General Information of Drug (ID: DMSI8N3)

Drug Name
CI-1033
Synonyms
Canertinib; Canertinib HCl; Canertinib dihydrochloride; Canertinib dihydrochloride [USAN]; CI1033; PD 183805; Canertinib dihydrochloride (USAN); PD-0183805; PD-183805; Canertinib, PD-183805, CI1033, PD183805; N-[4-(3-Chloro-4-fluorophenylamino)-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]acrylamide dihydrochloride; N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-[3-(4-morpholinyl)propoxy]-6-quinazolinyl]-2-propenamide dihydrochloride; N-[4-(3-chloro-4-fluoroanilino)-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]prop-2-enamide; N-[4-(3-chloro-4-fluoroanilino)-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]prop-2-enamide dihydrochloride; N-(4-(3-chloro-4-fluorophenyl)amino)-7-(3-morpholin-4-yl)propoxy)quinazolin-6-yl)prop-2-enamide dihydrochloride; N-{4-[(3-chloro-4-fluorophenyl)amino]-7-[3-(morpholin-4-yl)propoxy]quinazolin-6-yl}prop-2-enamide; N-(4-((3-Chloro-4-fluorophenyl)amino)-7-(3-(morpholin-4-yl)propoxy)quinazolin-6-yl)prop-2-enamide; 2-Propenamide, N-(4-((3-chloro-4-fluorophenyl) amino)-7-(3-(4-morpholinyl) propoxy)-6-quinazolinyl)-, dihydrochloride; 2-Propenamide, N-(4-((3-chloro-4-fluorophenyl)amino)-7-(3-(4-morpholinyl)propoxy)-6-quinazolinyl)-, dihydrochloride
Indication
Disease Entry ICD 11 Status REF
Lymphoma 2A80-2A86 Phase 2 [1]
Therapeutic Class
Anticancer Agents
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 485.9
Logarithm of the Partition Coefficient (xlogp) 3.9
Rotatable Bond Count (rotbonds) 9
Hydrogen Bond Donor Count (hbonddonor) 2
Hydrogen Bond Acceptor Count (hbondacc) 8
Chemical Identifiers
Formula
C24H25ClFN5O3
IUPAC Name
N-[4-(3-chloro-4-fluoroanilino)-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]prop-2-enamide
Canonical SMILES
C=CC(=O)NC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC(=C(C=C3)F)Cl)OCCCN4CCOCC4
InChI
InChI=1S/C24H25ClFN5O3/c1-2-23(32)30-21-13-17-20(14-22(21)34-9-3-6-31-7-10-33-11-8-31)27-15-28-24(17)29-16-4-5-19(26)18(25)12-16/h2,4-5,12-15H,1,3,6-11H2,(H,30,32)(H,27,28,29)
InChIKey
OMZCMEYTWSXEPZ-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
156414
ChEBI ID
CHEBI:61399
CAS Number
267243-28-7
UNII
C78W1K5ASF
DrugBank ID
DB05424
TTD ID
D0YB3W
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Epidermal growth factor receptor (EGFR) TTGKNB4 EGFR_HUMAN Inhibitor [2]
Erbb2 tyrosine kinase receptor (HER2) TT6EO5L ERBB2_HUMAN Inhibitor [2]
Erbb4 tyrosine kinase receptor (Erbb-4) TT0JESD ERBB4_HUMAN Inhibitor [2]
RAC-alpha serine/threonine-protein kinase (AKT1) TTWTSCV AKT1_HUMAN Inhibitor [2]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Epidermal growth factor receptor (EGFR) OTAPLO1S EGFR_HUMAN Gene/Protein Processing [3]
Interleukin-8 (CXCL8) OTS7T5VH IL8_HUMAN Gene/Protein Processing [4]
Transforming growth factor beta-1 proprotein (TGFB1) OTV5XHVH TGFB1_HUMAN Gene/Protein Processing [5]
Vascular endothelial growth factor A, long form OTIM9MZ3 VEGFA_HUMAN Gene/Protein Processing [4]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Lymphoma
ICD Disease Classification 2A80-2A86
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
RAC-alpha serine/threonine-protein kinase (AKT1) DTT AKT1 2.63E-29 0.65 1.45
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1 6.142 11.1946 2.2584 10.3437
NOS-1 [Human HNSCC] GDSC1 -0.3184 2.0416 -0.3466 57.6059
ES5 GDSC1 -0.0018 5.191 -0.6597 52.7865
EW-13 GDSC1 0.5832 3.0589 0.5044 46.9184
ES7 GDSC1 0.7018 3.4559 0.5695 45.6315
U2OS GDSC1 0.778 3.7819 0.5873 44.8882
ES4 GDSC1 0.8517 8.5196 -1.0811 46.5771
H-EMC-SS GDSC1 0.9143 3.5427 0.7831 43.1195
HuO9 GDSC1 1.0364 3.0686 0.9848 41.3254
EW-16 GDSC1 1.367 4.9532 0.905 39.1212
NY GDSC1 1.4 4.5856 1.0574 38.2536
ES1 GDSC1 1.4665 4.1744 1.2447 36.9064
EW-18 GDSC1 1.505 3.6049 1.4096 35.7706
MHH-ES-1 GDSC1 1.6058 2.8394 1.5969 34.007
EW-7 GDSC1 1.6525 5.1257 1.1554 36.0514
SK-ES-1 GDSC1 1.692 6.1477 0.8075 37.2665
A-673 GDSC1 1.7799 2.6253 1.7788 31.7824
CADO-ES1 GDSC1 1.8554 3.5197 1.7991 31.1835
A-673 CTRP2 2.0664 2.8476 2.0664 26.5021
SaOS-2 CTRP2 2.1791 4.0455 2.1613 25.8108
EW-3 GDSC1 2.2338 3.9987 2.1225 26.8151
TC71 CTRP2 2.2984 3.016 2.2983 24.9567
EW-22 GDSC1 2.3299 4.3028 2.1531 26.0458
SK-ES-1 CTRP2 2.3627 3.1409 2.3627 24.5282
EW-24 GDSC1 2.5202 17.5807 -3.863 42.2633
CAL-78 GDSC1 2.6276 3.3305 2.6244 21.1996
CHSA8926 GDSC1 2.7559 5.9197 2.014 24.5977
SaOS-2 GDSC1 2.8554 7.1297 1.5652 26.8775
HuO-3N1 GDSC1 2.8559 7.1647 1.5493 26.967
EW-1 GDSC1 2.8819 7.7634 1.2914 28.2701
SJSA-1 CTRP2 2.9228 14.911 -1.7521 31.1219
HOS GDSC1 3.24 6.7106 2.1387 21.3379
MG-63 CTRP2 3.2541 5.0303 3.2044 18.7576
SK-PN-DW GDSC1 3.3203 6.8485 2.1506 20.8781
SJSA-1 GDSC1 3.3551 4.3707 3.2531 12.7575
G-292 clone A141B1 CTRP2 3.4377 4.9108 3.4108 17.4569
G-292 clone A141B1 GDSC1 3.4974 5.457 2.9765 14.0276
MG-63 GDSC1 3.7242 5.0058 3.4086 9.7075
Hs 888.T CTRP2 3.8515 7.6394 3.0843 17.4399
CAL-78 CTRP2 3.9074 8.9036 2.5945 19.1805
ES8 GDSC1 4.4134 10.1841 1.4667 20.7149
CAL-72 GDSC1 5.1133 10.5645 1.8332 16.0584
ES6 GDSC1 5.2645 9.7494 2.348 12.1512
SK-N-MC CTRP2 5.4127 8.3657 3.6798 5.4246
TC-71 GDSC1 6.1053 8.0568 3.6486 1.3985
Hs 822.T CTRP2 6.6765 15.047 2.0585 15.1588
SW1353 CTRP2 8.3467 10.0113 5.5013 0.2361
HOS CTRP2 9.0065 14.8358 3.8032 4.9861
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 283 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 0.4888 2.6553 0.4695 32.5851
JM1 CTRP2 1.4044 3.0457 1.4014 30.9224
JM1 GDSC1 2.1247 3.5983 2.0758 27.7751
EoL-1 CTRP2 -4.571 -2.6564 -4.571 70.6842
DoHH2 GDSC1 -2.8068 1.2566 -2.8835 78.38
SU-DHL-6 CTRP2 -2.0377 5.3741 -2.6023 53.0918
MV4-11 CTRP2 -1.0979 2.0132 -1.1161 47.6075
BL-70 CTRP2 -1.0823 12.9334 -4.2934 48.6675
SU-DHL-6 GDSC1 -0.898 2.8214 -1.0464 62.4532
Mono-Mac-1 CTRP2 -0.7855 2.2566 -0.8053 45.543
MV4-11 GDSC1 -0.5001 1.0438 -0.5015 60.1893
SIG-M5 GDSC1 -0.4585 1.2843 -0.4623 59.6095
EoL-1 GDSC1 -0.3867 0.9032 -0.3871 58.834
GA-10 CTRP2 -0.2648 2.815 -0.2956 42.1173
MOLM-13 CTRP2 -0.2061 1.8475 -0.2085 41.6492
Ramos.2G6.4C10 GDSC1 -0.0674 4.1726 -0.4283 53.7736
Mono-Mac-6 CTRP2 -0.0483 18.6991 -5.8737 46.1168
LAMA-84 GDSC1 0.0578 2.9119 -0.0362 53.0095
MOLM-6 CTRP2 0.0703 2.071 0.0677 39.8085
Ku812 CTRP2 0.0745 2.2911 0.069 39.7898
OCI-AML-2 GDSC1 0.0875 2.0886 0.0702 52.8583
SU-DHL-5 GDSC1 0.1772 3.3896 0.0148 51.5886
MOLM-16 CTRP2 0.3 2.9561 0.2793 38.3352
ALL-PO GDSC1 0.3279 2.7775 0.2675 49.9297
ALL-SIL GDSC1 0.3615 1.7587 0.359 49.507
KMS-20 CTRP2 0.4169 3.9007 0.3283 37.7619
BV-173 GDSC1 0.4985 2.4424 0.4753 47.8408
PF-382 GDSC1 0.5395 3.2478 0.4299 47.485
NU-DUL-1 CTRP2 0.5961 2.4889 0.5931 36.3072
NU-DUL-1 GDSC1 0.5991 3.6031 0.4304 46.8897
EM-2 GDSC1 0.6393 3.0532 0.5649 46.2387
MY-M12 GDSC1 0.641 3.2688 0.5356 46.2867
SEM CTRP2 0.6765 4.1057 0.5794 36.0685
OCI-Ly19 GDSC1 0.6929 3.2063 0.6009 45.6393
CTV-1 GDSC1 0.7125 2.7187 0.6781 45.2418
HAL-01 GDSC1 0.7493 3.4022 0.6301 45.0408
MEG-01 GDSC1 0.7592 3.241 0.6667 44.8489
NK-92MI GDSC1 0.7749 2.3076 0.7664 44.3765
QIMR-WIL GDSC1 0.7827 2.4157 0.7701 44.296
Pfeiffer CTRP2 0.7951 2.0118 0.7951 34.9716
RS4;11 CTRP2 0.8401 2.8145 0.8236 30.0679
Karpas-620 GDSC1 0.8559 2.4701 0.8429 43.3878
Ku812 GDSC1 0.8741 3.1895 0.797 43.4145
SUP-B15 GDSC1 0.8951 2.9089 0.8526 43.0263
NCI-H929 CTRP2 0.9193 3.7649 0.8707 34.3032
SU-DHL-16 GDSC1 0.9736 1.7395 0.9735 41.8547
KE-37 GDSC1 1.0141 2.6381 0.9975 41.4363
MOLT-16 GDSC1 1.018 2.5719 1.0049 41.3701
MHH-CALL-4 CTRP2 1.0415 5.2572 0.7777 34.1698
PF-382 CTRP2 1.0682 2.8179 1.0651 33.1623
Daudi CTRP2 1.0922 2.7401 1.0902 32.9989
TALL-1 [Human adult T-ALL] CTRP2 1.1045 3.5228 1.0801 32.9914
NALM-6 CTRP2 1.1174 3.8353 1.0721 32.9741
MOLM-13 GDSC1 1.1322 2.5918 1.1213 39.934
EM-2 CTRP2 1.1459 2.3843 1.1457 32.6353
697 CTRP2 1.1489 2.2156 1.1489 32.6146
KE-37 CTRP2 1.165 2.1027 1.165 32.5072
OCI-AML-5 GDSC1 1.1664 4.5406 0.8161 40.9562
MOLT-16 CTRP2 1.1838 2.5357 1.1834 32.3833
P31/FUJ CTRP2 1.1888 2.1997 1.1888 32.3485
GDM-1 GDSC1 1.1977 3.438 1.1067 39.5276
MOLP-8 GDSC1 1.2086 2.868 1.1845 39.0534
ST486 CTRP2 1.2095 2.6117 1.2089 32.2129
Ri-1 CTRP2 1.2115 3.1531 1.2041 32.2223
A4/Fukuda GDSC1 1.231 3.4138 1.1462 39.0897
KMS-12-BM CTRP2 1.2461 2.7883 1.2446 31.9722
THP-1 CTRP2 1.251 2.927 1.2481 31.9439
CCRF-CEM GDSC1 1.2584 2.817 1.2398 38.4025
P30/OHK GDSC1 1.2801 2.9826 1.2502 38.1955
JVM-3 CTRP2 1.2842 2.8465 1.2824 31.7193
SU-DHL-8 CTRP2 1.3136 7.2128 0.228 30.4803
HDLM-2 CTRP2 1.3158 6.6547 0.7053 33.4301
KMS-11 CTRP2 1.3173 4.167 1.2513 31.712
Mino CTRP2 1.3414 2.6579 1.341 31.3333
OPM-2 CTRP2 1.3441 2.2724 1.3441 31.3142
MOLT-13 GDSC1 1.348 4.2379 1.099 38.4479
NKM-1 GDSC1 1.3849 3.6468 1.2725 37.3406
P32/ISH GDSC1 1.3876 3.4387 1.3104 37.1206
697 GDSC1 1.3927 3.0928 1.3584 36.8187
HuT 78 CTRP2 1.397 3.4106 1.3855 30.9999
KYO-1 CTRP2 1.4148 3.1302 1.4107 30.8568
RCH-ACV CTRP2 1.4201 3.5023 1.4058 30.8557
KMS-34 CTRP2 1.4371 2.767 1.4365 30.6967
AML-193 CTRP2 1.4421 3.1755 1.4375 30.6763
Loucy GDSC1 1.463 2.6987 1.456 35.7796
Karpas-231 GDSC1 1.4673 3.8686 1.3177 36.5274
EB1 CTRP2 1.4753 2.6875 1.475 30.4408
SUP-T1 CTRP2 1.4908 4.8435 1.3438 30.8275
OCI-AML-3 CTRP2 1.5179 2.4207 1.5179 30.1559
Hs 611.T CTRP2 1.5323 2.9691 1.5263 25.0897
OCI-M1 GDSC1 1.5395 2.8596 1.5279 34.8523
Kasumi-2 CTRP2 1.5663 3.6118 1.5512 29.884
JURL-MK1 CTRP2 1.5792 2.9825 1.578 29.7519
ML-2 GDSC1 1.5865 2.9885 1.5692 34.2997
HT CTRP2 1.5893 2.594 1.5893 29.6804
CA46 GDSC1 1.5948 5.4371 0.981 37.2143
RCH-ACV GDSC1 1.6032 4.059 1.4224 35.0364
SET-2 CTRP2 1.6242 2.915 1.6236 29.4501
KMS-21-BM CTRP2 1.6325 3.3889 1.6261 29.4143
KHM-1B CTRP2 1.6363 3.9148 1.6072 29.4649
DND-41 CTRP2 1.6376 4.828 1.5043 29.8067
MOLT-3 CTRP2 1.6445 2.3815 1.6445 29.313
SUP-T11 CTRP2 1.6474 3.6471 1.633 29.3418
NALM-6 GDSC1 1.6475 2.8817 1.638 33.4894
KMS-26 CTRP2 1.6588 3.1105 1.6571 29.2229
KMS-27 CTRP2 1.6693 2.442 1.6693 29.1477
