Details of the Drug-Related molecule(s) Activity Atlas

General Information of Drug (ID: DMM7ZXR)

• Drug Name: GSK2126458 Drug Info
• Synonyms: 1086062-66-9; Omipalisib; GSK-2126458; GSK 2126458; UNII-1X8F5A3NA0; 2,4-difluoro-N-(2-methoxy-5-(4-(pyridazin-4-yl)quinolin-6-yl)pyridin-3-yl)benzenesulfonamide; 2,4-difluoro-N-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide; 2,4-Difluoro-N-[2-methoxy-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl]benzenesulfonamide; 1X8F5A3NA0; Omipalisib (GSK2126458, GSK458); C25H17F2N5O3S; Omipalisib [USAN:INN]
• Cross-matching ID:
  PubChem CID: 25167777
  ChEBI ID: CHEMBL1236962
  CAS Number: CAS 1086062-66-9
  TTD ID: D03EZE

Molecule-level Activity Landscape of This Drug

IC50 (9) EC50 (3) Kd (1) Ki (9) Download

Molecule Name	Gene Name	UniProt ID	Type	IC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	EC50 (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Kd (nM)	Details
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Molecule Name	Gene Name	UniProt ID	Type	Ki (nM)	Details
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Experimental Drug Sensitivity Data Across Cancer Cell Lines

Cell Line	Related Disease	IC50 (Log₂ µM)	Original Dataset	Details
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Cytotoxic Activity Landscape of This Drug

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Cell Line	Disease	Value (nM)	ChEMBL Assay ID	Details
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