Details of the Drug

General Information of Drug (ID: DM63OD7)

Drug Name
Pifithrin-alpha
Synonyms P53 inhibitor, Univ of Illinois; PFT-alpha; PFT-beta; Pifithrin compounds, Quark; Pifithrin-beta
Indication
Disease Entry ICD 11 Status REF
Toxicity N.A. Terminated [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski):
0		 Molecular Weight 367.3
Logarithm of the Partition Coefficient Not Available
Rotatable Bond Count 3
Hydrogen Bond Donor Count 2
Hydrogen Bond Acceptor Count 3
Chemical Identifiers
Formula
C16H19BrN2OS
IUPAC Name
2-(2-imino-4,5,6,7-tetrahydro-1,3-benzothiazol-3-yl)-1-(4-methylphenyl)ethanone;hydrobromide
Canonical SMILES
CC1=CC=C(C=C1)C(=O)CN2C3=C(CCCC3)SC2=N.Br
InChI
InChI=1S/C16H18N2OS.BrH/c1-11-6-8-12(9-7-11)14(19)10-18-13-4-2-3-5-15(13)20-16(18)17;/h6-9,17H,2-5,10H2,1H3;1H
InChIKey
HAGVCKULCLQGRF-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
9929138
CAS Number
63208-82-2
TTD ID
D02NYK

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Cellular tumor antigen p53 (TP53) TT7SBF5 P53_HUMAN Inhibitor [2]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Apoptosis regulator BAX (BAX) OTAW0V4V BAX_HUMAN Gene/Protein Processing [3]
Apoptotic protease-activating factor 1 (APAF1) OTJWIVY0 APAF_HUMAN Gene/Protein Processing [4]
Aryl hydrocarbon receptor (AHR) OTFE4EYE AHR_HUMAN Protein Interaction/Cellular Processes [5]
Cadherin-1 (CDH1) OTFJMXPM CADH1_HUMAN Gene/Protein Processing [6]
Caspase-3 (CASP3) OTIJRBE7 CASP3_HUMAN Protein Interaction/Cellular Processes [4]
Cyclin-dependent kinase 1 (CDK1) OTW1SC2N CDK1_HUMAN Gene/Protein Processing [7]
Cyclin-dependent kinase inhibitor 1 (CDKN1A) OTQWHCZE CDN1A_HUMAN Gene/Protein Processing [3]
Cytochrome P450 1A1 (CYP1A1) OTE4EFH8 CP1A1_HUMAN Gene/Protein Processing [5]
Cytochrome P450 1A2 (CYP1A2) OTLLBX48 CP1A2_HUMAN Gene/Protein Processing [8]
Cytochrome P450 1B1 (CYP1B1) OTYXFLSD CP1B1_HUMAN Gene/Protein Processing [8]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Toxicity
ICD Disease Classification N.A.
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Cellular tumor antigen p53 (TP53) DTT TP53 7.01E-01 0.06 0.09
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 149 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 6.4275 10.7526 5.0897 14.6588
MEC1 CTRP2 9.2603 12.8721 6.3908 3.8685
JM1 CTRP2 8.8496 13.6772 5.7183 7.1826
SU-DHL-1 CTRP2 2.7584 7.4237 2.4031 35.0533
EoL-1 CTRP2 3.1618 6.5455 3.0213 31.7257
SK-MM-2 CTRP2 3.7264 13.7041 1.0386 35.1178
KMS-21-BM CTRP2 3.8013 14.0847 0.9402 35.0955
L-540 CTRP2 4.8901 7.2935 4.7523 20.1985
SUP-M2 CTRP2 5.2988 11.1923 3.7614 22.6798
HH [Human lymphoma] CTRP2 5.2991 7.8857 5.0554 17.8497
Peer CTRP2 5.4799 11.0153 4.0244 21.225
HT CTRP2 5.494 7.9992 5.2357 16.6046
Ku812 CTRP2 5.6735 11.8415 3.8386 21.4082
Daudi CTRP2 5.6774 7.5208 5.5595 14.8774
697 CTRP2 5.7629 8.2993 5.4344 15.0732
ALL-SIL CTRP2 5.9045 9.1336 5.2758 15.2736
A3/Kawakami CTRP2 5.9607 7.7296 5.819 13.0727
GA-10 CTRP2 6.1069 9.4648 5.3498 14.438
NU-DUL-1 CTRP2; CTRP1 6.1281 7.811 5.9836 12.0684
MOLT-16 CTRP2 6.1565 8.823 5.6666 13.0708
Karpas-620 CTRP2 6.2953 9.4264 5.5612 13.1071
MOLT-3 CTRP2 6.3575 10.4279 5.1726 14.4984
Mono-Mac-6 CTRP2 6.3824 17.4062 1.797 26.258
KE-97 CTRP2 6.3838 11.9588 4.4723 17.2264
Pfeiffer CTRP2 6.4506 12.0167 4.5078 16.9274
NCO2 CTRP2 6.458 13.1832 3.9474 19.071
OPM-2 CTRP2 6.4952 10.6389 5.2094 14.0111
KMS-11 CTRP2; CTRP1 6.5007 15.4766 2.8686 22.8433
PL21 CTRP2; CTRP1 6.5696 10.3507 5.4263 13.0492
OCI-AML-3 CTRP2; CTRP1 6.57 9.2342 5.9347 11.0099
