Details of the Drug

General Information of Drug (ID: DMSOB3U)

Drug Name
KH-CB19
Synonyms KH CB19
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 338.2
Logarithm of the Partition Coefficient (xlogp) 3.1
Rotatable Bond Count (rotbonds) 4
Hydrogen Bond Donor Count (hbonddonor) 1
Hydrogen Bond Acceptor Count (hbondacc) 4
Chemical Identifiers
Formula
C15H13Cl2N3O2
IUPAC Name
ethyl 3-[(E)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methylindole-2-carboxylate
Canonical SMILES
CCOC(=O)C1=C(C2=C(N1C)C(=C(C=C2)Cl)Cl)/C(=C\\N)/C#N
InChI
InChI=1S/C15H13Cl2N3O2/c1-3-22-15(21)14-11(8(6-18)7-19)9-4-5-10(16)12(17)13(9)20(14)2/h4-6H,3,18H2,1-2H3/b8-6-
InChIKey
CXJCGSPAPOTTSF-VURMDHGXSA-N
Cross-matching ID
PubChem CID
44237094
TTD ID
D00BAJ

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
CDC-like kinase 1 (CLK1) TTE6YDG CLK1_HUMAN Inhibitor [2]
CDC-like kinase 3 (CLK3) TTQPE1U CLK3_HUMAN Inhibitor [2]
Dual-specificity tyrosine-phosphorylation regulated kinase 1A (DYRK1A) TTSBVFO DYR1A_HUMAN Inhibitor [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 102 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 6.1383 7.498 3.6474 0.1472
JK1 CTRP2 6.9476 9.3632 3.2854 0.5234
JM1 CTRP2 6.4606 8.0264 3.5809 0.1668
OPM-2 CTRP2 4.4065 5.6457 3.5555 1.6885
SK-MM-2 CTRP2 4.512 69.1548 -28.0932 43.3318
EB1 CTRP2 4.6097 6.3446 3.3589 2.1869
HPB-ALL CTRP2 4.766 6.575 3.3535 1.993
Ci-1 CTRP2 4.9264 5.8786 3.7569 0.3888
SIG-M5 CTRP2 4.9377 6.2127 3.6219 0.8026
OCI-AML-2 CTRP2 4.9924 7.6002 3.0159 3.0247
MC116 CTRP2 5.1599 5.9526 3.8283 0.1198
SUP-T1 CTRP2 5.1633 9.1984 2.3636 5.4073
NU-DUL-1 CTRP2 5.1859 7.2214 3.3136 1.6438
HuNS1 CTRP2 5.2046 7.1331 3.3641 1.4424
Granta-519 CTRP2 5.2277 10.6547 1.6989 8.0105
KYO-1 CTRP2 5.2635 7.2176 3.3598 1.3985
KMS-34 CTRP2 5.2995 7.0167 3.467 1.0003
EoL-1 CTRP2 5.3426 9.9981 2.1016 6.2011
Karpas-299 CTRP2 5.3606 7.489 3.294 1.5341
AML-193 CTRP2 5.3837 7.1664 3.4469 0.9953
NB4 CTRP2 5.3955 8.3684 2.9141 2.9024
KMS-12-BM CTRP2 5.4018 7.0502 3.5051 0.7986
SKM-1 CTRP2 5.4195 7.075 3.5035 0.7903
BL-70 CTRP2 5.423 6.6056 3.6923 0.2877
MM1.S CTRP2 5.4459 7.0485 3.5274 0.7007
SUP-T11 CTRP2 5.4873 7.9303 3.1691 1.8497
HL-60 CTRP2 5.4975 6.8799 3.6188 0.4232
KMS-18 CTRP2 5.503 9.8146 2.3004 5.171
Raji CTRP2 5.5089 6.8857 3.6215 0.4106
Reh CTRP2 5.5468 11.1901 1.6666 7.6453
KO52 CTRP2 5.5938 6.7089 3.7228 0.1693
A4/Fukuda CTRP2 5.6035 8.64 2.9162 2.6496
U-937 CTRP2 5.625 7.1554 3.5674 0.4837
CMK CTRP2 5.6293 7.5591 3.4059 0.9319
MOLT-13 CTRP2 5.6409 7.0621 3.6105 0.3732
HEL 92.1.7 CTRP2 5.7037 6.9877 3.6643 0.2374
BV-173 CTRP2 5.7296 7.5133 3.4728 0.6712
Karpas-422 CTRP2 5.7337 10.123 2.3067 4.8323
REC-1 CTRP2 5.7695 9.1603 2.778 2.9768
SU-DHL-4 CTRP2 5.782 6.9962 3.6917 0.1675
Kasumi-2 CTRP2 5.8116 9.688 2.5604 3.7498
SET-2 CTRP2 5.84 6.9911 3.7152 0.1208
JJN-3 CTRP2 5.8599 7.6538 3.4763 0.587
RS4;11 CTRP2 5.8677 8.0984 3.2995 1.079
RL CTRP2 5.8889 7.5837 3.5163 0.4742
RPMI-6666 CTRP2 5.8912 7.2807 3.6311 0.2362
OCI-M1 CTRP2 5.9066 7.2756 3.639 0.2179
JeKo-1 CTRP2 5.9147 7.5125 3.5545 0.3772
DND-41 CTRP2 5.9206 7.9959 3.3673 0.8435
MOLM-6 CTRP2 5.9398 7.5862 3.5371 0.4042
Mino CTRP2 5.9447 7.084 3.7209 0.0947
AMO1 CTRP2 5.9535 7.2622 3.6618 0.1691
SU-DHL-6 CTRP2 5.9656 7.5278 3.5697 0.3257
THP-1 CTRP2 5.9832 7.6577 3.5282 0.405
Kasumi-1 CTRP2 5.9921 7.8071 3.4747 0.5224
TF-1 CTRP2 6.0029 7.1427 3.7215 0.085
MOLP-2 CTRP2 6.0168 8.3332 3.2754 1.0439
