 13.5775 -3.4708 40.2307
SF539 CTRP2 1.5928 2.1334 1.5928 24.0505
8-MG-BA CTRP2 1.616 2.1584 1.616 23.8959
U-251MG CTRP2 1.6255 2.1663 1.6255 23.8331
T98G CTRP2 1.7287 2.9135 1.7271 23.1521
D283 Med CTRP2 1.7808 2.935 1.7793 22.8053
TM-31 CTRP2 1.8457 2.2526 1.8457 22.3687
SNU-466 CTRP2 1.8923 2.9673 1.8912 22.0625
SF268 CTRP2 1.9646 4.0859 1.8998 21.7971
YH-13 CTRP2 2.8298 4.6971 2.7323 16.1578
Becker CTRP2 3.0383 5.0399 2.884 14.9728
Daoy CTRP2 3.1589 4.4858 3.1197 13.7685
SF295 CTRP2; CTRP1 3.3251 5.5433 3.0531 13.4959
GB-1 CTRP2 3.3736 4.5382 3.3415 12.3167
M059K CTRP2 3.3939 5.2512 3.2165 12.6942
LN-229 CTRP2; CTRP1 3.4341 5.0308 3.3176 12.2088
42-MG-BA CTRP2 3.4675 5.2161 3.3065 12.1462
ONS-76 CTRP2 3.5697 5.5276 3.324 11.7774
SNU-1105 CTRP2 3.6596 5.0788 3.5518 10.6799
DK-MG CTRP2 3.7205 5.6477 3.4468 10.8824
Hs 683 CTRP2 3.7324 5.5826 3.4821 10.7163
GOS-3 CTRP2 3.9158 5.7207 3.6312 9.6306
SNU-738 CTRP2 4.0503 5.6748 3.7926 8.6395
GMS-10 CTRP2 4.1532 6.1254 3.7221 8.6279
SNU-201 CTRP2 4.1554 5.4482 3.9861 8.1924
LN-18 CTRP2 4.1784 4.783 4.1657 6.8991
DBTRG-05MG CTRP2 4.2165 5.1778 3.7043 2.0044
SNB-75 CTRP2 4.3068 9.1472 2.4456 13.4369
SF126 CTRP2 4.3776 5.7243 4.1231 6.465
U-118MG CTRP2 4.3871 6.1096 3.9709 7.0341
CCF-STTG1 CTRP2 4.4171 6.2601 3.9345 7.1015
SW1088 CTRP2 4.432 6.1105 3.4085 2.9263
SNU-626 CTRP2 4.4721 5.3873 4.35 5.7458
KALS-1 CTRP2 4.6101 6.1718 3.5079 2.1867
KG-1-C CTRP2 4.6177 5.2097 4.5636 4.124
CAS-1 CTRP2 4.7236 5.9157 4.3997 4.4661
U-87MG ATCC CTRP2 4.7603 8.3446 3.2535 9.1136
KNS-81 CTRP2 4.8322 9.2002 2.1831 7.6654
KNS-60 CTRP2 4.8433 10.7916 1.4022 11.0635
SNU-489 CTRP2 5.0417 6.0297 4.6523 2.6823
GaMG CTRP2; CTRP1 5.1371 6.5543 4.4758 3.2203
NMC-G1 CTRP2 5.344 6.7235 4.5615 2.4703
A-172 CTRP2 6.2358 17.9457 -0.3249 19.6187
⏷ Show the Full List of 43 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
AN3-CA CTRP2 1.1552 1.975 1.1552 26.9607
JHUEM-2 CTRP2; CTRP1 1.5292 3.3195 1.5115 24.5326
HEC-50B CTRP2 1.8472 2.8496 1.8416 16.6132
JHUEM-1 CTRP2 1.8852 2.3286 1.8852 22.1059
HEC-108 CTRP2; CTRP1 2.1118 4.5095 1.9911 21.0114
HEC-151 CTRP2; CTRP1 2.212 4.0555 2.1662 20.0874
HEC-6 CTRP2; CTRP1 2.2717 3.5837 2.2631 19.5645
JHUEM-7 CTRP2 2.4188 4.2704 2.3595 18.758
HEC-59 CTRP2; CTRP1 2.4288 4.5661 2.3232 18.8519
JHUEM-3 CTRP2 2.5277 4.434 2.4522 18.0902
HEC-251 CTRP2; CTRP1 2.8064 4.2989 2.768 16.1095
HEC-1-A CTRP2 2.8776 5.4556 2.5934 16.5087
RL95-2 CTRP2 2.9174 4.1875 2.8958 15.3145
HEC-265 CTRP2; CTRP1 2.9452 3.9324 2.9394 15.0766
MFE-319 CTRP2; CTRP1 2.9525 4.7757 2.8498 15.3608
HEC-1-B CTRP2 3.1962 6.0943 2.7201 15.1127
MFE-296 CTRP2 3.2013 4.7052 3.1321 13.59
ESS-1 CTRP2 3.2099 5.0863 3.0597 13.8184
KLE CTRP2; CTRP1 3.6496 5.3755 3.4591 11.0447
EN CTRP2 4.2005 5.6556 3.9609 7.5781
EFE-184 CTRP2 4.4492 5.7906 3.5789 2.1386
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 2.8895 3.9811 2.8803 15.4582