Reh GDSC1 1.673 3.7215 1.5701 33.7356
SU-DHL-10 CTRP2 1.6965 3.49 1.6699 23.9919
H9 GDSC1 1.7019 4.0685 1.5276 33.7926
Karpas-45 GDSC1 1.7105 3.352 1.6665 32.915
SUP-B15 CTRP2 1.7332 3.0995 1.732 28.7259
PL-21 GDSC1 1.7419 5.2111 1.2217 35.1409
HEL GDSC1 1.7477 3.7366 1.6481 32.7892
MOTN-1 CTRP2 1.7518 2.6252 1.7518 28.5977
CA46 CTRP2 1.7689 4.4099 1.7022 28.7083
SR GDSC1 1.7704 3.5914 1.6974 32.3456
Jurkat GDSC1 1.7954 3.7491 1.6973 32.1882
RPMI-8402 GDSC1 1.7985 4.209 1.5981 32.7595
KG-1 GDSC1 1.8193 5.5554 1.177 34.852
K-562 GDSC1 1.8291 3.5357 1.7687 31.5371
DB CTRP2 1.8589 3.5498 1.8523 27.9064
OPM-2 GDSC1 1.8656 4.0683 1.706 31.6913
SU-DHL-4 CTRP2 1.8664 7.5422 0.6776 27.1337
BV-173 CTRP2 1.8862 5.2941 1.6871 28.3773
Farage GDSC1 1.9016 3.1223 1.8875 30.3423
NB4 GDSC1 1.9115 2.9071 1.9071 30.1583
DEL CTRP2 1.914 2.5025 1.914 27.517
BC-1 GDSC1 1.9237 3.2822 1.8986 30.1353
SKM-1 GDSC1 1.9411 4.1741 1.7625 30.8756
SU-DHL-10 GDSC1 1.951 2.4814 1.951 29.637
U-937 CTRP2 1.9735 4.0328 1.9494 27.2015
WIL2 NS GDSC1 1.9859 3.9034 1.8734 29.9099
KO52 CTRP2 1.9874 2.8885 1.9874 27.0283
L-363 GDSC1 1.9964 3.7484 1.9145 29.5863
CTB-1 GDSC1 2.0102 7.3351 0.6258 36.0011
HC-1 GDSC1 2.0127 3.4987 1.9696 29.1376
KCL-22 GDSC1 2.0143 4.3001 1.8095 30.1342
ST486 GDSC1 2.0279 3.8149 1.9364 29.2545
M-07e CTRP2 2.0285 6.1838 1.6229 28.1406
Granta-519 CTRP2 2.0298 3.146 2.0271 21.5266
SR CTRP2 2.0311 4.3388 1.9861 26.8886
L-363 CTRP2 2.0616 15.8455 -2.4722 37.6593
RS4;11 GDSC1 2.0683 4.7707 1.7268 30.3093
VAL GDSC1 2.0716 3.9836 1.9495 28.9044
MOLP-2 CTRP2 2.0934 6.2258 1.6817 27.7332
RPMI-8866 GDSC1 2.0995 3.5082 2.0607 28.0252
A3/Kawakami GDSC1 2.1046 3.846 2.0135 28.2954
SU-DHL-8 GDSC1 2.1081 5.3598 1.5602 31.0453
MHH-CALL-3 CTRP2 2.1118 8.5134 0.8946 30.246
JeKo-1 CTRP2 2.1257 2.8113 2.1257 26.1069
HDLM-2 GDSC1 2.1298 4.6633 1.8283 29.3154
L-540 CTRP2 2.1436 3.6109 2.1398 26.0004
HL-60 GDSC1 2.1556 3.6273 2.1048 27.4008
MLMA GDSC1 2.1703 2.9764 2.1683 26.9077
RPMI-6666 GDSC1 2.1999 3.9346 2.0991 27.1697
Kasumi-1 CTRP2 2.2078 5.3585 1.8575 21.5687
LP-1 GDSC1 2.2163 3.2617 2.205 26.3916
ME1 CTRP2 2.2222 7.2612 1.4873 27.9916
JJN-3 CTRP2 2.2457 14.7893 -1.7911 36.0898
NU-DHL-1 CTRP2 2.254 3.2367 2.2538 25.2531
Namalwa CTRP2 2.2653 3.4956 2.264 25.1809
L-428 CTRP2 2.2763 3.9007 2.2674 25.1333
SIG-M5 CTRP2 2.277 2.8324 2.277 25.0991
F-36P CTRP2 2.2921 3.5114 2.2908 25.0025
HD-MY-Z CTRP2 2.3016 3.4959 2.3005 24.9389
GA-10 GDSC1 2.3156 3.4782 2.2923 25.2264
HL-60 CTRP2 2.316 3.4856 2.315 24.8423
U266B1 CTRP2 2.3281 16.7829 -2.6673 37.2428
P12-Ichikawa CTRP2 2.3449 3.2697 2.3448 24.6468
SUP-T1 GDSC1 2.3621 3.4009 2.3473 24.5909
NOMO-1 GDSC1 2.3805 3.4952 2.3588 24.4047
MC116 CTRP2 2.4003 10.0533 0.0991 27.4844
JSC-1 GDSC1 2.4231 4.3094 2.2531 24.8412
PL21 CTRP2 2.4333 7.3798 1.6724 26.7108
MOLT-4 GDSC1 2.4457 3.5937 2.4177 23.6298
OCI-AML-5 CTRP2 2.4915 2.9106 2.4915 23.6699
JURL-MK1 GDSC1 2.5068 4.0237 2.4137 23.2896
KMS-18 CTRP2 2.5245 4.1949 2.5098 23.4995
RL CTRP2 2.5255 3.2107 2.5255 23.4433
HPB-ALL CTRP2 2.5301 4.0883 2.5202 23.4459
TUR GDSC1 2.5441 3.7392 2.5042 22.4764
A3/Kawakami CTRP2 2.5592 3.0022 2.5592 23.2191
OCI-M1 CTRP2 2.6082 3.0795 2.6082 22.8922
Hs 445 GDSC1 2.6405 4.003 2.5631 21.5162
KMOE-2 GDSC1 2.6704 4.584 2.4418 22.1588
ROS-50 GDSC1 2.697 5.9158 1.9549 25.2969
KY821 GDSC1 2.7171 3.3945 2.7137 20.0816
L-428 GDSC1 2.762 4.411 2.5944 20.6032
Mono-Mac-6 GDSC1 2.7702 5.1308 2.355 22.2074
RPMI-8226 GDSC1 2.7975 5.8136 2.1028 23.7881
SUP-M2 GDSC1 2.8372 4.1137 2.7534 19.1018
KOPN-8 GDSC1 2.843 4.8557 2.5362 20.5546
P12-Ichikawa GDSC1 2.8773 3.6546 2.8656 18.1317
SUP-HD1 GDSC1 2.9172 5.2766 2.4531 20.7422
THP-1 GDSC1 2.923 7.5784 1.4192 27.3696
IM-9 GDSC1 3.044 3.917 3.0133 16.1694
CESS GDSC1 3.0509 5.999 2.2806 21.2728
Daudi GDSC1 3.1191 10.9474 -0.0398 32.8564
HH [Human lymphoma] GDSC1 3.1675 7.6262 1.631 24.9549
BE-13 GDSC1 3.2212 4.5614 3.0477 14.9201
Sc-1 GDSC1 3.2483 5.8762 2.5354 18.4849
SU-DHL-1 GDSC1 3.2749 3.8931 3.2616 13.1715
LC4-1 GDSC1 3.2826 4.678 3.0737 14.4041
U266B1 GDSC1 3.2849 4.4256 3.1603 13.7881
EJM GDSC1 3.2971 4.9418 2.9893 14.9298
MC116 GDSC1 3.3795 4.0183 3.3576 11.9201
ME1 GDSC1 3.3867 6.4739 2.3933 18.8596
SCC-3 GDSC1 3.4342 4.0909 3.4051 11.2828
Jiyoye GDSC1 3.4747 4.5916 3.3118 11.6895
BALL-1 GDSC1 3.4791 4.6214 3.3059 11.7077
HT GDSC1 3.5002 4.2171 3.4515 10.587
U-698-M GDSC1 3.5554 5.7733 2.8886 14.4153
DEL GDSC1 3.568 6.6451 2.4847 17.3739
P3HR-1 CTRP2 3.5916 8.6487 1.9239 17.3068
KMS-11 GDSC1 3.6927 6.3339 2.7532 14.824
MHH-PREB-1 GDSC1 3.7548 7.5584 2.2098 18.5383
Raji GDSC1 3.7809 5.4548 3.2593 10.5699
RPMI-8226 CTRP2 3.7811 7.9016 2.9018 18.3337
P31/FUJ GDSC1 3.81 4.1668 3.7966 6.4846
YT GDSC1 3.8307 5.3588 3.3532 9.6268
KM-H2 GDSC1 3.8343 4.35 3.7819 6.4412
Granta-519 GDSC1 3.8386 4.5892 3.7033 6.9705
Toledo CTRP2 3.9023 10.5214 1.8411 22.011
L-1236 GDSC1 3.944 6.254 3.0253 11.6732
EJM CTRP2 4.0166 7.5059 3.3127 16.1089
OCI-Ly19 CTRP2 4.1604 7.2399 3.5722 14.714
GR-ST GDSC1 4.1804 7.6693 2.5289 14.5214
EHEB CTRP2 4.1967 10.0467 2.3523 19.371
JJN-3 GDSC1 4.2105 10.0574 1.3608 22.0872
BL-41 GDSC1 4.2874 5.9708 3.4686 6.856
KMS-12-BM GDSC1 4.3216 6.5999 3.1826 8.9806
SK-MM-2 GDSC1 4.3346 5.6759 3.6555 5.2102
SUP-HD1 CTRP2 4.3849 7.9844 2.9942 10.6902
TK [Human B-cell lymphoma] GDSC1 4.5495 5.9859 3.6711 4.3649
Karpas-422 CTRP2 4.5642 9.0632 2.6221 11.9244
ATN-1 GDSC1 4.6355 8.0519 2.7114 11.5183
SU-DHL-4 GDSC1 4.6996 6.5821 3.4891 5.3203
BC-3 GDSC1 4.771 6.7941 3.4371 5.5091
EB2 GDSC1 4.7767 6.7193 3.4778 5.1791
WSU-DLCL2 GDSC1 4.8156 6.8415 3.4461 5.31
LP-1 CTRP2 4.8258 8.2796 3.2412 8.5822
Karpas-299 CTRP2 4.8734 12.908 1.5937 20.5505
DG-75 GDSC1 5.0162 7.071 3.474 4.5503
VL51 GDSC1 5.2198 7.1014 3.5901 3.2157
OCI-AML-3 GDSC1 5.2266 8.0923 3.127 6.59
L-540 GDSC1 5.2324 9.6915 2.3529 12.214
DB GDSC1 5.2977 12.7718 0.8801 20.8752
MN-60 GDSC1 5.3068 8.349 3.0583 6.887
NOMO-1 CTRP2 5.6662 15.921 0.7875 21.5136
RPMI-6666 CTRP2 5.6933 7.0862 5.2082 4.2571
OCI-Ly3 CTRP2 5.8096 8.3379 3.9835 3.4078
Karpas-620 CTRP2 5.9033 12.0671 2.9147 13.3373
WSU-NHL GDSC1 5.9111 7.5359 3.7675 1.0192
RC-K8 GDSC1 6.2049 7.4247 3.9279 0.2297
Karpas-299 GDSC1 6.2375 7.7408 3.8272 0.5051
GDM-1 CTRP2 6.2609 14.4613 2.015 16.1071
Karpas-422 GDSC1 6.3265 13.3053 1.3712 15.2698
AMO1 GDSC1 6.3342 7.615 3.9087 0.2273
JVM-2 GDSC1 6.3551 9.414 3.2041 3.6198
RL GDSC1 6.4789 7.8577 3.8769 0.2483
JVM-3 GDSC1 6.6361 8.2384 3.8013 0.3738
EHEB GDSC1 6.6843 8.2298 3.8222 0.3007
DND-41 GDSC1 6.7692 13.6073 1.5262 13.2693
Raji CTRP2 6.7983 10.8115 4.2562 6.1783
ARH-77 GDSC1 7.0194 8.4082 3.8794 0.11
MM1.S CTRP2 7.049 9.0633 5.2673 1.7612
OCI-Ly10 CTRP2 7.2032 9.8992 4.0926 1.3911
CMK CTRP2 7.3073 13.5182 2.5125 7.4203
HEL 92.1.7 CTRP2 7.5376 8.7158 5.6564 0.2141
BL-41 CTRP2 7.5388 8.6767 5.6712 0.1874
TF-1 CTRP2 7.5867 8.9029 5.6068 0.293
NB4 CTRP2 7.6293 8.7459 5.681 0.1465
OCI-AML-2 CTRP2 7.8448 8.918 5.6997 0.0806
K-562 CTRP2 7.8558 9.2401 5.5902 0.2303
KE-97 CTRP2 7.9359 9.4495 5.5452 0.2855
Reh CTRP2 7.9651 15.995 2.5648 11.0735
Jurkat CTRP2 7.9975 9.431 5.576 0.2125
HEL CTRP2 8.2194 9.4847 5.6387 0.0868
LAMA-84 CTRP2 8.2247 13.1162 4.1182 4.7225
KMM-1 CTRP2 8.2269 12.8753 4.231 4.2926
KCL-22 CTRP2 8.2813 13.4513 3.9978 5.1119
KM-H2 CTRP2 8.3555 9.8754 5.5528 0.1603
AMO1 CTRP2 9.9275 24.6062 -0.2333 17.2121
⏷ Show the Full List of 283 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 -3.5912 9.1498 -5.4573 58.0257
TE8 CTRP2 0.2979 10.6084 -2.267 39.9124
OE21 CTRP2 -4.2299 3.7442 -4.6344 64.0322
TE-15 GDSC1 -3.1468 12.9683 -7.1346 61.3432
KYSE-450 GDSC1 -3.0482 4.7799 -3.8509 70.3199
TE-6 CTRP2 -1.2457 8.8971 -3.1541 46.7358
TE-4 CTRP2 -1.1007 12.1023 -3.9587 48.671
TE-6 GDSC1 -0.5972 9.5751 -3.0297 54.6634
KYSE-410 CTRP2 -0.554 6.8329 -1.3865 45.1404
OE19 GDSC1 -0.3999 9.0928 -2.6167 53.8948
EC-GI-10 CTRP2 -0.1759 13.8011 -3.7438 45.4759
TE-14 CTRP2 0.0423 7.6299 -0.9984 42.0788
TE-5 CTRP2 0.1444 6.3002 -0.4661 40.7418
KYSE-140 GDSC1 0.2104 13.9977 -4.2591 50.4299
TE-8 GDSC1 0.2486 7.0787 -1.0925 50.5198
KYSE-150 GDSC1 0.4739 4.356 0.1131 48.4586
TE-5 GDSC1 0.9409 3.0335 0.8877 42.5075
KYSE-140 CTRP2 1.1463 9.7265 -0.6165 37.278
EC-GI-10 GDSC1 1.1675 8.2482 -0.6387 44.1937
TE-11 CTRP2 1.2427 11.7289 -1.3767 38.3578
TE-4 GDSC1 1.2896 6.6258 0.1882 41.8701
KYSE-520 GDSC1 1.3934 8.3849 -0.4712 42.5878
KYSE-270 GDSC1 1.5492 11.2543 -1.6593 43.5268
COLO 680N GDSC1 2.1262 4.1913 1.9601 28.5064
KYSE-150 CTRP2 2.4145 4.0197 2.4044 24.2167
TE-9 GDSC1 2.5341 4.1694 2.4103 23.1514
KYSE-410 GDSC1 2.6694 9.2246 0.3865 33.3928
TE-10 GDSC1 2.906 6.4151 1.946 24.2665
KYSE-70 GDSC1 3.2123 4.3207 3.1113 14.5331
TE-11 GDSC1 3.2553 4.3547 3.1488 14.0337
KYSE-180 GDSC1 3.4063 6.5623 2.3702 18.9357
TE-1 GDSC1 3.5211 5.5006 2.9806 13.8842
T.T GDSC1 3.5448 4.4204 3.445 10.377
KYSE-30 CTRP2 4.3317 16.3865 -0.6152 28.3813
TE-10 CTRP2 4.563 16.4086 -0.4187 27.3603
OE33 GDSC1 4.9755 15.1778 -0.5714 27.9207
KYSE-520 CTRP2 5.3588 20.5342 -1.7795 28.7868
COLO 680N CTRP2 5.7364 16.8724 0.3716 22.6388
KYSE-510 CTRP2 5.7443 12.9502 2.3384 15.9217
TE-1 CTRP2 6.1377 13.6987 2.2947 15.2994
KYSE-510 GDSC1 6.8515 14.7329 1.0438 15.6804
OE19 CTRP2 7.5578 14.8979 2.8068 10.7939
OE33 CTRP2 7.6679 11.6282 4.4617 4.0929
TE-9 CTRP2 8.1113 9.3556 5.6445 0.0968
OE21 GDSC1 8.1354 16.6102 0.9904 13.0472
KYSE-180 CTRP2 8.5301 20.4352 0.8008 16.2804
KYSE-450 CTRP2 9.1138 24.8951 -0.9613 20.3138
KYSE-70 CTRP2 12.7766 28.4205 -0.1545 13.3809
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 66 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 9.6526 28.6137 -2.3926 22.7885
HuP-T4 CTRP2 -2.1922 8.4861 -3.7124 53.1552
HuP-T4 GDSC1 0.4704 4.6164 0.0346 48.5425
SU.86.86 CTRP2 1.5832 13.8837 -2.0143 38.3226
Capan-1 GDSC1 2.0717 5.1235 1.6086 30.9878
Panc 04.03 GDSC1 2.2352 10.2633 -0.5271 38.2781
Capan-1 CTRP2 2.3815 19.7306 -4.0484 38.8517