MOLM-6 CTRP2 6.5933 11.9927 4.6541 16.0118
SU-DHL-5 CTRP1 6.6228 7.5946 6.5722 18.0853
CA46 CTRP2 6.6319 10.1708 5.5634 12.2438
DB CTRP2 6.6353 10.2136 5.5466 12.3038
Namalwa CTRP2 6.6857 9.8668 5.7582 11.3223
KMS-34 CTRP2 6.7427 10.8351 5.3552 12.826
LAMA-84 CTRP2 6.8239 16.2017 2.1902 20.2284
RCH-ACV CTRP2 6.8894 12.0151 4.9187 14.2687
KM-H2 CTRP2 6.9132 13.7521 3.4895 15.0973
HuT 78 CTRP2 6.933 11.2772 5.3203 12.5291
THP-1 CTRP2; CTRP1 6.9654 10.4369 5.7683 10.7091
WSU-DLCL2 CTRP2; CTRP1 6.9735 9.1791 6.3698 8.2384
RS4;11 CTRP2 7.0024 12.0558 5.0022 13.6767
JVM-3 CTRP2 7.0843 10.4451 5.8673 9.9276
U-937 CTRP2; CTRP1 7.1219 11.602 5.3448 12.1016
MV4-11 CTRP2 7.1665 9.8284 6.2437 8.1834
SET-2 CTRP2 7.225 12.6152 4.9257 13.5027
KMS-27 CTRP2 7.2725 9.0392 6.723 5.9651
NOMO-1 CTRP2; CTRP1 7.2747 9.9245 6.3086 7.7689
NALM-6 CTRP2 7.2857 13.222 4.6776 14.3768
KMS-12-BM CTRP2 7.3379 13.6457 4.5122 14.9259
Toledo CTRP2 7.3465 10.9558 5.8571 9.3886
RPMI-8226 CTRP2; CTRP1 7.3652 10.4773 6.1208 8.3476
HD-MY-Z CTRP2 7.3774 10.8282 5.9481 8.942
EB1 CTRP2 7.4121 11.9094 5.442 10.98
LP-1 CTRP2; CTRP1 7.4206 11.3404 5.743 9.8047
OCI-Ly3 CTRP2 7.4304 13.5471 4.6418 14.216
TF-1 CTRP2 7.4862 10.6614 6.1279 7.9582
KE-37 CTRP2 7.5537 12.3842 5.3286 11.1577
MOLM-16 CTRP2; CTRP1 7.6168 9.1204 7.0188 4.0553
NCI-H929 CTRP2 7.6853 11.471 5.2366 6.04
HDLM-2 CTRP2 7.6925 10.1753 5.872 3.2564
OCI-AML-2 CTRP2 7.7032 9.3574 6.968 3.9797
SU-DHL-4 CTRP2; CTRP1 7.7361 9.1273 7.1221 3.3689
GDM-1 CTRP2; CTRP1 7.7561 9.8772 6.7653 4.826
EM-2 CTRP2 7.8113 19.9332 1.7731 23.2636
MOLP-2 CTRP2 7.8522 11.3603 6.0936 7.3629
P12-Ichikawa CTRP2 7.8755 15.5942 3.9961 15.827
KMS-20 CTRP2 7.8789 11.6581 5.9669 7.8441
BV-173 CTRP2 7.9222 9.7245 6.9691 3.5445
SKM-1 CTRP2; CTRP1 7.9941 10.2578 6.7729 4.3368
SU-DHL-6 CTRP2 7.997 14.1335 4.8268 12.3391
Jurkat CTRP2 8.0568 15.097 3.7262 11.8866
KHM-1B CTRP2 8.1352 14.1684 4.9221 11.691
SUP-T1 CTRP2 8.1768 12.9984 5.5397 9.0739
AMO1 CTRP2; CTRP1 8.1944 10.0917 7.0112 2.9899
TALL-1 [Human adult T-ALL] CTRP2 8.2337 12.7449 5.7113 8.2559
SEM CTRP2 8.3134 13.0732 5.6107 8.5324
MC116 CTRP2 8.3244 12.5774 5.8659 7.4502
Mino CTRP2 8.3659 13.8287 5.2757 9.8231
Ri-1 CTRP2 8.3728 10.8931 6.7357 3.7468
DEL CTRP2 8.3736 16.6359 3.8822 15.293
Reh CTRP2 8.3799 11.1245 6.6272 4.1847
HPB-ALL CTRP2 8.3997 11.324 6.5437 4.4987
L-428 CTRP2 8.4148 11.4691 6.4835 4.7239
SR CTRP2 8.419 11.1899 6.6238 4.136
NU-DHL-1 CTRP2 8.4195 12.257 6.0979 6.3193
KMS-26 CTRP2 8.444 11.755 6.3643 5.1706
EJM CTRP2; CTRP1 8.4945 18.4905 3.0658 18.0281
KCL-22 CTRP2 8.5032 19.0922 2.7604 18.9455
MOLM-13 CTRP2 8.5114 15.7069 4.4551 12.857
JURL-MK1 CTRP2 8.5265 17.7015 3.4729 16.4903
F-36P CTRP2 8.5402 12.1738 6.2295 5.5728
MM1.S CTRP2 8.5464 12.4681 6.0892 6.1441
L-363 CTRP2 8.5635 10.1609 7.2174 1.536
KO52 CTRP2 8.6199 13.9984 5.3882 8.9172
CML-T1 CTRP2 8.6285 14.5113 5.1405 9.9139
SUP-B15 CTRP2 8.6842 14.8297 5.0254 10.284
MOLT-13 CTRP2 8.7366 10.7474 7.0529 1.9569
SUP-T11 CTRP2 8.7417 11.1492 6.8675 2.6735
PF-382 CTRP2 8.756 11.5528 6.6848 3.3821
OCI-AML-5 CTRP2 8.7648 11.5732 6.6809 3.3853
JJN-3 CTRP2 8.7658 10.5535 7.1599 1.5184
Karpas-299 CTRP2 8.7927 14.8602 5.0929 9.826
HEL 92.1.7 CTRP2 8.9256 13.7019 5.7614 6.8861
KMS-18 CTRP2 8.9914 14.3003 5.5161 7.7824
OCI-M1 CTRP2 9.0082 11.7217 6.7694 2.7146
RPMI-6666 CTRP2 9.0169 11.79 6.743 2.8058
REC-1 CTRP2 9.0758 15.0968 5.1871 8.979
MHH-CALL-4 CTRP2 9.0781 11.2835 7.0126 1.7207
Ci-1 CTRP2 9.1124 15.0185 5.2522 8.6586
AML-193 CTRP2 9.1467 15.886 4.8514 10.2029