SU-DHL-8 CTRP2 6.0299 7.2004 3.7113 0.0913
U266B1 CTRP2 6.03 9.2335 2.8962 2.2723
RCH-ACV CTRP2 6.042 8.2127 3.3366 0.8516
L-540 CTRP2 6.0461 7.6743 3.5479 0.339
Pfeiffer CTRP2 6.0614 7.4768 3.6261 0.1957
P3HR-1 CTRP2 6.1092 7.4011 3.6706 0.1237
MOLT-16 CTRP2 6.1585 7.4718 3.6639 0.1225
GA-10 CTRP2 6.16 7.4236 3.6811 0.1028
KMS-20 CTRP2 6.1655 7.8323 3.5375 0.3162
Hs 611.T CTRP2 6.1795 8.7373 3.1879 1.1884
PL21 CTRP2 6.1815 7.7872 3.5604 0.2695
GDM-1 CTRP2 6.1956 8.6325 3.2388 1.0282
ST486 CTRP2 6.199 7.7667 3.5746 0.24
L-363 CTRP2 6.2006 7.4636 3.6818 0.0956
RPMI-8226 CTRP2 6.2287 7.9689 3.5124 0.3417
LP-1 CTRP2 6.2716 7.8604 3.5688 0.2292
NOMO-1 CTRP2 6.2733 7.7581 3.6059 0.1737
Karpas-620 CTRP2 6.2975 7.5617 3.6825 0.0813
MOLP-8 CTRP2 6.3186 7.9019 3.5719 0.2121
Daudi CTRP2 6.326 7.8819 3.5818 0.1956
OCI-AML-3 CTRP2 6.3591 7.5553 3.7059 0.0554
SUP-B15 CTRP2 6.3821 7.9941 3.563 0.2094
ME1 CTRP2 6.4297 7.6893 3.6853 0.0636
MOTN-1 CTRP2 6.487 7.9861 3.6045 0.1328
NU-DHL-1 CTRP2 6.4979 7.966 3.6153 0.119
SUP-HD1 CTRP2 6.5233 8.8982 3.2829 0.7184
SR CTRP2 6.5374 8.1587 3.5628 0.1744
L-428 CTRP2 6.538 8.0261 3.609 0.1193
F-36P CTRP2 6.5501 8.9937 3.2575 0.7673
DB CTRP2 6.5612 8.1354 3.5796 0.1486
MOLM-16 CTRP2 6.579 8.2411 3.5492 0.1835
HD-MY-Z CTRP2 6.6182 8.354 3.524 0.2094
MHH-CALL-4 CTRP2 6.7202 8.5345 3.4982 0.2221
M-07e CTRP2 6.7317 8.2362 3.6057 0.0949
OCI-Ly19 CTRP2 6.7884 18.5184 -1.0196 15.504
K-562 CTRP2 6.8 8.0002 3.7069 0.0253
HuT 78 CTRP2 6.8242 9.2458 3.2785 0.5881
TALL-1 [Human adult T-ALL] CTRP2 6.9044 8.9164 3.4319 0.2748
Mono-Mac-1 CTRP2 6.9508 9.5054 3.2331 0.6327
KMS-11 CTRP2 7.0756 8.9173 3.4947 0.1556
MHH-CALL-3 CTRP2 7.2956 9.4302 3.3964 0.2336
Ri-1 CTRP2 7.686 9.8822 3.3811 0.1793
OCI-Ly3 CTRP2 8.2617 21.036 -1.2111 13.9734
EJM CTRP2 9.2714 22.1887 -1.0937 12.3182
OCI-AML-5 CTRP2 12.4743 28.5472 -2.0615 11.4894
⏷ Show the Full List of 102 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 5.5469 7.7662 3.2748 1.4231
TE15 CTRP2 5.9997 10.0138 2.5257 3.6578
EC-GI-10 CTRP2 5.4275 8.2288 2.9984 2.5437
TE-5 CTRP2 5.5378 7.6821 3.3065 1.3246
TE-14 CTRP2 6.085 9.6295 2.751 2.7327
KYSE-70 CTRP2 6.1542 7.8092 3.5415 0.3125
TE-11 CTRP2 6.1972 8.1672 3.4243 0.5421
KYSE-150 CTRP2 6.2076 7.5515 3.6541 0.1252
KYSE-520 CTRP2 6.2096 8.1586 3.433 0.5164
KYSE-510 CTRP2 6.218 8.1201 3.4513 0.4718
TE-6 CTRP2 6.2235 8.7662 3.1974 1.1291
OE21 CTRP2 6.316 8.3073 3.4213 0.4949
KYSE-30 CTRP2 6.4572 7.6009 3.7239 0.0363
KYSE-450 CTRP2 6.5276 7.7944 3.6836 0.0553
TE-4 CTRP2 6.5526 8.311 3.5146 0.2393
OE19 CTRP2 6.6157 8.2409 3.5628 0.1587
KYSE-410 CTRP2 6.6351 8.1286 3.6084 0.1054
OE33 CTRP2 6.6624 8.245 3.5782 0.1325
TE-1 CTRP2 7.2608 9.1389 3.4846 0.1372
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 27 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 5.4017 7.0365 3.5107 0.7815
SU.86.86 CTRP2 5.4771 7.4443 3.3768 1.1446
DAN-G CTRP2 5.6216 7.1872 3.5534 0.521
YAPC CTRP2 5.7462 7.042 3.6612 0.2289
TCC-Pan2 CTRP2 5.7781 7.5472 3.4815 0.6191
Panc 05.04 CTRP2 5.7926 11.5684 1.6551 7.3269
PaTu 8902 CTRP2 5.8773 7.1827 3.6612 0.1898
PK-45H CTRP2 5.8932 8.1891 3.2743 1.1371
KP-2 CTRP2 5.9407 7.4446 3.5906 0.2942
PSN1 CTRP2 6.0037 8.4865 3.2051 1.2667
HuP-T4 CTRP2 6.0387 8.5162 3.2102 1.2242
PaTu 8988s CTRP2 6.0828 7.884 3.4841 0.4586
Hs 766T CTRP2 6.1561 7.9859 3.4762 0.444
SW1990 CTRP2 6.1873 7.9303 3.51 0.3615
PaTu 8988t CTRP2 6.1897 7.1987 3.7668 0.0313
