General Information of Drug (ID: DMPE7DQ)

Drug Name
STF-62247 Drug Info
Synonyms Renal cell carcinoma therapy, Stanford University
Cross-matching ID
PubChem CID
704473
ChEBI ID
CHEMBL125656
CAS Number
CAS 315702-99-9
TTD Drug ID
D01CIN

Consensus Signature of Drug Pharmacogenomic Perturbation (DPP)

Term Name NES FDR q-val Tag % Leading Edge Genes
Steroid hormone biosynthesis 2.18 8.44e-3 43/61 (70.49%) AKR1C2;UGT2B4;AKR1C1;...
Steroid biosynthesis 2.17 4.22e-3 19/20 (95%) EBP;MSMO1;FDFT1;...
Allograft rejection 2.17 2.81e-3 32/38 (84.21%) HLA-DQA1;HLA-F;HLA-G;...
Fat digestion and absorption 2.05 4.22e-3 35/43 (81.4%) CD36;ACAT2;PLPP3;...
Lysosome 2.02 3.38e-3 115/128 (89.84%) NEU1;LAMP1;MCOLN1;...
Graft-versus-host disease 2.01 2.81e-3 32/42 (76.19%) HLA-DQA1;HLA-F;HLA-G;...
Metabolism of xenobiotics by cytochrome P450 2.00 2.41e-3 49/77 (63.64%) ADH1B;UGT2B4;AKR1C1;...
Cholesterol metabolism 1.90 6.33e-3 44/50 (88%) CD36;NPC2;SOAT1;...
Retinol metabolism 1.89 5.63e-3 41/68 (60.29%) ADH1B;RDH11;UGT2B4;...
Type I diabetes mellitus 1.89 5.07e-3 38/43 (88.37%) HLA-DQA1;PTPRN2;HLA-F;...
PPAR signaling pathway 1.77 1.38e-2 66/74 (89.19%) SCD;CD36;FABP4;...
Complement and coagulation cascades 1.70 2.74e-2 76/85 (89.41%) CFB;C1R;C1S;...
Fatty acid degradation 1.68 3.44e-2 40/43 (93.02%) ADH1B;ACAT2;ACADSB;...
Primary bile acid biosynthesis 1.68 3.20e-2 15/17 (88.24%) CYP39A1;AMACR;AKR1C4;...
Tyrosine metabolism 1.67 3.49e-2 30/36 (83.33%) ADH1B;MAOB;TYRP1;...
Relaxin signaling pathway -1.67 5.00e-2 114/129 (88.37%) PIK3CA;MAPK11;INSL5;...
Leukocyte transendothelial migration -1.73 3.85e-2 90/114 (78.95%) ARHGAP35;ICAM1;CTNNA2;...
Proteoglycans in cancer -1.74 4.40e-2 172/205 (83.9%) CCND1;MAP2K1;PRKACA;...
Yersinia infection -1.76 3.61e-2 120/137 (87.59%) MAP2K1;MAPK1;ITGA5;...
Colorectal cancer -1.77 4.10e-2 84/86 (97.67%) MAPK9;SOS2;GADD45B;...
Adherens junction -1.78 4.84e-2 63/71 (88.73%) FER;CTNNA3;NLK;...
Focal adhesion -1.93 0.00e+0 180/201 (89.55%) RAF1;PAK4;PARVA;...
Tight junction -1.94 0.00e+0 130/169 (76.92%) CCND1;PRKACA;MYL6;...
Bacterial invasion of epithelial cells -2.08 0.00e+0 59/77 (76.62%) CTNNA2;ITGA5;ACTR3;...
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Pharmacogenomic Perturbation Across Diseases and Tissues

Fibroblast
Nasopharyngeal carcinoma
Cell Line Name Cellosaurus Accession Species of Origin Drug Dosage Time Point Details
FIBRNPC CVCL_UK07 Homo sapiens 10uM 6H, 24H