General Information of Drug (ID: DMPE7DQ)

Drug Name
STF-62247
Synonyms Renal cell carcinoma therapy, Stanford University
Indication
Disease Entry ICD 11 Status REF
Renal cell carcinoma 2C90 Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
Chemical Identifiers
Formula
C15H13N3S
Canonical SMILES
CC1=CC(=CC=C1)NC2=NC(=CS2)C3=CC=NC=C3
InChI
1S/C15H13N3S/c1-11-3-2-4-13(9-11)17-15-18-14(10-19-15)12-5-7-16-8-6-12/h2-10H,1H3,(H,17,18)
InChIKey
KATNUHQNJGNLPW-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
704473
ChEBI ID
CHEBI:125656
CAS Number
315702-99-9
TTD ID
D01CIN
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1 4.7554 8.2269 1.9647 6.7687
EW-24 GDSC1 3.2929 4.7757 2.593 6.2515
CHSA0108 GDSC1 3.3747 4.5736 2.7628 4.6126
ES7 GDSC1 3.6702 5.6734 2.4477 6.1032
ES5 GDSC1 3.7564 7.7698 1.4734 13.2325
EW-13 GDSC1 3.8865 8.6452 1.1395 15.1308
EW-7 GDSC1 3.9714 5.8679 2.5687 4.3034
ES6 GDSC1 4.4085 8.2846 1.7043 9.5443
ES1 GDSC1 4.455 6.4573 2.5974 2.9831
EW-1 GDSC1 4.554 7.5473 2.155 5.8922
A-673 GDSC1 4.7245 6.3746 2.7772 1.4069
NOS-1 [Human HNSCC] GDSC1 4.7395 8.5154 1.8182 7.8477
TC-71 GDSC1 4.7968 7.1553 2.4803 3.1124
SK-ES-1 GDSC1 4.9463 9.2122 1.6237 8.6906
ES8 GDSC1 5.2291 10.8188 1.0466 11.7943
HOS GDSC1 5.2586 6.563 2.9327 0.2952
CAL-78 GDSC1 5.2926 13.3154 -0.1164 18.2118
H-EMC-SS GDSC1 5.4345 9.1308 1.9618 5.3134
MG-63 GDSC1 5.4418 6.8759 2.8905 0.3273
ES4 GDSC1 5.4568 9.846 1.6499 7.3238
SK-PN-DW GDSC1 5.4832 7.702 2.5966 1.4487
HuO-3N1 GDSC1 5.492 7.5807 2.6483 1.1941
CAL-72 GDSC1 5.531 7.2289 2.7977 0.5621
CHSA0011 GDSC1 5.551 8.4881 2.306 2.9492
U2OS GDSC1 5.6841 7.9587 2.5853 1.2978
SaOS-2 GDSC1 5.7253 7.3504 2.8286 0.3682
MHH-ES-1 GDSC1 5.7665 7.6931 2.7207 0.6798
CADO-ES1 GDSC1 5.9173 7.6517 2.7938 0.3774
NY GDSC1 5.937 8.5012 2.485 1.5145
EW-16 GDSC1 5.9615 10.4083 1.6917 6.0321
CHSA8926 GDSC1 5.9667 7.5691 2.8405 0.2508
SJSA-1 GDSC1 6.1326 7.7692 2.831 0.2212
HuO9 GDSC1 6.2205 8.3612 2.6554 0.6271
EW-18 GDSC1 6.2268 8.096 2.752 0.358
G-292 clone A141B1 GDSC1 6.3333 8.848 2.5212 1.0226
EW-3 GDSC1 6.3817 8.5369 2.6541 0.5483
EW-11 GDSC1 6.791 9.1578 2.5875 0.5436
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 144 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JM1 GDSC1 4.5077 7.0097 2.3766 4.4113
SU-DHL-5 GDSC1 0.8206 4.4732 0.22 35.0229
EoL-1 GDSC1 0.8281 3.516 0.552 33.2498
DB GDSC1 0.9834 3.982 0.5723 32.1473
BE-13 GDSC1 1.5277 7.9092 -0.5793 34.2658
Karpas-299 GDSC1 1.9861 3.4523 1.8336 18.1328
ATN-1 GDSC1 2.0294 4.728 1.3929 21.0048
SUP-M2 GDSC1 2.2863 5.7271 1.1931 21.1416
DND-41 GDSC1 2.3098 6.7912 0.7041 24.2115
BC-3 GDSC1 2.3583 3.8786 2.0904 14.3077
RPMI-6666 GDSC1 2.5918 7.974 0.3829 24.8161
NALM-6 GDSC1 2.6867 10.3754 -0.7259 29.6251
YT GDSC1 2.7428 4.1978 2.3565 10.4282
OCI-M1 GDSC1 2.7523 4.682 2.1411 12.0169
SU-DHL-6 GDSC1 2.7898 6.6951 1.194 18.8835
THP-1 GDSC1 2.819 5.292 1.9109 13.4867
NU-DUL-1 GDSC1 2.8554 10.7064 -0.7442 29.0324
MOLM-13 GDSC1 2.9084 9.8824 -0.2872 26.8836
ST486 GDSC1 3.065 9.8934 -0.1581 25.6659
HC-1 GDSC1 3.1309 5.7062 1.9885 11.6112
SR GDSC1 3.1525 5.0717 2.3233 8.9132
WIL2 NS GDSC1 3.2585 4.465 2.7184 5.3948
ML-2 GDSC1 3.293 6.2806 1.8409 12.1312
K-562 GDSC1 3.3021 5.1361 2.4207 7.5747
LP-1 GDSC1 3.3576 4.9115 2.5797 6.1185
A3/Kawakami GDSC1 3.4098 4.5771 2.7898 4.2759
ALL-PO GDSC1 3.4244 5.5135 2.3338 7.8168
MHH-PREB-1 GDSC1 3.4387 9.2305 0.4874 20.8267
P12-Ichikawa GDSC1 3.4602 6.8138 1.7133 12.4905
Karpas-45 GDSC1 3.4607 8.3745 0.9335 17.9953
TUR GDSC1 3.4708 5.869 2.1939 8.7511
RPMI-8402 GDSC1 3.5354 9.0653 0.6495 19.5092
GR-ST GDSC1 3.582 5.9967 2.2191 8.1748
SU-DHL-10 GDSC1 3.6124 6.5577 1.9636 10.0541
P31/FUJ GDSC1 3.6381 5.4321 2.5427 5.4636
AMO1 GDSC1 3.66 9.3024 0.6323 19.1659
HEL GDSC1 3.6889 7.2157 1.6962 11.8236
CTV-1 GDSC1 3.7203 9.8259 0.4195 20.2036
NOMO-1 GDSC1 3.7413 4.9937 2.8319 2.9304
KY821 GDSC1 3.7553 5.7895 2.454 5.7921
697 GDSC1 3.7744 6.9812 1.8793 10.1606
BL-41 GDSC1 3.8017 7.9879 1.4003 13.6041
KMOE-2 GDSC1 3.8263 8.6327 1.0987 15.6091
P32/ISH GDSC1 3.8561 6.4774 2.19 7.5248
L-363 GDSC1 3.8708 8.5072 1.196 14.7995
EB2 GDSC1 3.9567 7.0399 1.9876 8.7652
OCI-AML-2 GDSC1 3.977 10.2158 0.429 19.2685
KG-1 GDSC1 3.9834 5.4677 2.7661 2.8116
LAMA-84 GDSC1 4.013 11.8805 -0.3718 23.2853
SIG-M5 GDSC1 4.0222 8.5094 1.3114 13.5054
MOLT-13 GDSC1 4.0298 8.2918 1.4248 12.684
ALL-SIL GDSC1 4.0371 6.9653 2.0828 7.8041
LC4-1 GDSC1 4.0438 9.8158 0.68 17.5623
CESS GDSC1 4.0586 6.154 2.4904 4.6622
KOPN-8 GDSC1 4.1353 6.4158 2.4168 5.0134
P30/OHK GDSC1 4.1446 5.7999 2.7121 2.834
KE-37 GDSC1 4.1525 7.4356 1.936 8.573
SUP-B15 GDSC1 4.1533 7.8364 1.7407 10.0181
SU-DHL-16 GDSC1 4.182 5.5916 2.8285 1.9549
HH [Human lymphoma] GDSC1 4.1901 13.6264 -1.1016 25.7922
SU-DHL-1 GDSC1 4.2039 5.4164 2.9172 1.3445
U266B1 GDSC1 4.2091 6.4598 2.4446 4.6212
Karpas-620 GDSC1 4.2326 5.8274 2.7519 2.373
Sc-1 GDSC1 4.2458 8.5151 1.4753 11.6566
MY-M12 GDSC1 4.2498 7.6816 1.8853 8.6705
VAL GDSC1 4.2997 9.3771 1.0912 14.1265
JSC-1 GDSC1 4.3155 8.7866 1.393 12.0259
CCRF-CEM GDSC1 4.3263 6.3161 2.5853 3.3342
OCI-Ly19 GDSC1 4.3602 8.0149 1.8011 8.9773
OCI-AML-5 GDSC1 4.3702 13.0802 -0.6888 23.5593
