General Information of Drug (ID: DMF3AN7)

Drug Name
Loratadine Drug Info
Synonyms
Aerotina; Alarin; Alavert; Alerpriv; Allertidin; Anhissen; Biloina; Bonalerg; Civeran; Claratyne; Clarinase; Claritin; Claritine; Clarityn; Clarityne; Clarium; Fristamin; Histaloran; Lergy; Lertamine; Lesidas; Lisino; Loracert; Loradex; Loradif; Loranox; Lorantis; Lorastine; Loratadina; Loratadinum; Loratidine; Loratyne; Loraver; Lorfast; Loritine; Lowadina; Nularef; Optimin; Polaratyne; Pylor; Restamine; Rhinase; Rinomex; Roletra; Sanelor; Sensibit; Sohotin; Tadine; Velodan; Versal; Zeos; Bedix Loratadina; Claratyne Cold; Claratyne Decongestant; Clarinase Reperabs; Claritin D; Claritin Hives Relief; Claritin Hives Relief Reditab; Claritin Reditabs; Claritin reditab; Clarityne Dy Repetabs; Loratadina [Spanish]; Loratadine Redidose; Loratadine Wyeth Brand; Loratadinum [Latin]; Sinhistan Dy; Talorat Dy; Wyeth Brand of Loratadine; L 9664; Sch 29851; Sch29851; Alavert (TN); AllergyX (TN); Children's Claritin; Claritin (TN); Claritine (TN); Clarityn (TN); Clarityne (TN); Clarityne-D; Flonidan (TN); Fristamin (TN); Lomilan (TN); Lorfast (TN); Rinolan (TN); Roletra (TN); Sch-29851; Symphoral (TN); Tidilor (TN); Alavert, Claritin, Loratadine; Loratadine [USAN:BAN:INN]; Loratadine (JAN/USAN/INN); Ethyl 4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)piperidine-1-carboxylate; Ethyl 4-(8-chloro-5,6-dihydro-11H-benzo(5,6)cyclohepta(1,2-b)pyridin-11-ylidene)-1-piperidinecarboxylate; 1-Piperidenecarboxylic acid, 4-(8-chloro-5,6-duhydro-11H-benzo [5,6]cyclohepta[1,2-b]-pyridin-11-ylidene)-, ethyl ester; 1-Piperidinecarboxylic acid, 4-(8-chloro-5,6-dihydro-11H-benzo(5,6)cyclohepta(1,2-b)pyridin-11-ylidene)-, ethyl ester; 1-Piperidinecarboxylic acid, 4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-, ethyl ester; 1-piperidinecarboxylic acid,4-(8-chloro-5,6-dihydro-11H-benzo(5,6)cyclohepta(1,2-b)pyridin-11-ylidene)-,ethyl ester; 4-(8-Chloro-5,6-dihydro-11H-benzo(5,6)cyclohepta(1,2-b)pyridin-11-ylidene)-1-piperidinecarboxylic Acid Ethyl Ester; 4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene-1-piperidinecarboxylic acidethyl ester; 4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cycloheptal[1,2-b]pyridin-11-ylidene-1-piperidinecarboxylic acid ethyl ester
Indication
Disease Entry ICD 11 Status REF
Allergy 4A80-4A85 Approved [1] , [2]
Allergic rhinitis CA08.0 Discontinued in Phase 2 [3]
Therapeutic Class
Antihistamines
Cross-matching ID
PubChem CID
3957
ChEBI ID
CHEBI:6538
CAS Number
79794-75-5
TTD ID
D06ABF
VARIDT ID
DR00541
INTEDE ID
DR0977
ACDINA ID
D00374

Full List of Drug Formulations Containing This Drug

Loratadine 10 mg tablet
Company Formulation ID FDA Description
Pfizer Consumer Healthcare F12496 Anhydrous citric acid; Maltodextrin; Ascorbic acid; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Sodium bicarbonate; Crospovidone; Silicon dioxide; Cellulose, microcrystalline
Pfizer Consumer Healthcare F12497 Anhydrous citric acid; Maltodextrin; Aspartame; Magnesium stearate; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Sodium bicarbonate; Crospovidone; Silicon dioxide; Cellulose, microcrystalline; Corn syrup; Icodextrin
Pfizer Consumer Healthcare F12500 Anhydrous citric acid; Maltodextrin; Aspartame; Magnesium stearate; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Sodium bicarbonate; Crospovidone; Silicon dioxide; Cellulose, microcrystalline; Corn syrup; Icodextrin
Cardinal Health F12502 Anhydrous citric acid; Sodium stearate; Lactose monohydrate; Sodium lauryl sulfate; Aspartame; Mannitol; Crospovidone; Povidone; Cellulose, microcrystalline; Colloidal silicon dioxide