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ACHN CTRP2 1.7327 2.1915 1.7327 23.1199
UO-31 CTRP2 2.0755 3.6573 2.0572 20.9021
VMRC-RCZ CTRP2 2.7683 3.6478 2.7665 16.2397
786-O CTRP2 3.3429 5.3655 3.1278 13.1693
VMRC-RCW CTRP2; CTRP1 3.4986 5.1869 3.3484 11.9008
TUHR10TKB CTRP2 3.7504 4.3814 3.6409 3.4253
Caki-2 CTRP2 3.7664 5.9595 3.3811 11.0002
KMRC-1 CTRP2 3.8768 5.4407 3.686 9.5387
OS-RC-2 CTRP2 4.1579 6.516 3.5568 9.2677
SNU-1272 CTRP2 4.1866 5.3213 4.0608 7.2456
A-498 CTRP2 4.2799 5.6282 4.0562 6.9927
769-P CTRP2 4.4342 6.2417 3.9602 6.9554
KMRC-2 CTRP2 4.5004 8.5257 2.9288 11.0239
KMRC-3 CTRP2 4.6122 5.6718 4.3917 4.7879
Caki-1 CTRP2 4.6348 7.8292 3.3945 8.7989
KMRC-20 CTRP2 4.6973 5.7499 4.4469 4.6768
RCC10RGB CTRP2; CTRP1 4.8058 5.8828 4.497 3.8703
TUHR14TKB CTRP2 4.8404 8.3286 3.3325 8.6151
BFTC-909 CTRP2 5.0121 6.0921 4.5945 2.987
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 49 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW620 CTRP2; CTRP1 0.4479 1.2715 0.4479 31.6643
SW480 CTRP1 0.9507 2.0669 0.9504 60.8086
SNU-C1 CTRP2 1.6905 2.7185 1.69 23.4024
NCI-H716 CTRP2 1.8904 4.1336 1.8142 22.3296
LS411N CTRP2; CTRP1 1.9162 3.6241 1.894 21.9744
SNU-175 CTRP1 1.9639 3.4906 1.951 46.4124
HCT 116 CTRP2; CTRP1 1.9725 2.8179 1.9724 21.526
SW48 CTRP2; CTRP1 2.1433 2.9789 2.143 20.3908
SNU-C4 CTRP2; CTRP1 2.1994 3.6268 2.1869 20.0586
LS180 CTRP2; CTRP1 2.3506 3.6548 2.341 19.0432
LS513 CTRP2; CTRP1 2.4312 3.2839 2.4306 18.4772
SNU-C5 CTRP2; CTRP1 2.4938 3.8676 2.4778 18.1124
HCT 15 CTRP2 2.5316 4.2441 2.4829 17.9721
NCI-H747 CTRP2 2.5666 4.8458 2.4157 18.0947
LoVo CTRP2; CTRP1 2.588 3.7636 2.5801 17.459
DLD-1 CTRP2; CTRP1 2.6677 3.9638 2.6521 16.9546
GP2d CTRP2; CTRP1 2.6956 3.5071 2.6948 16.7196
SK-CO-1 CTRP2; CTRP1 2.7876 4.4824 2.7235 16.3228
KM12 CTRP2; CTRP1 2.8476 4.7768 2.7358 16.0896
COLO205 CTRP2; CTRP1 2.8495 4.8646 2.7193 16.1416
HT-55 CTRP2; CTRP1 2.9669 5.056 2.8022 15.4843
SNU-C2A CTRP2; CTRP1 3.0003 4.89 2.8777 15.113
COLO 320 CTRP2; CTRP1 3.1059 5.914 2.6891 15.4865
CW-2 CTRP2; CTRP1 3.1274 4.3159 3.1048 13.9215
SNU-81 CTRP1 3.2031 4.6776 3.1387 29.1276
HCT 8 CTRP2; CTRP1 3.4048 4.8001 3.3347 12.2404
RCM-1 [Human ESC] CTRP2; CTRP1 3.4738 5.949 3.0721 12.9959
COLO 678 CTRP2; CTRP1 3.4962 6.3166 2.9533 13.3875
SNU-1033 CTRP2 3.5251 5.6791 3.2245 12.2766
SW948 CTRP2; CTRP1 3.5296 5.2833 3.3554 11.7817
SNU-1040 CTRP1 3.5955 5.9647 3.1966 26.0634
SW403 CTRP1 3.5974 5.6266 3.3209 24.5887
LS123 CTRP2; CTRP1 3.6087 4.7908 3.5564 10.8231
SW1417 CTRP2 3.615 5.6853 3.3196 11.6621
SNU-407 CTRP2 3.6349 4.8933 3.3028 5.1777
SNU-503 CTRP2 3.9439 6.0195 3.5459 9.8775
LS1034 CTRP2 3.9468 5.739 3.6577 9.4424
NCI-H508 CTRP2; CTRP1 4.1118 5.0588 4.0491 7.5155
C2BBe1 CTRP2; CTRP1 4.2723 5.6022 4.0579 7.0078
HCC-56 CTRP2 4.3103 5.3197 4.1961 6.3825
SNU-61 CTRP2; CTRP1 4.3823 5.5188 4.2068 6.1332