NB4 GDSC1 4.3846 6.8969 2.3519 4.8725
BC-1 GDSC1 4.3891 8.0967 1.7817 9.0381
JJN-3 GDSC1 4.4041 6.7471 2.4341 4.2352
Loucy GDSC1 4.4121 9.3451 1.1896 13.1291
HAL-01 GDSC1 4.4193 10.7441 0.5064 17.3942
OCI-AML-3 GDSC1 4.4259 8.7719 1.4797 11.0942
EJM GDSC1 4.4896 6.5658 2.5685 3.1105
Farage GDSC1 4.5221 7.1628 2.3145 4.821
KCL-22 GDSC1 4.5318 7.4374 2.1923 5.6759
SCC-3 GDSC1 4.5576 6.1282 2.797 1.5258
MC116 GDSC1 4.5635 5.5879 3.0158 0.4216
DEL GDSC1 4.5671 5.4996 3.0499 0.2973
JVM-2 GDSC1 4.59 10.6585 0.6753 15.8739
HT GDSC1 4.6143 7.5855 2.1754 5.6017
TK [Human B-cell lymphoma] GDSC1 4.6182 6.3656 2.7275 1.8498
SK-MM-2 GDSC1 4.6281 10.8039 0.6318 16.0214
L-1236 GDSC1 4.6298 7.0046 2.4523 3.6222
Daudi GDSC1 4.6456 6.7156 2.5903 2.6688
Karpas-422 GDSC1 4.6642 6.3705 2.749 1.652
EM-2 GDSC1 4.673 6.9477 2.5028 3.1958
JVM-3 GDSC1 4.681 7.5179 2.2484 4.9313
MN-60 GDSC1 4.6861 6.7529 2.5962 2.5588
Raji GDSC1 4.6983 7.418 2.3049 4.4983
RPMI-8226 GDSC1 4.7125 7.0364 2.4857 3.2345
SU-DHL-8 GDSC1 4.7135 6.1005 2.8829 0.8691
SUP-T1 GDSC1 4.7137 7.3164 2.3604 4.0815
RPMI-8866 GDSC1 4.7228 8.9777 1.5866 9.5221
KMS-12-BM GDSC1 4.7233 7.6577 2.2098 5.1093
Reh GDSC1 4.7339 10.3455 0.9325 13.8628
SUP-HD1 GDSC1 4.7471 7.8649 2.1286 5.6277
OPM-2 GDSC1 4.7929 10.6712 0.8159 14.423
RS4;11 GDSC1 4.8201 6.4638 2.7866 1.2356
CA46 GDSC1 4.8348 7.152 2.5028 2.8984
SU-DHL-4 GDSC1 4.8491 6.5651 2.7591 1.3461
JURL-MK1 GDSC1 4.8554 9.6016 1.3773 10.6096
MEG-01 GDSC1 4.8697 10.8245 0.7958 14.3281
PF-382 GDSC1 4.8722 6.7189 2.7071 1.6015
L-540 GDSC1 4.8848 6.545 2.784 1.1731
ROS-50 GDSC1 4.9141 9.3283 1.5473 9.2972
U-698-M GDSC1 4.9154 11.1805 0.655 15.0499
MOLT-4 GDSC1 4.9243 12.621 -0.0433 18.875
RC-K8 GDSC1 4.9333 6.8152 2.6971 1.576
KMS-11 GDSC1 4.9604 9.3348 1.5748 8.9913
QIMR-WIL GDSC1 4.9605 8.3139 2.0524 5.6831
ARH-77 GDSC1 4.9783 8.8669 1.8069 7.3453
MV4-11 GDSC1 4.9826 11.0432 0.7692 14.175
BALL-1 GDSC1 5.0007 10.0108 1.2795 10.8804
WSU-NHL GDSC1 5.0025 7.3806 2.4937 2.6714
MOLP-8 GDSC1 5.0532 6.3851 2.9178 0.4475
PL-21 GDSC1 5.066 11.2006 0.7513 14.0538
BV-173 GDSC1 5.123 7.0118 2.7069 1.2946
MOLT-16 GDSC1 5.1542 6.7316 2.8298 0.7049
Ramos.2G6.4C10 GDSC1 5.1584 6.457 2.9327 0.342
WSU-DLCL2 GDSC1 5.2712 6.4671 2.9709 0.1987
H9 GDSC1 5.2812 8.1226 2.3215 3.2819
HL-60 GDSC1 5.2964 6.3981 3.0034 0.1295
Mono-Mac-6 GDSC1 5.3083 15.1672 -1.0119 22.1983
KM-H2 GDSC1 5.326 8.0547 2.3743 2.8857
ME1 GDSC1 5.3368 6.7325 2.902 0.3437
RL GDSC1 5.4148 11.5854 0.8049 12.8096
Ku812 GDSC1 5.4296 7.093 2.8073 0.5927
DG-75 GDSC1 5.5603 7.7859 2.5981 1.3605
A4/Fukuda GDSC1 5.5649 6.9924 2.895 0.2667
Hs 445 GDSC1 5.5718 6.9599 2.9089 0.2333
HDLM-2 GDSC1 5.6385 7.633 2.6909 0.8827
L-428 GDSC1 5.684 7.3638 2.8083 0.4443
Granta-519 GDSC1 5.7026 7.8918 2.6193 1.1288
Namalwa GDSC1 5.7419 7.5063 2.7792 0.5016
VL51 GDSC1 5.8132 7.8885 2.6671 0.8445
NKM-1 GDSC1 6.0447 15.5083 -0.6514 18.7721
Jiyoye GDSC1 6.0594 7.7849 2.7993 0.3092
CTB-1 GDSC1 6.136 8.2559 2.6607 0.6578
GDM-1 GDSC1 7.1793 18.7687 -1.4439 19.3839
MLMA GDSC1 7.2698 19.7411 -1.8488 20.6493
⏷ Show the Full List of 144 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OACP4 C GDSC1 4.1682 15.7244 -2.165 29.4076
KYSE-50 GDSC1 4.7208 6.5012 2.7226 1.7243
FLO-1 GDSC1 5.1797 8.2529 2.2086 4.1842
KYAE-1 GDSC1 5.316 7.0978 2.7587 0.8661
ESO-51 GDSC1 5.4909 15.596 -1.0887 22.0203
KYSE-220 GDSC1 5.5742 7.5688 2.6883 0.9451
ESO-26 GDSC1 5.7706 7.6111 2.7524 0.5703
HCE-4 GDSC1 5.8383 7.5676 2.794 0.4113
OACM5.1 C GDSC1 5.9929 14.1488 -0.0324 15.9787
SK-GT-4 GDSC1 6.1443 8.5804 2.5437 1.077
TE-12 GDSC1 7.4062 9.608 2.6528 0.2181
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1 6.8741 8.7825 2.7466 0.1874
Cancer Drug Sensitivity Data Curated from 31 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SJNB-17 GDSC1 3.1563 9.3636 0.1843 23.5833
NB1 GDSC1 3.8034 6.8768 1.9532 9.5049
SK-N-DZ GDSC1 4.0703 6.6265 2.2711 6.2828
SK-N-MC-IXC GDSC1 4.2593 5.7351 2.8083 1.9445
SK-N-BE(2)-M17 GDSC1 4.3058 6.3049 2.5779 3.4305
SJNB-7 GDSC1 4.536 6.5178 2.6166 2.6972
NB69 GDSC1 4.6614 6.864 2.5335 3.0132
CHP-126 GDSC1 4.719 9.5795 1.2941 11.5418
LA-N-6 GDSC1 4.7788 7.1499 2.4726 3.1962
SK-N-FI GDSC1 4.9248 6.8098 2.6952 1.5978
SK-N-SH GDSC1 4.944 7.4027 2.4528 3.028
IMR-5 GDSC1 5.0503 6.7971 2.7592 1.1147
MHH-NB-11 GDSC1 5.0622 6.8675 2.7367 1.2131
KP-N-YS GDSC1 5.0887 7.4201 2.5218 2.3657
Kelly GDSC1 5.1031 6.4514 2.9132 0.4327
SJNB-14 GDSC1 5.1993 6.7525 2.8406 0.6285
GI-ME-N GDSC1 5.293 9.5654 1.6789 7.493
SK-N-AS GDSC1 5.3425 7.7682 2.5032 2.1107
TGW GDSC1 5.4476 6.9951 2.8501 0.4405
SJNB-13 GDSC1 5.5201 7.2096 2.8005 0.5596
SJNB-5 GDSC1 5.5207 7.2474 2.7868 0.606
GOTO GDSC1 5.5903 7.639 2.6683 1.0156
NB(TU)1 GDSC1 5.705 7.3988 2.8037 0.4471
CHP-212 GDSC1 5.7314 7.3746 2.8223 0.3823
SJNB-6 GDSC1 5.7389 7.2499 2.8688 0.2647
NH-12 GDSC1 5.761 7.686 2.7212 0.6818
CHP-134 GDSC1 5.8327 7.2167 2.9134 0.1529
SiMa GDSC1 5.8469 7.7465 2.733 0.5896
SJNB-10 GDSC1 6.0517 7.6732 2.8351 0.2361
KP-N-YN GDSC1 6.1057 8.2634 2.6461 0.7244
SJNB-12 GDSC1 6.568 8.3892 2.7731 0.2128