U266B1 CTRP2 9.2047 12.6578 6.4559 3.6857
SIG-M5 CTRP2 9.2107 10.1604 7.5368 0.12
KYO-1 CTRP2 9.2186 19.4555 3.1414 16.3918
BCP-1 CTRP2 9.238 13.1486 6.2453 4.4721
HL-60 CTRP2 9.2426 10.5626 7.4004 0.3739
HEL CTRP2 9.2644 20.2681 2.0746 15.9784
Hs 611.T CTRP2 9.2804 13.8531 5.937 5.6435
JeKo-1 CTRP2 9.296 12.7058 6.4916 3.4305
BL-70 CTRP2; CTRP1 9.2991 13.7084 6.0191 5.289
Raji CTRP2 9.3338 10.8955 7.3103 0.5512
NB4 CTRP2 9.3451 16.0645 4.9089 9.6575
M-07e CTRP2 9.3852 16.0403 4.9496 9.4336
Karpas-422 CTRP2 9.386 10.7596 7.3861 0.3407
Mono-Mac-1 CTRP2 9.4105 19.7351 3.1492 16.0348
MHH-CALL-3 CTRP2 9.5058 12.5405 6.6948 2.4224
CMK CTRP2 9.5283 13.0421 6.4797 3.196
RPMI-8402 CTRP2 9.5289 11.0984 7.3173 0.4315
RL CTRP2 9.5316 12.1898 6.8654 1.7897
MOTN-1 CTRP2 9.5559 12.0154 6.9543 1.467
SUP-HD1 CTRP2 9.65 12.6347 6.735 2.1303
DND-41 CTRP2 9.6561 14.6655 5.8007 5.6646
SU-DHL-8 CTRP2 9.6562 11.0102 7.4023 0.2122
ME1 CTRP2 9.67 11.8769 7.0708 1.0098
ST486 CTRP2 9.6799 11.8837 7.0728 0.997
Granta-519 CTRP2 9.7347 16.8491 4.8044 9.4637
A4/Fukuda CTRP2 9.8407 11.5175 7.2891 0.3598
Ki-JK CTRP2 9.8458 16.8522 4.8805 9.0033
K-562 CTRP2 9.9138 12.1724 7.0665 0.8609
MOLP-8 CTRP2 10.0611 11.3678 7.4262 0.0945
EHEB CTRP2 10.1266 12.0167 7.2194 0.3913
Kasumi-1 CTRP2 10.3184 11.9487 7.3181 0.1736
KMS-28BM CTRP2 10.4942 12.7067 7.1119 1.0002
OCI-Ly10 CTRP2; CTRP1 10.7699 21.972 3.0596 14.2322
Kasumi-2 CTRP2 11.3302 22.6337 3.1154 13.1679
P31/FUJ CTRP2 11.7747 23.4515 3.0242 12.8475
OCI-Ly19 CTRP2 11.7951 26.842 1.4035 17.5828
P3HR-1 CTRP2 11.993 25.3629 2.2558 14.9091
⏷ Show the Full List of 149 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 8.6117 11.8323 6.4489 4.5543
TE15 CTRP2 8.9602 12.2371 6.4947 3.859
TE-6 CTRP2 7.8641 11.1565 6.2054 6.8698
TE-10 CTRP2 8.6396 12.3775 5.4453 3.7334
TE-5 CTRP2 8.7151 14.7849 5.0712 10.0458
KYSE-140 CTRP2 8.7786 11.8493 6.5577 3.8617
KYSE-30 CTRP2 8.9214 12.033 6.5663 3.6269
TE-4 CTRP2 9.0773 13.2684 6.0793 5.3633
KYSE-70 CTRP2 9.2567 11.2341 7.1325 1.1372
KYSE-150 CTRP2 9.4204 12.7886 6.5306 3.1301
KYSE-410 CTRP2 9.6106 16.7108 4.7839 9.7326
OE19 CTRP2 9.6829 10.7348 7.5085 0.0681
TE-9 CTRP2 9.7658 12.0398 7.0502 1.0035
EC-GI-10 CTRP2 9.8644 18.9258 3.8845 12.715
COLO 680N CTRP2 9.9124 17.7187 4.5074 10.3329
KYSE-450 CTRP2 9.9391 15.6012 5.5429 6.2936
TE-11 CTRP2 9.9699 15.3468 5.683 5.7091
OE33 CTRP2 10.1237 16.6425 5.17 7.4886
TE-1 CTRP2 10.1327 15.9119 5.5219 6.12
OE21 CTRP2 10.1371 16.2621 5.3595 6.7398
KYSE-510 CTRP2 11.3782 17.695 5.4602 4.8943
KYSE-520 CTRP2 11.4258 20.9719 3.9725 10.1443
KYSE-180 CTRP2 11.9781 21.7527 3.9602 9.4814
TE-14 CTRP2 12.9127 26.9809 2.0997 14.1462
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 36 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 10.1142 12.2172 7.1383 0.5707
PSN1 CTRP2 6.2901 9.7748 5.4025 13.7493
MIA PaCa-2 CTRP2 7.0562 9.9485 6.0808 9.1121
PaTu 8988s CTRP2 8.1183 12.9953 5.4942 9.3706
Panc 04.03 CTRP2 8.2627 12.3653 5.9232 7.3197
SNU-410 CTRP2 8.3275 12.6107 5.8517 7.5039
SU.86.86 CTRP2 8.7685 11.5337 6.7024 3.2941
YAPC CTRP2 8.8105 10.0522 7.4047 0.6284
TCC-Pan2 CTRP2 8.8336 11.4226 6.7982 2.8254
Capan-2 CTRP2 8.9394 12.9944 6.1159 5.4183
HPAC CTRP2 8.98 10.7299 7.203 1.146
Panc 03.27 CTRP2 9.0452 14.7832 5.3186 8.4979
SW1990 CTRP2 9.0867 16.1515 4.6761 10.9921
PK-59 CTRP2 9.1372 13.317 6.097 5.2055
HuP-T3 CTRP2 9.2107 20.1902 2.7707 17.6292
KP-4 CTRP2 9.2483 11.62 6.9594 1.7368
HuP-T4 CTRP2 9.4031 12.7786 6.5245 3.1735
HPAF-II CTRP2 9.4292 13.4145 6.2443 4.2233
PaTu 8902 CTRP2; CTRP1 9.4296 12.6198 6.6137 2.8057