RKO CTRP2; CTRP1 4.4665 5.4126 4.3353 5.4099
HT115 CTRP2; CTRP1 4.6931 5.5371 4.5318 4.0259
CL-34 CTRP1 4.7453 6.289 4.2468 10.8093
MDST8 CTRP2; CTRP1 4.8686 5.9996 4.5038 3.6901
HT-29 CTRP2; CTRP1 5.1167 5.8335 4.8171 1.834
CL-11 CTRP2 5.1194 7.005 3.4437 1.7519
OUMS-23 CTRP2 5.2809 6.1087 4.8178 1.5106
CL-40 CTRP1 5.6526 7.1042 4.6011 3.8974
⏷ Show the Full List of 49 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHH-5 CTRP2 1.4769 2.347 1.4768 24.8216
Hep 3B2.1-7 CTRP2 1.7831 6.0022 1.2271 24.7367
JHH-2 CTRP2 1.7881 3.0749 1.7847 22.7628
SNU-398 CTRP2; CTRP1 1.9366 4.5046 1.8025 22.2224
SNU-886 CTRP2 2.2338 5.2577 1.2868 11.6733
PLC/PRF/5 CTRP2 2.6516 5.6773 2.2775 18.3368
SK-HEP-1 CTRP2 2.8385 4.31 2.8007 15.8943
HLF CTRP2 2.905 5.192 2.6993 16.042
SNU-423 CTRP2 2.974 5.2501 2.7586 15.6189
JHH-4 CTRP2 3.0596 4.6966 2.9807 14.5655
SNU-387 CTRP2 3.3698 5.0812 3.2353 12.6999
SNU-449 CTRP2; CTRP1 3.5087 5.7241 3.1912 12.4484
SNU-182 CTRP2 3.5204 5.6352 3.2345 12.2532
JHH-1 CTRP2 3.7057 5.4891 3.4843 10.7859
SNU-878 CTRP2 3.8428 5.4102 3.6587 9.7397
SNU-761 CTRP2 3.9816 6.5357 2.8267 6.4556
Li-7 CTRP2 4.1125 6.0171 3.7247 8.7269
SNU-475 CTRP2 4.5453 5.1238 4.5061 4.5517
JHH-6 CTRP2; CTRP1 4.7112 4.9711 4.7078 3.3248
HuH-1 CTRP2 4.7861 6.2546 4.3026 4.7076
Hep-G2 CTRP2; CTRP1 5.0703 6.6773 4.3566 3.8556
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 155 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1341 CTRP2 0.5582 1.6762 0.5581 30.931
NCI-H1963 CTRP1 0.5724 2.192 0.5697 65.8446
NCI-H1930 CTRP1 0.6266 3.7415 0.5189 61.8534
NCI-H1155 CTRP2 1.3585 2.799 1.3548 25.6211
NCI-H1048 CTRP1 1.3833 2.5984 1.3822 53.4931
NCI-H810 CTRP2; CTRP1 1.4394 2.58 1.4386 25.0733
NCI-H82 CTRP1 1.5125 2.2278 1.5125 51.6985
NCI-H1573 CTRP1 1.5174 3.8805 1.4501 51.5165
NCI-H1092 CTRP2 1.525 3.6439 1.4836 24.6407
NCI-H211 CTRP2 1.5794 2.3308 1.5794 24.1394
NCI-H1869 CTRP2 1.5846 2.53 1.5844 24.1054
NCI-H1568 CTRP2; CTRP1 1.6131 3.7616 1.5649 24.0778
NCI-H1694 CTRP2; CTRP1 1.7047 3.5753 1.6774 23.3977
NCI-H2171 CTRP2 1.7113 2.8071 1.7104 23.2652
SBC-5 CTRP2 1.7651 2.1374 1.7651 22.905
NCI-H1563 CTRP2 1.7836 2.4387 1.7836 22.7817
NCI-H2029 CTRP2; CTRP1 1.8425 2.5182 1.8425 22.3899
RERF-LC-MS CTRP2 1.8742 2.9896 1.8728 22.1838
DMS 53 CTRP2 1.901 3.0994 1.8984 22.0097
NCI-H1581 CTRP2 1.9077 3.1537 1.9043 21.9678
VMRC-LCD CTRP2; CTRP1 1.9306 3.4106 1.9203 21.8385
LK2 CTRP2 1.9941 4.2504 1.9081 21.674
Lu-65 CTRP2; CTRP1 2.0303 3.895 1.9911 21.2731
SHP-77 CTRP2; CTRP1 2.0835 3.8638 2.05 20.8998
MOR/CPR CTRP2 2.1196 3.5856 2.1067 20.5907
NCI-H596 CTRP1 2.1427 3.3322 2.139 43.832
NCI-H1666 CTRP2; CTRP1 2.193 3.6318 2.1801 20.1025
NCI-H1395 CTRP2 2.2404 6.2898 1.6211 21.958
NCI-H661 CTRP2; CTRP1 2.2406 4.3463 2.1577 20.0242
SW1573 CTRP2 2.2529 3.9863 2.125 14.1702
DMS 273 CTRP2; CTRP1 2.372 3.5066 2.3678 18.8829