⏷ Show the Full List of 31 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuCC-T1 GDSC1 4.4867 7.1952 2.2771 5.1717
Cancer Drug Sensitivity Data Curated from 51 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MRK-nu-1 GDSC1 3.0602 6.1697 1.6958 14.131
DU4475 GDSC1 3.3579 5.0427 2.5143 6.6323
HCC202 GDSC1 3.517 7.4769 1.4283 14.3899
HCC1806 GDSC1 3.7825 6.915 1.9183 9.8382
CAMA-1 GDSC1 3.8142 5.6497 2.5651 4.7624
HCC2157 GDSC1 3.8909 7.6447 1.6396 11.5769
OCUB-M GDSC1 3.9531 7.9949 1.5136 12.2944
CAL-85-1 GDSC1 4.1273 8.1369 1.5741 11.3109
HCC2218 GDSC1 4.1338 5.9946 2.615 3.5554
JIMT-1 GDSC1 4.2174 6.8796 2.2502 6.0422
HCC1419 GDSC1 4.2382 10.6698 0.4059 18.5436
ZR-75-30 GDSC1 4.2445 6.1927 2.5921 3.4659
Evsa-T GDSC1 4.4347 6.2206 2.6916 2.3901
UACC-893 GDSC1 4.4692 7.1714 2.2771 5.213
MDA-MB-468 GDSC1 4.4791 7.2337 2.2543 5.3547
MDA-MB-453 GDSC1 4.4929 6.3263 2.6772 2.3778
UACC-812 GDSC1 4.5622 6.4521 2.6602 2.3648
CAL-120 GDSC1 4.8595 6.5297 2.7784 1.2317
BT-20 GDSC1 4.8687 6.2354 2.8982 0.6549
COLO 824 GDSC1 4.8949 7.8362 2.2314 4.5917
CAL-148 GDSC1 4.9844 6.701 2.7675 1.1449
MDA-MB-175-VII GDSC1 5.0493 6.7761 2.7671 1.0779
HCC70 GDSC1 5.1536 13.9546 -0.5299 20.5604
MFM-223 GDSC1 5.2556 7.194 2.6949 1.2114
HCC1954 GDSC1 5.2849 7.6658 2.5173 2.1097
HCC1599 GDSC1 5.3118 10.868 1.0784 11.3828
YMB-1-E GDSC1 5.355 7.5349 2.6044 1.5518
MDA-MB-157 GDSC1 5.4199 7.4167 2.6805 1.1156
EFM-192A GDSC1 5.4215 7.1708 2.7751 0.7168
HDQ-P1 GDSC1 5.4899 7.7541 2.5788 1.5292
MCF-7 GDSC1 5.5249 7.3445 2.7525 0.7281
Hs 578T GDSC1 5.5309 7.2323 2.7964 0.5666
BT-483 GDSC1 5.5758 7.2239 2.817 0.474
AU565 GDSC1 5.5884 7.655 2.6614 1.047
HCC1569 GDSC1 5.6068 12.9805 0.2659 15.3933
HCC1428 GDSC1 5.7091 7.5978 2.7329 0.674
HCC1500 GDSC1 5.7147 7.2373 2.8644 0.2834
MDA-MB-436 GDSC1 5.7416 7.5505 2.7631 0.5525
MDA-MB-330 GDSC1 5.7478 7.5577 2.7629 0.5495
BT-474 GDSC1 5.7821 7.0464 2.953 0.1054
BT-549 GDSC1 5.8457 8.0873 2.6055 1.0649
MDA-MB-415 GDSC1 5.8462 7.4873 2.8253 0.327
HCC38 GDSC1 5.9208 7.76 2.7566 0.4775
MDA-MB-361 GDSC1 5.9386 7.6226 2.8118 0.3241
CAL-51 GDSC1 5.9534 7.4786 2.8668 0.2034
MDA-MB-231 GDSC1 6.0989 13.1051 0.534 12.7146
HCC1395 GDSC1 6.1003 8.0965 2.7045 0.5408
T-47D GDSC1 6.1593 8.2099 2.6864 0.5648
HCC1187 GDSC1 6.1879 15.218 -0.413 17.3441
HCC1937 GDSC1 6.2294 8.0757 2.76 0.3383
EFM-19 GDSC1 6.4437 8.4616 2.7038 0.3911
⏷ Show the Full List of 51 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 54 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D-247MG GDSC1 2.7984 24.3857 -7.6269 41.4437
8-MG-BA GDSC1 3.4357 5.1297 2.5348 6.1951
GaMG GDSC1 3.4944 6.1791 2.0581 9.7279
U-251MG GDSC1 3.7632 5.1804 2.7569 3.4395
MOG-G-CCM GDSC1 4.1793 7.4005 1.9721 8.2263
YKG-1 GDSC1 4.1918 6.1103 2.5975 3.5468
D-566MG GDSC1 4.2187 6.0091 2.661 3.0337
GI-1 GDSC1 4.2866 6.9255 2.2747 5.6805
D-263MG GDSC1 4.315 6.4533 2.515 3.8581
Daoy GDSC1 4.3187 6.0353 2.7082 2.4995
NMC-G1 GDSC1 4.4315 7.9848 1.8651 8.3143
KNS-42 GDSC1 4.4411 5.8844 2.8407 1.4402
SF539 GDSC1 4.5145 8.1798 1.8281 8.3599
KALS-1 GDSC1 4.6747 7.7266 2.1477 5.6589
DK-MG GDSC1 4.7106 7.4567 2.2945 4.544
DBTRG-05MG GDSC1 4.7314 7.6446 2.2208 5.0138
Hs 683 GDSC1 4.8097 7.2619 2.4403 3.3519
42-MG-BA GDSC1 4.829 6.7975 2.6526 1.9777
D-423MG GDSC1 4.8616 7.7403 2.2553 4.4968
AM-38 GDSC1 4.8929 8.8277 1.7706 7.8032
CAS-1 GDSC1 4.9408 6.6825 2.7547 1.2588
LN-18 GDSC1 4.9828 5.9551 3.0439 0.1383
SK-MG-1 GDSC1 5.018 6.88 2.7111 1.3945
U-87MG ATCC GDSC1 5.0333 7.4861 2.4645 2.8022
M059J GDSC1 5.047 7.3042 2.5495 2.2635
PFSK-1 GDSC1 5.0519 7.2464 2.5764 2.0981
LN-405 GDSC1 5.0602 6.5742 2.8501 0.6973
GB-1 GDSC1 5.1012 6.7553 2.7981 0.8839
D283 Med GDSC1 5.1118 6.4615 2.913 0.4284
SF295 GDSC1 5.166 6.5268 2.9104 0.4057
D-336MG GDSC1 5.1884 8.5452 2.0827 5.0003
LNZTA3WT4 GDSC1 5.214 8.0404 2.3211 3.3985
MOG-G-UVW GDSC1 5.2552 7.3344 2.6387 1.4915
A-172 GDSC1 5.3746 7.112 2.7779 0.7411
U-118MG GDSC1 5.3964 7.2807 2.7229 0.9495
LN-229 GDSC1 5.4152 7.3826 2.6917 1.0696
D-392MG GDSC1 5.4311 10.3948 1.3792 9.1592
KS-1 [Human Krukenberg tumour] GDSC1 5.4543 8.0169 2.455 2.2299
Becker GDSC1 5.476 7.9958 2.4743 2.0943
D-502MG GDSC1 5.5358 8.1691 2.4319 2.2494
D-542MG GDSC1 5.5794 7.1579 2.8421 0.3977
KINGS-1 GDSC1 5.5831 8.1364 2.4682 1.9916
T98G GDSC1 5.6232 8.2279 2.45 2.039
H4 GDSC1 5.6711 7.9849 2.5694 1.3845
SF268 GDSC1 5.6754 8.1923 2.4889 1.7739
SF126 GDSC1 5.6976 7.0023 2.9388 0.1425
SNB-75 GDSC1 5.7214 8.7922 2.2643 2.9415
ONS-76 GDSC1 5.9505 7.4877 2.8627 0.2119
YH-13 GDSC1 5.975 7.1845 2.9722 0.0588
SW1088 GDSC1 5.9798 7.7548 2.7806 0.385
KNS-81-FD GDSC1 6.0216 7.9188 2.7382 0.4816
Onda 10 GDSC1 6.105 7.9027 2.7749 0.3493
SW1783 GDSC1 6.1373 8.2057 2.6794 0.5977
Onda 11 GDSC1 6.3914 8.702 2.5983 0.7131
⏷ Show the Full List of 54 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ETK-1 GDSC1 3.4234 6.2727 1.9535 10.7888
TGBC1TKB GDSC1 5.3709 7.1614 2.7576 0.8251
TGBC24TKB GDSC1 5.7861 7.6052 2.7606 0.5355
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MFE-280 GDSC1 4.4821 6.8754 2.4228 4.1403
RL95-2 GDSC1 4.5496 6.2279 2.7506 1.817
MFE-296 GDSC1 4.6908 6.909 2.5301 2.9811
KLE GDSC1 5.3903 12.5188 0.3393 15.5579