PaTu 8988s CTRP2 2.4017 4.575 2.3531 24.4319
SNU-213 CTRP2 2.4371 10.3665 0.4464 30.5674
KP-4 CTRP2 2.4865 3.2488 2.4865 23.7034
HuP-T3 CTRP2 2.4934 4.8729 2.4148 23.9238
MIA PaCa-2 CTRP2 2.5735 3.1855 2.5735 23.1234
SW1990 CTRP2 2.5967 11.3076 0.1831 30.8219
Panc 03.27 GDSC1 2.775 8.1514 1.0032 30.2582
HPAC GDSC1 2.8816 8.3636 1.0035 29.7287
Capan-2 CTRP2 2.9067 8.3399 1.8035 24.8501
SUIT-2 GDSC1 2.9651 8.3923 1.069 29.0026
MZ-PC-1 GDSC1 3.0283 5.335 2.5459 19.5067
KP-4 GDSC1 3.0751 4.6728 2.8515 17.0896
BxPC-3 CTRP2 3.1397 10.2792 1.1973 26.2594
BxPC-3 GDSC1 3.3132 11.0429 0.0877 31.5874
HuP-T3 GDSC1 3.4198 4.7382 3.199 12.7826
KP-1N GDSC1 3.5704 5.8968 2.8452 14.6737
MIA PaCa-2 GDSC1 3.6517 4.4697 3.5454 9.0895
SU.86.86 GDSC1 3.718 4.3524 3.6543 7.969
KP-2 CTRP2 3.7475 5.7228 3.6177 15.7501
CFPAC-1 GDSC1 3.7519 4.3306 3.6974 7.4836
L3.3 CTRP2 3.7809 12.2075 0.9202 25.4422
QGP-1 GDSC1 4.0043 5.2701 3.5627 7.2474
Panc 08.13 GDSC1 4.0229 6.5645 2.9427 11.9929
Panc 04.03 CTRP2 4.0385 6.8196 3.6036 14.9357
PSN1 CTRP2 4.0428 6.2773 3.7922 14.221
Capan-2 GDSC1 4.0762 10.5115 1.0201 24.439
PaTu 8902 GDSC1 4.2836 5.9867 3.4574 6.958
PL4 GDSC1 4.3654 6.8873 3.0753 9.6625
Hs 766T GDSC1 4.6021 6.1718 3.6188 4.6095
HPAF-II GDSC1 4.7425 15.6721 -1.0066 30.0239
Hs 766T CTRP2 5.039 17.9857 -0.7835 27.2163
HPAF-II CTRP2 5.0795 12.6962 1.8837 19.0466
PaTu 8988t GDSC1 5.1389 7.6883 3.2613 5.8208
KP-3 GDSC1 5.2371 12.51 0.9634 20.6449
Panc 10.05 CTRP2 5.351 14.5887 1.1815 20.9049
PaTu 8902 CTRP2 5.5586 6.9128 5.1599 4.7756
KP-3 CTRP2 5.5796 11.4706 2.9348 13.9178
PSN1 GDSC1 6.5567 8.4636 3.6879 0.7961
Panc 03.27 CTRP2 6.6531 14.9529 2.0867 15.0979
DAN-G GDSC1 6.7406 8.1781 3.8604 0.2003
PK-45H CTRP2 6.7419 10.8528 4.1938 6.5289
Panc 10.05 GDSC1 6.9287 8.6699 3.758 0.3624
AsPC-1 CTRP2 6.9731 18.2605 0.6919 19.2646
PK-59 CTRP2 7.1125 20.9171 -0.5217 22.4865
SNU-410 CTRP2 7.2112 14.9518 2.5218 12.4652
Panc 02.03 GDSC1 7.287 25.771 -4.043 30.7151
SW1990 GDSC1 7.2986 9.0006 3.7767 0.2053
DAN-G CTRP2 7.3303 18.0661 1.0687 17.4217
PaTu 8988t CTRP2 7.5533 8.7969 5.6328 0.2534
YAPC CTRP2 7.7188 9.9993 5.2264 1.2563
HPAC CTRP2 7.9701 9.522 5.5321 0.2983
QGP-1 CTRP2 8.3596 10.0685 5.4857 0.2575
TCC-Pan2 CTRP2 8.4134 9.8648 5.5774 0.1202
Panc 05.04 CTRP2 8.4651 39.1281 -8.5259 33.2872
CFPAC-1 CTRP2 8.527 10.3008 5.4664 0.2428
SUIT-2 CTRP2 8.5653 9.8582 5.6325 0.0537
Panc 02.03 CTRP2 8.593 15.7761 3.1035 8.1203
YAPC GDSC1 9.2982 19.7905 0.2364 14.2157
AsPC-1 GDSC1 9.3839 20.5126 -0.0445 15.2139
⏷ Show the Full List of 66 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 105 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 6.668 17.2146 0.2537 17.1467
CHL-1 GDSC1 -1.8205 8.3377 -3.7857 60.7526
A-431 GDSC1 -0.7506 3.9105 -1.1071 59.778
SK-MEL-2 GDSC1 0.7318 2.8647 0.6848 45.0453
A-388 GDSC1 1.1533 6.4392 0.1211 42.9582
DJM-1 GDSC1 1.2674 2.8764 1.2452 38.311
Hs 940.T GDSC1 1.3041 4.8382 0.8743 39.6996
IGR-1 GDSC1 1.4012 2.7482 1.3909 36.5718
COLO 800 GDSC1 1.4899 2.5805 1.4866 35.4209
HT-144 GDSC1 1.4979 2.7174 1.4911 35.342
A-375 GDSC1 1.5883 3.4952 1.5169 34.6003
WM115 GDSC1 1.662 2.6067 1.6602 33.2604
VMRC-MELG GDSC1 1.711 4.7791 1.3357 34.7752
CP50-MEL-B GDSC1 1.8401 2.9368 1.8332 31.0657
MZ-MEL-2 GDSC1 1.853 2.511 1.8528 30.863
MMAc-SF GDSC1 2.0006 2.9064 1.9977 29.0347
Mel JuSo GDSC1 2.006 2.7617 2.0052 28.9545
Mel Ho GDSC1 2.006 2.8373 2.0044 28.9593
Hs 934.T CTRP2 2.1155 3.9922 2.0985 26.2315
WM793 GDSC1 2.1465 3.6489 2.0919 27.5391
COLO 792 GDSC1 2.1647 2.8867 2.1638 26.9714
RPMI-7951 GDSC1 2.171 3.5225 2.1349 27.1151
Hs 688(A).T CTRP2 2.1975 5.2279 2.0376 26.174
RVH-421 GDSC1 2.2442 5.7726 1.542 30.3401
WM1552C GDSC1 2.3125 3.5633 2.2801 25.3226
WM115 CTRP2 2.3128 2.8484 2.3128 24.8604
LOX-IMVI GDSC1 2.3156 3.5684 2.2827 25.2876
WM35 GDSC1 2.3504 3.659 2.3084 24.9106
WM266-4 CTRP2 2.3557 2.8194 2.3557 24.5744
SK-MEL-5 GDSC1 2.4223 3.8047 2.3637 24.12
SK-MEL-30 GDSC1 2.4289 3.2389 2.4246 23.6894
G-361 GDSC1 2.4303 3.6871 2.3899 23.9018
451Lu GDSC1 2.4424 3.5307 2.4207 23.6312
IPC-298 GDSC1 2.4628 3.5622 2.439 23.39
CJM [Human melanoma] CTRP2 2.4826 2.9886 2.4826 23.7294
SK-MEL-24 CTRP2 2.4858 3.7565 2.4834 23.7159
HT-144 CTRP2 2.4906 3.0813 2.4906 23.6758
WM278 GDSC1 2.493 3.4388 2.4809 22.9377
IGR-37 CTRP2 2.5372 2.9712 2.5372 23.3653
Hs 940.T CTRP2 2.5512 10.1611 0.6539 29.6319
Hs 944.T CTRP2 2.556 4.7638 2.4955 23.4446
MeWo CTRP2 2.5593 4.0771 2.5504 23.2481
SK-MEL-28 GDSC1 2.5942 3.0181 2.5941 21.5973
A101D GDSC1 2.5987 3.0742 2.5986 21.5411
Malme-3M CTRP2 2.6207 5.2913 2.4834 23.2788
WM983B CTRP2 2.6239 4.5558 2.5887 22.9064
IST-MEL1 GDSC1 2.6291 3.9098 2.5685 21.549
RPMI-7951 CTRP2 2.6341 3.4238 2.634 22.7204
COLO 783 GDSC1 2.6388 3.7922 2.5979 21.2999
IGR-37 GDSC1 2.7363 3.2135 2.736 19.8221
LB373-MEL-D GDSC1 2.8772 3.4484 2.8752 18.0714
COLO 679 GDSC1 2.9272 4.0696 2.8606 17.8636
SK-MEL-1 GDSC1 2.972 3.5321 2.9695 16.8896
SK-MEL-1 CTRP2 3.001 3.8989 3.0005 20.2774
WM88 CTRP2 3.0028 5.2276 2.907 20.5901
COLO 800 CTRP2 3.0668 5.4337 2.9389 20.2757
RVH-421 CTRP2 3.0754 5.1367 2.9993 20.0384
UACC-62 GDSC1 3.0757 3.5169 3.0749 15.583
A2058 GDSC1 3.0992 3.8046 3.0852 15.3726
Hs 938.T GDSC1 3.1066 3.7987 3.0935 15.2743
SK-MEL-24 GDSC1 3.1434 4.3219 3.0358 15.4375
LB2518-MEL GDSC1 3.2191 3.9619 3.1941 13.9447
G-mel GDSC1 3.2324 4.5776 3.0544 14.8119
MZ-MEL-7 GDSC1 3.2949 4.5496 3.1316 13.9312
Hs 895.T CTRP2 3.3276 5.4893 3.2105 18.5012
UACC-62 CTRP2 3.3908 5.2653 3.318 17.9263
COLO 829 GDSC1 3.4195 4.6069 3.2468 12.4457
M14 GDSC1 3.4287 4.6058 3.2571 12.3232
UACC-257 GDSC1 3.4391 4.0804 3.412 11.2087
SH-4 GDSC1 3.6333 4.3885 3.5512 9.152
SK-MEL-3 GDSC1 3.6875 4.1564 3.6667 8.0636
MeWo GDSC1 3.7625 4.213 3.7373 7.1549
CP66-MEL GDSC1 3.7972 4.3314 3.7467 6.8909
GAK GDSC1 3.8145 4.2913 3.7762 6.5926
HMV-II GDSC1 4.2341 5.4625 3.6769 5.4142
Hs 294T CTRP2 4.3348 8.1198 3.3793 15.0029
SK-MEL-3 CTRP2 4.3788 5.8195 4.2828 11.4276
UACC-257 CTRP2 4.6628 7.7863 3.8618 12.2428
WT2-iPS CTRP2 4.6818 7.0272 4.2085 10.8274
COLO 792 CTRP2 4.8386 10.6943 2.6513 16.6742
WT2-iPS GDSC1 4.8656 7.9753 2.9262 9.1468
Hs 839.T CTRP2 5.4751 13.0366 2.0633 17.5237
SK-MEL-28 CTRP2 6.8283 8.7733 5.2648 2.0368
IGR-1 CTRP2 6.8339 8.5795 5.3588 1.6669
SK-MEL-2 CTRP2 7.0713 16.4032 1.694 15.757
A2058 CTRP2 7.1849 8.1392 5.7279 0.2022
WM793 CTRP2 7.3742 9.6822 5.1778 1.7383
K029AX CTRP2 7.3985 11.8978 4.1548 5.6735
LOX-IMVI CTRP2 7.5149 12.3527 4.0157 6.0638
IPC-298 CTRP2 7.652 9.0907 5.563 0.3593
WM1799 CTRP2 7.6578 9.5882 5.368 0.8656
SK-MEL-30 CTRP2 7.7348 9.0734 5.6034 0.2456
SK-MEL-5 CTRP2 7.8504 9.2156 5.5969 0.2203
HMCB CTRP2 7.8919 9.1348 5.6416 0.1411
Hs 936.T CTRP2 7.8986 9.3043 5.5835 0.2287
MDA-MB-435S CTRP2 7.988 9.3908 5.5868 0.1979
A101D CTRP2 8.0009 9.4998 5.5524 0.2511
IGR-39 CTRP2 8.0271 9.3256 5.6245 0.1351
Mel Ho CTRP2 8.182 9.7011 5.5497 0.2046
Mel JuSo CTRP2 8.2072 10.5522 5.2365 0.8803
A-375 CTRP2 8.3565 9.6727 5.6229 0.0832
Hs 852.T CTRP2 8.3638 9.5679 5.6606 0.0526
SK-MEL-31 CTRP2 8.4542 10.1587 5.4895 0.2263
G-361 CTRP2 8.4762 10.1168 5.5126 0.188
COLO 829 CTRP2 10.6882 26.0451 -0.4004 16.6132
⏷ Show the Full List of 105 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ESO-26 GDSC1 -3.8968 6.6891 -5.3896 69.6581
KYAE-1 GDSC1 -1.6953 3.5337 -2.0477 66.7619
TE-12 GDSC1 -0.1423 9.101 -2.3549 52.5659
KYSE-220 GDSC1 1.3077 11.5465 -2.0314 45.0292
FLO-1 GDSC1 1.8253 4.0542 1.6654 32.1909
OACP4 C GDSC1 1.8442 9.8538 -0.7071 40.5977
HCE-4 GDSC1 2.5691 3.7334 2.5317 22.148
OACM5.1 C GDSC1 2.6184 3.9063 2.5576 21.6841
KYSE-50 GDSC1 3.1345 4.7557 2.8862 16.5236
SK-GT-4 GDSC1 3.9101 12.189 0.0401 29.3899
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1 2.9287 4.0488 2.8664 17.8167
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CHP-212 GDSC1 -0.204 2.1076 -0.2321 56.2758
SK-N-SH GDSC1 0.1944 1.9869 0.1841 51.5703
MHH-NB-11 CTRP2 0.384 3.1362 0.357 37.7958
IMR-5 GDSC1 1.0487 2.8422 1.0197 41.0671
NB69 GDSC1 1.3158 3.4832 1.2263 38.0705
NH-12 GDSC1 1.5569 4.0696 1.3694 35.6363
KP-N-YS GDSC1 1.5763 3.1587 1.5451 34.5112
NB1 GDSC1 1.6227 4.0319 1.45 34.7535
MHH-NB-11 GDSC1 1.7025 5.4725 1.0833 36.0477
SJNB-12 GDSC1 1.7063 3.6044 1.6265 33.1846
SJNB-14 GDSC1 1.729 2.9896 1.7167 32.4882
SJNB-10 GDSC1 1.8211 3.6129 1.7485 31.7123
NB(TU)1 GDSC1 1.9012 4.4515 1.6436 31.8397
SK-N-FI GDSC1 1.9058 3.2522 1.8824 30.3484
GOTO GDSC1 1.9207 3.3291 1.8911 30.2013
GI-ME-N GDSC1 1.9726 3.6739 1.9014 29.8154
SK-N-BE(2) CTRP2 2.0577 7.6323 1.1761 29.5327
SiMa GDSC1 2.1676 4.012 2.0477 27.6951
CHP-134 GDSC1 2.2973 4.0875 2.1717 26.1168
SK-N-DZ CTRP2 2.3123 3.1372 2.3122 24.864
SK-N-AS CTRP2 2.4012 3.9725 2.3924 24.3009
Kelly GDSC1 2.4498 3.585 2.4229 23.5723
CHP-212 CTRP2 2.4502 3.1802 2.4502 23.9449
SK-N-MC-IXC GDSC1 2.6216 3.1689 2.6211 21.2572
KP-N-YN GDSC1 2.774 4.1972 2.6649 20.0593
SJNB-17 GDSC1 2.9088 4.5993 2.696 19.0838
SK-N-SH CTRP2 2.9252 8.3965 1.7996 24.8108
SJNB-13 GDSC1 3.2622 4.168 3.2035 13.6261
LA-N-6 GDSC1 3.4313 4.7539 3.2054 12.6764
SJNB-7 GDSC1 3.5685 4.3148 3.5016 9.8566
SK-N-BE(2)-M17 GDSC1 3.5882 14.8756 -1.5781 35.2877
SJNB-5 GDSC1 3.5976 4.4145 3.5044 9.673
TGW GDSC1 3.8073 4.3512 3.752 6.7976
SK-N-AS GDSC1 3.8964 4.3679 3.8442 5.6651
KP-N-YN CTRP2 4.028 8.5708 2.8661 17.8148
SJNB-6 GDSC1 4.2811 5.5303 3.6834 5.1861
SK-N-DZ GDSC1 4.7087 8.0936 2.7479 10.9986
Kelly CTRP2 7.7157 12.9548 3.8632 6.3854
NB1 CTRP2 7.8974 9.1824 5.6268 0.1606
KP-N-SI9s CTRP2 8.532 21.3682 0.3439 17.6667
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-478 CTRP2 -1.3884 6.391 -2.1645 49.6215
SNU-308 CTRP2 0.5364 10.464 -1.5618 41.0211
HuCC-T1 CTRP2 2.129 6.069 1.7647 27.3353
SNU-869 CTRP2 2.329 4.9054 2.2343 25.0738
HuCC-T1 GDSC1 2.5244 3.885 2.4599 22.8822
HuH-28 CTRP2 3.7671 10.1742 1.8711 22.2515
SNU-1196 CTRP2 6.6392 13.4264 2.8366 12.247
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 112 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