NCI-H841 CTRP2; CTRP1 2.3868 3.4046 2.3847 18.7772
DMS 454 CTRP2 2.4099 5.1993 2.157 19.4992
HCC2108 CTRP1 2.4141 4.0803 2.377 40.1593
EKVX CTRP2 2.4908 5.4954 2.1597 19.2451
Lu-99 CTRP2; CTRP1 2.5037 3.5892 2.4996 18.0067
NCI-H1703 CTRP2 2.5237 4.9163 2.3529 18.45
COR-L279 CTRP1 2.5298 3.3473 2.5292 37.4764
NCI-H2342 CTRP2; CTRP1 2.5705 5.3311 2.2954 18.5133
HCC44 CTRP2; CTRP1 2.5826 3.8886 2.5684 17.516
NCI-H1373 CTRP2; CTRP1 2.651 4.1375 2.6209 17.1146
NCI-H23 CTRP2; CTRP1 2.6593 4.9566 2.4911 17.5402
NCI-H2286 CTRP1 2.6616 4.0774 2.6374 35.7927
NCI-H1836 CTRP1 2.6854 4.3466 2.6336 36.4053
NCI-H2141 CTRP2; CTRP1 2.7638 4.0011 2.7493 16.312
NCI-H2196 CTRP2 2.7746 4.4067 2.7206 16.3743
NCI-H2087 CTRP2 2.7752 4.438 2.567 10.7584
NCI-H522 CTRP2; CTRP1 2.7778 5.3797 2.5074 17.1205
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 2.7874 4.5374 2.7148 16.3534
NCI-H2106 CTRP2 2.8131 5.2021 2.5962 16.6926
NCI-H1944 CTRP2; CTRP1 2.833 4.9305 2.6865 16.3091
NCI-H1355 CTRP2; CTRP1 2.8833 4.878 2.7531 15.9172
ChaGo-K-1 CTRP2; CTRP1 2.9156 5.7723 2.5326 16.6204
HCC78 CTRP2; CTRP1 2.9218 4.1035 2.9067 15.2632
NCI-H1435 CTRP1 2.9328 5.2449 2.7152 33.2942
NCI-H1876 CTRP1 2.944 4.3745 2.9051 32.6391
T3M-10 CTRP2; CTRP1 2.9481 4.8223 2.8354 15.4249
COLO 699 CTRP2; CTRP1 2.973 4.5795 2.9074 15.095
NCI-H1299 CTRP2; CTRP1 3.0175 4.6188 2.9488 14.81
NCI-H1437 CTRP1 3.0193 4.7521 2.9268 31.2722
DV-90 CTRP2; CTRP1 3.0207 4.1599 3.0057 14.6054
NCI-H1105 CTRP2; CTRP1 3.0424 5.0394 2.8887 14.9436
COLO 668 CTRP2; CTRP1 3.0555 5.4433 2.791 15.2563
NCI-H2081 CTRP2; CTRP1 3.0677 5.4093 2.8146 15.1337
NCI-H446 CTRP2 3.0697 4.7102 2.7881 8.9601
NCI-H647 CTRP2 3.1136 5.1352 2.942 14.5345
HOP-62 CTRP2 3.1205 5.1047 2.9575 14.4577
NCI-H526 CTRP2 3.1238 4.8507 3.0203 14.225
HCC15 CTRP2; CTRP1 3.1458 4.6025 3.0893 13.9148
LXF 289 CTRP2; CTRP1 3.1504 4.3652 3.1243 13.7802
NCI-H3255 CTRP1 3.1792 4.814 3.0879 29.6624
NCI-H2170 CTRP2 3.2186 5.1856 3.0433 13.8503
HCC4006 CTRP2; CTRP1 3.2233 4.5367 3.1817 13.3484
RERF-LC-Ad2 CTRP2 3.2303 6.3015 2.6772 15.1802
A-549 CTRP2; CTRP1 3.2659 5.0484 3.1301 13.3947
NCI-H1792 CTRP2; CTRP1 3.3436 5.2708 3.1561 13.0645
NCI-H2085 CTRP2 3.3607 5.6725 2.6706 8.6431
LUDLU-1 CTRP2 3.3661 5.4053 3.141 13.0517
HCC1438 CTRP2 3.382 5.1932 3.2195 12.7196
HOP-92 CTRP2 3.3826 5.3358 3.1799 12.8606
HCC2935 CTRP2; CTRP1 3.3883 4.8793 3.3014 12.4085
HCC2279 CTRP2 3.4088 5.2057 3.2454 12.5446
NCI-H520 CTRP2 3.4223 5.0829 3.2921 12.3362
SCLC-21H CTRP1 3.4398 4.5791 3.4067 25.5205
NCI-H358 CTRP2; CTRP1 3.4434 5.8724 3.0676 13.0991
NCI-H1651 CTRP2 3.4475 5.8604 3.0764 13.0543
IA-LM CTRP2 3.4552 5.6199 3.169 12.6864
Calu-3 CTRP2; CTRP1 3.4615 4.8498 3.3867 11.8797
LC-1/sq-SF CTRP2; CTRP1 3.4661 5.3403 3.2695 12.2844
DMS 114 CTRP2 3.4756 5.7652 3.1408 12.7322
NCI-H2009 CTRP2; CTRP1 3.4986 5.3147 3.3125 12.9467
COR-L95 CTRP2 3.5221 6.3394 2.9715 13.2465