MFE-319 GDSC1 5.4312 6.8281 2.9034 0.2982
EN GDSC1 5.6139 7.1319 2.8642 0.3228
AN3-CA GDSC1 5.7207 7.6566 2.7158 0.7277
ESS-1 GDSC1 6.0649 7.577 2.8724 0.1663
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 31 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KTCTL-26A GDSC1 1.7493 3.8252 1.4553 22.0514
KTCTL-1M GDSC1 2.3517 4.6216 1.7697 16.6837
NCC021 GDSC1 3.1109 8.1453 0.7543 20.4711
KTCTL-140 GDSC1 3.3308 4.5189 2.7535 4.8458
KTCTL-21 GDSC1 3.4156 8.5316 0.8178 18.9049
769-P GDSC1 3.4751 5.4635 2.3998 7.1209
KTCTL-195 GDSC1 3.9338 6.4359 2.2671 6.7013
VMRC-RCW GDSC1 4.2227 6.0856 2.6282 3.2571
KTCTL-13 GDSC1 4.3711 8.8672 1.3938 11.8547
RXF 393L GDSC1 4.3835 9.1777 1.2508 12.8012
A-498 GDSC1 4.4762 6.2183 2.7155 2.1596
786-O GDSC1 4.4769 11.5426 0.1553 19.1741
SN12C GDSC1 4.5725 7.5808 2.1511 5.8758
KMRC-20 GDSC1 4.687 6.8156 2.5692 2.7318
VMRC-RCZ GDSC1 4.7679 7.441 2.3358 4.1383
BFTC-909 GDSC1 4.8214 6.5663 2.7453 1.4562
LB1047-RCC GDSC1 4.916 7.8839 2.2222 4.6109
KMRC-1 GDSC1 4.9594 6.4453 2.8565 0.7548
BB65-RCC GDSC1 5.009 7.0281 2.6461 1.7589
SW156 GDSC1 5.1091 7.916 2.3182 3.6006
LB2241-RCC GDSC1 5.3803 7.5086 2.6266 1.4121
SW13 GDSC1 5.3974 6.8647 2.8777 0.3837
UO-31 GDSC1 5.476 8.4455 2.2854 3.1878
OS-RC-2 GDSC1 5.5237 7.1628 2.819 0.4966
ACHN GDSC1 5.6502 11.4571 1.0207 10.9139
HA7-RCC GDSC1 6.0633 7.7954 2.7971 0.3128
TK-10 GDSC1 6.1766 8.2912 2.6637 0.6253
RCC10RGB GDSC1 6.2205 12.8609 0.726 11.3514
CAL-54 GDSC1 6.3634 8.0823 2.8055 0.2072
LB996-RCC GDSC1 6.6041 8.5383 2.735 0.2715
Caki-1 GDSC1 8.6932 19.7951 -0.9561 14.4935
⏷ Show the Full List of 31 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H747 GDSC1 3.8268 7.6724 1.5766 12.2473
LS411N GDSC1 3.9859 9.7704 0.6575 17.8914
HT-29 GDSC1 4.049 7.1212 2.0152 8.2807
SW620 GDSC1 4.3178 6.7578 2.3744 4.8695
HCT 116 GDSC1 4.4038 8.3234 1.6822 9.7166
RKO GDSC1 4.4548 7.5925 2.0688 6.7653
NCI-H716 GDSC1 4.4714 7.5352 2.107 6.4436
LoVo GDSC1 4.5192 7.4363 2.1848 5.7608
COLO 320HSR GDSC1 4.5336 7.6714 2.0832 6.4608
SW48 GDSC1 4.5535 6.6613 2.5626 3.025
SNU-1040 GDSC1 4.566 8.4777 1.72 8.9986
KM12 GDSC1 4.6083 7.5935 2.1679 5.6695
HT115 GDSC1 4.8198 6.2888 2.8563 0.8871
SW948 GDSC1 4.8266 6.4576 2.7921 1.199
LS123 GDSC1 4.9553 6.5478 2.8149 0.9464
SNU-81 GDSC1 5.0003 6.618 2.8074 0.9372
LS1034 GDSC1 5.0364 11.8203 0.4296 16.0177
SW1116 GDSC1 5.0375 6.9765 2.6811 1.53
MDST8 GDSC1 5.0722 6.5916 2.8485 0.6941
C2BBe1 GDSC1 5.0918 7.339 2.5576 2.1501
CCK-81 GDSC1 5.1055 8.3131 2.1392 4.7886
CW-2 GDSC1 5.1486 7.4894 2.523 2.2693
CaR-1 GDSC1 5.1617 8.0796 2.2753 3.7833
HCT 15 GDSC1 5.205 6.7068 2.8599 0.5531
SNU-C1 GDSC1 5.2369 7.1335 2.7103 1.1566
T84 GDSC1 5.2519 7.3182 2.6437 1.4696
SW1417 GDSC1 5.318 7.3523 2.6604 1.3129
SNU-C5 GDSC1 5.4004 7.537 2.6245 1.4007
SNU-175 GDSC1 5.4026 7.1619 2.7707 0.7482
RCM-1 [Human ESC] GDSC1 5.4266 6.7309 2.9357 0.2234
HCC2998 GDSC1 5.4443 7.5229 2.6498 1.2337
HT-55 GDSC1 5.4451 6.7194 2.9463 0.195
LS180 GDSC1 5.4623 6.9479 2.8726 0.367
SW626 GDSC1 5.6466 8.1123 2.5077 1.7116
SNU-61 GDSC1 5.6659 7.6495 2.6961 0.8412
LS513 GDSC1 5.6718 7.3082 2.8235 0.4064
COLO205 GDSC1 5.7106 7.0602 2.9238 0.1644
SW1463 GDSC1 5.8399 7.4076 2.8507 0.2703
GP5d GDSC1 5.9101 7.489 2.8478 0.2534
CL-11 GDSC1 5.9941 7.7983 2.7706 0.4051
SNU-C2B GDSC1 6.3309 8.8837 2.5068 1.0799
COLO 678 GDSC1 6.3622 8.1381 2.7861 0.2421
SW837 GDSC1 6.4697 8.4854 2.705 0.3787
SNU-407 GDSC1 8.8962 22.7856 -2.2207 18.7273
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1 4.3354 6.5082 2.5022 3.9037
Cancer Drug Sensitivity Data Curated from 16 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-423 GDSC1 3.9387 5.5663 2.6907 3.4754
HLE GDSC1 4.2253 8.1341 1.6471 10.4869
SK-HEP-1 GDSC1 4.2953 6.3201 2.5645 3.5491
JHH-6 GDSC1 4.5092 5.4835 3.0326 0.3969
JHH-1 GDSC1 4.5358 5.738 2.9461 0.7495
JHH-4 GDSC1 4.6752 6.8627 2.5418 2.9325
SNU-475 GDSC1 4.8907 6.4945 2.8069 1.0515
Hep 3B2.1-7 GDSC1 4.9058 6.6204 2.7634 1.2548
Hep-G2/C3A GDSC1 5.0017 6.6683 2.7883 1.0255
HuH-1 GDSC1 5.1462 6.6384 2.8615 0.5876
SNU-398 GDSC1 5.1495 7.1913 2.6469 1.5743
SNU-387 GDSC1 5.2946 7.052 2.7671 0.8488
Huh-7 GDSC1 5.5584 12.0316 0.6881 13.1398
JHH-7 GDSC1 5.9646 7.3295 2.9209 0.1157
JHH-2 GDSC1 6.2393 7.6886 2.8948 0.1035
SNU-449 GDSC1 6.3456 8.1313 2.7826 0.2535
⏷ Show the Full List of 16 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 171 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H196 GDSC1 2.2602 3.5702 2.0955 14.7995
NCI-H2731 GDSC1 3.0523 10.6691 -0.5565 27.5085
NCI-H2795 GDSC1 3.1568 30.7741 -10.5193 42.5589
COR-L303 GDSC1 3.4958 5.2684 2.5138 6.154
NCI-H226 GDSC1 3.5052 5.2356 2.5376 5.9353
Lu-65 GDSC1 3.5895 6.1022 2.1724 8.5136
LB647-SCLC GDSC1 3.6559 12.3122 -0.8746 26.6439
LC-2/ad GDSC1 3.7321 5.9112 2.3768 6.4615
NCI-H64 GDSC1 3.741 6.7796 1.9536 9.7034
PC-14 GDSC1 3.7694 5.7529 2.4823 5.5308
CAL-12T GDSC1 3.8977 6.3204 2.2975 6.5741
EMC-BAC-1 GDSC1 3.9527 10.8206 0.1087 21.1107
HOP-62 GDSC1 4.0016 6.0211 2.5157 4.6223
HCC44 GDSC1 4.0198 6.9888 2.0588 8.036
EPLC-272H GDSC1 4.0383 6.0074 2.5469 4.293
LCLC-97TM1 GDSC1 4.151 6.8944 2.1977 6.614
BEN GDSC1 4.1955 8.2379 1.5745 11.1003