HuP-T3 CTRP2 6.214 7.9284 3.5215 0.3295
MIA PaCa-2 CTRP2 6.277 7.4585 3.7102 0.0605
Panc 03.27 CTRP2 6.2928 7.76 3.6124 0.1606
HPAC CTRP2 6.3804 7.9458 3.5795 0.1861
L3.3 CTRP2 6.5339 7.8896 3.6539 0.0772
Panc 02.03 CTRP2 6.5632 8.2739 3.5318 0.2112
AsPC-1 CTRP2 6.5856 9.7153 2.9819 1.5136
Capan-2 CTRP2 6.6125 8.3666 3.5174 0.2202
PK-59 CTRP2 6.6994 8.6186 3.4603 0.2852
SNU-410 CTRP2 6.7263 8.647 3.4605 0.2775
Panc 08.13 CTRP2 6.7484 8.368 3.5666 0.1309
Panc 04.03 CTRP2 6.9632 8.8294 3.4845 0.1882
⏷ Show the Full List of 27 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 10.9588 28.7365 -3.0889 15.694
SK-MEL-2 CTRP2 4.807 6.7947 3.2763 2.2432
Hs 940.T CTRP2 4.9071 6.8437 3.3178 1.9511
Hs 839.T CTRP2 5.0683 7.1196 3.2899 1.8636
Hs 934.T CTRP2 5.1268 6.5091 3.5938 0.7341
WM115 CTRP2 5.1372 7.8729 2.9818 2.9661
G-361 CTRP2 5.1936 7.9864 2.9647 2.9596
Hs 852.T CTRP2 5.209 7.5649 3.1707 2.1489
Hs 936.T CTRP2 5.4643 7.142 3.4977 0.7752
SK-MEL-28 CTRP2 5.4779 7.089 3.5262 0.6826
WM1799 CTRP2 5.4976 7.1236 3.5214 0.6831
WM266-4 CTRP2 5.5078 6.6652 3.7049 0.2289
RVH-421 CTRP2 5.5884 7.5365 3.3949 0.9966
A2058 CTRP2 5.5898 6.54 3.7811 0.0878
UACC-257 CTRP2 5.6961 7.0764 3.6282 0.3112
IGR-39 CTRP2 5.7169 6.9925 3.6678 0.2266
CJM [Human melanoma] CTRP2 5.7494 7.2429 3.5875 0.3762
SK-MEL-5 CTRP2 5.8658 7.4876 3.5434 0.4229
A101D CTRP2 5.966 10.055 2.486 3.8476
HMCB CTRP2 5.995 6.9498 3.7836 0.0356
SK-MEL-3 CTRP2 6.0407 7.3393 3.667 0.1418
LOX-IMVI CTRP2 6.0544 7.8621 3.4804 0.4797
WT2-iPS CTRP2 6.0756 7.2431 3.7129 0.0829
SK-MEL-30 CTRP2 6.0781 7.5013 3.6237 0.195
Hs 944.T CTRP2 6.1456 7.8237 3.5327 0.3323
UACC-62 CTRP2 6.184 7.9308 3.5085 0.3657
Hs 895.T CTRP2 6.2167 7.7304 3.5945 0.2039
IPC-298 CTRP2 6.2448 7.4949 3.6867 0.0845
WM88 CTRP2 6.2457 11.1295 2.1614 4.7444
IGR-37 CTRP2 6.27 10.6284 2.4072 3.7902
COLO 792 CTRP2 6.2945 8.0562 3.5066 0.3298
MDA-MB-435S CTRP2 6.307 7.9314 3.5569 0.2386
WM793 CTRP2 6.3501 7.7568 3.6344 0.1226
Hs 294T CTRP2 6.3946 7.6821 3.6756 0.0753
A-375 CTRP2 6.4058 7.6986 3.6739 0.0754
Malme-3M CTRP2 6.4141 8.8654 3.2469 0.8696
COLO 829 CTRP2 6.4232 8.6739 3.3264 0.6637
MeWo CTRP2 6.4301 7.8253 3.6394 0.1043
SK-MEL-31 CTRP2 6.4563 8.526 3.3972 0.4876
COLO 800 CTRP2 6.5174 8.4894 3.4359 0.3858
Mel JuSo CTRP2 6.7307 8.1647 3.6294 0.075
HT-144 CTRP2 6.8539 8.2364 3.6475 0.0513
WM983B CTRP2 7.0553 13.4018 1.6098 5.8438
K029AX CTRP2 8.6285 17.6966 0.5916 7.6517
IGR-1 CTRP2 12.1886 31.4205 -3.5619 15.4404
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 5.7683 7.8554 3.3514 0.9947
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IMR-32 CTRP2 5.281 6.4464 3.6926 0.3537
SK-N-DZ CTRP2 5.849 7.3793 3.5775 0.3556
KP-N-SI9s CTRP2 5.9735 7.8663 3.4434 0.6086
NH-6 CTRP2 6.1321 8.8853 3.102 1.4898
SK-N-FI CTRP2 6.2233 7.5171 3.6715 0.1028
KP-N-YN CTRP2 6.2382 9.5401 2.8762 2.1434
Kelly CTRP2 6.2546 7.6049 3.6525 0.1186
CHP-126 CTRP2 6.3116 7.737 3.6274 0.1378
SK-N-SH CTRP2 6.3501 8.0447 3.5326 0.2661
NB1 CTRP2 6.3783 7.8803 3.6018 0.1567
SK-N-BE(2) CTRP2 6.7449 9.2703 3.2352 0.7225
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-869 CTRP2 6.2844 22.8722 -3.5427 23.1597
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Hs 822.T CTRP2 5.306 6.8175 3.5545 0.7193
SK-N-MC CTRP2 5.4499 6.5516 3.7236 0.2135
TC71 CTRP2 5.7052 6.826 3.7233 0.1395
A-673 CTRP2 5.9416 7.364 3.6205 0.239
MG-63 CTRP2 6.089 8.2131 3.3583 0.7642