AU565 GDSC1 -6.7067 4.5171 -7.7678 78.88
BT-474 GDSC1 -6.6172 2.3989 -7.1516 83.0432
SK-BR-3 CTRP2 -6.2335 14.2298 -10.2256 61.9382
HCC2218 CTRP2 -4.9615 2.3091 -5.1912 68.3487
MDA-MB-175-VII GDSC1 -4.5312 10.3779 -7.4719 66.7294
EFM-192A CTRP2 -3.4478 4.0905 -3.8542 60.4607
ZR-75-30 CTRP2 -3.3737 8.9949 -5.1678 57.3802
HCC2218 GDSC1 -2.9841 12.24 -6.6476 61.4093
HCC1419 GDSC1 -2.4765 7.5534 -4.176 64.0507
OCUB-M GDSC1 -2.3331 1.8866 -2.4496 74.2508
AU565 CTRP2 -1.8604 8.2678 -3.2777 51.7883
HCC1419 CTRP2 -1.3426 7.5561 -2.4755 49.4263
HCC202 GDSC1 -1.3301 10.8406 -4.3371 57.1021
UACC-893 GDSC1 -1.1156 6.4832 -2.3165 59.2728
HCC1954 CTRP2 -0.5733 5.6484 -1.0735 44.8784
CAL-85-1 CTRP2 -0.445 12.6152 -3.4976 46.224
MDA-MB-361 CTRP2 0.2726 24.8898 -8.5346 46.2775
MDA-MB-468 GDSC1 0.6203 4.5522 0.217 46.9938
MDA-MB-453 GDSC1 0.7677 5.8814 -0.0717 46.1282
HCC1806 GDSC1 0.9796 4.8252 0.5254 43.324
HCC1187 GDSC1 1.0101 3.1701 0.9447 41.7096
MDA-MB-330 GDSC1 1.1171 15.8582 -4.2948 47.1248
BT-483 GDSC1 1.1479 6.1782 0.2197 42.7794
DU4475 GDSC1 1.1651 2.4226 1.1605 39.4881
EFM-192A GDSC1 1.1761 13.733 -3.2074 46.4146
HCC1599 GDSC1 1.1932 2.6645 1.1807 39.1818
HCC38 GDSC1 1.1981 4.2721 0.9263 40.3013
BT-474 CTRP2 1.3323 14.0628 -2.3461 39.5289
Hs 578T GDSC1 1.3538 3.3646 1.285 37.4935
MDA-MB-453 CTRP2 1.4127 4.0192 1.3658 31.0137
UACC-812 GDSC1 1.4161 9.5874 -1.0012 43.3167
MRK-nu-1 GDSC1 1.6571 3.0976 1.6349 33.448
HCC38 CTRP2 1.6751 6.109 1.2582 30.5004
DU4475 CTRP2 1.7405 2.7719 1.7404 28.6734
HCC1806 CTRP2 1.7564 4.1487 1.7148 28.7069
EFM-19 GDSC1 1.7854 6.0663 0.9391 36.1344
CAL-148 GDSC1 1.8028 3.2175 1.7775 31.6471
HCC1569 GDSC1 1.8093 5.867 1.0446 35.5254
MDA-MB-468 CTRP2 1.8439 12.1551 -1.4352 33.3607
CAL-51 CTRP2 1.9167 3.3825 1.914 27.5084
Hs 578Bst CTRP2 1.9205 4.2642 1.8768 27.6208
HCC2157 GDSC1 1.9587 6.7683 0.8238 35.5343
HDQ-P1 GDSC1 2.1091 3.7118 2.0421 28.0856
HCC1954 GDSC1 2.1279 9.2598 -0.15 37.8385
CAMA-1 GDSC1 2.2084 5.6151 1.5677 30.4037
COLO 824 GDSC1 2.2314 4.6655 1.9382 28.0185
MDA-MB-157 CTRP2 2.3617 3.9917 2.3514 24.569
CAL-85-1 GDSC1 2.3869 13.0642 -1.7507 40.0651
BT-549 GDSC1 2.4737 5.1649 2.0252 26.0606
MDA-MB-361 GDSC1 2.5093 14.0441 -2.1217 40.1829
T-47D CTRP2 2.6453 7.8904 1.7069 25.9541
HCC202 CTRP2 2.7089 15.4956 -1.6845 34.6624
HCC1500 GDSC1 2.7413 3.3624 2.7392 19.7706
HCC70 GDSC1 2.7807 3.9752 2.7203 19.6532
MCF-7 GDSC1 2.7837 4.3087 2.6468 20.1244
BT-20 CTRP2 2.8677 6.0043 2.5885 22.1368
BT-20 GDSC1 2.981 4.2794 2.8699 17.4887
MFM-223 GDSC1 2.9868 4.5212 2.8059 17.8922
CAL-51 GDSC1 3.0115 5.7905 2.3332 21.1013
HCC1395 GDSC1 3.0354 4.2315 2.9415 16.6939
CAL-120 CTRP2 3.06 4.5249 3.045 19.9329
HCC1937 GDSC1 3.2914 4.6643 3.0882 14.2545
CAL-120 GDSC1 3.3365 6.4874 2.3382 19.4874
HCC1428 CTRP2 3.3622 7.2299 2.7255 20.1704
MDA-MB-436 GDSC1 3.4502 6.5995 2.3945 18.5595
MDA-MB-231 GDSC1 3.4701 6.0387 2.6804 16.3691
KPL-1 CTRP2 3.5146 4.3132 3.514 16.8559
Evsa-T GDSC1 3.6186 4.3481 3.5471 9.2622
YMB-1-E GDSC1 3.6219 4.581 3.4743 9.75
MDA-MB-415 GDSC1 3.6974 4.8047 3.4671 9.4087
T-47D GDSC1 3.8367 12.8467 -0.3513 31.044
HCC1428 GDSC1 3.9199 6.3929 2.9349 12.4711
MDA-MB-157 GDSC1 5.2284 9.8084 2.2926 12.6451
HCC1500 CTRP2 5.3839 18.0813 -0.533 25.8621
HDQ-P1 CTRP2 5.4092 15.2106 0.9218 21.6288
Hs 578T CTRP2 5.5605 13.1559 1.4103 14.9627
HCC1143 CTRP2 5.7528 19.5537 -0.9547 26.1513
CAL-148 CTRP2 6.7136 15.1542 2.0345 15.1788
ZR-75-30 GDSC1 6.999 20.2587 -1.5404 25.5228
HCC1937 CTRP2 7.2666 19.6309 0.2409 20.0966
JIMT-1 CTRP2 7.5727 9.2572 5.4625 0.6522
MCF-7 CTRP2 7.8443 14.0542 3.4222 7.9454
CAMA-1 CTRP2 8.1109 9.5297 5.5838 0.1719
HMC-1-8 CTRP2 8.2077 9.4982 5.63 0.0971
ZR-75-1 CTRP2 8.3965 23.0178 -0.5707 20.4345
BT-549 CTRP2 8.6077 17.6368 2.2205 11.3704
MDA-MB-231 CTRP2 8.8886 20.7095 0.9258 15.3329
HCC1395 CTRP2 9.1105 18.4912 2.1535 10.8883
BT 145 CTRP2 -2.3377 3.5065 -2.5561 55.1762
BT 179 CTRP2 -1.7285 17.2208 -6.8555 50.7308
BT 239 CTRP2 -0.0954 12.5403 -3.1049 44.8013
BT 231 CTRP2 -0.0585 9.06 -1.6279 43.3204
BT164 CTRP2 0.0646 4.9869 -0.2262 40.5755
BT 428 CTRP2 0.1549 3.9359 0.0461 39.5479
BT 416 CTRP2 0.2568 3.4426 0.2042 38.718
BT 172 CTRP2 0.9395 4.6582 0.7813 34.5166
BT 248 CTRP2 1.0216 4.9253 0.8229 34.1002
BT147 CTRP2 1.4696 5.0145 1.2906 31.074
BT 271 CTRP2 1.4931 6.6095 0.9123 32.2034
BT 228 CTRP2 1.9732 11.5333 -0.547 34.4609
BT 139 CTRP2 2.0775 14.7663 -1.9434 36.8063
BT 112 CTRP2 2.1281 11.2447 -0.2602 33.3318
BT 286 CTRP2 2.3606 2.9853 2.3605 24.5423
BT 444 CTRP2 2.4358 2.9341 2.4358 24.0407
BT 131 CTRP2 2.4807 3.012 2.4807 23.7418
BT 482 CTRP2 2.4861 3.0367 2.4861 23.7056
BT 422 CTRP2 2.6119 2.9566 2.6119 22.8677
BT 187 CTRP2 2.9349 10.889 0.7134 28.3492
BT 328 CTRP2 4.105 8.3367 3.0487 16.9012
BT 320 CTRP2 6.0256 13.1226 2.4896 14.7717
BT 159 CTRP2 7.0993 35.3806 -7.7542 34.3572
BT 224 CTRP2 9.4671 22.8348 0.3024 16.363
⏷ Show the Full List of 112 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 -3.6404 2.0825 -3.7638 62.8254
Cancer Drug Sensitivity Data Curated from 97 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-466 CTRP2 1.1231 3.2566 1.1109 32.8269
PFSK-1 GDSC1 1.4376 3.904 1.2776 36.9431
KS-1 [Human Krukenberg tumour] GDSC1 1.6717 5.3038 1.1125 36.1202
D283 Med GDSC1 1.9426 4.5817 1.65 31.5426
KNS-60 CTRP2 1.9668 3.8846 1.9169 22.1475
SF539 CTRP2 2.2483 3.3525 2.2477 25.2922
D283 Med CTRP2 2.2525 3.0544 2.2525 25.2621
DK-MG GDSC1 2.3533 3.9862 2.255 25.2402
CAS-1 CTRP2 2.4457 5.0778 2.3324 24.3608
SF268 CTRP2 2.4595 3.4823 2.4591 23.8844
SF539 GDSC1 2.4652 3.7912 2.412 23.5484
U-251MG CTRP2 2.5331 4.5916 2.4899 23.5384
D-336MG GDSC1 2.5339 4.6482 2.2727 24.0746
GB-1 GDSC1 2.5908 6.3992 1.6341 27.8592
MOG-G-CCM GDSC1 2.6085 4.386 2.4341 22.5623
Hs 683 CTRP2 2.7554 3.3442 2.7554 21.9118
YKG-1 GDSC1 2.7901 4.0292 2.7201 19.599
GI-1 GDSC1 2.8655 5.0739 2.4786 20.8357
Daoy CTRP2 2.8696 4.3546 2.8574 21.1919
SW1783 GDSC1 2.8787 3.8071 2.8518 18.2116
GB-1 CTRP2 2.9184 4.8935 2.8645 21.0082
SF126 GDSC1 2.9509 3.9189 2.9133 17.3777
YH-13 GDSC1 3.051 4.7173 2.8098 17.512
8-MG-BA GDSC1 3.1437 5.2724 2.6927 17.8611
GaMG GDSC1 3.1759 5.0211 2.8293 16.7109
YKG-1 CTRP2 3.1876 5.6257 3.0302 19.5752
ONS-76 GDSC1 3.2412 4.2741 3.1552 14.071
Daoy GDSC1 3.2714 5.4137 2.765 16.693
AM-38 GDSC1 3.2774 4.3787 3.166 13.7913
U-251MG GDSC1 3.2781 4.4702 3.1391 13.9723
42-MG-BA GDSC1 3.3137 4.2838 3.2318 13.138
D-566MG GDSC1 3.315 4.3879 3.2044 13.3169
42-MG-BA CTRP2 3.3163 4.7824 3.2943 18.2486
SW1783 CTRP2 3.3954 14.7641 -0.681 30.8098
D-502MG GDSC1 3.452 10.0953 0.6816 28.608
NMC-G1 GDSC1 3.4757 5.2149 3.0619 13.4974
LN-18 GDSC1 3.4912 4.1033 3.4643 10.5566
M059J GDSC1 3.5317 4.9603 3.2289 11.9883
KALS-1 CTRP2 3.5891 9.9259 1.8092 22.9415
H4 GDSC1 3.642 4.8858 3.3754 10.3597
LNZTA3WT4 GDSC1 3.7249 4.5451 3.5982 8.3211
Onda 10 GDSC1 3.7483 4.3371 3.6917 7.543
Onda 11 GDSC1 3.793 5.2854 3.3506 9.8189
CAS-1 GDSC1 3.796 8.9668 1.5479 22.6569
D-423MG GDSC1 3.8189 8.3447 1.8774 20.5142
SF126 CTRP2 3.8298 6.6744 3.4303 16.1867
Becker GDSC1 3.8462 4.3194 3.8034 6.2273
SK-MG-1 GDSC1 3.8561 5.1898 3.4575 8.7159
U-87MG ATCC GDSC1 3.8955 4.3905 3.8362 5.7249
D-263MG GDSC1 3.9126 6.9758 2.6401 14.7496
DK-MG CTRP2 3.9164 10.8604 1.6944 22.4993
LN-229 GDSC1 3.9743 9.8159 1.2801 23.4607
MOG-G-UVW GDSC1 4.0966 5.6901 3.442 7.8008
KNS-81 CTRP2 4.1226 26.27 -5.7115 37.0469
Hs 683 GDSC1 4.1812 4.8573 3.9295 3.6453
SNB-75 GDSC1 4.4633 6.9239 3.1368 8.8373
SW1088 CTRP2 4.4906 9.6472 2.8271 16.8045
KINGS-1 GDSC1 4.5417 7.7723 2.7763 11.3486
KNS-42 CTRP2 4.5428 7.4499 3.8859 12.4607
D-542MG GDSC1 4.5908 7.1206 3.1398 8.3828
D-392MG GDSC1 4.6746 9.6723 1.9346 16.8752
SF295 GDSC1 4.8398 6.5159 3.6208 3.9113
D-247MG GDSC1 4.847 7.0661 3.359 5.888
LN-405 GDSC1 4.8696 6.4082 3.6923 3.2971
CCF-STTG1 CTRP2 5.1487 10.3454 3.1084 14.146
SF268 GDSC1 5.3984 8.5586 3.0196 6.9314
SW1088 GDSC1 5.4768 8.8673 2.9247 7.4208
KNS-81-FD GDSC1 5.5126 7.8315 3.4321 3.6965
U-118MG GDSC1 5.928 11.3641 2.0328 12.3688
LN-229 CTRP2 5.9624 14.0472 1.9745 16.8457
T98G GDSC1 6.0798 7.9176 3.6925 1.2057
U-118MG CTRP2 6.1775 14.8057 1.7742 17.1465
A-172 GDSC1 6.4276 8.5176 3.612 1.2331
KALS-1 GDSC1 6.4558 14.4375 0.9133 17.3608
GaMG CTRP2 6.5644 11.6362 3.6691 9.0062
Becker CTRP2 6.5953 10.2976 3.5704 4.0316
A-172 CTRP2 6.614 13.0209 2.2765 9.4704
KNS-42 GDSC1 6.6928 7.8671 3.9483 0.0787
SNU-1105 CTRP2 6.968 9.3308 5.0924 2.5306
SNU-626 CTRP2 7.0418 12.3942 3.6576 8.2415
SNU-201 CTRP2 7.213 13.4972 3.2414 9.6429
T98G CTRP2 7.2801 11.4793 3.4439 3.685
SNU-489 CTRP2 7.3097 12.8478 3.6309 7.9214
NMC-G1 CTRP2 7.3773 10.8158 4.6571 3.7043
SF295 CTRP2 7.4135 9.2068 5.4058 0.9313
DBTRG-05MG GDSC1 7.4262 14.2847 1.6286 11.1839
M059K CTRP2 7.4866 14.0723 3.1597 9.5272
ONS-76 CTRP2 7.6528 9.6926 5.3223 1.007
U-87MG ATCC CTRP2 7.679 9.2417 5.5166 0.4534
LN-18 CTRP2 7.6791 8.6262 5.7408 0.064
GMS-10 CTRP2 7.7087 16.8293 1.9683 13.6831
SNU-738 CTRP2 7.8886 9.286 5.5863 0.227
8-MG-BA CTRP2 7.9451 12.5977 4.1839 4.8177
DBTRG-05MG CTRP2 8.5844 14.2079 3.8353 5.358
YH-13 CTRP2 9.1283 17.8778 2.4584 9.7763
GOS-3 CTRP2 10.5791 23.4154 0.7853 13.3848
TM-31 CTRP2 10.9902 20.1096 2.5808 7.1089
⏷ Show the Full List of 97 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ETK-1 GDSC1 2.1334 4.9619 1.7325 29.8813
TGBC24TKB GDSC1 7.0533 20.1065 -1.4259 25.054
TGBC1TKB GDSC1 7.153 8.8001 3.7938 0.2121
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-3 CTRP2 -0.4431 6.8484 -1.2704 44.5144
AN3-CA GDSC1 0.3692 2.8279 0.3056 49.4409
RL95-2 GDSC1 0.9507 6.2942 -0.0354 44.7
MFE-280 GDSC1 1.1853 4.2077 0.9293 40.3882
JHUEM-7 CTRP2 1.7296 3.3664 1.725 28.7611
JHUEM-1 CTRP2 1.7634 2.9327 1.7631 28.5218
HEC-151 CTRP2 1.7662 4.6941 1.6628 28.85
HEC-1-A CTRP2 1.8295 3.9538 1.8051 28.1618
KLE CTRP2 2.3349 4.2014 2.3136 24.7846
EN GDSC1 2.6622 3.4476 2.6554 20.7891
MFE-296 CTRP2 2.7722 4.4895 2.7488 21.8783
MFE-319 GDSC1 3.2191 4.0784 3.1751 14.0678