COR-L321 GDSC1 4.2374 5.7858 2.7733 2.2184
LXF 289 GDSC1 4.2642 6.8204 2.3098 5.4782
NCI-H526 GDSC1 4.2796 6.9014 2.2815 5.6485
DMS 273 GDSC1 4.283 6.8698 2.2987 5.5124
NCI-H810 GDSC1 4.2905 7.6966 1.9067 8.3976
SBC-5 GDSC1 4.4395 5.8882 2.8383 1.4571
NCI-H1694 GDSC1 4.464 8.9685 1.4111 11.4626
SHP-77 GDSC1 4.4822 6.4299 2.6252 2.7417
COR-L23 GDSC1 4.4832 8.9379 1.4397 11.2093
NCI-H345 GDSC1 4.5014 5.4674 3.0354 0.392
NCI-H1963 GDSC1 4.5067 6.8022 2.4713 3.7463
NCI-H661 GDSC1 4.5429 6.9498 2.4256 3.9886
NCI-H2141 GDSC1 4.5474 6.6481 2.565 3.0207
NCI-H720 GDSC1 4.5666 7.6115 2.1328 6.0214
NCI-H69 GDSC1 4.6573 11.3712 0.3745 17.4244
NCI-H2444 GDSC1 4.6793 5.808 2.9809 0.4709
NCI-H1581 GDSC1 4.6807 6.6655 2.6314 2.3442
NCI-H841 GDSC1 4.6905 6.8301 2.5647 2.7546
SK-MES-1 GDSC1 4.699 6.858 2.5572 2.7884
NCI-H2196 GDSC1 4.7178 6.7369 2.6203 2.3514
NCI-H187 GDSC1 4.7214 6.1691 2.8592 0.9769
NCI-H211 GDSC1 4.7369 7.2239 2.4157 3.6572
A-427 GDSC1 4.7831 8.9711 1.6303 9.059
NCI-H1915 GDSC1 4.7832 9.0844 1.5763 9.4348
NCI-H2171 GDSC1 4.7881 6.6717 2.6849 1.8474
NCI-H2085 GDSC1 4.7971 9.6232 1.327 11.1055
LK-2 GDSC1 4.8177 6.8389 2.6291 2.1357
LCLC-103H GDSC1 4.8345 9.766 1.2839 11.2938
NCI-H1648 GDSC1 4.8475 7.3577 2.4191 3.4216
NCI-H2081 GDSC1 4.8479 7.4956 2.3578 3.8294
NCI-H2595 GDSC1 4.9112 8.0595 2.1393 5.19
COR-L95 GDSC1 4.9618 6.6192 2.7897 1.0602
NCI-H520 GDSC1 5.0103 7.0281 2.6467 1.7538
DMS 114 GDSC1 5.0139 7.2642 2.5495 2.3131
NCI-H1838 GDSC1 5.0173 7.2215 2.5694 2.19
SK-LU-1 GDSC1 5.0174 7.2314 2.5652 2.2147
NCI-H1793 GDSC1 5.0267 6.7553 2.7651 1.1112
NCI-H2818 GDSC1 5.0314 7.21 2.5814 2.0986
NCI-H510A GDSC1 5.0316 8.5658 1.9799 6.0278
SW1573 GDSC1 5.0343 7.4799 2.4678 2.7804
NCI-H1734 GDSC1 5.0582 7.0871 2.6457 1.6961
NCI-H1573 GDSC1 5.0641 7.0031 2.683 1.4873
NCI-H1048 GDSC1 5.0953 6.8839 2.7452 1.1354
UMC-11 GDSC1 5.1222 6.9397 2.7353 1.1555
NCI-H2029 GDSC1 5.1359 6.5822 2.8782 0.5331
NCI-H1437 GDSC1 5.1366 8.4566 2.0925 5.0393
DMS 79 GDSC1 5.1535 6.9109 2.7605 1.0046
IA-LM GDSC1 5.2011 6.8816 2.7925 0.8206
NCI-H847 GDSC1 5.2031 6.5121 2.9299 0.3281
NCI-H1944 GDSC1 5.2322 7.2131 2.6766 1.3254
COR-L105 GDSC1 5.2497 10.7716 1.083 11.5111
DMS 53 GDSC1 5.2675 6.9847 2.7813 0.812
NCI-H2591 GDSC1 5.268 11.2655 0.859 12.8602
NCI-H2172 GDSC1 5.2832 6.6048 2.9271 0.2993
NCI-H2135 GDSC1 5.2882 6.7876 2.8633 0.4884
NCI-H446 GDSC1 5.2939 6.9344 2.8113 0.6715
SBC-3 GDSC1 5.2959 7.254 2.6893 1.1966
NCI-H460 GDSC1 5.2984 6.4762 2.9775 0.1765
NCI-H209 GDSC1 5.3072 7.9041 2.4287 2.59
NCI-H1155 GDSC1 5.3152 6.9651 2.8085 0.6666
NCI-H2373 GDSC1 5.3326 7.091 2.7683 0.8125
NCI-H1688 GDSC1 5.3338 7.258 2.7045 1.0881
NCI-H838 GDSC1 5.3352 7.2599 2.7044 1.0874
NCI-H2803 GDSC1 5.3658 7.2235 2.7317 0.9383
NCI-H3255 GDSC1 5.3703 7.4905 2.6292 1.4098
COR-L88 GDSC1 5.3721 7.5697 2.5984 1.5631
NCI-H1703 GDSC1 5.3737 7.0698 2.7933 0.6823
NCI-H2722 GDSC1 5.3766 7.0884 2.7875 0.7023
NCI-H2369 GDSC1 5.3914 6.8377 2.8851 0.3655
NCI-H522 GDSC1 5.4157 8.2471 2.3388 2.9605
NCI-H1869 GDSC1 5.4328 7.531 2.6415 1.2845
SW1271 GDSC1 5.4381 7.5304 2.6441 1.2668
NCI-H524 GDSC1 5.4504 7.5687 2.6345 1.2998
RERF-LC-MS GDSC1 5.4527 7.2344 2.7641 0.7362
NCI-H2087 GDSC1 5.459 7.7397 2.5704 1.6064
NCI-H358 GDSC1 5.4744 7.7817 2.5607 1.6384
NCI-H1563 GDSC1 5.4893 7.0041 2.8628 0.3819
Lu-165 GDSC1 5.5081 7.1213 2.8279 0.4769
NCI-H1436 GDSC1 5.5098 6.9841 2.8776 0.332
NCI-H650 GDSC1 5.5123 7.2906 2.7675 0.6812
NCI-H82 GDSC1 5.5206 7.6813 2.6215 1.29
Ms-1 GDSC1 5.5277 7.0383 2.8652 0.3575
HOP-92 GDSC1 5.5288 7.6388 2.6418 1.1883
LOU-NH91 GDSC1 5.5372 7.5626 2.6749 1.0334
NCI-H322M GDSC1 5.5401 10.9705 1.1788 10.1886
NCI-H1975 GDSC1 5.5484 7.7367 2.6122 1.3063
NCI-H1792 GDSC1 5.5598 7.5381 2.6939 0.9336
NCI-H1781 GDSC1 5.5614 6.7458 2.978 0.1117
NCI-H2170 GDSC1 5.5655 7.7272 2.6234 1.2371
HCC33 GDSC1 5.5716 6.9485 2.9127 0.225
NCI-H1836 GDSC1 5.5761 6.8793 2.938 0.1736
NCI-H1092 GDSC1 5.5793 7.0162 2.892 0.2685
NCI-H727 GDSC1 5.6196 10.3191 1.5313 7.746
SBC-1 GDSC1 5.6212 6.9429 2.9323 0.1721
NCI-H292 GDSC1 5.6306 7.0567 2.8966 0.2403
NCI-H1435 GDSC1 5.6309 7.0975 2.8825 0.2718
NCI-H1693 GDSC1 5.6379 7.5538 2.7205 0.7681
NCI-H1770 GDSC1 5.6586 7.0592 2.9058 0.2122
NCI-H2342 GDSC1 5.7045 7.6189 2.7233 0.7115
NCI-H2869 GDSC1 5.706 7.6967 2.6949 0.8162
NCI-H1650 GDSC1 5.7218 8.2563 2.4847 1.7431
NCI-H2122 GDSC1 5.7386 7.3656 2.8282 0.3636
Lu-99A GDSC1 5.7621 8.3113 2.4813 1.7153
IST-SL1 GDSC1 5.7697 7.6604 2.734 0.6321
ChaGo-K-1 GDSC1 5.7872 7.7928 2.6922 0.7687
HCC827 GDSC1 5.7924 7.4426 2.8211 0.3592
CPC-N GDSC1 5.8157 7.5205 2.8022 0.399
HCC15 GDSC1 5.8359 7.8351 2.6961 0.7217
NCI-H596 GDSC1 5.8374 7.2826 2.8927 0.187
NCI-H1355 GDSC1 5.8404 8.0357 2.6229 0.9977
NCI-H2009 GDSC1 5.8463 7.6871 2.7542 0.5228
NCI-H2227 GDSC1 5.851 7.3157 2.8862 0.1952
NCI-H1876 GDSC1 5.8523 7.878 2.6869 0.744
NCI-H2804 GDSC1 5.8769 8.395 2.4999 1.5046
NCI-H2347 GDSC1 5.8889 9.1497 2.1986 3.0784
RERF-LC-KJ GDSC1 5.8926 7.5872 2.8073 0.353
NCI-H513 GDSC1 5.9035 7.6657 2.7837 0.4099
EBC-1 GDSC1 5.9146 7.8305 2.7289 0.5646
Lu-139 GDSC1 5.9406 12.0198 0.9421 10.7158
RERF-LC-Sq1 GDSC1 5.9474 8.7225 2.402 1.9053