Panc 10.05 CTRP2 9.4297 14.7558 5.6049 6.7584
DAN-G CTRP2 9.4595 13.9723 6.0003 5.1429
Capan-1 CTRP2 9.498 13.1729 6.4007 3.5322
SNU-213 CTRP2 9.5543 10.7387 7.4606 0.148
QGP-1 CTRP2 9.5632 10.805 7.4404 0.1764
L3.3 CTRP2 9.6776 12.9966 6.5891 2.6241
BxPC-3 CTRP2 9.7109 23.8524 1.3385 20.9736
PaTu 8988t CTRP2 9.8371 10.9631 7.4851 0.0743
Panc 08.13 CTRP2 10.1836 18.5497 4.2945 10.7242
CFPAC-1 CTRP2 10.3867 11.8724 7.369 0.104
KP-2 CTRP2 10.4067 14.5658 6.3034 2.9028
Panc 02.03 CTRP2 11.083 19.8732 4.2685 9.5525
Panc 05.04 CTRP2 11.4597 19.3796 4.7399 7.3807
AsPC-1 CTRP2 11.6341 26.1735 1.6147 17.2392
Hs 766T CTRP2 11.6927 24.5711 2.4312 14.8029
SUIT-2 CTRP2 12.8531 28.4164 1.3747 16.2202
PK-45H CTRP2 13.0803 32.6776 -0.5248 20.4493
⏷ Show the Full List of 36 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 47 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 9.2629 13.9383 5.8841 5.8811
SK-MEL-1 CTRP2; CTRP1 7.8362 9.216 7.1639 2.9912
A-375 CTRP2; CTRP1 8.1623 10.963 6.5546 4.9501
UACC-257 CTRP2 8.2206 16.3042 3.9245 15.425
SK-MEL-24 CTRP2 8.2341 12.8982 5.6352 8.5724
Hs 688(A).T CTRP2 8.3803 11.2278 6.5767 4.3933
RVH-421 CTRP2 8.398 12.5919 5.9156 7.1153
UACC-62 CTRP2 8.6389 13.0565 5.868 6.9075
SK-MEL-28 CTRP2; CTRP1 8.6759 9.7161 7.4939 0.5211
Hs 895.T CTRP2 8.6812 15.3022 4.7886 11.2388
HT-144 CTRP2 8.7176 12.7288 6.087 5.8773
IGR-37 CTRP2 8.7587 11.6193 6.6547 3.499
WT2-iPS CTRP2 8.8328 12.5136 6.2743 4.9328
SK-MEL-30 CTRP2 8.8544 10.3028 7.3208 0.862
IPC-298 CTRP2 8.9644 11.0415 7.0556 1.6852
SK-MEL-2 CTRP2 9.0088 10.1407 7.4622 0.3419
WM793 CTRP2 9.0226 11.2695 6.9866 1.8755
SK-MEL-31 CTRP2 9.0816 11.8671 6.7478 2.7076
WM115 CTRP2 9.1918 13.8553 5.8752 6.0202
WM266-4 CTRP2 9.194 13.7197 5.9421 5.7473
G-361 CTRP2 9.2085 17.3089 4.1961 12.6343
WM1799 CTRP2 9.2251 14.069 5.795 6.2948
COLO 829 CTRP2 9.2374 12.1194 6.727 2.6014
MeWo CTRP2 9.264 15.611 5.0721 9.139
HMCB CTRP2 9.313 16.0014 4.9165 10.3183
Hs 839.T CTRP2 9.3573 10.2266 7.567 0.0572
A2058 CTRP2 9.3901 15.0742 5.4235 8.0556
Hs 940.T CTRP2 9.3948 11.3182 7.1672 0.919
IGR-39 CTRP2 9.5296 10.846 7.4125 0.2498
CJM [Human melanoma] CTRP2 9.6355 15.4799 5.3975 7.2856
Hs 936.T CTRP2 9.6843 11.4959 7.2308 0.5618
COLO 800 CTRP2 9.7057 12.0726 7.007 1.1769
MDA-MB-435S CTRP2 9.7394 11.5949 7.2165 0.5687
WM88 CTRP2 9.7723 17.6411 4.4458 10.7805
Hs 944.T CTRP2 9.7742 16.4701 5.0155 8.5845
LOX-IMVI CTRP2 9.7763 11.3719 7.3172 0.328
A101D CTRP2 9.7881 17.3776 4.5854 10.2251
SK-MEL-5 CTRP2; CTRP1 9.8576 15.8145 5.4013 7.0407
Hs 852.T CTRP2; CTRP1 9.8923 16.7603 4.9571 8.6387
COLO 792 CTRP2 10.369 13.3276 6.8126 1.3728
SK-MEL-3 CTRP2 10.5794 16.2096 5.6627 5.0397
WM983B CTRP2 10.9039 16.3758 5.779 4.2573
Mel Ho CTRP2 11.7853 21.9913 3.7248 10.5257
Mel JuSo CTRP2 12.1448 21.3748 4.2396 8.324
Hs 294T CTRP2 12.1764 22.8198 3.5866 10.4906
IGR-1 CTRP2 12.454 25.3388 2.577 13.3345
K029AX CTRP2 12.9903 26.7709 2.2503 13.6147
⏷ Show the Full List of 47 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 7.5629 11.9686 5.5439 10.2434
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CHP-212 CTRP2 8.2564 13.1464 5.5292 8.973
CHP-126 CTRP2 8.5141 11.0637 6.7538 3.4537
KP-N-YN CTRP2 8.6576 19.0701 2.8948 18.2199
IMR-32 CTRP2 8.658 13.1344 5.8439 6.976
SK-N-AS CTRP2 8.7324 13.3593 5.7883 7.0839
MHH-NB-11 CTRP2 9.0359 11.7758 6.7617 2.7102
Kelly CTRP2 9.0451 11.898 6.7104 2.8968
SK-N-BE(2) CTRP2 9.1071 13.7158 5.8837 6.111
SK-N-DZ CTRP2 9.4285 10.7136 7.4209 0.2523
SK-N-FI CTRP2 9.693 11.6128 7.1886 0.6646