HOS CTRP2 6.1518 8.0655 3.444 0.518
SK-ES-1 CTRP2 6.2869 7.7685 3.6073 0.1687
G-292 clone A141B1 CTRP2 6.3534 8.8534 3.2237 0.9689
SJSA-1 CTRP2 6.5566 8.1793 3.5627 0.1706
CAL-78 CTRP2 6.637 8.4349 3.5023 0.2363
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 56 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Hs 578Bst CTRP2 3.8556 5.8003 3.0309 4.905
EFM-192A CTRP2 5.1144 8.5336 2.6511 4.3153
ZR-75-1 CTRP2 5.3342 6.7945 3.5777 0.6306
HCC1419 CTRP2 5.3833 10.8751 1.7036 7.7469
BT-549 CTRP2 5.5451 9.0875 2.6727 3.6476
BT-474 CTRP2 5.6815 7.2186 3.5676 0.454
HCC1428 CTRP2 6.03 7.7303 3.5203 0.4023
DU4475 CTRP2 6.0396 7.3944 3.6472 0.1695
T-47D CTRP2 6.155 8.4187 3.3063 0.8648
MDA-MB-157 CTRP2 6.1684 8.4152 3.314 0.8359
ZR-75-30 CTRP2 6.1925 8.1481 3.4297 0.5319
MDA-MB-361 CTRP2 6.2186 8.3106 3.3781 0.642
CAL-85-1 CTRP2 6.2348 9.279 2.9873 1.7751
HCC202 CTRP2 6.2373 9.4116 2.9315 1.9576
MDA-MB-231 CTRP2 6.3686 8.0839 3.5256 0.2724
CAL-51 CTRP2 6.4951 8.0662 3.5796 0.1614
SK-BR-3 CTRP2 6.5017 8.1563 3.5504 0.199
BT-20 CTRP2 6.5409 8.2687 3.5252 0.2262
HCC1500 CTRP2 6.5959 8.5679 3.4383 0.3544
Hs 578T CTRP2 6.6425 8.7654 3.384 0.4414
HCC2218 CTRP2 6.674 8.3309 3.5526 0.16
MDA-MB-468 CTRP2 6.7988 8.2393 3.6278 0.0692
HCC38 CTRP2 6.9312 8.7687 3.494 0.1827
HCC1143 CTRP2 6.9883 9.5023 3.2499 0.5807
BT 416 CTRP2 4.914 8.9738 2.2942 6.0765
BT 498 CTRP2 5.374 6.5509 3.6925 0.309
BT 139 CTRP2 5.3887 6.6278 3.6692 0.3561
BT 482 CTRP2 5.4336 7.8583 3.1706 1.9004
BT164 CTRP2 5.451 7.134 3.4945 0.7945
BT 228 CTRP2 5.458 8.0944 3.0782 2.2117
BT 340 CTRP2 5.6015 7.0285 3.6065 0.4009
BT 231 CTRP2 5.665 8.5052 3.0136 2.2248
BT 179 CTRP2 5.6899 7.2133 3.5733 0.4362
BT 239 CTRP2 5.7179 7.1805 3.5979 0.367
BT 320 CTRP2 5.7239 6.701 3.7737 0.0737
BT 504 CTRP2 5.7945 7.0938 3.6613 0.2136
BT147 CTRP2 5.7988 7.3063 3.5842 0.3622
BT 422 CTRP2 5.9269 7.2213 3.6663 0.169
BT 359 CTRP2 5.9493 7.6535 3.5155 0.448
BT 112 CTRP2 5.9594 7.6105 3.5361 0.3979
BT 131 CTRP2 5.9816 7.1586 3.7084 0.1024
BT 444 CTRP2 6.0275 7.3009 3.6756 0.1333
BT 172 CTRP2 6.0463 7.2884 3.6869 0.1158
BT 145 CTRP2 6.0713 7.975 3.4441 0.5564
BT 271 CTRP2 6.0721 7.5068 3.6194 0.2031
BT 224 CTRP2 6.0891 7.7193 3.5486 0.3219
BT 333 CTRP2 6.1617 7.3056 3.7218 0.0639
BT 245 CTRP2 6.1646 7.4356 3.6786 0.1047
BT 286 CTRP2 6.2389 7.7004 3.6134 0.171
BT 328 CTRP2 6.2475 7.7019 3.6161 0.1654
BT 330 CTRP2 6.2984 7.4575 3.7178 0.0527
BT 440 CTRP2 6.4502 7.5656 3.7332 0.032
BT 248 CTRP2 6.4557 8.0639 3.5659 0.1879
BT 232 CTRP2 6.4901 7.7972 3.6699 0.0692
BT 159 CTRP2 6.6465 8.1474 3.606 0.1061
BT 216 CTRP2 6.6796 8.8351 3.3731 0.4491
⏷ Show the Full List of 56 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 27 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW1783 CTRP2 2.8315 35.8851 -12.8698 39.9495
M059K CTRP2 5.2712 7.1123 3.4104 1.2152
KNS-60 CTRP2 5.4502 6.6282 3.6952 0.2703
KNS-81 CTRP2 5.4792 6.4547 3.7702 0.1258
SF268 CTRP2 5.5401 8.3445 3.0131 2.3611
GMS-10 CTRP2 5.5819 6.7307 3.7103 0.1941
KG-1-C CTRP2 5.618 6.9843 3.6305 0.3389
CCF-STTG1 CTRP2 5.6915 6.7548 3.7433 0.115
DK-MG CTRP2 5.7221 7.1286 3.6193 0.3192
SF539 CTRP2 5.8489 7.6591 3.4692 0.611
DBTRG-05MG CTRP2 5.8733 7.4692 3.5536 0.3968
Hs 683 CTRP2 5.9338 8.1337 3.3173 0.9785
YH-13 CTRP2 5.9851 8.7404 3.0873 1.661
TM-31 CTRP2 6.0804 7.7514 3.5331 0.3555
T98G CTRP2 6.2043 11.6078 1.9112 5.7567
SW1088 CTRP2 6.2099 10.1328 2.5969 3.1587