NCI-H441 GDSC1 5.9564 8.0637 2.66 0.7712
NCI-H1299 GDSC1 5.9953 7.9168 2.7289 0.5218
NCI-H1755 GDSC1 6.0216 7.8599 2.7591 0.4236
Calu-6 GDSC1 6.0232 7.7198 2.8088 0.3004
NCI-H2023 GDSC1 6.0465 7.5523 2.8744 0.1673
NCI-H647 GDSC1 6.0555 7.9004 2.7575 0.4132
Lu-135 GDSC1 6.0574 8.0391 2.7087 0.5504
ABC-1 GDSC1 6.1096 8.0832 2.7128 0.5118
COLO 668 GDSC1 6.1174 7.9493 2.7632 0.373
NCI-H3122 GDSC1 6.1189 8.0093 2.7426 0.4249
NCI-H2291 GDSC1 6.1244 8.3011 2.6396 0.7349
NCI-H1568 GDSC1 6.1343 7.9858 2.7566 0.3826
NCI-H748 GDSC1 6.1344 8.7109 2.4898 1.3093
EMC-BAC-2 GDSC1 6.1437 8.2511 2.6655 0.6381
HCC78 GDSC1 6.1611 8.102 2.7256 0.4519
A-549 GDSC1 6.2269 8.163 2.7286 0.4157
NCI-H23 GDSC1 6.2571 9.9347 2.0543 3.3736
NCI-H2461 GDSC1 6.2863 8.063 2.7849 0.2662
Calu-3 GDSC1 6.2867 7.9551 2.8219 0.198
NCI-H1666 GDSC1 6.3291 8.0728 2.7967 0.2315
LC-1/sq GDSC1 6.401 8.6454 2.6225 0.6318
NCI-H1623 GDSC1 6.4222 8.3253 2.7433 0.3097
NCI-H1304 GDSC1 6.4341 7.8915 2.8932 0.0797
NCI-H1651 GDSC1 6.4659 8.7082 2.6249 0.5915
IST-SL2 GDSC1 6.5034 8.3021 2.78 0.2166
EKVX GDSC1 6.575 8.4304 2.7616 0.2308
NCI-H2110 GDSC1 6.5827 8.5917 2.7091 0.3304
PaCa-3 GDSC1 6.7979 8.889 2.6838 0.3155
NCI-H1993 GDSC1 6.879 22.6816 -3.5511 26.4663
NCI-H2405 GDSC1 6.9005 9.1218 2.6403 0.3736
NCI-H2228 GDSC1 7.7747 22.5131 -2.8369 22.7413
HARA [Human squamous cell lung carcinoma] GDSC1 8.0202 16.3164 0.2265 10.425
Lu-134-A GDSC1 8.4969 22.8695 -2.5206 20.4107
NCI-H2030 GDSC1 8.7059 20.4899 -1.2689 15.7017
⏷ Show the Full List of 171 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1 3.5962 6.9392 1.7606 11.6566
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE-15 GDSC1 4.495 6.6484 2.5344 3.3333
TE-9 GDSC1 4.5298 6.2771 2.7188 2.0464
KYSE-450 GDSC1 4.7426 6.4473 2.756 1.5015
TE-6 GDSC1 4.9213 7.2707 2.498 2.7797
TE-8 GDSC1 4.998 8.7269 1.8846 6.7611
OE19 GDSC1 5.0838 6.7083 2.8088 0.8526
TE-5 GDSC1 5.1418 6.7973 2.7995 0.8416
KYSE-520 GDSC1 5.1693 9.1572 1.7914 7.0115
TE-4 GDSC1 5.2087 7.525 2.5382 2.0959
TE-11 GDSC1 5.3159 7.2278 2.7084 1.0877
TE-10 GDSC1 5.3342 7.3913 2.6523 1.3354
KYSE-150 GDSC1 5.3727 6.5541 2.9772 0.1562
OE21 GDSC1 5.4718 7.378 2.7177 0.9074
T.T GDSC1 5.4884 7.2979 2.7549 0.7453
COLO 680N GDSC1 5.5399 7.2929 2.7777 0.6259
EC-GI-10 GDSC1 5.602 7.3903 2.7666 0.6247
TE-1 GDSC1 5.6563 7.363 2.7979 0.4899
KYSE-270 GDSC1 5.8112 8.4741 2.4387 1.8742
KYSE-510 GDSC1 5.8687 7.5671 2.8055 0.3674
KYSE-70 GDSC1 5.9409 7.9024 2.7131 0.6002
KYSE-410 GDSC1 5.9884 7.708 2.8002 0.3329
KYSE-140 GDSC1 6.2727 8.8714 2.4872 1.2035
OE33 GDSC1 6.9454 16.9469 -0.7311 17.0243
KYSE-180 GDSC1 8.5458 20.7459 -1.488 16.8212
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OVTOKO GDSC1 3.5631 5.8562 2.2741 7.8081
A2780 GDSC1 3.6043 5.858 2.3055 7.4254
SK-OV-3 GDSC1 3.6326 5.7291 2.3914 6.6622
TOV-112D GDSC1 4.0929 6.1958 2.4934 4.5513
OV56 GDSC1 4.2617 6.4918 2.4635 4.3551
RMG-I GDSC1 4.346 6.479 2.5223 3.7364
OAW28 GDSC1 4.4316 7.2726 2.2053 5.8263
OVKATE GDSC1 4.617 9.9642 1.0349 13.5454
DOV13 GDSC1 4.7585 7.3402 2.3759 3.8843
TOV-21G GDSC1 4.8333 6.3037 2.8565 0.8729
OAW42 GDSC1 4.8655 6.0029 2.9835 0.3413
FU-OV-1 GDSC1 4.9596 7.1912 2.5525 2.3792
TYK-nu GDSC1 4.9789 9.2965 1.6051 8.7374
EFO-21 GDSC1 5.0442 10.7254 0.9658 12.7914
OVCAR-5 GDSC1 5.1181 6.9613 2.7248 1.2108
OVCAR-8 GDSC1 5.2196 7.9636 2.3574 3.1608
OC 314 GDSC1 5.2242 7.3005 2.6379 1.5319
ES-2 GDSC1 5.2271 6.5857 2.9128 0.3661
EFO-27 GDSC1 5.2533 6.9671 2.782 0.8209
OV-90 GDSC1 5.4605 7.3313 2.7307 0.8629
JHOS-2 GDSC1 5.536 7.0394 2.8679 0.3465
Caov-3 GDSC1 5.5562 7.1726 2.828 0.4509
OVCAR-3 GDSC1 5.7303 7.3461 2.832 0.3571
Kuramochi GDSC1 5.9008 7.9804 2.6685 0.7778
OVCAR-4 GDSC1 6.042 7.9769 2.7252 0.5092
OVISE GDSC1 6.0496 16.4394 -1.0994 20.6427
IGROV-1 GDSC1 6.4641 8.3961 2.7339 0.316
OVK18 GDSC1 7.0484 15.9596 -0.1984 14.3822
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HPAC GDSC1 3.4314 4.6229 2.7843 4.2444
HuP-T4 GDSC1 3.7986 8.5298 1.1282 15.5043
MIA PaCa-2 GDSC1 4.334 6.0353 2.7171 2.4103
Panc 02.03 GDSC1 4.5927 6.5325 2.6416 2.4306
DAN-G GDSC1 4.5983 6.5075 2.6556 2.3308
PaTu 8902 GDSC1 4.7722 8.0419 2.062 6.0405
Panc 10.05 GDSC1 4.8013 8.2258 1.9945 6.4488
PaTu 8988t GDSC1 4.9067 6.5658 2.7858 1.1392
KP-4 GDSC1 5.0102 6.5044 2.8556 0.7156
HuP-T3 GDSC1 5.1774 7.2069 2.6538 1.5045
KP-2 GDSC1 5.293 7.6557 2.5255 2.0527
SU.86.86 GDSC1 5.3282 7.3494 2.6662 1.274
PL4 GDSC1 5.3393 7.1348 2.7544 0.8644
YAPC GDSC1 5.3885 6.6732 2.9419 0.2226
SW1990 GDSC1 5.4689 7.393 2.7108 0.9389
PSN1 GDSC1 5.4839 11.5759 0.8557 12.3282
SUIT-2 GDSC1 5.6254 12.8311 0.3504 14.8862
QGP-1 GDSC1 5.6522 7.0625 2.9023 0.2212
Panc 08.13 GDSC1 5.7064 7.6848 2.6995 0.7983
Capan-1 GDSC1 5.7087 7.3724 2.8145 0.4143
Panc 03.27 GDSC1 5.7248 7.3775 2.8188 0.3949
MZ-PC-1 GDSC1 5.7638 7.9502 2.6231 1.0597
Capan-2 GDSC1 5.9106 7.8325 2.7266 0.5741
HPAF-II GDSC1 5.9974 7.6564 2.8215 0.2813
CFPAC-1 GDSC1 6.0173 7.6465 2.832 0.2526
Hs 766T GDSC1 6.0497 7.7138 2.8204 0.2664
Panc 04.03 GDSC1 6.1775 7.7862 2.8409 0.1921
KP-3 GDSC1 6.1994 8.8277 2.4727 1.3257
BxPC-3 GDSC1 6.3713 8.7555 2.5708 0.8169
AsPC-1 GDSC1 6.4816 9.2979 2.4129 1.3382