SiMa CTRP2 9.7868 12.6784 6.7907 1.8094
NH-6 CTRP2 9.8306 14.577 5.9553 4.8344
SK-N-SH CTRP2 10.1859 12.3541 7.1165 0.6287
KP-N-SI9s CTRP2 10.5679 21.8638 2.9553 14.8083
NB1 CTRP2 12.1039 22.4542 3.7118 10.1645
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuCC-T1 CTRP2 2.4506 3.1716 2.4506 36.006
SNU-308 CTRP2 7.963 10.9897 5.6643 3.7421
SNU-478 CTRP2 8.2704 9.9742 6.3053 0.8778
SNU-1196 CTRP2 9.8391 11.2472 7.3872 0.1864
HuH-28 CTRP2 10.1121 11.3201 7.46 0.059
SNU-1079 CTRP2 10.6193 22.1415 2.8566 15.0482
SNU-869 CTRP2 11.4473 23.2642 2.8921 13.7208
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-ES-1 CTRP2 8.6214 12.5394 6.1096 5.9374
Hs 888.T CTRP2 8.6577 13.2015 5.8106 7.1138
A-673 CTRP2 8.768 14.155 5.4227 8.5265
Hs 822.T CTRP2 8.9182 13.2573 5.9731 6.0323
SJSA-1 CTRP2 9.132 13.2491 6.1261 5.0959
TC71 CTRP2 9.1852 10.713 7.3147 0.6309
SK-N-MC CTRP2 9.5345 10.4845 7.5415 0.0575
SW1353 CTRP2 9.6923 11.7651 7.1272 0.8315
HOS CTRP2 9.7832 15.4276 5.5223 6.5857
G-292 clone A141B1 CTRP2 9.9569 14.666 5.9931 4.5333
MHH-ES-1 CTRP2 9.973 15.6327 5.5502 6.2201
SaOS-2 CTRP2 10.6609 18.0034 4.8775 7.8788
MG-63 CTRP2 12.0525 21.5153 4.1175 8.8527
CAL-78 CTRP2 13.6322 57.2211 -12.2011 34.0342
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 71 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 CTRP2 4.759 8.0123 4.4302 21.7541
CAL-148 CTRP2 7.1417 8.6126 6.241 2.5406
BT-20 CTRP2 7.1777 10.9574 5.7032 10.3983
MDA-MB-453 CTRP2 7.5769 12.7287 5.1766 11.7392
KPL-1 CTRP2 7.6185 12.531 5.311 11.0993
HCC1954 CTRP2 7.9735 10.3676 6.6895 4.6258
HCC1500 CTRP2 8.0087 11.6672 6.0689 7.1702
MCF-7 CTRP2; CTRP1 8.1808 13.4579 5.3257 10.0453
HCC1937 CTRP2 8.4008 14.1195 4.457 8.2323
Hs 578Bst CTRP2 8.7451 13.6926 5.6336 7.6995
CAL-51 CTRP2 8.7652 13.0728 5.9531 6.3529
HCC2218 CTRP2 8.8498 10.6516 7.1647 1.4097
AU565 CTRP2 8.9677 14.4003 5.4498 8.0898
HCC1395 CTRP2 9.053 13.9339 4.9802 5.09
MDA-MB-361 CTRP2 9.1061 13.8078 5.8383 6.2963
CAL-85-1 CTRP2 9.1849 15.2392 5.1968 8.7659
ZR-75-1 CTRP2 9.239 10.6292 7.3729 0.4427
HCC1143 CTRP2 9.3264 14.6246 5.5967 6.9429
HCC1569 CTRP2 9.3628 11.6665 7.0021 1.4784
SK-BR-3 CTRP2 9.3752 13.9174 5.9703 5.3774
T-47D CTRP2 9.3883 15.7292 5.1037 8.8193
MDA-MB-157 CTRP2 9.4512 17.9376 4.0671 12.713
BT-474 CTRP2 9.5355 10.9306 7.3836 0.2861
HCC1419 CTRP2 9.6534 13.3478 6.4152 3.294
HCC1428 CTRP2 9.7714 13.6037 6.3691 3.3317
ZR-75-30 CTRP2 9.8115 16.3373 5.1053 8.1796
UACC-812 CTRP2 9.8257 11.4124 7.322 0.301
BT-549 CTRP2 9.9302 12.0838 7.1094 0.7366
CAMA-1 CTRP2 10.1346 11.4269 7.4318 0.0793
JIMT-1 CTRP2 10.166 11.5271 7.4089 0.0965
HCC38 CTRP2 10.3004 18.3746 4.4597 9.9389
EFM-192A CTRP2 10.3035 11.7545 7.3798 0.1053
MDA-MB-468 CTRP2 10.304 12.314 7.1808 0.4019
Hs 578T CTRP2 10.3958 18.4116 4.5071 9.6258
MDA-MB-415 CTRP2 10.8744 18.5413 4.7621 8.0293
HMC-1-8 CTRP2 11.0481 18.7328 4.7832 7.7295
HCC202 CTRP2 11.5662 24.8476 2.2101 15.6406
HCC1806 CTRP2 11.6586 20.8501 4.1799 9.1214
MDA-MB-231 CTRP2 11.7687 29.4117 0.1315 20.7773
BT 239 CTRP2 8.603 10.4474 7.1086 1.9074
BT 286 CTRP2 8.6568 11.2408 6.7672 3.1909
BT 320 CTRP2 8.8852 11.2829 6.8967 2.3754
BT 359 CTRP2 8.9357 10.9261 7.0909 1.587
BT 328 CTRP2 8.9776 12.1588 6.5436 3.6404
BT 416 CTRP2 8.9794 20.2043 2.5838 18.6349
BT 248 CTRP2 8.9859 13.594 5.8573 6.4012
BT 330 CTRP2 9.0788 10.483 7.3578 0.5781
BT 231 CTRP2 9.1254 12.7191 6.3751 4.1095
BT 131 CTRP2 9.146 10.5284 7.3708 0.5005
BT 245 CTRP2 9.2615 12.7935 6.4285 3.7194
BT 216 CTRP2 9.2662 14.4802 5.6246 6.9203
BT 498 CTRP2 9.377 16.8101 4.5667 10.942