NCI-H1755 CTRP2; CTRP1 3.5427 5.2351 3.3834 11.641
NCI-H2405 CTRP2; CTRP1 3.549 5.1929 3.4018 11.5554
Calu-6 CTRP2; CTRP1 3.5582 4.6772 3.5199 11.1104
HCC1833 CTRP2; CTRP1 3.5688 5.8687 3.2038 12.229
NCI-H1184 CTRP2 3.5914 5.0934 3.1679 5.8762
RERF-LC-A1 CTRP2 3.6023 4.7528 3.5558 10.8455
KNS-62 CTRP2; CTRP1 3.6287 5.1205 3.5078 10.9318
COR-L51 CTRP1 3.6427 5.2243 3.4955 23.482
NCI-H1793 CTRP2; CTRP1 3.6575 5.9125 3.2827 11.6796
NCI-H441 CTRP1 3.6678 6.26 3.1573 25.8971
COR-L105 CTRP2 3.6751 6.2303 3.177 12.0353
NCI-H727 CTRP2; CTRP1 3.6991 6.461 3.1071 12.2416
PC-14 CTRP2 3.7212 6.1925 2.764 7.3311
NCI-H2228 CTRP2 3.7347 6.0787 2.8323 6.9946
NCI-H1975 CTRP1 3.7425 6.0037 3.3385 23.5574
NCI-H838 CTRP2 3.7692 5.4453 3.5674 10.2928
NCI-H1339 CTRP2 3.7782 5.4702 3.5693 10.2593
HCC33 CTRP1 3.7808 4.9565 3.7114 20.4795
HCC827 CTRP2; CTRP1 3.8064 5.234 3.6715 9.802
SK-MES-1 CTRP2 3.8288 5.3478 3.6628 9.7662
COR-L88 CTRP1 3.8379 5.6216 3.5828 21.0942
LCLC-97TM1 CTRP2; CTRP1 3.8514 5.0113 3.7765 9.2889
HCC1195 CTRP2; CTRP1 3.8569 5.3144 3.7035 9.5338
RERF-LC-KJ CTRP1 3.866 5.3438 3.7045 19.9819
NCI-H460 CTRP2; CTRP1 3.888 5.3302 3.7326 9.3351
NCI-H2110 CTRP2; CTRP1 3.9002 6.4467 3.3225 10.8641
HCC1588 CTRP2 3.9688 4.6813 3.955 8.2966
NCI-H2023 CTRP2; CTRP1 3.9771 5.4939 3.7774 8.9068
NCI-H2122 CTRP2; CTRP1 3.9975 5.0429 3.9283 8.298
NCI-H2073 CTRP1 4.0009 6.2428 3.5138 21.1053
NCI-H196 CTRP2 4.0109 5.6705 3.7518 8.9052
EPLC-272H CTRP2; CTRP1 4.022 5.2483 3.9028 8.3139
NCI-H2030 CTRP2; CTRP1 4.0326 5.8634 3.7019 9.034
EBC-1 CTRP2; CTRP1 4.0332 5.1657 3.9374 8.1555
HCC95 CTRP2 4.0408 6.4861 3.4504 10.7525
HCC366 CTRP2 4.0587 6.4742 3.474 9.8522
NCI-H1650 CTRP2 4.0688 6.0891 3.1248 4.9242
NCI-H292 CTRP2 4.0785 5.5031 3.8842 8.2149
LCLC-103H CTRP2; CTRP1 4.1146 4.9385 4.0761 7.412
NCI-H1623 CTRP2 4.1391 8.1005 2.7975 12.3847
NCI-H1838 CTRP2 4.1616 6.4969 3.5692 9.209
CAL-12T CTRP2; CTRP1 4.267 5.6137 4.0479 7.0606
NCI-H226 CTRP2 4.2767 5.7056 3.4891 2.8546
SW1271 CTRP2 4.3124 6.574 3.0845 4.6055
LOU-NH91 CTRP2 4.3204 5.5422 3.6048 2.252
HCC1359 CTRP1 4.3685 4.9658 4.3449 12.1864
Calu-1 CTRP2 4.3715 8.6278 2.76 12.0057
NCI-H1781 CTRP1 4.3897 5.406 4.2544 12.7478
NCI-H322 CTRP2 4.4083 7.1283 3.5215 8.7932
SK-LU-1 CTRP2; CTRP1 4.4215 5.2936 4.3251 5.5798
NCI-H650 CTRP2; CTRP1 4.4404 6.0397 4.0562 6.5584
NCI-H1915 CTRP2; CTRP1 4.4514 5.5619 4.2649 5.7183
NCI-H2291 CTRP2 4.5781 6.3885 4.0365 6.2899
NCI-H2444 CTRP2 4.5887 7.6416 2.7695 5.4963
COR-L23 CTRP1 4.69 6.2707 4.2017 11.4883
NCI-H2126 CTRP2; CTRP1 4.8098 6.7838 4.0686 5.6167
NCI-H889 CTRP2 4.9135 6.4394 3.5787 1.4623
NCI-H2172 CTRP1 4.9646 6.1181 4.5378 7.1492
Sq-1 CTRP2; CTRP1 5.1404 6.7959 4.358 3.7079
RERF-LC-Ad1 CTRP2 5.198 5.9879 4.8106 1.6956
HCC1171 CTRP2 5.378 8.3422 3.7813 5.6751
BEN CTRP2; CTRP1 5.4527 8.9019 3.5618 6.4577
Hs 888.Lu CTRP2 3.5359 8.5853 1.983 17.1031