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H2052 GDSC1 4.7997 7.2962 2.4194 3.51
NCI-H28 GDSC1 5.3511 7.1689 2.7464 0.8882
MSTO-211H GDSC1 5.7037 7.9001 2.6166 1.1394
MPP 89 GDSC1 5.778 7.4524 2.8122 0.3889
IST-Mes1 GDSC1 5.8134 7.4325 2.8324 0.3224
NCI-H2452 GDSC1 6.1251 8.316 2.6344 0.7521
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PC-3 GDSC1 4.917 7.8738 2.2274 4.5737
DU145 GDSC1 5.1035 8.0181 2.27 3.9244
LNCaP clone FGC GDSC1 5.2795 12.5125 0.265 16.2612
VCaP GDSC1 5.7052 7.127 2.8991 0.2117
22Rv1 GDSC1 5.8931 7.7654 2.744 0.5292
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 GDSC1 6.0018 7.7016 2.8074 0.3112
Cancer Drug Sensitivity Data Curated from 56 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-7951 GDSC1 3.7991 6.2228 2.2732 7.0582
IGR-1 GDSC1 3.8169 5.2662 2.7525 3.3283
WM115 GDSC1 3.8428 5.2662 2.7699 3.1292
GAK GDSC1 3.9779 6.2484 2.3897 5.6404
WM35 GDSC1 4.0127 5.8642 2.5981 3.9768
CP50-MEL-B GDSC1 4.0238 5.5063 2.7734 2.666
Mel Ho GDSC1 4.0533 7.2677 1.9466 8.7844
UACC-62 GDSC1 4.0799 5.8402 2.653 3.4064
SK-MEL-28 GDSC1 4.1186 6.2638 2.4781 4.5997
MZ-MEL-7 GDSC1 4.2539 6.2137 2.5882 3.4725
LB373-MEL-D GDSC1 4.2702 5.8535 2.7618 2.2326
G-361 GDSC1 4.3617 6.7708 2.3964 4.6042
SK-MEL-1 GDSC1 4.3685 6.5467 2.5048 3.8106
MeWo GDSC1 4.5176 6.909 2.429 4.0191
Hs 938.T GDSC1 4.533 7.2742 2.2695 5.1179
CP66-MEL GDSC1 4.5353 6.3381 2.6953 2.1861
IPC-298 GDSC1 4.6075 6.3576 2.7253 1.8799
VMRC-MELG GDSC1 4.6208 6.0291 2.8688 1.0428
451Lu GDSC1 4.6229 6.7915 2.544 3.0161
SK-MEL-24 GDSC1 4.6486 6.8302 2.5413 2.9856
A2058 GDSC1 4.6849 6.0469 2.8912 0.8589
SK-MEL-5 GDSC1 4.7331 6.0227 2.9219 0.6708
SK-MEL-30 GDSC1 4.7533 6.2263 2.851 0.9828
Mel JuSo GDSC1 4.8081 8.3084 1.9602 6.6755
COLO 829 GDSC1 4.8105 7.039 2.5389 2.7093
SK-MEL-3 GDSC1 4.8215 11.4859 0.4384 16.5798
A101D GDSC1 4.8387 6.0739 2.9467 0.4857
M14 GDSC1 4.8676 7.2031 2.4984 2.8694
LB2518-MEL GDSC1 4.9018 6.7893 2.6924 1.6439
SK-MEL-2 GDSC1 4.9043 6.2541 2.9061 0.5942
A-375 GDSC1 4.9153 6.3961 2.8565 0.7945
IGR-37 GDSC1 5.0584 9.6859 1.4727 9.4408
WT2-iPS GDSC1 5.1171 6.2632 2.9858 0.2191
Hs 940.T GDSC1 5.2443 6.734 2.8656 0.5078
SH-4 GDSC1 5.2685 6.9362 2.8001 0.7344
G-mel GDSC1 5.2731 6.9921 2.7808 0.8091
COLO 679 GDSC1 5.2863 7.2085 2.7029 1.1422
MMAc-SF GDSC1 5.2893 7.1482 2.7277 1.0249
COLO 783 GDSC1 5.3056 6.656 2.9174 0.3155
COLO 800 GDSC1 5.4257 7.7819 2.5377 1.8157
CHL-1 GDSC1 5.5314 7.3549 2.7513 0.7281
HT-144 GDSC1 5.5322 6.9549 2.8962 0.2762
WM1552C GDSC1 5.5679 7.1308 2.8474 0.3882
LOX-IMVI GDSC1 5.6394 7.2506 2.8318 0.3985
WM793 GDSC1 5.6698 7.172 2.8707 0.285
COLO 792 GDSC1 5.7714 16.9325 -1.5395 23.0076
MZ-MEL-2 GDSC1 5.8382 7.7302 2.7355 0.5864
UACC-257 GDSC1 5.87 7.0323 2.9872 0.0568
WM278 GDSC1 5.8924 7.7653 2.7438 0.5302
HMV-II GDSC1 6.0047 7.9945 2.7044 0.5919
DJM-1 GDSC1 6.1084 8.1048 2.7046 0.5363
RVH-421 GDSC1 6.3019 15.4377 -0.441 17.2009
IST-MEL1 GDSC1 6.3444 7.877 2.8679 0.1194
A-431 GDSC1 6.4991 8.2899 2.7827 0.2132
A-388 GDSC1 6.7293 8.6797 2.731 0.2454
EquiPSC Line K2 GDSC1 5.8489 8.2504 2.5441 1.3285
⏷ Show the Full List of 56 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1 4.4559 7.7835 1.9783 7.4236
Cancer Drug Sensitivity Data Curated from 20 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-LMS-1 GDSC1 3.8576 5.2974 2.7649 3.129
Hs 633.T GDSC1 4.5458 6.4511 2.6515 2.4501
HT-1080 GDSC1 4.6603 6.5322 2.6781 2.0856
GCT GDSC1 4.7648 6.6474 2.6833 1.8913
RKN GDSC1 4.8273 8.8863 1.7001 8.4583
Rh30 GDSC1 4.8613 6.702 2.7087 1.6069
SW684 GDSC1 4.9244 6.0483 2.9898 0.2913
A-204 GDSC1 4.9727 9.0929 1.6971 8.1186
VA-ES-BJ GDSC1 5.0681 6.5362 2.8677 0.6206
EW-8 GDSC1 5.0803 6.9734 2.7026 1.3655
RD GDSC1 5.087 7.1968 2.6145 1.8311
MES-SA GDSC1 5.217 6.4234 2.9664 0.2277
KYM-1 GDSC1 5.5353 6.7742 2.9594 0.1463
MFH-ino GDSC1 5.5863 7.5672 2.694 0.9118
G-402 GDSC1 5.5909 9.799 1.7516 6.3747
SW982 GDSC1 5.8128 6.9095 3.0084 0.0453
Rh41 GDSC1 5.9697 7.5259 2.8564 0.2183
SK-UT-1 GDSC1 6.0265 7.5559 2.8662 0.1857
G-401 GDSC1 6.0537 8.494 2.5384 1.1719
SW872 GDSC1 6.1268 7.5877 2.8902 0.1278
⏷ Show the Full List of 20 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 26 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NUGC-4 GDSC1 1.2637 5.3853 0.3181 31.8178
TGBC11TKB GDSC1 4.3496 6.2262 2.6402 2.9024
Hs 746.T GDSC1 4.4408 6.1752 2.715 2.2257
MKN45 GDSC1 4.4824 5.7956 2.8981 1.0567
ECC10 GDSC1 4.5882 9.1634 1.4042 11.1564
HSC-39 GDSC1 4.6584 7.8558 2.0769 6.2023
HGC-27 GDSC1 4.7798 7.7449 2.2042 5.0241
Fu97 GDSC1 4.7913 6.9248 2.5782 2.4931
SCH GDSC1 4.8464 6.1722 2.9129 0.6126
SNU-5 GDSC1 4.8807 6.2335 2.904 0.6214
RF-48 GDSC1 4.9183 8.2328 2.0641 5.6953
GCIY GDSC1 5.0579 7.4807 2.4799 2.6668
MKN7 GDSC1 5.1785 7.4139 2.5695 1.9604
MKN1 GDSC1 5.284 6.8947 2.8221 0.6379
MKN28 GDSC1 5.3239 8.8601 2.0195 5.1512
AGS GDSC1 5.4457 6.7104 2.9496 0.1883
SNU-16 GDSC1 5.5575 6.6818 2.998 0.086
NUGC-3 GDSC1 5.5644 8.4494 2.3292 2.7934
SNU-1 GDSC1 5.687 8.2784 2.4596 1.911
23132/87 GDSC1 5.7028 7.5424 2.7508 0.6161
OCUM-1 GDSC1 5.7924 7.674 2.738 0.6048
RERF-GC-1B GDSC1 5.812 8.2785 2.5168 1.4905