MFE-296 GDSC1 3.2647 4.6536 3.0631 14.5755
KLE GDSC1 3.3701 9.7336 0.787 28.4848
HEC-50B CTRP2 3.4849 11.2688 0.5531 22.9582
ESS-1 GDSC1 3.7519 4.2323 3.7218 7.3199
RL95-2 CTRP2 4.1256 15.8891 -0.5561 28.7185
HEC-1-B CTRP2 4.4375 16.5289 -0.5906 28.0774
AN3-CA CTRP2 4.4757 9.4488 2.352 13.3122
HEC-251 CTRP2 5.7478 23.6934 -3.0285 30.4006
EN CTRP2 6.363 10.7492 3.202 5.9275
EFE-184 CTRP2 6.7414 21.4355 -1.0783 24.5575
HEC-6 CTRP2 7.7718 9.096 5.6098 0.2222
HEC-265 CTRP2 7.9671 9.1782 5.654 0.1105
ESS-1 CTRP2 8.0783 15.3762 2.9456 9.4536
HEC-59 CTRP2 8.3545 15.6803 2.9892 8.8856
JHUEM-2 CTRP2 8.4534 13.2965 4.175 4.24
MFE-319 CTRP2 8.5471 17.6571 2.1684 11.6476
HEC-108 CTRP2 10.6624 27.0804 -0.918 17.9871
Ishikawa (Heraklio) 02 ER- CTRP2 7.3447 21.4173 -0.5871 22.2456
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 51 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
769-P GDSC1 -0.4859 11.13 -3.6095 53.6418
TK-10 GDSC1 -0.1633 8.0401 -1.9218 52.9673
CAL-54 CTRP2 0.3758 12.8207 -2.7456 42.9443
KTCTL-140 GDSC1 0.5588 6.7425 -0.6292 48.1911
SW13 GDSC1 0.6068 3.9079 0.3726 46.9062
UO-31 CTRP2 0.7823 5.9127 0.3371 36.3731
769-P CTRP2 1.3916 9.9425 -0.4498 36.0997
KTCTL-21 GDSC1 1.8793 4.3154 1.6579 31.8937
VMRC-RCZ GDSC1 2.0239 8.2652 0.2148 37.327
KTCTL-26A GDSC1 2.105 5.1967 1.6178 30.7328
TUHR14TKB CTRP2 2.4326 5.0031 2.3305 24.4094
LB996-RCC GDSC1 2.501 8.294 0.6702 33.1315
LB2241-RCC GDSC1 2.5111 6.6449 1.4434 29.3827
KMRC-2 CTRP2 2.7154 5.7482 2.4877 22.9659
KTCTL-195 GDSC1 2.7453 5.0729 2.3506 22.3725
HA7-RCC GDSC1 2.7698 5.1543 2.3455 22.2753
KTCTL-13 GDSC1 2.808 5.8442 2.1004 23.7493
KMRC-3 CTRP2 2.9248 5.2009 2.8275 21.1148
786-O GDSC1 3.033 5.2106 2.602 19.0819
CAL-54 GDSC1 3.1002 10.1222 0.3498 31.527
LB1047-RCC GDSC1 3.1139 5.364 2.6232 18.514
NCC021 GDSC1 3.1191 8.0761 1.3676 26.7023
A-704 GDSC1 3.1648 4.7294 2.9284 16.0632
BB65-RCC GDSC1 3.2245 4.5908 3.0414 14.9459
ACHN GDSC1 3.3687 35.1192 -11.8781 44.7812
KTCTL-1M GDSC1 3.5565 5.2806 3.1156 12.7048
RXF 393L GDSC1 3.5932 5.8965 2.8677 14.4
OS-RC-2 GDSC1 3.6684 4.5742 3.5268 9.13
SN12C GDSC1 3.6792 9.2765 1.2905 24.6163
KMRC-1 GDSC1 3.7465 4.1746 3.7271 7.317
KMRC-20 GDSC1 3.7934 4.7901 3.5735 8.1459
UO-31 GDSC1 3.8803 8.4454 1.8815 20.2336
VMRC-RCW GDSC1 4.1729 5.8443 3.4333 7.567
A-498 GDSC1 4.6017 5.8792 3.7623 3.4975
BFTC-909 GDSC1 4.6074 6.812 3.3061 7.0324
RCC10RGB GDSC1 4.6167 5.7564 3.833 2.9101
SW156 GDSC1 4.9671 11.8049 1.1036 20.7939
VMRC-RCZ CTRP2 5.3465 17.4013 -0.2257 25.1372
TUHR4TKB CTRP2 6.2028 11.2576 3.5686 10.0839
Caki-1 GDSC1 7.1048 24.3735 -3.4896 30.0298
TUHR10TKB CTRP2 7.5494 12.2087 4.1083 5.6449
VMRC-RCW CTRP2 7.7939 12.5364 4.115 5.2835
KMRC-20 CTRP2 8.1928 15.1695 3.1243 8.5996
786-O CTRP2 8.5564 11.922 4.8409 1.8092
OS-RC-2 CTRP2 8.6316 19.1465 1.5043 13.8351
SNU-1272 CTRP2 8.9853 18.0788 2.2665 10.6621
ACHN CTRP2 9.2407 23.3046 -0.8694 16.5202
KMRC-1 CTRP2 9.5907 17.5196 2.0645 6.2824
RCC10RGB CTRP2 9.9709 20.0666 1.9733 10.3591
Caki-1 CTRP2 10.2194 27.368 -1.37 19.7015
Caki-2 CTRP2 15.6996 39.6929 -3.5747 17.9236
⏷ Show the Full List of 51 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 90 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW48 CTRP2 -4.366 8.4303 -6.0475 60.8384
CCK-81 GDSC1 -4.0492 4.4408 -4.8464 74.0246
CCK-81 CTRP2 -3.5382 6.0212 -4.4071 59.5609
GP2d CTRP2 -1.8327 9.3222 -3.6266 51.5577
HT115 CTRP2 -1.7787 3.2072 -1.9187 51.9683
SW1116 CTRP2 -1.4968 18.66 -7.7648 48.794
NCI-H508 CTRP2 -1.1472 7.5145 -2.2496 48.4536
NCI-H747 CTRP2 -0.9544 7.9453 -2.1858 47.5426
COLO 678 CTRP2 -0.4116 13.9074 -4.0311 46.3739
T84 CTRP2 -0.2579 6.1628 -0.8662 43.1539
CW-2 CTRP2 -0.1902 9.6978 -2.375 41.8246
HT-55 CTRP2 -0.1427 14.2459 -3.9095 45.4665
HT115 GDSC1 0.3796 5.7814 -0.4518 49.5161
SNU-175 GDSC1 0.4174 5.9234 -0.4632 49.2092
SK-CO-1 CTRP2 0.4343 8.0521 -0.7236 40.067
LoVo CTRP2 0.5254 5.224 0.2239 37.6407
SNU-C4 CTRP2 0.732 5.6002 0.3618 36.4925
C2BBe1 CTRP2 0.9371 8.8341 -0.4791 37.7286
LoVo GDSC1 1.163 5.2073 0.5977 41.689
SNU-407 CTRP2 1.5052 4.5959 1.3978 30.5998
COLO 320 CTRP2 1.8798 7.5717 1.0069 30.6365
SNU-1033 CTRP2 2.1174 18.5515 -3.722 39.1148
SW1116 GDSC1 2.273 14.3613 -2.4931 41.5825
CL-11 CTRP2 2.3867 5.1135 2.2629 24.7899
HCT 15 CTRP2 2.3933 3.6503 2.3914 24.3304
SNU-C5 CTRP2 2.4178 4.2936 2.3938 24.2414
SW948 CTRP2 2.4505 3.3131 2.4504 23.9436
HCT 8 CTRP2 2.4611 2.9373 2.4611 23.8725
NCI-H747 GDSC1 2.4679 7.2513 1.1246 31.2752
SNU-C2A CTRP2 2.7565 8.0578 1.7591 25.4437
LS1034 CTRP2 2.8111 4.5061 2.7881 21.618
SNU-61 GDSC1 2.8651 6.864 1.6986 26.0338
DLD-1 CTRP2 2.8842 3.4266 2.8842 21.0535
SNU-81 GDSC1 2.9163 6.4553 1.938 24.2668
SNU-C1 CTRP2 3.1334 5.1517 3.0592 19.6454
HCC2998 GDSC1 3.1568 4.58 2.9716 15.8038
C2BBe1 GDSC1 3.1658 4.8203 2.8961 16.2865
SNU-1040 GDSC1 3.2092 9.132 0.9365 28.5015
SW1417 GDSC1 3.2139 6.6506 2.1417 21.4412
SNU-61 CTRP2 3.3912 10.1613 1.5034 24.544
RKO GDSC1 3.5964 6.5034 2.5801 16.5441
SNU-407 GDSC1 3.6338 4.5329 3.5043 9.4745
CL-11 GDSC1 3.6367 4.4524 3.5348 9.2455
LS180 GDSC1 3.7286 10.6377 0.6569 27.5661
COLO205 GDSC1 3.7704 4.1821 3.7516 7.0146
SW626 GDSC1 3.7966 4.5696 3.6661 7.4574
GP5d GDSC1 3.93 11.2247 0.5387 27.2901
LS123 GDSC1 3.9515 11.5604 0.3895 27.8464
LS513 GDSC1 4.0365 8.9963 1.7428 20.4883
SW1417 CTRP2 4.0734 7.9451 3.1872 16.4431
LS123 CTRP2 4.1759 8.0056 3.2669 15.8603
HT-29 GDSC1 4.179 6.8975 2.9132 11.6122
LS411N GDSC1 4.1913 5.8335 3.4547 7.3277
CW-2 GDSC1 4.2707 13.2675 -0.1936 28.9342
CaR-1 GDSC1 4.2789 6.11 3.3918 7.4924
SW48 GDSC1 4.2966 5.6422 3.6406 5.4663
NCI-H716 GDSC1 4.3103 5.5096 3.7184 4.8017
HCT 116 GDSC1 4.4149 6.17 3.4741 6.3567
KM12 GDSC1 4.4567 5.7789 3.7025 4.4184
LS513 CTRP2 4.7203 11.2504 2.2696 18.4249
COLO 678 GDSC1 4.8518 6.4173 3.6762 3.4632
COLO 320HSR GDSC1 5.2084 7.2208 3.5278 3.6859
SNU-C2B GDSC1 5.2372 20.893 -3.2138 33.7848
SNU-503 CTRP2 5.3522 19.2816 -1.1595 27.4455
SNU-C5 GDSC1 5.3652 7.2669 3.6012 2.8347
SW620 GDSC1 5.4404 7.3272 3.6173 2.581
KM12 CTRP2 5.5578 9.4294 3.931 9.8664
HCC-56 CTRP2 5.6475 15.4287 1.0175 20.8157
T84 GDSC1 5.8275 10.1041 2.5688 9.0469
LS1034 GDSC1 5.849 7.3556 3.8106 0.8779
SW948 GDSC1 6.075 7.6521 3.7939 0.7479
HCT 15 GDSC1 6.158 8.087 3.6608 1.2781
SW837 GDSC1 6.2574 16.7591 -0.3666 23.4898
SNU-C1 GDSC1 6.5396 8.2075 3.7756 0.4977
MDST8 GDSC1 6.7483 7.9922 3.9256 0.0967
NCI-H716 CTRP2 7.0799 10.1484 4.778 3.6249
HT-55 GDSC1 7.2204 19.5699 -1.0422 23.4507
HT-29 CTRP2 7.3295 9.209 5.3612 1.1453
LS411N CTRP2 7.4504 8.6105 5.6603 0.2372
OUMS-23 CTRP2 7.6078 8.7775 5.6614 0.1833
COLO205 CTRP2 7.7623 9.0253 5.6317 0.1881
SW1463 GDSC1 7.7836 23.0871 -2.3554 26.016
HCT 116 CTRP2 7.8243 9.4114 5.5136 0.3929
COLO201 CTRP2 7.924 10.6998 5.0336 1.7139
MDST8 CTRP2 7.9511 9.2263 5.6314 0.142
RCM-1 [Human ESC] CTRP2 8.4591 18.7613 1.5687 13.8822
SW620 CTRP2 8.8244 14.1933 3.9875 4.515
LS180 CTRP2 8.8385 19.494 1.4819 13.598
RCM-1 [Human ESC] GDSC1 8.85 21.3484 -0.7778 19.0194
RKO CTRP2 8.9682 21.1619 0.7621 15.7239
⏷ Show the Full List of 90 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1 2.4697 4.0676 2.3639 23.836
Cancer Drug Sensitivity Data Curated from 38 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-182 CTRP2 -0.3225 4.2536 -0.5097 42.8376
JHH-5 CTRP2 0.4402 45.4535 -18.5054 47.7075
JHH-2 GDSC1 0.6344 3.3754 0.5109 46.4005
JHH-4 GDSC1 0.7932 6.4321 -0.2571 46.1638
SNU-761 CTRP2 0.8344 30.9752 -11.5774 45.03
SNU-423 GDSC1 1.0903 3.1521 1.0322 40.6919
SNU-449 GDSC1 1.1561 7.3775 -0.2684 43.6855
SNU-475 GDSC1 1.5553 2.2192 1.5552 34.5838
HuH-6 CTRP2 1.6059 2.726 1.6057 29.5707
JHH-1 GDSC1 1.7309 28.3566 -9.9176 47.1225
SNU-398 GDSC1 1.8926 2.9119 1.8877 30.3971
Li-7 CTRP2 1.9885 4.7035 1.899 27.3234
SNU-878 CTRP2 2.1368 5.1984 1.9776 26.5753
JHH-2 CTRP2 2.1706 6.8018 1.5881 27.8108
SNU-449 CTRP2 2.3296 4.9709 2.2249 25.104
Huh-7 GDSC1 2.4557 4.2226 2.3115 24.2643
SNU-423 CTRP2 2.4707 4.0803 2.4597 23.8452
Hep 3B2.1-7 GDSC1 2.7122 4.3405 2.5601 21.1188
HLE GDSC1 2.7601 3.6042 2.7472 19.6039
SNU-886 CTRP2 3.024 4.7377 2.9922 43.385
SNU-387 GDSC1 3.2638 4.1041 3.2185 13.5177
JHH-7 GDSC1 3.2678 4.1062 3.2224 13.4685
SK-HEP-1 GDSC1 3.606 4.0861 3.59 9.051
JHH-6 GDSC1 3.8834 4.6512 3.7257 6.5775
Hep-G2/C3A GDSC1 3.9737 5.0482 3.6393 6.7932
JHH-4 CTRP2 4.9065 10.7328 2.0845 13.5163
HuH-1 GDSC1 4.9088 7.6612 3.1126 7.5945
SNU-398 CTRP2 5.1338 7.6069 3.8369 5.2556
SNU-387 CTRP2 6.1115 17.8368 0.204 22.3724
SK-HEP-1 CTRP2 6.6071 9.636 3.8832 2.7454
JHH-6 CTRP2 7.2398 8.2441 5.7112 0.2149
HuH-1 CTRP2 7.6314 9.3499 5.4525 0.6436
Hep-G2 CTRP2 7.8881 9.3166 5.575 0.2469
Hep 3B2.1-7 CTRP2 8.1595 9.4354 5.6343 0.1
HLF CTRP2 8.715 15.5572 3.287 7.2647
JHH-1 CTRP2 9.2284 22.3941 0.3472 16.5849
SNU-475 CTRP2 9.5134 17.4634 2.902 7.677
PLC/PRF/5 CTRP2 10.2165 19.2292 2.5194 8.1824
⏷ Show the Full List of 38 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 309 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HCC4006 CTRP2 -12.6145 1.9265 -13.3603 82.4933
HCC827 CTRP2 -11.8587 -0.5922 -12.1618 85.6412
COR-L105 CTRP2 -9.0643 10.6169 -11.8858 69.0993
PC-14 CTRP2 -8.2142 -4.7198 -8.2146 89.8606
NCI-H1975 CTRP2 -6.7629 0.5439 -6.9013 76.5776
HCC827 GDSC1 -5.6104 23.8933 -14.6089 60.7927
NCI-H1666 CTRP2 -5.5675 10.3669 -8.0247 62.7524
HCC2935 CTRP2 -4.7622 4.5702 -5.3818 65.1911
NCI-H1623 GDSC1 -4.648 19.0522 -11.4037 61.1979
Calu-3 GDSC1 -4.0335 9.0604 -6.4186 66.9434
NCI-H3255 GDSC1 -2.9356 8.8744 -5.1804 64.1128
Calu-3 CTRP2 -2.5877 5.0011 -3.1131 55.9541
NCI-H1623 CTRP2 -2.3864 12.1536 -5.3265 53.1611
NCI-H322 CTRP2 -2.3195 11.8498 -5.132 52.9951
EPLC-272H CTRP2 -1.9794 9.0701 -3.6916 52.186
NCI-H358 CTRP2 -1.8342 2.8356 -1.9361 52.3463
NCI-H1781 GDSC1 -0.9544 4.418 -1.4628 60.6204
CAL-12T GDSC1 -0.9267 8.98 -3.1141 56.4683
NCI-H1568 GDSC1 -0.8588 35.0786 -15.5618 51.795
DV-90 CTRP2 -0.5941 4.7187 -0.8862 44.7317
NCI-H1648 GDSC1 -0.5576 10.6659 -3.4725 54.0888
