Details of the Drug-Related molecule(s) Activity Atlas

General Information of Drug (ID: DMCGX9U)

• Drug Name: PHA-665752 Drug Info
• Synonyms: PHA-665752; 477575-56-7; PHA 665752; PHA665752; TCMDC-125885; UNII-0VXU5T5R3J; (2R)-1-[[5-[(Z)-[5-[[(2,6-DICHLOROPHENYL)METHYL]SULFONYL]-1,2-DIHYDRO-2-OXO-3H-INDOL-3-YLIDENE]METHYL]-2,4-DIMETHYL-1H-PYRROL-3-YL]CARBONYL]-2-(1-PYRROLIDINYLMETHYL)PYRROLIDINE; 0VXU5T5R3J; CHEMBL450786; CHEBI:90197; (R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimethyl-4-(2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl)-1H-pyrrol-2-yl)methylene)indolin-2-one; PHA-665752 hydrate
• Cross-matching ID:
  PubChem CID: 10461815
  ChEBI ID: CHEMBL90197
  CAS Number: CAS 477575-56-7
  TTD ID: D00TBD

Molecule-level Activity Landscape of This Drug

IC50 (12) EC50 (5) Kd (216) Ki (1) Download

Molecule Name	Gene Name	UniProt ID	Type	IC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	EC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Kd (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Ki (nM)	Details
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Experimental Drug Sensitivity Data Across Cancer Cell Lines

Cell Line	Related Disease	IC50 (Log₂ µM)	Original Dataset	Details
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Cytotoxic Activity Landscape of This Drug

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Cell Line	Disease	Value (nM)	ChEMBL Assay ID	Details
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