IM95 GDSC1 6.0173 8.0129 2.7027 0.5904
TMK-1 GDSC1 6.0603 7.7531 2.8107 0.2837
NCI-N87 GDSC1 6.4535 8.6395 2.6447 0.5407
SNG-M GDSC1 5.8355 7.234 2.9085 0.1602
⏷ Show the Full List of 26 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 16 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
K5 GDSC1 4.653 6.5834 2.6521 2.26
WRO GDSC1 4.7074 6.1843 2.8467 1.0561
CAL-62 GDSC1 4.7479 6.4716 2.7485 1.5366
FTC-133 GDSC1 4.7897 6.868 2.6019 2.3475
B-CPAP GDSC1 5.0205 6.5875 2.8281 0.8246
ASH-3 GDSC1 5.0616 6.6898 2.8063 0.8838
8505C GDSC1 5.067 6.93 2.7138 1.323
KMH-2 GDSC1 5.3107 7.696 2.5175 2.0735
8305C GDSC1 5.4379 7.0189 2.8378 0.4849
TT GDSC1 5.4935 6.9956 2.8675 0.3669
IHH-4 GDSC1 5.5091 6.8355 2.9292 0.2103
CGTH-W-1 GDSC1 5.5378 6.9249 2.9087 0.2452
ML-1 [Human leukemia] GDSC1 5.5925 7.2001 2.832 0.4204
TT2609-C02 GDSC1 5.7095 7.5007 2.7687 0.5529
HTC-C3 GDSC1 6.0016 8.0151 2.6957 0.6214
BHT-101 GDSC1 7.5188 24.1532 -3.8106 25.8111
⏷ Show the Full List of 16 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SCC-9 GDSC1 4.2856 6.7975 2.3347 5.2401
OSC-20 GDSC1 4.5455 6.8163 2.488 3.5495
BHY GDSC1 4.7223 6.9339 2.5366 2.8804
FaDu GDSC1 4.9809 6.8878 2.6903 1.5517
Ca9-22 GDSC1 5.0202 7.569 2.4215 3.095
PCI-04B GDSC1 5.029 7.5318 2.4425 2.9472
Detroit 562 GDSC1 5.0387 6.9564 2.6899 1.4813
LB771-HNC GDSC1 5.0675 8.3122 2.1173 5.0126
SAS GDSC1 5.0705 7.9277 2.2915 3.8447
HSC-3 GDSC1 5.0788 6.4789 2.8935 0.5164
CAL-27 GDSC1 5.1409 6.6149 2.8681 0.5667
HO-1-N-1 GDSC1 5.1448 7.1476 2.6625 1.4979
HO-1-u-1 GDSC1 5.1473 7.7324 2.4188 2.899
SCC-15 GDSC1 5.2112 7.4869 2.5553 1.9959
HSC-4 GDSC1 5.2279 6.7038 2.8702 0.5021
BB49-HNC GDSC1 5.2923 7.5921 2.5514 1.91
BB30-HNC GDSC1 5.3165 7.8124 2.4719 2.3244
HSC-2 GDSC1 5.5078 6.7653 2.9528 0.1647
BICR 22 GDSC1 5.5449 7.0458 2.8689 0.3397
PCI-06A GDSC1 5.5518 7.6561 2.6452 1.1514
SCC-4 GDSC1 5.5808 7.0718 2.8731 0.3138
KON GDSC1 5.5968 7.1474 2.8524 0.3611
PE/CA-PJ15 GDSC1 5.7274 7.3893 2.8156 0.4026
PCI-30 GDSC1 5.7316 7.709 2.7008 0.7757
OSC-19 GDSC1 5.7717 7.3945 2.8303 0.3442
PCI-38 GDSC1 5.8456 11.8112 0.9794 10.7085
KOSC-2 GDSC1 5.8985 8.2971 2.5476 1.2675
PCI-15A GDSC1 5.9021 7.5913 2.8094 0.344
SKN-3 GDSC1 5.929 7.8073 2.7428 0.5143
NCI-H3118 GDSC1 5.9681 7.6477 2.8139 0.3084
JHU-011 GDSC1 5.9704 8.6763 2.431 1.7375
JHU-022 GDSC1 5.9786 8.4632 2.5181 1.3248
BICR 31 GDSC1 5.9926 7.4444 2.8921 0.1514
DOK GDSC1 6.0015 8.1091 2.6613 0.7373
SCC-25 GDSC1 6.002 7.7484 2.7911 0.3498
SAT [Human HNSCC] GDSC1 6.0239 11.1137 1.4106 7.6652
BICR 10 GDSC1 6.0443 7.6422 2.8431 0.2228
CAL-33 GDSC1 6.0478 7.842 2.7752 0.371
BICR 78 GDSC1 6.3185 8.1047 2.7821 0.2622
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 16 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW1710 GDSC1 3.5008 6.3967 1.9547 10.5058
639V GDSC1 3.882 5.5897 2.6414 3.9928
UM-UC-3 GDSC1 3.9249 5.6612 2.6362 3.9185
647V GDSC1 4.2593 6.3403 2.5328 3.8576
KU-19-19 GDSC1 4.3829 6.8244 2.3848 4.6385
5637 GDSC1 4.6439 6.8133 2.5461 2.9625
J82 GDSC1 5.41 7.4283 2.6716 1.1659
T24 GDSC1 5.4883 7.5167 2.6715 1.0923
BFTC-905 GDSC1 5.5174 6.8306 2.9339 0.1982
HT-1197 GDSC1 5.5325 6.9336 2.9037 0.2583
CAL-29 GDSC1 5.5777 6.9758 2.9055 0.2386
SW780 GDSC1 5.6652 7.3366 2.8108 0.4462
TCCSUP GDSC1 5.6681 7.1195 2.8884 0.2457
HT-1376 GDSC1 6.07 7.8183 2.7916 0.3231
RT-112 GDSC1 6.1128 7.3472 2.9646 0.0518
RT-4 GDSC1 6.2438 7.6834 2.898 0.0992
⏷ Show the Full List of 16 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PA-1 GDSC1 3.479 7.8708 1.2004 16.1367
C-33 A GDSC1 3.9169 5.9389 2.497 4.9936
ACC-OV7 GDSC1 3.9951 6.4721 2.2932 6.3259
OV17R GDSC1 4.1427 6.3579 2.4493 4.7528
PEO1 GDSC1 4.1953 7.2372 2.0627 7.5037
NEC8 GDSC1 4.3041 8.5579 1.4968 11.3303
BPH-1 GDSC1 4.3865 6.5653 2.5073 3.7533
HeLa GDSC1 4.4097 5.5241 2.9738 0.7481
JAR GDSC1 4.4277 6.3423 2.6332 2.7935
NT2-D1 GDSC1 4.9527 8.8875 1.7809 7.5867
HEC-1 GDSC1 4.9719 6.5115 2.8364 0.8321
OVCA433 GDSC1 5.0038 6.8184 2.7293 1.3165
OVCA420 GDSC1 5.0393 8.6694 1.9368 6.3072
KGN GDSC1 5.0567 8.3397 2.0984 5.1629
SW954 GDSC1 5.0879 7.7802 2.3661 3.3306
C-4-I GDSC1 5.1713 7.0955 2.6957 1.2975
OVMIU GDSC1 5.1995 9.1037 1.8346 6.6504
LB831-BLC GDSC1 5.2068 7.3359 2.6152 1.6726
SKN GDSC1 5.25 7.3885 2.6143 1.6243
SiHa GDSC1 5.2628 6.5521 2.9381 0.2793
NCC-IT GDSC1 5.2667 6.9166 2.8067 0.7095
SKG-IIIa GDSC1 5.3032 7.193 2.7164 1.0633
Ca Ski GDSC1 5.3129 10.0175 1.4807 8.7695
DoTc2 4510 GDSC1 5.3267 7.1368 2.7483 0.901
OMC-1 [Human cervical carcinoma] GDSC1 5.3442 7.3283 2.6816 1.1843
HT-3 GDSC1 5.4721 7.6056 2.6297 1.3006
JEG-3 GDSC1 5.5599 6.9916 2.8935 0.2721
MS751 GDSC1 5.6923 7.3842 2.8041 0.4524
UWB1.289 GDSC1 5.6942 11.3523 1.0981 10.3318
DSH1 GDSC1 5.7847 7.5607 2.7761 0.4887
HEY GDSC1 5.8305 7.934 2.6571 0.87
SW962 GDSC1 5.8557 7.4674 2.8356 0.2988
ME-180 GDSC1 5.8612 8.119 2.6 1.0751
SW756 GDSC1 5.9037 7.3356 2.8979 0.1618
CAL-39 GDSC1 5.9439 8.1845 2.6098 0.9695
JHOS-3 GDSC1 5.9552 8.2061 2.6063 0.9744
SiSo GDSC1 6.1767 8.5079 2.5842 0.8974
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug

References

1 The ChEMBL database in 2017. Nucleic Acids Res. 2017 Jan 4;45(D1):D945-D954.