COR-L105 GDSC1 -0.471 16.6638 -6.1887 52.4856
EKVX CTRP2 -0.4598 12.1117 -3.2961 46.1684
NCI-H1693 CTRP2 0.0245 10.414 -2.0779 43.4954
SK-MES-1 CTRP2 0.1383 7.7368 -0.9314 41.5855
CAL-12T CTRP2 0.1602 18.4951 -5.5739 45.4585
PaCa-3 GDSC1 0.3429 14.0238 -4.1437 49.9187
NCI-H322M GDSC1 0.378 20.7217 -7.359 49.851
NCI-H661 CTRP2 0.4722 5.4921 -0.0745 34.4424
NCI-H661 GDSC1 0.6287 7.5263 -0.8794 47.8422
NCI-H522 CTRP2 0.7214 6.25 0.1778 37.0178
NCI-H2087 CTRP2 0.7378 5.3697 0.4225 36.3027
NCI-H1184 CTRP2 0.9004 4.4618 0.7702 34.6879
NCI-H1734 CTRP2 0.9903 10.3637 -1.0457 38.6257
NCI-H1975 GDSC1 1.0035 7.8075 -0.6121 45.1667
EPLC-272H GDSC1 1.013 3.7215 0.8553 42.0398
HOP-92 CTRP2 1.1569 7.6824 0.188 35.4065
NCI-H1341 CTRP2 1.2492 2.7106 1.2482 31.9496
NCI-H1869 GDSC1 1.2999 5.9018 0.4895 41.0029
RERF-LC-Sq1 GDSC1 1.3038 18.8565 -5.5919 46.9933
NCI-H358 GDSC1 1.4574 7.4406 0.0148 41.1959
NCI-H1694 CTRP2 1.4788 3.8548 1.4475 30.5213
Sq-1 CTRP2 1.48 5.3536 1.2333 31.2278
NCI-H1755 CTRP2 1.4896 3.832 1.4602 30.443
NCI-H1838 CTRP2 1.5363 6.3879 1.0266 31.7031
NCI-H2444 CTRP2 1.5366 30.3828 -10.655 43.5295
SW1271 CTRP2 1.5929 7.0022 0.8947 31.9229
IST-SL2 GDSC1 1.6566 4.3629 1.4019 34.7889
NCI-H211 CTRP2 1.7291 3.5165 1.721 28.776
NCI-H146 CTRP2 1.7371 2.8097 1.7369 28.6964
NCI-H2170 CTRP2 1.7434 6.6167 1.1827 30.5214
NCI-H1385 CTRP2 1.7434 4.9763 1.5931 29.1607
NCI-H1869 CTRP2 1.757 13.1086 -1.4829 36.9515
NCI-H2342 GDSC1 1.7653 4.4262 1.5026 33.5207
NCI-H1355 CTRP2 1.7838 7.8764 0.7916 31.6051
NCI-H1155 CTRP2 1.8003 3.1675 1.799 28.2792
NCI-H524 GDSC1 1.8152 4.1164 1.6396 32.4086
ABC-1 GDSC1 1.8403 4.3624 1.6025 32.4666
COLO 668 CTRP2 1.8541 3.9464 1.831 27.9939
NCI-H847 GDSC1 1.8777 4.612 1.57 32.4163
HCC44 CTRP2 1.9012 4.1514 1.8659 27.7209
NCI-H1573 CTRP2 1.9247 5.6617 1.6469 28.3904
NCI-H1581 CTRP2 1.9304 3.0473 1.9301 27.4088
NCI-H810 CTRP2 1.9392 3.0954 1.9388 27.3505
Lu-135 GDSC1 1.9535 3.4898 1.9077 29.8935
NCI-H2106 CTRP2 1.9729 3.5235 1.9685 27.1398
NCI-H1703 CTRP2 1.9747 3.233 1.9738 27.1158
EBC-1 CTRP2 1.9961 4.3356 1.9496 27.127
SBC-3 GDSC1 2.0126 4.7122 1.6853 30.8994
Ms-1 GDSC1 2.0132 4.4421 1.7685 30.3931
PC-14 GDSC1 2.0287 9.2855 -0.2585 38.6368
NCI-H446 CTRP2 2.09 5.1176 1.942 26.848
SW1271 GDSC1 2.1315 5.1087 1.6783 30.2176
NCI-H1650 CTRP2 2.1321 15.7265 -2.3475 37.2874
NCI-H1105 CTRP2 2.1712 3.5695 2.1683 25.8136
NCI-H292 CTRP2 2.1891 12.0316 -0.5564 33.8333
COR-L95 CTRP2 2.1917 3.4456 2.1904 25.6716
COLO 699 CTRP2 2.194 3.8141 2.1861 25.6784
LCLC-97TM1 CTRP2 2.25 4.7813 2.1675 25.5581
NCI-H2171 GDSC1 2.2644 3.3838 2.2468 25.8302
NCI-H1563 CTRP2 2.2686 4.3139 2.237 25.261
EKVX GDSC1 2.2777 7.2272 0.9448 33.1642
NCI-H1568 CTRP2 2.2963 16.1623 -2.3987 36.93
NCI-H2141 CTRP2 2.3009 6.0477 1.9581 26.1233
NCI-H1915 CTRP2 2.3065 3.2344 2.3064 24.9025
NCI-H1092 CTRP2 2.3189 4.5641 2.2669 24.995
Lu-99 CTRP2 2.3371 3.2665 2.337 24.6989
NCI-H2196 CTRP2 2.3393 4.196 2.3185 24.7535
NCI-H1694 GDSC1 2.3394 5.7161 1.6653 29.0739
ChaGo-K-1 CTRP2 2.3426 4.463 2.3018 24.7994
NCI-H1048 GDSC1 2.3519 3.8528 2.2795 25.089
NCI-H1581 GDSC1 2.4378 3.7626 2.387 23.8752
NCI-H2029 CTRP2 2.448 3.9772 2.4401 23.9861
HCC1438 CTRP2 2.4502 12.0548 -0.3067 32.4897
DMS 114 CTRP2 2.4856 3.7843 2.4827 23.7189
DMS 454 CTRP2 2.493 3.872 2.4886 23.6748
NCI-H1793 CTRP2 2.5059 4.0674 2.4962 23.6065
HOP-62 CTRP2 2.5267 9.2862 1.0096 28.6225
COR-L51 CTRP2 2.5393 3.6504 2.5383 23.3547
NCI-H1876 GDSC1 2.5409 4.6708 2.2729 24.033
VMRC-LCD CTRP2 2.5701 4.9392 2.4874 23.4267
NCI-H810 GDSC1 2.5948 4.6136 2.3501 23.2078
NCI-H23 GDSC1 2.5993 3.7789 2.5576 21.7983
NCI-H1304 GDSC1 2.6111 4.5489 2.3882 22.8575
HCC78 GDSC1 2.6307 3.4984 2.6199 21.2082
HCC33 GDSC1 2.6627 3.9136 2.6041 21.1158
NCI-H2810 GDSC1 2.678 3.6312 2.6589 20.6698
NCI-H2795 GDSC1 2.6792 4.1347 2.5766 21.1992
LK2 CTRP2 2.6983 3.0292 2.6983 22.2924
T3M-10 CTRP2 2.705 9.7417 0.9963 28.1392
NCI-H2066 GDSC1 2.7113 3.8185 2.6716 20.3859
NCI-H889 CTRP2 2.7121 11.7529 0.0932 30.7301
NCI-H69 GDSC1 2.7182 5.0769 2.3201 22.73
NCI-H2869 GDSC1 2.7426 4.9851 2.3807 22.1791
NCI-H290 GDSC1 2.744 5.4147 2.2144 23.3145
RERF-LC-A1 CTRP2 2.7998 3.9243 2.798 21.6218
NCI-H510A GDSC1 2.8067 3.9462 2.7537 19.2798
NCI-H2009 CTRP2 2.8074 7.8676 1.8884 24.8379
NCI-H2369 GDSC1 2.8104 3.3167 2.8098 18.8976
CPC-N GDSC1 2.8311 4.4361 2.6624 19.7494
NCI-H650 GDSC1 2.8396 3.9802 2.7831 18.892
NCI-H647 CTRP2 2.8414 5.674 2.6426 22.0255
NCI-H1688 GDSC1 2.8427 5.8138 2.1495 23.2368
COR-L88 GDSC1 2.8445 3.3987 2.8431 18.4767
HOP-62 GDSC1 2.8448 4.1787 2.7466 19.1025
NCI-H835 GDSC1 2.8533 3.6768 2.8387 18.4495
NCI-H1703 GDSC1 2.8546 5.371 2.3487 21.8027
UMC-11 GDSC1 2.8877 4.0212 2.8274 18.3153
A-427 GDSC1 2.8887 3.971 2.8377 18.2421
NCI-H2081 GDSC1 2.9094 4.6163 2.691 19.1147
COR-L303 GDSC1 2.9173 4.2974 2.7956 18.355
NCI-H513 GDSC1 2.9203 10.5894 -0.0449 33.74
LB647-SCLC GDSC1 2.9439 4.0151 2.8893 17.5764
NCI-H596 GDSC1 2.9458 3.6132 2.9393 17.2427
NCI-H1792 GDSC1 2.9601 3.6834 2.9498 17.088
SBC-5 GDSC1 2.983 3.7487 2.9683 16.8293
NCI-H841 CTRP2 3.0102 9.1544 1.5665 25.3816
NCI-H2818 GDSC1 3.0236 4.3124 2.9076 16.9896
NCI-H727 GDSC1 3.024 8.0414 1.2943 27.557
LC-2/ad GDSC1 3.0253 4.2409 2.9281 16.8418
NCI-H2110 CTRP2 3.0284 7.8061 2.1473 23.265
Lu-139 GDSC1 3.0309 5.3032 2.5618 19.3796
NCI-H2081 CTRP2 3.038 6.1411 2.4814 16.4997
NCI-H1915 GDSC1 3.0476 3.9559 3.0114 16.1605
NCI-H1838 GDSC1 3.0748 9.3594 0.701 30.1965
NCI-H1105 GDSC1 3.0763 3.9284 3.0462 15.7623
NCI-H2347 GDSC1 3.0902 4.6298 2.8827 16.7887
COR-L311 GDSC1 3.1041 4.0634 3.0535 15.5483
NCI-H2030 GDSC1 3.1133 5.692 2.4808 19.5418
NCI-H2444 GDSC1 3.1177 6.6354 2.0546 22.4957
NCI-H196 CTRP2 3.1325 4.7295 3.1065 19.4869
HCC1171 CTRP2 3.1466 9.7536 1.4417 25.4255
LCLC-97TM1 GDSC1 3.1504 6.61 2.0986 22.04
NCI-H2591 GDSC1 3.1814 8.85 1.0491 28.0797
NCI-H1435 GDSC1 3.1894 7.7597 1.5873 25.1119
NCI-H522 GDSC1 3.194 7.0252 1.9445 22.8589
NCI-H1836 GDSC1 3.2028 4.363 3.0891 14.738
NCI-H1395 CTRP2 3.2225 7.6164 2.428 21.6775
NCI-H1436 GDSC1 3.2454 4.8996 2.9509 15.4749
Calu-6 GDSC1 3.2673 4.4598 3.1306 14.0907
NCI-H1155 GDSC1 3.2725 4.6271 3.0809 14.4083
NCI-H2228 CTRP2 3.2747 16.052 -1.4208 32.7134
HARA [Human squamous cell lung carcinoma] CTRP2 3.2915 5.1789 3.2245 18.5679
NCI-H187 GDSC1 3.3193 4.317 3.2291 13.1247
NCI-H441 GDSC1 3.3202 4.3471 3.2217 13.1693
NCI-H720 GDSC1 3.3388 4.5048 3.1941 13.2548
NCI-H1944 GDSC1 3.3695 7.5524 1.8575 22.604
NCI-H2087 GDSC1 3.3857 4.7254 3.1673 13.1891
NCI-H64 GDSC1 3.3897 4.1877 3.3378 11.9887
NCI-H2291 GDSC1 3.4046 5.2346 2.9801 14.4524
NCI-H2135 GDSC1 3.4212 4.946 3.1188 13.3532
NCI-H1734 GDSC1 3.4599 4.9897 3.1415 12.9906
BEN GDSC1 3.4707 6.5387 2.4434 18.1122
NCI-H1793 GDSC1 3.4766 8.3205 1.5808 23.8352
NCI-H526 GDSC1 3.5056 4.7404 3.2899 11.6808
HCC15 CTRP2 3.5146 5.2456 3.4535 17.0614
EMC-BAC-1 GDSC1 3.5166 15.1397 -1.772 35.953
Lu-99A GDSC1 3.526 5.3895 3.0358 13.4469
NCI-H520 GDSC1 3.5276 5.1788 3.1311 12.73
IA-LM CTRP2 3.5333 6.8277 3.0562 18.4421
NCI-H1563 GDSC1 3.5355 9.9413 0.8326 27.559
NCI-H2196 GDSC1 3.5416 5.2626 3.1085 12.8297
EMC-BAC-2 GDSC1 3.5475 5.0168 3.2215 11.9636
LOU-NH91 GDSC1 3.5578 4.4387 3.4534 10.2468
COR-L321 GDSC1 3.571 4.2863 3.5119 9.7731
NCI-H2722 GDSC1 3.5777 6.6815 2.4762 17.3929
NCI-H2731 GDSC1 3.6094 4.7055 3.414 10.2468
LXF 289 GDSC1 3.6405 4.3325 3.5753 8.9462
NCI-H1770 GDSC1 3.6605 4.2999 3.606 8.6247
DMS 114 GDSC1 3.6825 4.2477 3.6429 8.2502
SBC-5 CTRP2 3.6852 4.2997 3.6851 15.7174
NCI-H209 GDSC1 3.7071 5.1522 3.3259 10.4084
IST-SL1 GDSC1 3.7214 6.881 2.513 16.4968
NCI-H520 CTRP2 3.7223 6.3984 3.4054 16.5938
COLO 668 GDSC1 3.7262 4.4342 3.638 8.0358
NCI-H196 GDSC1 3.7542 4.497 3.647 7.8193
NCI-H226 GDSC1 3.7653 4.1695 3.7482 7.0673
RERF-LC-MS GDSC1 3.7669 5.0023 3.4538 9.1635
IA-LM GDSC1 3.7869 4.309 3.7415 6.9851
Lu-134-A GDSC1 3.796 5.099 3.4397 9.1307
KNS-62 GDSC1 3.803 4.225 3.7788 6.6426
NCI-H3122 GDSC1 3.8034 4.5535 3.6794 7.3263
NCI-H841 GDSC1 3.8132 4.3986 3.7441 6.819
NCI-H446 GDSC1 3.8312 4.8315 3.5948 7.8009
NCI-H2595 GDSC1 3.8634 6.8623 2.6519 14.8632
NCI-H211 GDSC1 3.8682 6.8807 2.6472 14.8792
NCI-H2804 GDSC1 3.8772 5.737 3.2165 10.4728
SK-LU-1 GDSC1 3.8906 5.9314 3.1345 11.0504
NCI-H1355 GDSC1 3.923 4.8034 3.7013 6.5617
NCI-H2009 GDSC1 3.9381 6.5405 2.8785 12.8308
NCI-H1435 CTRP2 3.9438 24.3498 -4.9129 36.5188
NCI-H2029 GDSC1 3.9443 4.9153 3.6723 6.6781
NCI-H2373 GDSC1 3.962 5.6291 3.3486 9.087
NCI-H23 CTRP2 4.0138 6.7065 3.2515 10.4927
NCI-H2085 CTRP2 4.0232 12.4721 0.4486 21.9891
NCI-H2141 GDSC1 4.0443 6.4622 3.0124 11.367
DMS 53 GDSC1 4.0676 5.361 3.5777 6.86
Lu-165 GDSC1 4.0855 4.9497 3.7943 5.105
LUDLU-1 CTRP2 4.0927 13.0291 0.8168 24.9839
NCI-H1651 GDSC1 4.1093 5.6978 3.4496 7.6899
NCI-H1573 GDSC1 4.1209 5.3462 3.6339 6.2009
NCI-H2803 GDSC1 4.1307 4.9723 3.8262 4.662
LK-2 GDSC1 4.2002 6.399 3.1803 9.4496
LCLC-103H GDSC1 4.214 6.2972 3.243 8.9052
NCI-H146 GDSC1 4.2295 7.378 2.7162 12.9308
HCC15 GDSC1 4.2467 5.2561 3.7908 4.4696
NCI-H1650 GDSC1 4.2504 6.2157 3.3148 8.204
NCI-H1092 GDSC1 4.2546 5.6449 3.6035 5.9144
COR-L23 GDSC1 4.3233 6.8547 3.0567 9.9601
COR-L95 GDSC1 4.3273 5.8806 3.547 6.0919
NCI-H82 GDSC1 4.5246 7.517 2.89 10.5389
SBC-1 GDSC1 4.5743 8.0655 2.6561 12.1419
NCI-H1993 GDSC1 4.6052 15.9682 -1.2668 31.1919
ChaGo-K-1 GDSC1 4.6108 6.5461 3.4404 5.9727
NCI-H1944 CTRP2 4.6868 10.1945 2.7522 16.6304
NCI-H441 CTRP2 4.7045 14.0108 0.896 23.2765
NCI-H460 GDSC1 4.758 6.0209 3.8026 2.7595
NCI-H345 GDSC1 4.7693 7.6339 3.0224 8.7132
NCI-H1755 GDSC1 4.8108 6.2105 3.7474 3.036
NCI-H1666 GDSC1 4.8134 20.0895 -3.1561 34.7663
NCI-H2342 CTRP2 4.8752 14.4511 0.1993 20.8991
SK-LU-1 CTRP2 4.8783 11.0871 2.4957 17.191
SHP-77 GDSC1 4.8897 6.9619 3.4399 5.1477
NCI-H647 GDSC1 5.0752 8.3051 2.9179 8.5775
NCI-H1299 GDSC1 5.1255 6.6962 3.7189 2.5138
EBC-1 GDSC1 5.1873 7.5277 3.3701 4.8871
NCI-H1651 CTRP2 5.197 15.7687 0.4592 23.5198
LC-1/sq-SF CTRP2 5.3847 12.4541 2.2744 16.9212