⏷ Show the Full List of 155 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 1.953 3.6403 1.9312 21.728
P-STS CTRP2 2.6883 4.5092 2.6128 17.0224
SYO-1 CTRP2 4.7669 5.5224 4.6158 3.5002
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 3.0038 5.0858 2.835 15.2536
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 4.239 6.139 3.8054 8.074
OVKATE CTRP1 -0.0969 1.5817 -0.0984 74.6874
TOV-21G CTRP2 1.304 2.0641 1.304 25.9709
TOV-112D CTRP2 1.744 3.0823 1.7399 23.0588
OVCAR-5 CTRP2 1.7924 3.3643 1.7804 22.7633
RMUG-S CTRP1 2.2326 4.7239 2.0792 43.1994
COV434 CTRP2; CTRP1 2.4126 3.9966 2.3834 18.6973
A2780 CTRP2; CTRP1 2.5421 3.6613 2.5367 17.7557
DOV13 CTRP2 2.5668 5.3387 2.2891 18.547
OC 314 CTRP2 2.587 4.2184 2.5448 17.5814
OVCAR-4 CTRP2; CTRP1 2.6216 4.6965 2.507 17.6017
OVK18 CTRP2; CTRP1 2.6305 4.0924 2.6035 17.2404
OV-90 CTRP2; CTRP1 2.714 4.4017 2.6566 16.7892
TYK-nu CTRP2; CTRP1 2.7633 4.2189 2.7311 16.3754
HEY A8 CTRP2; CTRP1 2.8036 3.6488 2.8021 16.0039
ONCO-DG-1 CTRP2 2.9776 8.4067 1.5109 20.34
OV56 CTRP2 3.2393 4.8404 3.1477 13.4158
SNU-119 CTRP2 3.2849 5.1732 3.119 13.3764
JHOM-1 CTRP2; CTRP1 3.3298 4.7715 3.259 12.7413
Kuramochi CTRP2 3.5812 7.8569 2.367 15.4716
SK-OV-3 CTRP2; CTRP1 3.5987 4.9935 3.5055 11.0325
IGROV-1 CTRP2; CTRP1 3.6077 5.7236 3.2983 11.7627
OVMANA CTRP1 3.685 4.5634 3.6677 21.44
OVSAHO CTRP2 3.685 5.4791 3.4651 10.9177
OV7 CTRP2; CTRP1 3.7253 5.4984 3.5026 10.6609
JHOS-2 CTRP2 3.7763 6.4374 3.1977 11.6819
RMG-I CTRP2; CTRP1 3.7812 6.557 3.1519 11.8478
MCAS CTRP2 3.8067 4.4454 3.675 3.1178
JHOS-4 CTRP1 3.8562 5.1868 3.7388 19.7838
OAW28 CTRP2 3.8571 5.7302 3.5646 10.0488
SNU-840 CTRP2; CTRP1 3.9398 7.371 2.9482 12.2537
COV362 CTRP2; CTRP1 3.9552 6.4355 3.3842 10.477
Caov-3 CTRP2; CTRP1 4.0443 4.9195 4.0037 7.8869
JHOC-5 CTRP2; CTRP1 4.0755 5.2127 3.971 7.9056
SNU-8 CTRP2 4.1005 4.9729 4.0546 8.105
EFO-27 CTRP2; CTRP1 4.2444 6.4557 3.6717 8.5893
OVCAR-8 CTRP2; CTRP1 4.27 5.8519 3.958 7.3965
OVISE CTRP2 4.4936 5.8023 4.2132 5.8016
OVTOKO CTRP2 4.4953 5.9509 4.1514 6.0391
ES2 CTRP2 4.5691 5.7448 4.3161 5.198
COV644 CTRP2; CTRP1 4.583 5.8015 4.3066 5.1982
OAW42 CTRP2; CTRP1 4.6916 5.5591 4.5215 4.0698
EFO-21 CTRP2; CTRP1 4.7178 6.4042 4.1654 5.4298
COV318 CTRP1 5.1672 7.0959 4.2307 8.8042
FU-OV-1 CTRP2 6.2207 20.1764 -2.1951 21.226
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 4.8596 5.3638 4.7767 2.6268
Aska-SS CTRP2 4.9568 5.5628 4.7947 2.2971
KYM-1 CTRP2 1.6025 2.1713 1.6025 23.9859
SK-UT-1 CTRP2 1.6333 3.4213 1.6134 23.8478
GCT CTRP2 1.7307 3.3027 1.7197 23.1702
Rh41 CTRP2 1.8354 2.463 1.8354 24.1459
A-204 CTRP2 2.2547 4.0972 2.2066 19.8112
G-402 CTRP2 2.3392 4.0388 2.3022 19.2115
G-401 CTRP2; CTRP1 2.4006 3.8295 2.3835 18.7359
MES-SA CTRP2 2.9184 4.5824 2.8482 15.4743
SK-LMS-1 CTRP2 3.0713 4.8018 2.9734 14.5544
HT-1080 CTRP2; CTRP1 3.0962 4.2139 3.0804 14.1059
RD CTRP2 3.1662 5.9782 2.7308 15.1574