8-MG-BA CTRP2 6.3136 7.8851 3.576 0.2072
U-251MG CTRP2 6.4061 7.7345 3.6619 0.086
42-MG-BA CTRP2 6.4799 8.0963 3.5634 0.1859
GOS-3 CTRP2 6.5328 8.6696 3.3748 0.5036
GaMG CTRP2 6.5514 8.05 3.6056 0.1209
U-118MG CTRP2 6.6917 13.0637 1.5397 6.5518
KALS-1 CTRP2 6.752 8.5103 3.5186 0.1873
Becker CTRP2 6.7719 8.2857 3.6029 0.0922
SNB-75 CTRP2 7.475 9.6215 3.3952 0.1997
D283 Med CTRP2 7.7707 19.8531 -0.9771 13.9277
A-172 CTRP2 11.0444 31.0962 -4.1518 18.0287
⏷ Show the Full List of 27 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-3 CTRP2 5.6741 12.0173 1.3545 8.6939
EFE-184 CTRP2 5.7998 8.0068 3.3038 1.1169
EN CTRP2 5.8019 10.8512 2.0056 5.9261
AN3-CA CTRP2 5.846 7.7369 3.4369 0.6979
JHUEM-1 CTRP2 5.9541 9.3696 2.7921 2.7218
JHUEM-7 CTRP2 6.2152 7.6387 3.6263 0.1586
ESS-1 CTRP2 6.2762 7.7158 3.6218 0.1518
MFE-319 CTRP2 6.4226 7.9159 3.6055 0.1433
MFE-296 CTRP2 6.4387 8.1847 3.5163 0.2674
HEC-151 CTRP2 6.6601 8.0797 3.6336 0.0795
HEC-1-A CTRP2 6.7115 8.3 3.5768 0.126
HEC-50B CTRP2 7.0809 8.6487 3.5875 0.071
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 13 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TUHR10TKB CTRP2 4.9491 7.0261 3.2592 2.1253
TUHR14TKB CTRP2 5.4099 8.1878 3.0066 2.5334
KMRC-1 CTRP2 5.8207 7.5841 3.4862 0.5832
RCC10RGB CTRP2 5.8912 7.1553 3.6763 0.163
VMRC-RCZ CTRP2 5.9905 8.8526 3.0416 1.8088
Caki-1 CTRP2 5.9948 8.8243 3.0562 1.7561
KMRC-2 CTRP2 6.0122 16.0598 -0.3802 14.6218
786-O CTRP2 6.1468 8.1364 3.4144 0.5901
Caki-2 CTRP2 6.2958 8.8774 3.1867 1.1109
VMRC-RCW CTRP2 6.4021 7.8064 3.636 0.1123
ACHN CTRP2 6.6031 8.2598 3.5515 0.1754
KMRC-3 CTRP2 7.0064 12.9146 1.8041 5.1847
UO-31 CTRP2 7.0694 8.8693 3.509 0.1413
⏷ Show the Full List of 13 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-C5 CTRP2 4.2598 6.2915 3.1255 3.7191
CCK-81 CTRP2 4.8535 10.7359 1.3781 9.9344
SNU-61 CTRP2 5.0007 7.1683 3.2253 2.1916
SW948 CTRP2 5.0747 6.6212 3.518 1.03
LoVo CTRP2 5.0916 8.0261 2.879 3.4336
HCT 8 CTRP2 5.0995 6.6953 3.4991 1.0718
SW1417 CTRP2 5.1085 8.4431 2.6906 4.1645
CW-2 CTRP2 5.2644 7.8929 3.0533 2.5289
MDST8 CTRP2 5.4602 7.3266 3.4182 1.0245
HCC-56 CTRP2 5.4851 6.5157 3.7506 0.1547
SNU-503 CTRP2 5.4937 8.0092 3.1375 1.9567
LS123 CTRP2 5.5276 10.5522 1.9623 6.4885
SNU-1033 CTRP2 5.5523 8.1902 3.09 2.0669
NCI-H747 CTRP2 5.5839 11.0977 1.7376 7.3057
T84 CTRP2 5.6639 7.8764 3.2894 1.2718
COLO201 CTRP2 5.7443 7.4132 3.5193 0.5407
NCI-H716 CTRP2 5.759 10.2147 2.2798 4.9045
CL-11 CTRP2 5.8003 7.8143 3.384 0.8756
C2BBe1 CTRP2 5.8906 8.3757 3.1942 1.3915
SNU-C4 CTRP2 5.9678 6.9508 3.774 0.0442
SNU-407 CTRP2 5.9894 8.3658 3.2484 1.1443
NCI-H508 CTRP2 6.0629 7.4445 3.6382 0.177
HCT 15 CTRP2 6.0742 8.1753 3.3666 0.7509
COLO 320 CTRP2 6.0971 9.0834 2.9987 1.8575
HT-55 CTRP2 6.2111 7.6279 3.6287 0.1564
LS1034 CTRP2 6.3709 7.8022 3.6262 0.1283
GP2d CTRP2 6.4541 8.4141 3.4383 0.4041
SW620 CTRP2 6.4699 8.0455 3.5776 0.1691
KM12 CTRP2 6.5256 7.8787 3.6548 0.0775
RCM-1 [Human ESC] CTRP2 6.5786 8.0333 3.6209 0.1012
SNU-C1 CTRP2 6.6539 8.4939 3.4877 0.2543
RKO CTRP2 7.074 8.6751 3.5763 0.0798
COLO 678 CTRP2 7.6902 20.0245 -1.1151 14.4706
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 18 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-886 CTRP2 -0.0247 2.3758 -4.7157 0.4258
SNU-761 CTRP2 5.0634 6.6737 3.4886 1.143
JHH-6 CTRP2 5.1873 6.3267 3.6978 0.3909
SNU-387 CTRP2 5.207 14.4156 -0.1758 15.271
HuH-6 CTRP2 5.686 10.6305 2.0332 5.9783