NCI-H1341 GDSC1 5.4136 18.6802 -1.969 30.6775
SK-MES-1 GDSC1 5.4471 7.5559 3.5185 3.2354
NCI-H226 CTRP2 5.5927 30.1828 -7.0708 34.199
NCI-H2461 GDSC1 5.6952 10.2859 2.3923 10.6131
NCI-H2170 GDSC1 5.7212 8.6449 3.1854 4.9694
DMS 273 GDSC1 5.8113 8.0083 3.5221 2.5403
KNS-62 CTRP2 5.914 11.0241 3.4451 11.1545
A-549 GDSC1 5.9387 8.4481 3.3994 3.0998
SW1573 GDSC1 5.9893 13.0811 1.2422 16.9059
HCC95 CTRP2 5.9992 16.1679 0.9449 20.3305
NCI-H2023 GDSC1 6.0852 7.7608 3.7565 0.9001
DMS 273 CTRP2 6.3044 14.5879 1.9873 16.1245
HCC1195 CTRP2 6.3541 12.8623 2.8899 12.562
Calu-1 CTRP2 6.3738 13.2559 2.7093 13.2405
RERF-LC-KJ GDSC1 6.3767 8.3708 3.6469 1.1214
NCI-H2228 GDSC1 6.3885 11.0636 2.4782 8.3061
RERF-LC-MS CTRP2 6.4433 9.1469 4.0084 2.4438
NCI-H2110 GDSC1 6.5224 9.6638 3.1852 3.4599
NCI-H838 GDSC1 6.5586 7.9493 3.874 0.2277
HCC44 GDSC1 6.5642 8.7857 3.5675 1.3053
NCI-H2286 CTRP2 6.6257 11.9758 3.5481 9.3961
NCI-H2122 GDSC1 6.682 8.2363 3.8192 0.309
NCI-H2405 GDSC1 6.6953 12.6404 1.9352 11.0398
BEN CTRP2 6.7435 8.8334 5.1807 2.4819
NCI-H2030 CTRP2 6.7937 15.8422 1.755 16.0434
Lu-65 GDSC1 6.8143 13.6603 1.5307 13.1343
NCI-H1437 GDSC1 6.8395 8.6154 3.7439 0.4388
NCI-H2291 CTRP2 6.8805 23.2934 -1.8936 26.1533
NCI-H2172 GDSC1 6.9692 8.472 3.8408 0.1764
RERF-LC-Ad1 CTRP2 7.0998 8.0677 5.7194 0.2559
MOR/CPR CTRP2 7.1004 8.0258 5.7356 0.2198
HCC1588 CTRP2 7.2581 19.6921 0.2038 20.2202
HCC366 CTRP2 7.3429 16.9019 1.6562 15.4115
HARA [Human squamous cell lung carcinoma] GDSC1 7.5311 20.8712 -1.4546 24.0451
LOU-NH91 CTRP2 7.6185 24.0142 -1.6647 24.3774
NCI-H727 CTRP2 7.6902 17.3567 1.6944 14.6859
NCI-H1792 CTRP2 7.7772 15.6253 2.6101 11.1973
NCI-H460 CTRP2 7.7871 9.0463 5.6336 0.1783
NCI-H292 GDSC1 7.8459 22.2182 -1.8865 24.622
LCLC-103H CTRP2 7.8649 9.6077 5.4556 0.5072
NCI-H838 CTRP2 7.8773 9.1864 5.6179 0.1789
NCI-H2122 CTRP2 7.8797 9.0423 5.6695 0.1082
HCC2279 CTRP2 7.9928 23.9894 -1.3605 23.0561
Calu-6 CTRP2 8.202 10.4132 5.2895 0.7429
NCI-H2405 CTRP2 8.2315 10.5665 5.242 0.8508
NCI-H1339 CTRP2 8.2787 16.9311 2.332 11.457
HCC1833 CTRP2 8.3007 16.8477 2.388 11.218
NCI-H2023 CTRP2 8.303 10.1939 5.4172 0.4012
SHP-77 CTRP2 8.3555 9.752 5.5955 0.1101
NCI-H2126 CTRP2 8.4403 9.7907 5.6122 0.0822
NCI-H650 CTRP2 8.4551 15.694 3.0507 8.51
LXF 289 CTRP2 8.5478 17.9214 2.0407 12.1027
NCI-H1299 CTRP2 8.6691 10.5465 5.4326 0.2579
HCC78 CTRP2 8.8959 10.4948 5.5328 0.0954
HCC2108 CTRP2 9.1871 11.0329 5.4522 0.1313
Lu-65 CTRP2 9.5146 23.535 -0.0047 17.1741
NCI-H1373 CTRP2 9.5233 19.387 2.0021 10.8502
A-549 CTRP2 10.6259 22.6595 1.1745 12.1261
NCI-H2172 CTRP2 11.8089 22.7724 1.8561 8.5891
RERF-LC-Ad2 CTRP2 13.1695 34.9494 -2.9879 19.4913
Hs 888.Lu CTRP2 3.5753 7.7726 2.7391 19.5192
⏷ Show the Full List of 309 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1 2.2125 7.9682 0.5395 35.1811
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 -0.5381 27.4451 -10.5378 48.2403
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
P-STS CTRP2 5.5882 10.3132 3.5188 11.5142
H-STS CTRP2 7.8003 19.4515 0.742 17.6548
SYO-1 CTRP2 8.3066 9.6671 5.6072 0.1055
Cancer Drug Sensitivity Data Curated from 70 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 6.9687 26.6404 -3.4938 29.0469
SNU-840 CTRP2 0.2272 18.0911 -5.3178 45.1635
SNU-119 CTRP2 0.2443 3.8628 0.1498 38.9195
TOV-112D GDSC1 0.6617 5.1079 0.0881 46.7896
JHOS-4 GDSC1 1.009 5.2912 0.402 43.3939
FU-OV-1 CTRP2 1.1574 15.8502 -3.3529 41.2079
RMG-I GDSC1 1.3264 12.9888 -2.7054 45.4923
A2780 CTRP2 1.5149 3.7058 1.4939 30.2462
IGROV-1 CTRP2 1.5472 9.1617 0.0367 34.4509
OVCAR-5 CTRP2 1.605 6.5751 1.0449 31.4169
OVISE GDSC1 1.7799 4.5508 1.482 33.5399
COV434 CTRP2 2.168 4.4589 2.1186 25.9914
TOV-112D CTRP2 2.2083 4.5158 2.1552 25.7355
Caov-3 CTRP2 2.2306 13.2915 -1.0991 34.8569
Caov-3 GDSC1 2.2516 5.1135 1.8059 28.7312
OC 314 CTRP2 2.3303 3.4992 2.3293 24.7472
TYK-nu CTRP2 2.3725 3.7759 2.3685 24.4761
JHOS-2 CTRP2 2.4935 4.8335 2.4202 23.9048
OAW42 CTRP2 2.8064 3.5054 2.8063 21.5724
A2780 GDSC1 2.829 6.0527 2.0308 24.1041
OAW28 GDSC1 2.865 7.6022 1.3517 28.0305
Caov-4 GDSC1 3.0245 6.7198 1.9233 23.8203
DOV13 GDSC1 3.0798 4.4743 2.9218 16.5752
RMG-I CTRP2 3.0963 25.7067 -6.3401 39.5447
ONCO-DG-1 CTRP2 3.1853 13.57 -0.3037 30.4479
TYK-nu GDSC1 3.2133 4.0381 3.176 14.0965
JHOS-2 GDSC1 3.4214 11.4952 -0.0403 31.5964
DOV13 CTRP2 3.4833 4.6001 3.4768 17.084
EFO-27 CTRP2 3.5554 11.2742 1.1473 25.2985
JHOM-1 CTRP2 3.5853 6.1597 3.3284 17.2853
OVCAR-3 GDSC1 3.6579 9.2482 1.2857 24.7332
OVK18 GDSC1 3.6853 4.2814 3.6378 8.268
TOV-21G GDSC1 3.7132 5.5986 3.1253 11.8988
ES-2 GDSC1 3.7658 4.8794 3.5067 8.7759
OVKATE GDSC1 3.9167 4.4375 3.8435 5.558
OVISE CTRP2 4.3313 5.1889 4.3217 11.4452
OAW42 GDSC1 4.4175 6.2866 3.418 6.7897
COV362 CTRP2 4.6799 8.9096 3.3606 14.2133
IGROV-1 GDSC1 4.7308 9.7083 1.9615 16.5039
ES2 CTRP2 4.9985 15.8213 0.2591 24.5423
OV-90 GDSC1 5.1144 6.6908 3.7146 2.5669
EFO-21 CTRP2 5.2436 6.5109 5.0101 6.1911
JHOC-5 CTRP2 5.2662 12.1952 2.2986 17.0853
Kuramochi GDSC1 5.3687 15.9004 -0.6198 26.8942
OVCAR-4 GDSC1 5.4961 18.8393 -1.9829 30.4904
OVTOKO CTRP2 5.5318 13.6597 1.8016 18.3641
SK-OV-3 GDSC1 5.5881 9.1533 2.8625 7.5846
OVCAR-8 GDSC1 5.7361 8.6331 3.1998 4.8364
OV56 GDSC1 5.8159 6.7371 4.0254 0.1465
OAW28 CTRP2 6.2015 17.188 0.603 21.004
OVCAR-5 GDSC1 6.3965 11.2864 2.3794 8.9356
FU-OV-1 GDSC1 6.8485 19.0315 -1.0482 24.3593
Kuramochi CTRP2 7.3735 14.4054 2.9132 10.679
TOV-21G CTRP2 7.3775 11.3561 4.4006 4.719
EFO-21 GDSC1 7.4284 14.9935 1.2996 12.978
OV-90 CTRP2 7.5076 9.6831 4.3178 0.5641
HEY A8 CTRP2 7.6408 9.7784 5.2801 1.1481
OV56 CTRP2 7.6994 12.4623 4.0878 5.5183
COV644 CTRP2 7.7105 21.0569 -0.8632 18.8742
OVCAR-8 CTRP2 7.8142 14.0165 3.4195 8
OVTOKO GDSC1 7.8566 16.5738 0.8317 14.4116
OVK18 CTRP2 8.1908 9.9782 5.452 0.3741
OV7 CTRP2 8.2244 21.2838 0.1564 18.7101
SK-OV-3 CTRP2 8.3631 21.1949 0.304 18.0546
OC 314 GDSC1 8.5963 18.5939 0.3558 15.0567
OVCAR-4 CTRP2 8.9438 19.1433 1.7256 12.6161
SNU-8 CTRP2 9.09 20.8185 1.0159 14.7446
EFO-27 GDSC1 10.2084 33.7657 -5.8293 28.6538
MCAS CTRP2 11.0626 23.6043 1.0113 12.0827
OVSAHO CTRP2 11.4542 23.1811 1.455 10.2423
⏷ Show the Full List of 70 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 43 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Aska-SS CTRP2 8.0193 9.2374 5.6523 0.1033
Yamato-SS CTRP2 8.0461 9.3579 5.6202 0.1368
TE 617.T CTRP2 -2.663 2.5978 -2.7859 57.3172
Rh41 GDSC1 -0.7878 1.3781 -0.7988 63.3011
A-204 CTRP2 0.4597 5.1819 0.1617 38.0558
GCT GDSC1 1.0618 4.2945 0.7715 41.9357
Hs 633.T GDSC1 1.1983 3.1411 1.1481 39.3192
TE 441.T CTRP2 1.4376 2.8145 1.4368 30.6938
Rh30 GDSC1 1.4511 2.9503 1.4311 36.0064
G-402 GDSC1 1.5449 4.8204 1.1418 36.8493
G-401 GDSC1 1.5844 4.4509 1.2982 35.819
G-401 CTRP2 1.6463 3.8014 1.6244 29.3738
EW-8 GDSC1 1.8368 3.5631 1.773 31.4616
SW684 GDSC1 1.92 5.2044 1.416 33.0021
GCT CTRP2 1.9307 3.9251 1.9113 27.4709
KYM-1 CTRP2 2.2295 3.9439 2.2178 25.4544
KYM-1 GDSC1 2.285 2.9766 2.2841 25.4674
Hs 729.T CTRP2 2.4393 3.1359 2.4393 24.0174
Rh18 CTRP2 2.4482 6.5199 1.9803 25.5891
SK-UT-1 GDSC1 2.4891 3.378 2.4805 22.964
SW872 GDSC1 2.628 3.9052 2.5681 21.5584
SW982 GDSC1 2.75 4.0673 2.6687 20.1744
SK-LMS-1 GDSC1 2.7596 4.7301 2.4902 21.3299
A-204 GDSC1 3.0583 5.075 2.6832 18.3707
Rh18 GDSC1 3.1102 4.0548 3.0617 15.4581
VA-ES-BJ GDSC1 3.3887 4.4204 3.275 12.4187
HT-1080 GDSC1 3.5821 4.201 3.5441 9.4935
MFH-ino GDSC1 3.6432 4.635 3.4772 9.6162
RD GDSC1 3.8503 9.7448 1.2081 24.3533
MES-SA GDSC1 4.0363 4.6569 3.8819 4.6657
HT-1080 CTRP2 4.1474 5.4595 4.0996 12.8005
G-402 CTRP2 5.0526 9.5906 3.3894 13.2186
RKN GDSC1 5.8893 7.8475 3.6305 1.7704
BT-12 CTRP2 6.979 7.9021 5.7311 0.2873
BT-16 CTRP2 7.0891 9.4478 5.1145 2.2924
RKN CTRP2 7.3759 9.1656 5.404 0.9669
RD CTRP2 7.6066 14.1046 2.4302 7.3314
SK-UT-1 CTRP2 7.7789 12.46 3.2913 3.713
SW982 CTRP2 7.7853 8.9049 5.6829 0.1096
MES-SA CTRP2 7.8132 9.001 5.6595 0.1341
Tm87-16 CTRP2 8.0404 9.3699 5.6139 0.1462
TTC-709 CTRP2 8.2039 9.7407 5.5438 0.2078
SK-LMS-1 CTRP2 8.3635 18.3669 1.6927 13.6053
⏷ Show the Full List of 43 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2 1.2965 4.844 1.1343 32.1665
NCI-H28 CTRP2 2.032 2.9356 2.032 26.7312
NCI-H2452 CTRP2 2.402 6.2744 1.7513 21.3763
MPP 89 CTRP2 2.4948 3.7463 2.4925 23.6555
MPP 89 GDSC1 2.8899 3.7413 2.8711 18.0195
IST-Mes1 GDSC1 3.491 4.8748 3.2212 12.2519
MSTO-211H GDSC1 4.2508 5.6014 3.6219 5.7839
NCI-H2452 GDSC1 4.5129 5.8666 3.7024 4.2369
NCI-H2052 GDSC1 4.8483 7.5681 3.1139 7.7663
NCI-H28 GDSC1 4.8967 8.1336 2.8713 9.4656
NCI-H2052 CTRP2 6.576 16.2386 0.6668 15.8616
JL-1 CTRP2 7.4174 13.3204 3.4775 8.3706
ACC-MESO-1 CTRP2 8.4205 13.9124 3.8703 5.4257
IST-Mes1 CTRP2 9.862 25.6846 -0.8046 18.814
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
VCaP GDSC1 2.1683 5.2339 1.672 30.0344
VCaP CTRP2 2.5178 4.8297 2.4465 23.736
LNCaP clone FGC CTRP2 2.6432 4.9097 2.5696 22.9086
PC-3 GDSC1 2.7625 3.962 2.7031 19.8745
22Rv1 CTRP2 3.021 5.7566 2.8188 20.8428
DU145 CTRP2 3.1436 11.2441 0.7568 27.638
PaCa-3 CTRP2 3.3285 5.0706 3.2786 18.2625
22Rv1 GDSC1 3.4423 4.4274 3.3312 11.7331
LNCaP clone FGC GDSC1 3.5328 5.0734 3.1821 12.3274
DU145 GDSC1 3.7855 7.5167 2.2581 18.069
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 -0.4476 6.9881 -1.319 44.5902
A-253 GDSC1 6.8705 15.061 0.8992 16.3681
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1 3.0364 4.988 2.6939 18.409
Cancer Drug Sensitivity Data Curated from 59 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-N87 CTRP2 -6.5716 -3.5619 -6.5719 82.5855
NCC-StC-K140 CTRP2 -5.301 7.2967 -6.7005 64.3435
NUGC-4 CTRP2 -2.698 13.8271 -6.3516 53.7957
SNU-216 CTRP2 -1.8079 5.8318 -2.468 51.8338
GCIY GDSC1 -1.1771 3.8523 -1.5579 62.9425
NUGC-4 GDSC1 -0.3278 10.2343 -3.0459 53.1927
HSC-39 GDSC1 -0.2014 1.6302 -0.2087 56.4279
AGS GDSC1 0.6485 5.8414 -0.1847 47.1896
MKN7 CTRP2 0.9787 6.8124 0.2887 35.7826
SNU-1 GDSC1 1.2214 2.2992 1.2196 38.7672