TTC-709 CTRP2 3.7124 5.0731 3.6108 10.3068
Rh18 CTRP2 3.7564 4.2411 3.6974 3.1791
TE 617.T CTRP2 3.821 5.2609 3.6798 9.728
RKN CTRP2; CTRP1 4.28 4.8799 4.2625 6.24
BT-16 CTRP2 4.2826 5.3878 4.1442 6.6555
Hs 729.T CTRP2 4.3445 6.9342 3.5513 8.825
BT-12 CTRP2 4.5943 6.1808 4.1489 5.7966
Tm87-16 CTRP2 4.7559 5.8986 4.4399 4.2238
TE 441.T CTRP2 4.8978 5.4905 4.766 2.5635
SW982 CTRP2 5.1954 6.3423 4.6312 2.4532
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2; CTRP1 2.4199 3.3859 2.4184 18.5552
NCI-H28 CTRP2; CTRP1 3.1442 6.1847 2.6304 15.599
NCI-H2052 CTRP2; CTRP1 3.4734 4.7687 3.4144 11.7455
NCI-H2452 CTRP2 4.0754 7.9565 2.1973 9.0838
IST-Mes1 CTRP2 4.2846 6.5018 3.6915 8.4079
ACC-MESO-1 CTRP2 4.4298 5.6 4.2272 5.9219
JL-1 CTRP2 4.6098 5.0877 4.5838 4.0766
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LNCaP clone FGC CTRP2 2.696 4.4231 2.6343 16.9234
DU145 CTRP2 2.7778 4.6147 2.6912 16.4659
NCI-H660 CTRP2 2.7815 4.7092 2.6777 16.5011
PaCa-3 CTRP2; CTRP1 3.792 4.8737 3.7396 9.6047
22Rv1 CTRP2 3.8548 6.0047 3.4575 10.4624
VCaP CTRP2 4.0024 5.0838 3.9243 8.2968
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 CTRP2 3.6627 6.9426 2.8621 13.2992
YD-15 CTRP2 4.1046 4.816 4.0839 7.4174
Cancer Drug Sensitivity Data Curated from 32 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-16 CTRP2 1.029 1.7593 1.029 27.7998
HGC-27 CTRP2 1.536 2.6669 1.5352 24.4311
SNU-1 CTRP2 1.6352 2.366 1.6352 23.7684
SNU-601 CTRP2 1.8283 2.4169 1.8283 22.4845
SNU-620 CTRP2 2.0081 3.3817 2.0007 21.3135
GSS CTRP2 2.0608 3.6388 2.0431 20.9979
LMSU CTRP2 2.4765 3.5229 2.4735 18.1841
HuG1-N CTRP2 2.4838 4.5741 2.3811 18.4763
IM95 CTRP2 2.8571 4.9286 2.7131 16.1399
Fu97 CTRP2; CTRP1 2.9516 4.3555 2.9153 15.137
SNU-5 CTRP2 3.0709 4.956 2.9396 14.6743
MKN1 CTRP2 3.2198 5.6204 2.9134 14.3209
NUGC-4 CTRP2; CTRP1 3.3177 4.5998 3.2737 12.7291
MKN74 CTRP2; CTRP1 3.3343 6.0958 2.8675 14.1649
SNU-216 CTRP2 3.3492 5.9863 2.9246 13.9065
SNU-719 CTRP2 3.4192 5.3063 3.2285 12.5743
ECC10 CTRP2 3.4541 4.7569 3.1762 6.2218
23132/87 CTRP2 3.4669 4.6203 3.4302 12.6038
KE-39 CTRP2 3.473 6.0653 3.0273 13.1682
MKN7 CTRP2; CTRP1 3.4757 4.9277 3.3862 11.837
NCC-StC-K140 CTRP2 3.7467 5.7105 3.4528 10.7845
NUGC-3 CTRP2 3.8686 4.7707 3.5923 3.3027
NCI-N87 CTRP2 4.0624 5.5855 3.838 8.434
SH-10-TC CTRP2; CTRP1 4.1301 5.8764 3.8003 8.3875
SNU-668 CTRP2 4.1925 5.7724 3.9076 7.803
ECC12 CTRP2 4.2336 5.7393 3.9643 8.041
AGS CTRP2; CTRP1 4.2544 5.0577 4.2044 6.5231
Hs 746.T CTRP2 4.7449 5.256 4.689 3.2863
MKN45 CTRP2 5.3676 7.5235 4.1814 4.018
SNG-M CTRP2; CTRP1 3.4479 4.6836 3.4009 11.8736
SNU-1077 CTRP2 3.5636 4.5432 3.5419 11.0179
SNU-685 CTRP2 3.7243 5.3313 3.5538 10.4763
⏷ Show the Full List of 32 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
FTC-133 CTRP2 2.8355 4.9711 2.6797 16.3254
FTC-238 CTRP2 2.9655 4.4904 2.9128 15.1009
8505C CTRP2 3.0439 4.5234 2.9919 14.5769