Hep-G2 CTRP2 5.7505 6.9456 3.6978 0.1663
SK-HEP-1 CTRP2 5.7822 7.1825 3.6238 0.287
HuH-1 CTRP2 5.8179 7.3767 3.5654 0.3949
JHH-1 CTRP2 5.9366 7.3309 3.6306 0.2232
SNU-475 CTRP2 5.9434 7.3612 3.6223 0.2354
JHH-5 CTRP2 6.0148 8.3515 3.2669 1.0704
JHH-4 CTRP2 6.2483 8.0061 3.5065 0.346
SNU-449 CTRP2 6.3969 10.1895 2.6782 2.6765
SNU-423 CTRP2 6.4668 9.5774 2.9801 1.6094
SNU-398 CTRP2 6.475 8.3493 3.4706 0.3355
JHH-2 CTRP2 6.6286 9.082 3.2576 0.7266
HLF CTRP2 9.157 18.343 0.6099 7.0189
PLC/PRF/5 CTRP2 13.3564 31.6744 -2.9608 12.8492
⏷ Show the Full List of 18 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 91 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1184 CTRP2 4.6168 6.6851 3.199 2.8254
NCI-H810 CTRP2 4.873 6.5881 3.4154 1.6184
NCI-H2126 CTRP2 5.0378 6.6732 3.4743 1.2189
DV-90 CTRP2 5.1394 6.733 3.5043 1.017
NCI-H2196 CTRP2 5.1916 7.1159 3.3643 1.4547
LUDLU-1 CTRP2 5.2223 8.0271 2.9641 2.9254
LK2 CTRP2 5.2791 6.268 3.7598 0.205
NCI-H2081 CTRP2 5.3182 11.8325 1.1867 9.9221
HCC4006 CTRP2 5.3302 10.5992 1.8002 7.4391
NCI-H1568 CTRP2 5.3597 9.3454 2.4283 4.8608
NCI-H2444 CTRP2 5.3891 6.95 3.5404 0.702
NCI-H2342 CTRP2 5.3981 9.0023 2.6177 4.0545
NCI-H1694 CTRP2 5.4279 8.179 3.0215 2.4565
NCI-H1092 CTRP2 5.4515 7.1689 3.4803 0.8372
NCI-H1105 CTRP2 5.5341 8.953 2.7287 3.4449
HCC2935 CTRP2 5.5375 7.4856 3.3905 1.0505
NCI-H1915 CTRP2 5.5803 7.6214 3.3548 1.1298
NCI-H1703 CTRP2 5.645 8.192 3.1418 1.7886
NCI-H1355 CTRP2 5.6673 8.9825 2.7977 3.0205
NCI-H1341 CTRP2 5.6904 8.0572 3.2256 1.4597
NCI-H1339 CTRP2 5.7664 7.3135 3.5677 0.4131
NCI-H226 CTRP2 5.8016 7.0453 3.6816 0.178
NCI-H522 CTRP2 5.8063 14.9546 0.0114 13.5818
LOU-NH91 CTRP2 5.8428 7.8133 3.4046 0.7887
NCI-H2286 CTRP2 5.8444 7.503 3.5283 0.4676
VMRC-LCD CTRP2 5.8681 7.7077 3.4587 0.6276
Sq-1 CTRP2 5.9186 8.2666 3.2545 1.1786
NCI-H2172 CTRP2 5.9567 7.6305 3.5274 0.4181
SW1573 CTRP2 5.9811 8.0683 3.3664 0.8074
Calu-1 CTRP2 6.0392 7.6275 3.5625 0.3129
NCI-H460 CTRP2 6.0676 7.2479 3.7084 0.0885
NCI-H2170 CTRP2 6.0755 8.4854 3.2412 1.1037
HCC1438 CTRP2 6.0772 7.2719 3.7036 0.092
DMS 273 CTRP2 6.0775 7.7663 3.5264 0.3704
EBC-1 CTRP2 6.0946 8.0763 3.4149 0.6157
SK-MES-1 CTRP2 6.1025 15.7794 -0.176 13.7668
NCI-H1793 CTRP2 6.1277 7.9661 3.4718 0.4661
NCI-H520 CTRP2 6.1508 8.3318 3.3392 0.7788
Calu-6 CTRP2 6.2066 7.8152 3.56 0.2624
HOP-62 CTRP2 6.2327 7.6926 3.6139 0.1718
NCI-H1869 CTRP2 6.2329 7.9816 3.5094 0.3459
IA-LM CTRP2 6.2349 7.5049 3.6798 0.0925
SK-LU-1 CTRP2 6.2477 7.7999 3.5814 0.2159
NCI-H647 CTRP2 6.2497 15.8484 -0.1029 13.2765
COLO 668 CTRP2 6.2553 8.1999 3.4366 0.4878
NCI-H1755 CTRP2 6.2554 8.3144 3.3927 0.5884
ChaGo-K-1 CTRP2 6.2904 9.2205 3.0411 1.5564
COR-L88 CTRP2 6.3007 14.9431 0.3753 11.4783
LC-1/sq-SF CTRP2 6.318 7.7574 3.6226 0.1425
NCI-H1563 CTRP2 6.3273 15.235 0.2521 11.8868
DMS 454 CTRP2 6.3296 8.6295 3.3022 0.7735
DMS 53 CTRP2 6.349 8.0756 3.521 0.2862
COR-L95 CTRP2 6.3713 7.7566 3.6421 0.1107
NCI-H2085 CTRP2 6.3721 8.3237 3.4385 0.4351
SW1271 CTRP2 6.3769 7.9859 3.564 0.2093
NCI-H2023 CTRP2 6.4147 8.1428 3.5222 0.2647
NCI-H1666 CTRP2 6.4231 8.0537 3.5573 0.2078
NCI-H2122 CTRP2 6.4402 7.8509 3.6343 0.1081
NCI-H1651 CTRP2 6.4466 8.1804 3.5209 0.2578
NCI-H1435 CTRP2 6.4635 8.2486 3.5028 0.6043
NCI-H1395 CTRP2 6.487 17.1048 -0.5459 14.4274
RERF-LC-MS CTRP2 6.5012 8.4456 3.4456 0.373
DMS 114 CTRP2 6.5129 7.9061 3.6411 0.0911
NCI-H838 CTRP2 6.5369 7.8563 3.6662 0.067
NCI-H446 CTRP2 6.549 8.3245 3.5084 0.2497