Pfizer Consumer Healthcare F12501 Anhydrous citric acid; Aspartame; Magnesium stearate; Mannitol; Sodium bicarbonate; Crospovidone; Silicon dioxide; Cellulose, microcrystalline; Corn syrup
Mylan Pharamceuticals F12498 Anhydrous lactose; Sodium lauryl sulfate; Magnesium stearate; Hypromellose; Povidone; Silicon dioxide; Cellulose, microcrystalline; Starch, corn
American Sales Company; CVS Pharmacy; Chain Drug Consortium; Chain Drug Marketing Association; Fred's; Good Neighbor Pharmacy; Health Mart; Major Pharmaceuticals; Meijer; Safeway; Select Brand; Shopko; Sunmark; SuperValu; Target Corporation; TopCare; Topco Associates; Valu Merchandisers Company; Walgreens Company F12503 Sodium stearyl fumarate; Aspartame; Magnesium stearate; Mannitol; Croscarmellose sodium
Cardinal Health F12504 Sodium stearyl fumarate; Aspartame; Magnesium stearate; Mannitol; Croscarmellose sodium
Ohm Laboratories F12505 Sodium stearyl fumarate; Aspartame; Magnesium stearate; Mannitol; Croscarmellose sodium
Mylan Pharamceuticals F12509 Anhydrous lactose; Sodium lauryl sulfate; Magnesium stearate; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Starch, corn
Cardinal Health F12510 Anhydrous lactose; Sodium lauryl sulfate; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Povidones; Starch, corn
Bayer HealthCare F12499 Anhydrous citric acid; Mannitol; Gelatin
Marc Glassman, Inc.; Selder, S.A. de C.V. F12512 Lactose monohydrate; Magnesium stearate; Croscarmellose sodium; Silicon dioxide; Microcrystalline cellulose
Allegiant Health; Apotex; AvPAK; Blenheim Phamacal; Cardinal Health; DLC Laboratories; Gericare Pharmaceuticals; Major Pharmaceuticals; NuCare Pharmaceuticals; Rugby Laboratories F12525 Lactose monohydrate; Magnesium stearate; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline
A-S Medication Solutions F12526 Lactose monohydrate; Magnesium stearate; Croscarmellose sodium; Silicon dioxide; Microcrystalline cellulose
DirectRX; H. J. Harkins Company; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Melaleuca; RemedyRepack F12515 Lactose monohydrate; Magnesium stearate; Povidone; Starch, corn
International Laboratories F12516 Lactose monohydrate; Magnesium stearate; Povidone; Starch, pregelatinized corn
McKesson; Walgreens Company F12517 Lactose monohydrate; Magnesium stearate; Povidone
RemedyRepack F12523 Lactose monohydrate; Magnesium stearate; Povidone; Starch, corn
Novartis Consumer Health; Target Brands F12511 Lactose monohydrate; Magnesium stearate; Cellulose, microcrystalline; Sodium starch glycolate type a potato
Novartis Consumer Health F12513 Lactose monohydrate; Magnesium stearate; Cellulose, microcrystalline; Sodium starch glycolate type a corn
Cardinal Health; Contract Pharmacal; Health Mart; Innovative Manufacturing and Distribution Services; Lake Eire Medical & Surgical Supply DBA Quality Care Products; McKesson; NCS HealthCare of KY, Inc dba Vangard Labs; NorthStar Rx; NuCare Pharmaceuticals; Physicians Total Care; RemedyRepack; Sandoz; St Marys Medical Park Pharmacy; State of Florida DOH Central Pharmacy; Sunmark; Wal-Mart Stores F12514 Lactose monohydrate; Magnesium stearate; Cellulose, microcrystalline; Sodium starch glycolate type a potato
A-S Medication Solutions; Proficient Rx; Unit Dose Services F12518 Lactose monohydrate; Magnesium stearate; Povidone, unspecified
Bryant Ranch Prepack; Cardinal Health; Unit Dose Services F12519 Lactose monohydrate; Magnesium stearate; Povidones; Starch, corn