NCI-N87 GDSC1 1.3155 15.4493 -3.9103 46.2652
SCH GDSC1 1.3741 3.5935 1.2705 37.4274
ECC10 CTRP2 1.4361 3.4961 1.4225 30.7464
NUGC-3 CTRP2 1.6056 20.3553 -5.0792 41.6289
IM95 GDSC1 1.6118 4.9303 1.1783 36.2191
SNU-1 CTRP2 1.914 3.3799 1.9112 27.5266
MKN1 GDSC1 1.9468 6.3296 0.9993 34.8641
SNU-16 CTRP2 1.9486 2.8129 1.9486 27.2868
MKN28 GDSC1 2.0211 3.4452 1.9849 28.9882
RERF-GC-1B GDSC1 2.054 4.6079 1.7632 30.1755
HGC-27 CTRP2 2.1041 3.2281 2.1037 26.2521
KATO III GDSC1 2.1179 4.8857 1.742 29.9173
Fu97 GDSC1 2.2734 3.4478 2.2507 25.7501
LMSU CTRP2 2.3859 3.9992 2.3759 24.407
KE-39 CTRP2 2.4473 15.2892 -1.8353 35.6208
HuG1-N CTRP2 2.4647 3.8046 2.4613 23.8597
Hs 746.T CTRP2 2.5307 4.1542 2.5181 23.4509
TGBC11TKB GDSC1 2.6453 3.8145 2.6016 21.237
ECC10 GDSC1 2.6935 4.4383 2.5117 21.5536
NUGC-3 GDSC1 2.7644 3.2694 2.7639 19.4724
HGC-27 GDSC1 2.8135 3.2814 2.8131 18.8577
MKN7 GDSC1 2.8149 4.8041 2.5243 20.7904
MKN1 CTRP2 2.8666 4.4396 2.8499 21.227
23132/87 GDSC1 2.8705 3.3853 2.8695 18.1489
SNU-601 CTRP2 2.9981 16.8219 -2.0544 34.5836
MKN74 CTRP2 3.0332 11.8067 0.3854 29.031
Hs 746.T GDSC1 3.1789 6.8655 2.0059 22.526
MKN45 GDSC1 3.4708 4.1527 3.4332 10.8817
RF-48 GDSC1 3.7065 4.4524 3.6106 8.3341
SNU-16 GDSC1 4.8996 6.1481 3.8336 2.1933
IM95 CTRP2 4.9091 17.667 -1.38 25.5776
Fu97 CTRP2 4.9139 6.3222 4.2938 3.6602
KATO III CTRP2 4.9978 10.008 3.1347 14.3795
SH-10-TC CTRP2 5.2862 9.1366 3.8285 10.8857
SNU-5 GDSC1 6.0782 7.3888 3.893 0.3824
OCUM-1 GDSC1 6.3182 8.3598 3.6252 1.2814
GSU CTRP2 7.0178 7.7702 5.7972 0.1292
MKN45 CTRP2 7.2285 8.5831 5.5735 0.5616
SNU-620 CTRP2 7.5709 8.8147 5.6332 0.2461
23132/87 CTRP2 7.6359 9.2829 5.4813 0.5643
AGS CTRP2 7.9417 16.112 2.4909 11.3876
SNU-5 CTRP2 8.1909 14.5895 3.4012 7.5327
ECC12 CTRP2 8.1916 9.7184 5.5471 0.206
SNU-719 CTRP2 10.1584 22.6091 0.8889 13.6276
SNU-668 CTRP2 11.5213 23.6044 1.3006 10.6444
SNG-M GDSC1 -0.7055 3.8187 -1.0359 59.5357
SNG-M CTRP2 3.1383 8.9461 1.789 24.243
SNU-1077 CTRP2 8.2456 9.8737 5.512 0.2469
SNU-685 CTRP2 8.3293 13.0155 4.2289 4.1813
⏷ Show the Full List of 59 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 27 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ML-1 [Human leukemia] CTRP2 0.2437 11.7009 -2.3912 43.0359
KMH-2 GDSC1 1.199 3.1866 1.1434 39.3378
IHH-4 GDSC1 1.8093 3.504 1.7521 31.7638
HTC-C3 GDSC1 1.8843 4.5304 1.602 32.19
B-CPAP GDSC1 2.0332 3.0773 2.0256 28.6565
TT2609-C02 GDSC1 2.2202 3.1335 2.2149 26.3048
SW579 CTRP2 2.377 2.9127 2.377 24.4329
8505C CTRP2 2.9824 4.4295 2.9699 20.4416
CGTH-W-1 GDSC1 2.992 4.1319 2.9177 17.1049
8505C GDSC1 2.9949 3.9932 2.9484 16.8856
ML-1 [Human leukemia] GDSC1 3.2128 4.3473 3.1044 14.577
FTC-133 GDSC1 3.2454 3.9734 3.2207 13.6136
CAL-62 GDSC1 3.3629 4.3391 3.2705 12.5953
8305C GDSC1 3.5992 4.3816 3.5161 9.5834
BHT-101 GDSC1 3.6243 4.6882 3.4366 10.0065
ASH-3 GDSC1 3.7135 4.2762 3.6698 7.8903
K5 GDSC1 3.7207 5.5778 3.1425 11.7338
WRO GDSC1 3.8218 4.2646 3.7906 6.4538
TT2609-C02 CTRP2 3.8277 6.0368 3.6273 15.4687
FTC-133 CTRP2 4.1342 7.0433 3.6218 14.5963
8305C CTRP2 5.4239 11.1024 2.9814 14.0593
TT GDSC1 6.0336 7.9194 3.6705 1.3687
TT CTRP2 7.034 19.8285 -0.0413 21.324
FTC-238 CTRP2 7.1693 13.1124 3.3984 9.0841
B-CPAP CTRP2 7.7227 14.6277 3.0583 9.5558
CGTH-W-1 CTRP2 8.0764 13.3706 3.9047 5.7311
BHT-101 CTRP2 8.6438 9.9095 5.642 0.0419
⏷ Show the Full List of 27 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 68 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 -5.6912 5.1808 -6.5379 67.411
SNU-1214 CTRP2 -2.8739 7.6786 -4.1792 56.1272
PE/CA-PJ34 (clone C12) CTRP2 -2.6762 6.9774 -3.7428 55.5948
SNU-1076 CTRP2 -2.5518 7.0758 -3.6376 55.0344
SCC-25 CTRP2 -2.526 6.317 -3.3846 55.179
CAL-27 CTRP2 -2.2682 15.1033 -6.4582 52.3759
BICR 56 CTRP2 -1.7698 5.7521 -2.4055 51.6453
SCC-9 GDSC1 -1.167 4.1964 -1.6345 62.3482
HSC-2 CTRP2 -0.9836 8.3999 -2.3769 47.7581
SCC-15 GDSC1 -0.9724 3.1915 -1.1912 62.4933
BHY CTRP2 -0.575 9.4007 -2.3099 46.0024
PCI-04B GDSC1 -0.5472 6.4618 -1.6985 56.0146
SCC-4 CTRP2 -0.37 7.2606 -1.3221 44.2526
BB30-HNC GDSC1 0.296 7.3519 -1.1544 50.1795
NCI-H3118 GDSC1 0.3646 13.4741 -3.8608 49.8275
BICR 6 CTRP2 0.4995 6.4582 -0.1247 38.597
PE/CA-PJ15 GDSC1 0.5141 9.1383 -1.7004 48.8719
BICR 31 CTRP2 0.5737 9.4583 -1.1113 40.2076
HSC-4 CTRP2 0.5912 9.3777 -1.0606 40.0604
PE/CA-PJ15 CTRP2 0.6776 13.7654 -2.8642 42.1088
SAT [Human HNSCC] GDSC1 0.9595 9.8248 -1.5642 46.3503
BHY GDSC1 1.0536 9.3523 -1.2532 45.5748
CAL-33 CTRP2 1.0651 7.8131 0.0421 36.0968
DOK GDSC1 1.1314 6.696 -0.0068 43.3714
CAL-27 GDSC1 1.1901 5.3351 0.5822 41.531
SCC-25 GDSC1 1.2075 5.6896 0.4715 41.718
BICR 16 CTRP2 1.2724 13.2549 -2.0342 39.2787
PE/CA-PJ41 (clone D2) CTRP2 1.2991 23.5277 -6.9101 43.5116
PCI-06A GDSC1 1.3876 10.2264 -1.3284 43.9017
Ca9-22 GDSC1 1.5078 5.1972 0.974 37.8412
SKN-3 GDSC1 1.5765 6.7608 0.4313 39.3147
BICR 22 CTRP2 1.9299 4.7904 1.8239 27.7696
PE/CA-PJ49 CTRP2 1.9316 13.1175 -1.3135 36.1332
HO-1-N-1 GDSC1 1.9846 3.6511 1.918 29.6365
OSC-20 GDSC1 2.0077 4.3411 1.791 30.2885
BICR 31 GDSC1 2.0675 6.7488 0.9443 34.3775
FaDu CTRP2 2.2385 11.2648 -0.1577 32.7516
KOSC-2 GDSC1 2.3946 3.6408 2.3578 24.3251
JHU-011 GDSC1 2.4671 4.7419 2.1692 25.1471
BICR 18 CTRP2 2.4974 4.316 2.4749 23.7058
JHU-022 GDSC1 2.5732 3.6995 2.5405 22.0666
PCI-15A GDSC1 2.6288 3.5179 2.6166 21.2412
SCC-4 GDSC1 2.8001 3.6214 2.7876 19.1013
OSC-19 GDSC1 3.0162 7.89 1.3598 27.2396
HSC-3 GDSC1 3.3131 4.1218 3.2684 12.8978
BICR 10 GDSC1 3.3209 4.1964 3.261 12.9008
CAL-33 GDSC1 3.5418 6.9375 2.3182 18.6952
BICR 78 GDSC1 3.7996 4.5097 3.6915 7.261
Detroit 562 GDSC1 3.8182 4.4645 3.7275 6.9068
FaDu GDSC1 4.0209 4.5135 3.9267 4.413
LB771-HNC GDSC1 4.1296 5.2083 3.7098 5.5726
SNU-1066 CTRP2 4.5294 17.5264 -1.0033 28.8516
HO-1-u-1 GDSC1 4.5504 5.7838 3.7716 3.5802
BICR 22 GDSC1 4.5629 5.9857 3.6813 4.2439
YD-8 CTRP2 4.6837 12.8364 1.457 21.4636
SCC-9 CTRP2 4.9676 21.1206 -2.4088 30.8096
PCI-30 GDSC1 5.088 14.8838 -0.3349 26.7442
HSC-4 GDSC1 5.8823 7.3863 3.8133 0.8336
HSC-2 GDSC1 6.2247 7.493 3.9113 0.2622
PCI-38 GDSC1 6.4253 8.0322 3.7947 0.5013
SAS GDSC1 6.4603 8.3898 3.6756 0.9218
KON GDSC1 6.7959 8.3338 3.8266 0.2516
HSC-3 CTRP2 6.801 18.7679 0.3017 20.7644
BB49-HNC GDSC1 6.9944 8.8209 3.7292 0.409
SNU-1041 CTRP2 7.2007 19.0262 0.4902 19.4724
SNU-46 CTRP2 7.9647 10.6117 5.0928 1.484
SNU-899 CTRP2 8.2579 9.7157 5.5728 0.1545
Detroit 562 CTRP2 10.3598 25.0186 -0.1315 16.3297
⏷ Show the Full List of 68 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 36 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-BLC1 CTRP2 -7.1387 -0.298 -7.2277 78.955
SCaBER CTRP2 -3.3306 25.9017 -12.476 53.4183
5637 CTRP2 -0.1203 5.068 -0.444 41.8181
VM-CUB-1 CTRP2 0.7613 6.3883 0.1813 36.8599
CAL-29 CTRP2 1.3225 4.5499 1.2089 31.8348
5637 GDSC1 1.6665 7.337 0.2747 39.22
CAL-29 GDSC1 1.9742 4.9705 1.5574 31.8821
RT-4 GDSC1 2.2003 4.0513 2.0744 27.3272
HT-1197 CTRP2 2.2636 3.35 2.2631 25.1897
UM-UC-3 GDSC1 2.3911 3.599 2.3593 24.3366
BFTC-905 GDSC1 2.729 3.3713 2.7265 19.9269
639V GDSC1 2.8212 4.4928 2.6345 19.9952
RT-112 GDSC1 2.8364 3.3053 2.836 18.5722
HT-1197 GDSC1 2.9289 4.4957 2.7509 18.5939
TCCSUP CTRP2 2.949 4.8565 2.9013 20.7831
KU-19-19 GDSC1 3.0356 3.6239 3.0312 16.1065
647V GDSC1 3.0874 7.0134 1.8469 24.0035
SW1710 GDSC1 3.1376 4.122 3.078 15.1895
253J-BV CTRP2 3.1722 4.3717 3.1665 19.1539
HT-1376 GDSC1 3.3435 9.9361 0.6629 29.1594
UM-UC-3 CTRP2 3.5187 5.7514 3.3621 17.3683
HT-1376 CTRP2 3.6727 20.3283 -3.159 34.7881
T24 GDSC1 3.9016 5.5336 3.338 9.4287
SW780 GDSC1 4.1024 4.9303 3.8198 4.8337
J82 GDSC1 4.1397 5.5756 3.5374 6.8804
TCCSUP GDSC1 4.8356 12.2149 0.7949 22.809
KMBC-2 CTRP2 4.8823 18.5796 -1.2162 28.562
T24 CTRP2 5.1939 8.8287 3.8925 10.8305
BC-3C CTRP2 5.6376 11.0126 3.2136 12.6663
253J CTRP2 6.9273 15.6221 1.9699 15.0257
SW1710 CTRP2 6.9339 15.0404 2.2645 13.924
639V CTRP2 7.14 8.5184 5.5571 0.6719
KU-19-19 CTRP2 7.5861 8.7361 5.668 0.1786
RT-112 CTRP2 8.1578 9.5778 5.5843 0.1606
647V CTRP2 8.268 21.1692 0.2457 18.3795
J82 CTRP2 9.7326 19.9032 1.0635 9.6601
⏷ Show the Full List of 36 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DSH1 GDSC1 -2.7403 1.852 -2.8781 76.2535
BPH-1 GDSC1 -1.7567 5.2973 -2.6017 64.0326
UWB1.289 GDSC1 -1.2509 12.535 -5.0178 56.0345
OVMIU GDSC1 -0.3333 5.3767 -1.0812 55.2802
C-33 A GDSC1 -0.143 4.8362 -0.7003 54.1057
HT-3 GDSC1 0.0422 4.1574 -0.3047 52.7553
ME-180 GDSC1 0.0545 4.9662 -0.5259 52.3842
Ca Ski GDSC1 0.6599 2.391 0.6449 45.8295
SW954 GDSC1 0.8609 3.566 0.7211 43.7803
KGN GDSC1 0.9969 5.3792 0.3581 43.5898
PA-1 GDSC1 1.5831 2.9183 1.5698 34.3174
NEC8 GDSC1 1.6194 2.5836 1.6175 33.7934
TC-YIK GDSC1 1.7617 4.0064 1.6073 32.9428
C-4-I GDSC1 2.0429 4.9914 1.6244 31.0725
SKN GDSC1 2.0581 3.6976 1.9896 28.7314
OMC-1 [Human cervical carcinoma] GDSC1 2.0763 3.2707 2.0591 28.179
NCC-IT GDSC1 2.1665 3.5646 2.1249 27.2066
DoTc2 4510 GDSC1 2.6888 9.4899 0.2765 33.702
PEO1 GDSC1 2.7486 8.7327 0.6991 31.7591
NT2-D1 GDSC1 2.7937 4.1139 2.7059 19.6714
CAL-39 GDSC1 2.8916 6.2332 2.014 23.8936
SiHa GDSC1 2.9035 3.3344 2.9032 17.7321
PWR-1E GDSC1 2.9447 5.1852 2.519 20.1325
HEC-1 GDSC1 3.0429 3.9367 3.0093 16.2024
JAR GDSC1 3.2717 4.2689 3.1899 13.6622
SiSo GDSC1 3.2866 4.5647 3.1176 14.0744
LB831-BLC GDSC1 3.3474 4.416 3.2313 12.9499
MS751 GDSC1 3.3727 4.2657 3.3008 12.334
SW962 GDSC1 3.5243 5.1327 3.1477 12.6231
SW756 GDSC1 3.5266 7.5089 2.0252 20.7941
JEG-3 GDSC1 3.6059 4.3415 3.5351 9.4163
HeLa GDSC1 3.8055 4.0734 3.8021 6.4768
HEY GDSC1 3.8106 5.7754 3.1349 11.3913
SKG-IIIa GDSC1 3.8171 4.2759 3.7828 6.5334
ACC-OV7 GDSC1 4.4786 7.9194 2.6521 12.5063
OV17R GDSC1 5.0131 7.7325 3.1526 6.9857
OVCA433 GDSC1 5.0257 10.9396 1.5798 17.9078
OVCA420 GDSC1 5.793 21.7566 -3.2018 32.4018
JHOS-3 GDSC1 5.9746 19.7591 -2.0663 29.4545
HeLa CTRP2 7.3704 8.389 5.71 0.1719
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug

References

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