RERF-LC-Ad2 CTRP2 6.5578 13.3223 1.331 7.519
NCI-H1792 CTRP2 6.6175 8.1261 3.603 0.1133
KNS-62 CTRP2 6.6502 8.3142 3.5498 0.1681
PC-14 CTRP2 6.6522 8.4535 3.5015 0.2338
NCI-H322 CTRP2 6.6597 8.0311 3.6498 0.0669
NCI-H841 CTRP2 6.676 8.0347 3.6542 0.0621
NCI-H661 CTRP2 6.6963 8.4815 3.5081 0.2138
NCI-H2228 CTRP2 6.709 20.4978 -2.0486 18.6947
NCI-H2110 CTRP2 6.7575 9.368 3.2028 0.7943
NCI-H1650 CTRP2 6.772 8.5998 3.4945 0.2154
LCLC-97TM1 CTRP2 6.8772 9.0356 3.3783 0.3713
EPLC-272H CTRP2 6.8879 8.652 3.5188 0.1609
COR-L105 CTRP2 6.9326 9.2204 3.3324 0.4368
NCI-H2087 CTRP2 6.9354 8.7709 3.4947 0.1809
NCI-H1623 CTRP2 6.947 13.9765 1.2745 7.223
HCC1195 CTRP2 6.9626 15.8468 0.397 10.432
LXF 289 CTRP2 6.9811 8.5899 3.5729 0.0928
NCI-H441 CTRP2 7.0093 8.9644 3.4542 0.218
NCI-H1373 CTRP2 7.0377 8.7279 3.546 0.1094
NCI-H23 CTRP2 7.1221 14.5707 1.1076 7.6196
A-549 CTRP2 7.143 8.7717 3.5677 0.0793
NCI-H1944 CTRP2 7.1568 13.1047 1.8073 5.004
EKVX CTRP2 7.4579 9.4899 3.4344 0.1588
NCI-H2141 CTRP2 7.9847 30.2427 -5.9013 25.3207
Lu-65 CTRP2 8.368 20.3971 -0.8352 12.6719
T3M-10 CTRP2 9.3188 22.0548 -1.0005 11.9795
⏷ Show the Full List of 91 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 5.1341 6.2425 3.7071 0.3971
P-STS CTRP2 6.3612 8.2315 3.4685 0.3789
SYO-1 CTRP2 6.661 8.2547 3.5744 0.137
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 6.1748 7.4806 3.6667 0.1163
Aska-SS CTRP2 6.1926 7.9894 3.4901 0.3997
GCT CTRP2 4.6882 6.2711 3.4465 1.7297
TE 441.T CTRP2 4.7112 6.9582 3.1328 2.9539
HT-1080 CTRP2 5.3118 7.3887 3.311 1.5227
BT-16 CTRP2 5.3298 6.9378 3.516 0.8192
BT-12 CTRP2 5.3521 6.2083 3.8098 0.0991
SW982 CTRP2 5.6243 7.1488 3.5697 0.4784
Hs 729.T CTRP2 5.7485 8.8435 2.9096 2.5137
RKN CTRP2 5.8849 7.1496 3.676 0.165
MES-SA CTRP2 6.0462 7.2765 3.6909 0.1111
G-401 CTRP2 6.1818 10.9322 2.2132 4.6251
TE 617.T CTRP2 6.3509 8.0562 3.5288 0.2723
SK-LMS-1 CTRP2 6.3649 8.4033 3.4054 0.5086
A-204 CTRP2 6.6181 9.0836 3.2523 0.7447
Tm87-16 CTRP2 6.652 8.2367 3.5773 0.1352
G-402 CTRP2 6.7648 8.9988 3.3468 0.4695
TTC-709 CTRP2 6.8373 8.5397 3.5394 0.1462
Rh18 CTRP2 7.2369 8.5986 3.656 0.0255
RD CTRP2 9.6813 21.1038 -0.3342 9.5015
SK-UT-1 CTRP2 12.9169 27.5723 -1.3691 9.2504
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 6.4565 7.7495 3.6743 0.0693
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 6.6689 20.4378 -2.0488 18.7583
COV362 CTRP2 5.3533 11.9295 1.1649 9.9514
OVCAR-5 CTRP2 5.4055 7.2986 3.4017 1.1242
OAW42 CTRP2 5.4145 6.6653 3.6659 0.3514
OV7 CTRP2 5.6014 8.7319 2.8729 2.8143
JHOM-1 CTRP2 5.6333 7.5088 3.4287 0.8602
JHOS-2 CTRP2 5.7494 8.7079 2.9712 2.2892
COV434 CTRP2 5.8329 11.2896 1.8167 6.6296
TOV-21G CTRP2 5.8464 7.2704 3.6171 0.2767
OV56 CTRP2 5.8644 7.0991 3.6862 0.1551
FU-OV-1 CTRP2 5.8981 7.6468 3.4959 0.5182
Caov-3 CTRP2 5.9165 7.3083 3.631 0.2286
RMG-I CTRP2 5.9622 11.7099 1.7027 6.8968
OAW28 CTRP2 6.0103 8.8406 3.0574 1.7381
OC 314 CTRP2 6.2005 7.4097 3.7001 0.0779
TOV-112D CTRP2 6.2014 8.1402 3.4365 0.5122
SK-OV-3 CTRP2 6.2419 9.1367 3.0517 1.5614
EFO-21 CTRP2 6.2877 8.2382 3.4357 0.4758
COV644 CTRP2 6.3423 8.3474 3.4172 0.4928
OVK18 CTRP2 6.4288 7.8289 3.6378 0.1062
OV-90 CTRP2 6.5526 8.1251 3.5801 0.1497
MCAS CTRP2 6.5878 8.1363 3.5889 0.1331
EFO-27 CTRP2 6.6171 8.4224 3.4993 0.246
IGROV-1 CTRP2 6.7146 8.3726 3.5529 0.1521
TYK-nu CTRP2 6.8443 8.3913 3.5925 0.0925
HEY A8 CTRP2 6.8537 8.2194 3.653 0.048
OVCAR-4 CTRP2 6.9329 8.5884 3.5566 0.1136
