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Drug Information

Drug General Information
Drug ID
D0L5FB
Former ID
DNCL002924
Drug Name
TAK-329
Indication Diabetes [ICD9: 253.5, 588.1; ICD10:E23.2, N25.1] Phase 1 [523386]
Company
Takeda Pharmaceuticals U.S.A.
Target and Pathway
Target(s) Glucokinase Target Info Inhibitor [551984]
KEGG Pathway Glycolysis / Gluconeogenesis
Galactose metabolism
Starch and sucrose metabolism
Amino sugar and nucleotide sugar metabolism
Butirosin and neomycin biosynthesis
Metabolic pathways
Biosynthesis of antibiotics
Carbon metabolism
Insulin signaling pathway
Insulin secretion
Prolactin signaling pathway
Glucagon signaling pathway
Type II diabetes mellitus
Maturity onset diabetes of the young
Central carbon metabolism in cancer
Pathway Interaction Database FOXA2 and FOXA3 transcription factor networks
HIF-1-alpha transcription factor network
PathWhiz Pathway Nucleotide Sugars Metabolism
Starch and Sucrose Metabolism
Galactose Metabolism
Trehalose Degradation
Reactome Regulation of gene expression in beta cells
Glucose transport
Glycolysis
WikiPathways SIDS Susceptibility Pathways
Glycolysis and Gluconeogenesis
MAPK Signaling Pathway
Regulation of beta-cell development
Metabolism of carbohydrates
Hexose transport
References
Ref 523386ClinicalTrials.gov (NCT01311076) TAK-329 Glucose Clamp Study. U.S. National Institutes of Health.
Ref 551984Clinical pipeline report, company report or official report of Takeda.
Cite DrugMAP

Fengcheng Li, Minjie Mou, ..., Jiayi Yin*, Yang Zhang*, Feng Zhu*. DrugMAP 2.0: molecular atlas and pharma-information of all drugs. Nucleic Acids Research.
DOI: 10.1093/nar/gkae791 (2024). PMID: 39271119
Learn more about DrugMAP >
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Correspondence

Prof. Feng Zhu 
College of Pharmaceutical Sciences, Zhejiang University

Dr. Yang Zhang 
School of Pharmacy, Hebei Medical University

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