B-CPAP CTRP2 3.1491 5.4677 2.8855 15.7465
TT CTRP2 3.5984 4.9776 3.5087 11.0223
CGTH-W-1 CTRP2 3.7415 6.2107 3.2551 12.4322
SW579 CTRP2 3.782 5.615 3.5246 10.414
CAL-62 CTRP2 3.7969 4.8663 3.7462 9.5662
8305C CTRP2 4.9137 6.5952 4.2569 4.6054
ML-1 [Human leukemia] CTRP2 4.9921 7.9438 2.9165 4.1574
TT2609-C02 CTRP2 5.2685 8.9918 3.3672 7.6147
BHT-101 CTRP2 5.3676 6.4173 4.7317 1.7196
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SCC-4 CTRP2 2.0555 5.1569 1.7817 21.926
FaDu CTRP2 2.2885 3.9068 2.2611 19.516
HSC-2 CTRP2; CTRP1 2.778 3.8278 2.7722 16.1883
PE/CA-PJ15 CTRP2 2.9202 4.8988 2.7885 15.6774
PE/CA-PJ34 (clone C12) CTRP2 3.1248 4.9449 3.0008 14.2907
HSC-3 CTRP2 3.3161 5.1816 3.1508 13.167
PE/CA-PJ49 CTRP2 3.4349 5.3819 3.2231 12.5468
YD-10B CTRP2 3.5977 5.1638 3.4628 11.1878
SNU-1214 CTRP2 3.6187 5.2523 3.4615 11.1287
SNU-46 CTRP2 3.6941 6.113 3.2441 11.725
CAL-27 CTRP2 3.8427 5.1485 3.734 9.4668
SNU-1041 CTRP2 3.8668 5.0844 3.7763 9.2417
BICR 6 CTRP2 3.8704 5.6417 3.6109 9.8366
CAL-33 CTRP2 3.8704 6.1239 3.4262 10.5404
HSC-4 CTRP2 3.8821 5.2287 3.3849 4.1827
SNU-1076 CTRP2 3.9067 4.7707 3.879 8.757
SNU-899 CTRP2 3.9789 5.5467 3.7614 8.9614
SCC-25 CTRP2 4.059 5.3373 3.4914 3.2962
PE/CA-PJ41 (clone D2) CTRP2 4.1028 6.2387 3.6215 9.1557
SCC-9 CTRP2; CTRP1 4.2694 5.3207 4.1512 6.6685
BICR 22 CTRP2 4.3284 5.7544 4.059 6.8472
SNU-1066 CTRP2 4.3719 5.6126 4.1606 6.3376
BHY CTRP2 4.4411 5.7922 4.1625 6.6073
YD-8 CTRP2 4.5615 7.6092 2.7648 5.5676
BICR 18 CTRP2 4.6323 6.6425 3.9693 6.4335
BICR 56 CTRP2 4.7502 5.5501 4.5868 3.658
BICR 31 CTRP2 4.9885 8.194 3.5293 7.4865
BICR 16 CTRP2 5.2302 6.7552 4.4538 3.1306
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UM-UC-1 CTRP2 1.627 2.4142 1.627 23.8232
UM-UC-3 CTRP2; CTRP1 1.8582 3.1846 1.8535 22.3013
SCaBER CTRP2 1.9284 2.5283 1.9284 21.8191
HT-1376 CTRP2; CTRP1 2.2098 3.5681 2.2002 19.9797
HT-1197 CTRP2 2.3239 3.8075 2.3054 19.2508
RT-4 CTRP2; CTRP1 2.4571 3.5085 2.4541 18.313
KMBC-2 CTRP2; CTRP1 2.6388 4.0213 2.618 17.1647
5637 CTRP2; CTRP1 2.7089 4.4786 2.6397 16.8636
J82 CTRP2 2.9085 6.242 2.3565 17.3002
BC-3C CTRP2 3.0945 5.9313 2.6706 15.5884
639V CTRP2 3.4853 5.2342 3.321 12.0397
T24 CTRP2 3.4948 5.368 3.2926 12.1142
JMSU-1 CTRP2 3.5413 5.3812 3.3393 12.704
253J CTRP2 3.6254 4.5008 3.6108 10.5828
VM-CUB-1 CTRP2 3.7055 5.9149 3.3331 11.3535
U-BLC1 CTRP2 3.7758 5.7134 3.4832 10.5868
TCCSUP CTRP2 3.8783 5.9932 3.487 10.2845
RT-112 CTRP2 4.2337 5.2181 3.698 1.9986
647V CTRP2 4.2645 5.4322 4.1098 6.8354
BFTC-905 CTRP2 4.3592 5.5921 4.1548 6.3953
KU-19-19 CTRP2 4.4794 6.3537 3.9547 6.8637
CAL-29 CTRP2 4.7228 5.8038 4.4493 4.2704
253J-BV CTRP2 4.8113 6.2193 4.3437 4.4802
SW1710 CTRP2 7.0032 8.855 3.5713 0.2052
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 4.2155 5.3894 4.0708 7.1233

References

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