A2780 CTRP2 6.9345 8.6703 3.5292 0.1412
SNU-840 CTRP2 7.0561 8.7765 3.5359 0.1163
OVCAR-8 CTRP2 7.1088 8.9332 3.5011 0.1434
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 4 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JL-1 CTRP2 5.895 8.5073 3.1401 1.5646
IST-Mes1 CTRP2 6.1032 8.3589 3.3062 0.8976
NCI-H2452 CTRP2 6.2447 8.2856 3.3991 0.5783
NCI-H2052 CTRP2 7.1117 8.9543 3.4949 0.1495
Cancer Drug Sensitivity Data Curated from 4 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU145 CTRP2 6.0448 10.0002 2.5592 3.48
PaCa-3 CTRP2 6.1356 7.353 3.6966 0.0904
LNCaP clone FGC CTRP2 6.2068 8.3148 3.3712 0.6653
VCaP CTRP2 6.2195 8.0725 3.4699 0.431
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 CTRP2 5.4274 10.6392 1.85 7.0894
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-16 CTRP2 4.3287 5.5032 3.5692 1.753
HGC-27 CTRP2 5.7197 8.6866 2.9636 2.3479
SH-10-TC CTRP2 5.7961 7.1699 3.6341 0.2623
NUGC-3 CTRP2 5.9309 7.7337 3.4765 0.5489
Hs 746.T CTRP2 6.0394 8.0116 3.4157 0.643
HuG1-N CTRP2 6.1131 8.108 3.4106 0.6166
LMSU CTRP2 6.1536 8.563 3.2471 1.0325
Fu97 CTRP2 6.1813 7.8075 3.5529 0.2827
SNU-601 CTRP2 6.1979 7.9257 3.516 0.3458
SNU-1 CTRP2 6.2316 8.4396 3.3331 0.7485
ECC10 CTRP2 6.2462 7.8412 3.566 0.2408
IM95 CTRP2 6.4467 9.5831 2.9675 1.6648
SNU-216 CTRP2 6.4949 7.9845 3.6079 0.1276
MKN7 CTRP2 6.9095 8.4695 3.5887 0.0879
MKN74 CTRP2 7.0696 8.9542 3.4798 0.1738
NCC-StC-K140 CTRP2 7.0896 9.2927 3.3676 0.3262
KE-39 CTRP2 7.7924 9.966 3.3901 0.1538
SNU-685 CTRP2 6.2641 7.7234 3.6147 0.1637
SNG-M CTRP2 6.3489 7.9962 3.5496 0.2386
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW579 CTRP2 5.4802 7.6259 3.2998 1.3994
FTC-238 CTRP2 5.7028 12.4621 1.1581 9.4229
ML-1 [Human leukemia] CTRP2 5.9002 8.4446 3.1697 1.4628
FTC-133 CTRP2 6.0335 7.4497 3.6251 0.2046
TT2609-C02 CTRP2 6.7344 9.3727 3.1907 0.8362
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
BICR 18 CTRP2 5.0484 7.0685 3.3013 1.8438
PE/CA-PJ15 CTRP2 5.4186 8.4956 2.8694 3.0459
HSC-2 CTRP2 5.4406 6.941 3.5686 0.5869
PE/CA-PJ41 (clone D2) CTRP2 5.6593 8.5224 3.0025 2.2707
PE/CA-PJ49 CTRP2 5.7209 7.3178 3.5463 0.4859
BICR 31 CTRP2 5.8306 9.6052 2.6106 3.5361
PE/CA-PJ34 (clone C12) CTRP2 5.9002 7.6952 3.478 0.5611
CAL-27 CTRP2 6.0553 7.3911 3.6542 0.1559
BICR 6 CTRP2 6.0701 7.4016 3.6561 0.1502
SCC-9 CTRP2 6.0889 7.7932 3.521 0.3769
FaDu CTRP2 6.1594 7.8148 3.5415 0.3107
SCC-4 CTRP2 6.1935 13.7411 0.8832 9.7409
BICR 16 CTRP2 6.2996 7.8416 3.5862 0.1956
SCC-25 CTRP2 6.3599 8.5523 3.3459 0.6484
BICR 56 CTRP2 6.3841 7.8334 3.6202 0.133
CAL-33 CTRP2 6.4001 8.2262 3.486 0.3321
BICR 22 CTRP2 6.4523 8.0062 3.5849 0.1633
YD-8 CTRP2 6.7149 8.5451 3.4925 0.2316
HSC-4 CTRP2 6.7391 8.1476 3.638 0.0676
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HT-1376 CTRP2 4.5819 6.5881 1.4088 0.4347
HT-1197 CTRP2 5.6734 7.8409 3.3095 1.1988
KMBC-2 CTRP2 5.7022 7.67 3.3958 0.9094
BC-3C CTRP2 5.8699 13.7185 0.6645 11.0659
UM-UC-1 CTRP2 6.1077 8.5029 3.2496 1.0563
647V CTRP2 6.117 8.0037 3.4528 0.5138
SCaBER CTRP2 6.1864 7.6581 3.6088 0.1901
UM-UC-3 CTRP2 6.317 7.8297 3.5969 0.1763
RT-4 CTRP2 6.6318 8.7342 3.3913 0.4309
RT-112 CTRP2 6.7892 8.0697 3.6807 0.0374
T24 CTRP2 6.8029 8.4364 3.5626 0.1267
J82 CTRP2 10.2891 21.7689 -0.2759 8.6676
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 6.0184 7.2195 3.7006 0.1049

References

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