BT 139 CTRP2 9.3773 10.574 7.4518 0.212
BT 112 CTRP2 9.3842 10.9952 7.2937 0.566
BT 444 CTRP2 9.4321 14.8051 5.5828 6.8435
BT 422 CTRP2 9.4481 10.6182 7.4634 0.1711
BT 504 CTRP2 9.4976 13.4655 6.2641 4.0588
BT 172 CTRP2 9.5138 15.4684 5.319 7.7744
BT 232 CTRP2 9.5656 15.4875 5.3456 7.5923
BT 340 CTRP2 9.5974 10.6588 7.5043 0.0846
BT164 CTRP2 9.608 11.205 7.3102 0.4113
BT 333 CTRP2 9.6535 11.7717 7.1061 0.9175
BT 228 CTRP2 9.6567 11.0682 7.3813 0.2484
BT 179 CTRP2 9.8181 15.5932 5.4666 6.756
BT 145 CTRP2 9.8259 15.1307 5.6916 5.8649
BT 482 CTRP2 9.8677 11.1278 7.4396 0.111
BT 159 CTRP2 9.9195 11.4069 7.3607 0.2062
BT 271 CTRP2 9.9551 11.5599 7.3192 0.2641
BT147 CTRP2 10.4045 17.4393 4.977 7.8455
BT 440 CTRP2 10.5445 17.1548 5.202 6.8103
BT 224 CTRP2 12.3284 20.7795 4.6223 6.8038
⏷ Show the Full List of 71 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 7.9879 9.186 6.4926 0.5009
Cancer Drug Sensitivity Data Curated from 42 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LN-18 CTRP2 7.7551 8.9724 6.4659 0.7727
LN-229 CTRP2; CTRP1 7.7774 10.9899 6.2275 7.0444
SF295 CTRP2 8.2156 9.4537 6.4894 0.3752
D283 Med CTRP2 8.6052 14.6813 5.0382 10.3691
KNS-60 CTRP2 8.7285 13.0293 5.9476 6.4342
U-118MG CTRP2 8.7943 11.4696 6.7501 3.0684
KNS-81 CTRP2 8.8538 11.0467 6.9868 2.0684
SNU-466 CTRP2 9.1386 10.1223 7.5229 0.1619
42-MG-BA CTRP2 9.1985 13.0904 6.2469 4.5198
SNU-738 CTRP2 9.2124 10.2553 7.5033 0.1731
GMS-10 CTRP2 9.217 11.0008 7.2111 0.9824
Hs 683 CTRP2 9.2336 13.8757 5.8941 5.883
SNU-626 CTRP2 9.4061 10.4045 7.5233 0.0962
SNU-1105 CTRP2 9.4097 10.4881 7.4953 0.1325
KNS-42 CTRP2 9.4364 16.1272 4.944 9.3758
Daoy CTRP2 9.4378 17.4796 4.2824 11.9292
ONS-76 CTRP2 9.4469 12.2987 6.7694 2.2136
YKG-1 CTRP2 9.4655 15.4817 5.2787 8.0065
SF268 CTRP2 9.4676 16.4267 4.8201 9.8132
SF539 CTRP2 9.5423 15.6948 5.2292 8.0879
SW1783 CTRP2 9.5464 18.0401 4.0869 12.4839
DK-MG CTRP2 9.6558 11.2938 7.2966 0.4204
SNB-75 CTRP2 9.7157 15.3725 5.5034 6.7537
M059K CTRP2 9.7653 15.3595 5.5429 6.5294
CCF-STTG1 CTRP2 9.8143 14.5312 5.9664 4.8122
SW1088 CTRP2 9.8529 17.3729 4.6333 9.9437
Becker CTRP2 9.9043 11.7367 7.2329 0.4525
GaMG CTRP2; CTRP1 10.248 16.7944 5.18 7.2821
GOS-3 CTRP2 10.4979 16.189 5.6224 5.6458
KG-1-C CTRP2 10.5939 17.3762 5.1297 7.0197
DBTRG-05MG CTRP2 10.7808 17.773 5.0627 7.0334
U-251MG CTRP2 10.814 17.5036 5.2092 6.4472
8-MG-BA CTRP2 10.8214 17.113 5.3944 6.1381
GB-1 CTRP2 11.1172 18.8878 4.7545 7.7476
KALS-1 CTRP2 12.3342 25.651 2.3485 14.1751
T98G CTRP2 12.3486 27.6258 1.4101 16.7973
TM-31 CTRP2 12.8788 21.7068 4.5241 6.9602
YH-13 CTRP2 12.9656 26.7599 2.2393 14.3397
U-87MG ATCC CTRP2 14.2029 31.5515 0.7799 16.0531
SNU-201 CTRP2 14.2862 31.5605 0.8302 15.83
A-172 CTRP2 14.4874 28.3393 2.4625 11.2455
SF126 CTRP2 15.2507 32.1149 1.1869 13.8391
⏷ Show the Full List of 42 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-151 CTRP2; CTRP1 6.4545 9.8002 5.5653 12.7773
JHUEM-1 CTRP2 6.8845 10.7058 5.5525 11.6861
HEC-251 CTRP2 8.5008 10.9351 6.8069 3.2571
JHUEM-2 CTRP2; CTRP1 8.5744 14.5443 5.095 10.2818
JHUEM-3 CTRP2 8.7472 20.829 2.0891 20.5644
EFE-184 CTRP2 8.9889 12.2062 6.5286 3.6846
HEC-59 CTRP2; CTRP1 9.1429 12.5036 6.4886 3.6379
HEC-50B CTRP2 9.1475 14.1129 5.7194 6.7157
HEC-6 CTRP2 9.2442 17.4928 4.1322 12.8144
KLE CTRP2; CTRP1 9.2595 13.5909 6.0486 5.2264
AN3-CA CTRP2 9.3225 14.0976 5.8483 5.9392
HEC-108 CTRP2; CTRP1 9.4099 13.8181 6.0408 5.0499
HEC-1-A CTRP2 9.5761 15.4644 5.3641 7.504
HEC-1-B CTRP2 9.7185 11.1696 7.3687 0.2512
ESS-1 CTRP2 9.7639 15.5951 5.4294 6.9774
