Target General Information
Target ID T25005
Target Name Tyrosine-protein kinase BTK
Synonyms ATK; Agammaglobulinaemia tyrosine kinase; B cell progenitor kinase; BPK; Bruton's tyrosine kinase; BTK
Target Type Successful
Gene Name BTK
Biochemical Class Kinase
UniProt ID BTK_HUMAN
Target Gene Expression Profiles in Other Tissues of Healthy Individuals
Reference
Ref 531450Antiarthritis effect of a novel Bruton's tyrosine kinase (BTK) inhibitor in rat collagen-induced arthritis and mechanism-based pharmacokinetic/pharmacodynamic modeling: relationships between inhibition of BTK phosphorylation and efficacy. J Pharmacol Exp Ther. 2011 Jul;338(1):154-63.
Ref 1572592NCBI GEO: archive for functional genomics data sets--update.