7-Eleven; American Sales Company; Amerisource Bergen; Aphena Pharma Solutions-Tennessee; Army & Air Force Exchange Service; BJWC; Big Lots Stores; CVS Pharmacy; Cardinal Health; Costco Wholesale; DZA Brands; Dolgencorp; Family Dollar; First Aid Direct; Greenbrier International; Harmon Stores; Harris Teeter; Humana Pharmacy; Hy-Vee; Kinray; Kmart Corporation; Kroger Company; L. Perrigo Company; Major Pharmaceuticals; McKesson; Meijer; NuCare Pharmaceuticals; Perrigo New York; Preferred Pharamaceuticals; Procter & Gamble Manufacturing Company; RemedyRepack; Rite Aid; Safeway; Sam's West; Save-A-Lot Food Stores; Shopko; SuperValu; Target Corporation; Topco Associates; Wakefern Food Corporation; Wal-Mart Stores; Walgreens Company F12520 Lactose monohydrate; Magnesium stearate; Povidones
Medicine Shoppe International F12521 Lactose monohydrate; Magnesium stearate; Starch, corn; Starch, pregelatinized corn
Moore Medical; Unifirst First Aid F12522 Lactose monohydrate; Magnesium stearate; Starch, corn
Select Corporation F12524 Lactose; Magnesium stearate; Starch, corn
Help Remedies; Rebel Distributors F12527 Lactose monohydrate; Magnesium stearate; Starch, corn; Starch, corn
Amerisource Bergen; Cardinal Health; Chain Drug Marketing Association; Family Dollar; Fred's; Major Pharmaceuticals; Medline Industries; Publix Super Markets; Select Brand; Shopko; Valu Merchandisers Company F12528 Lactose monohydrate; Magnesium stearate; Starch, corn; Starch, pregelatinized corn
SuperValu F12529 Lactose monohydrate; Magnesium stearate; Starch, corn; Starch, pregelatinized corn
American Health Packaging; Bayer HealthCare; CVS Pharmacy; Cardinal Health; Clinical Solutions Wholesale; Contract Pharmacal; DLC Laboratories; Kaiser Foundation Hospitals; Kinray; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Major Pharmaceuticals; Mylan Pharamceuticals; Navajo Manufacturing; NuCare Pharmaceuticals; Ohm Laboratories; Premier Value; Proficient Rx; Safeway; TYA Pharmaceuticals; Walgreens Company; WinCo Foods F12530 Lactose monohydrate; Magnesium stearate; Starch, corn
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⏷ Show the Full List of 32 Formulation(s)
Loratadine 5 mg tablet
Company Formulation ID FDA Description
Bayer HealthCare F12531 Anhydrous citric acid; Stearic acid; Aspartame; D&c red no. 27; Fd&c blue no. 2; Magnesium stearate; Mannitol; Silicon dioxide; Aluminum oxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
MSD Consumer Care F12533 Anhydrous citric acid; Stearic acid; Aspartame; D&c red no. 27; Fd&c blue no. 2; Magnesium stearate; Mannitol; Silicon dioxide; Aluminum oxide; Cellulose, microcrystalline
Bayer HealthCare F12532 Stearic acid; Aspartame; Magnesium stearate; Mannitol; Silicon dioxide; Cellulose, microcrystalline
Bayer HealthCare F12534 Anhydrous citric acid; Mannitol; Gelatin
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Loratadine 10 mg capsule
Company Formulation ID FDA Description
Marksans Pharma F12506 Capric acid; Fd&c blue no. 1; Sorbitol; Water; Polysorbate 80; Povidone k30; Gelatin; Sorbitan
CVS Pharmacy; Cardinal Health; KMART; Kroger Company; Time Cap Labs; Walgreens Company F12508 Fd&c blue no. 1; Sorbitol; Water; Polysorbate 80; Povidone; Caprylic/capric mono/diglycerides; Gelatin
Bayer HealthCare F12507 Fd&c blue no. 1; Sorbitol; Glycerin; Water; Polysorbate 80; Gelatin; Povidones
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References

1 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 7216).
2 Desloratadine treatment for intermittent and persistent allergic rhinitis: a review. Clin Ther. 2007 Sep;29(9):1795-802.
3 Trusted, scientifically sound profiles of drug programs, clinical trials, safety reports, and company deals, written by scientists. Springer. 2015. Adis Insight (drug id 800015252)