MFE-296 CTRP2 9.7776 16.027 5.2315 7.735
RL95-2 CTRP2 9.8195 10.9717 7.476 0.0802
MFE-319 CTRP2 10.0684 16.3196 5.2871 7.1121
JHUEM-7 CTRP2 10.2441 11.4402 7.4649 0.0441
EN CTRP2 11.018 18.1129 5.0532 6.7754
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 9.0762 11.771 6.789 2.5565
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 20 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TUHR14TKB CTRP2 7.2957 16.6394 2.9823 34.1177
VMRC-RCZ CTRP2 7.4036 10.69 6.04 8.502
CAL-54 CTRP2 7.9297 15.2241 4.2261 14.843
TUHR10TKB CTRP2 8.5511 13.2235 5.7195 7.6685
KMRC-2 CTRP2 8.8876 15.6621 4.768 10.9648
UO-31 CTRP2 9.0097 19.555 2.9304 17.4635
VMRC-RCW CTRP2 9.0385 12.2032 6.5626 3.4837
786-O CTRP2 9.1175 13.6395 5.9278 5.9168
KMRC-3 CTRP2 9.1445 12.5123 6.4856 3.6476
KMRC-20 CTRP2 9.3829 11.6196 7.0333 1.3557
TUHR4TKB CTRP2 9.6069 10.8766 7.4314 0.1788
SNU-1272 CTRP2 9.7453 19.9844 2.5559 13.5348
RCC10RGB CTRP2; CTRP1 9.7835 13.5224 6.4282 3.1783
OS-RC-2 CTRP2 10.0622 16.1213 5.3771 6.7722
A-498 CTRP2 10.1089 11.3863 7.4366 0.0783
ACHN CTRP2 10.2903 16.0647 5.5508 5.8087
KMRC-1 CTRP2 10.5806 18.4299 4.6225 8.9382
Caki-1 CTRP2 11.3732 22.9761 2.98 13.5447
Caki-2 CTRP2 13.0944 23.1354 4.0054 8.5081
769-P CTRP2 16.2658 41.7167 -2.6908 20.8588
⏷ Show the Full List of 20 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW480 CTRP1 6.3611 9.0921 5.7789 25.8821
SNU-175 CTRP1 6.8868 8.7265 6.481 17.1794
OUMS-23 CTRP2 6.9686 8.9796 6.4474 7.8358
SNU-C5 CTRP2; CTRP1 7.0828 10.675 5.7635 10.4593
C2BBe1 CTRP2 7.3385 10.9701 5.8429 9.4654
COLO 320 CTRP2; CTRP1 7.3924 11.6068 5.5856 10.5201
CL-11 CTRP2 7.7242 12.2113 5.5607 9.8487
CL-34 CTRP1 7.846 9.0131 7.2736 5.3805
NCI-H747 CTRP2 7.9369 15.9185 3.8849 16.1222
SNU-C4 CTRP2; CTRP1 7.9571 9.1825 7.2798 2.2756
CW-2 CTRP2; CTRP1 7.9925 10.4998 6.6507 4.853
CL-40 CTRP1 8.0212 9.1217 7.36 3.9171
HT115 CTRP2; CTRP1 8.0914 9.3043 7.3225 1.867
CCK-81 CTRP2 8.0973 9.5967 7.1699 2.3935
SNU-81 CTRP1 8.1214 9.754 7.1231 5.6695
T84 CTRP2 8.1807 11.3871 6.3457 5.696
SW948 CTRP2; CTRP1 8.2136 9.6933 7.2208 2.0931
SW1116 CTRP2 8.3033 13.4187 5.4306 9.2968
SNU-407 CTRP2 8.4289 11.644 6.4078 5.0149
HT-29 CTRP2; CTRP1 8.4765 10.3329 7.0941 2.2221
RCM-1 [Human ESC] CTRP2; CTRP1 8.5552 10.5354 7.0501 2.2893
LoVo CTRP2; CTRP1 8.5581 10.7454 6.9516 2.6791
SNU-61 CTRP2; CTRP1 8.5605 11.2195 6.7243 3.597
HT-55 CTRP2; CTRP1 8.5913 10.1188 7.2686 1.3929
RKO CTRP2; CTRP1 8.8289 12.6419 6.2227 5.2396
HCT 116 CTRP2; CTRP1 8.8832 13.6189 5.7844 6.9485
KM12 CTRP2; CTRP1 8.9912 13.3076 6.0139 5.8452
SNU-1040 CTRP1 9.0055 14.6991 5.3438 16.8248
SW620 CTRP2; CTRP1 9.0455 12.2364 6.5656 3.5495
NCI-H508 CTRP2; CTRP1 9.0767 13.444 6.0076 5.743
COLO 678 CTRP2; CTRP1 9.0842 14.0189 5.7337 6.8422
SNU-C1 CTRP2 9.2046 12.5683 6.4979 3.5214
SW48 CTRP2 9.2411 23.1604 1.3177 21.8332
HCT 8 CTRP2; CTRP1 9.2585 12.9652 6.3599 4.0781
SNU-503 CTRP2 9.3306 18.2357 3.8302 13.7835
MDST8 CTRP2; CTRP1 9.3476 12.8569 6.4681 3.5414
DLD-1 CTRP2 9.3511 10.261 7.553 0.0719
COLO205 CTRP2 9.5316 10.8843 7.3992 0.2574
HCC-56 CTRP2 9.5549 10.556 7.5243 0.0706
SNU-C2A CTRP2 9.5723 11.5583 7.1544 0.8327
GP2d CTRP2 9.5777 11.6228 7.1306 0.8979
LS180 CTRP2; CTRP1 9.6342 11.7399 7.1258 0.9344
SW1417 CTRP2 9.6766 17.9379 4.232 11.7347
LS1034 CTRP2 9.8743 15.3785 5.6059 6.1345
SK-CO-1 CTRP2 9.9873 16.0359 5.3683 6.9076
NCI-H716 CTRP2 10.0629 12.1939 7.1251 0.6266
HCT 15 CTRP2 10.0796 11.3728 7.4309 0.0873
LS123 CTRP2; CTRP1 10.3912 16.0716 5.6254 5.4817
COLO201 CTRP2 13.5457 25.8132 3.0508 10.5586
SNU-1033 CTRP2 13.5481 37.2798 -2.4323 23.5132
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-886 CTRP2 5.1107 44.0372 -12.577 43.4233
HuH-6 CTRP2 5.7693 9.9036 4.8117 17.4409
JHH-5 CTRP2 5.973 8.8827 5.4482 14.42
SNU-878 CTRP2 6.2972 13.1757 3.801 19.9974
SNU-761 CTRP2 7.4568 11.8415 5.5149 10.5832
SNU-398 CTRP2; CTRP1 8.0356 12.6665 5.6034 9.1641
Hep-G2 CTRP2; CTRP1 8.3935 10.4723 6.9695 2.8474
JHH-6 CTRP2; CTRP1 8.7608 13.9445 5.5211 8.1352
SNU-387 CTRP2 9.4998 12.0402 6.9135 1.6544
Hep 3B2.1-7 CTRP2 9.5861 11.0413 7.3629 0.3082
SNU-449 CTRP2; CTRP1 9.6237 19.0133 3.6654 13.8888
Li-7 CTRP2 9.6557 11.9871 7.0178 1.1816
JHH-1 CTRP2 9.6647 11.5559 7.1984 0.701
SNU-182 CTRP2 9.865 18.0384 4.3183 11.1172
SK-HEP-1 CTRP2 9.8809 11.7063 7.2346 0.4589
HuH-1 CTRP2 9.9477 11.2471 7.4272 0.119
JHH-4 CTRP2 9.9628 15.4195 5.6443 5.8684
JHH-2 CTRP2 9.9796 12.8684 6.8105 1.5799
SNU-423 CTRP2 10.2292 18.5049 4.3478 10.459
PLC/PRF/5 CTRP2 10.2946 17.251 4.9939 7.9303
SNU-475 CTRP2 10.7185 18.5864 4.6392 8.689
HLF CTRP2 11.8893 23.7212 2.9722 12.8583
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 151 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1963 CTRP1 2.0419 6.751 1.7756 71.1722
NCI-H1184 CTRP2 2.167 4.3165 -0.8595 1.2664
NCI-H647 CTRP2 5.6942 9.5324 4.8911 17.3355
RERF-LC-Ad1 CTRP2 5.8386 7.0369 4.4366 0.6967
SK-MES-1 CTRP2 5.9853 12.075 4.0335 19.8901
NCI-H810 CTRP2 6.012 8.198 5.7383 13.2128
DV-90 CTRP2 6.2243 13.0091 3.8135 20.1264
COR-L88 CTRP2 6.2773 13.9166 3.4211 21.4174
DMS 53 CTRP2 6.6332 12.28 4.5516 16.3262
NCI-H1930 CTRP1 6.727 15.686 1.6516 26.6246
NCI-H2170 CTRP2 6.7635 9.9589 5.792 10.9943
RERF-LC-KJ CTRP1 6.9797 10.8388 4.2329 10.4159
COLO 668 CTRP2; CTRP1 6.9806 11.3961 5.3064 12.4787
NCI-H3255 CTRP1 7.0228 10.0272 6.0201 20.2317
NCI-H1944 CTRP2 7.0914 14.7968 3.7229 18.4736
SCLC-21H CTRP1 7.1075 8.1327 6.9518 11.9941
COR-L51 CTRP2; CTRP1 7.1618 22.1855 0.1091 28.6825
NCI-H1105 CTRP2; CTRP1 7.2308 11.3121 5.5868 10.8622
NCI-H211 CTRP2 7.2934 12.4784 5.0542 12.832
EKVX CTRP2 7.3494 13.0176 4.8352 13.6061
NCI-H1573 CTRP2 7.4054 26.1302 -1.6662 31.4257
NCI-H1693 CTRP2 7.451 11.9597 5.4511 10.8609
HCC1195 CTRP2; CTRP1 7.5182 18.3114 2.3486 22.2499
NCI-H1341 CTRP2 7.526 12.9663 5.0142 12.5102
HCC1833 CTRP2; CTRP1 7.5309 10.7912 6.1135 8.0241
DMS 454 CTRP2 7.5342 11.6867 5.6596 9.8192
NCI-H526 CTRP2 7.5402 9.1153 6.2753 1.7658
NCI-H2342 CTRP2; CTRP1 7.5966 12.8278 5.1551 11.8807
NCI-H2291 CTRP2 7.6133 11.4878 5.1752 6.4349
SK-LU-1 CTRP2; CTRP1 7.6322 10.1829 6.5054 6.1705
NCI-H1836 CTRP1 7.7222 11.4227 5.9643 17.2953
EBC-1 CTRP2 7.7259 12.4821 5.4268 10.4032
LCLC-97TM1 CTRP2 7.7266 15.1254 4.106 15.7075
NCI-H522 CTRP2 7.7275 13.129 5.1048 11.732
NCI-H69 CTRP2 7.7386 11.4903 5.2659 5.821
NCI-H1581 CTRP2 7.788 13.6122 4.9141 12.3918
NCI-H2122 CTRP2; CTRP1 7.8098 10.5616 6.469 5.9653
NCI-H146 CTRP2 7.8433 14.4391 4.5469 13.7585
NCI-H358 CTRP2 7.906 12.029 5.8039 8.4763
NCI-H1734 CTRP2 7.9819 9.8576 6.2019 1.5188
NCI-H596 CTRP1 8.0548 13.4018 5.2516 20.9882
NCI-H889 CTRP2 8.0827 12.3328 5.7963 8.1762
NCI-H520 CTRP2 8.1288 13.4911 5.2551 10.3409
NCI-H2141 CTRP1 8.1305 9.3729 7.3175 3.9108
ChaGo-K-1 CTRP2 8.1684 13.5186 5.2733 10.1925
NCI-H1781 CTRP1 8.1773 11.3399 6.3788 12.0015
HCC1359 CTRP1 8.1878 10.1587 6.9731 6.7659
HCC44 CTRP2 8.2068 24.2244 -0.0448 26.9388
NCI-H1694 CTRP2; CTRP1 8.2809 13.048 5.6099 8.6866
CAL-12T CTRP2; CTRP1 8.294 10.8476 6.7127 4.0655
NCI-H1838 CTRP2 8.3462 15.4328 4.4606 13.138
NCI-H1876 CTRP1 8.4139 11.3135 6.5724 9.4775
NCI-H1355 CTRP2 8.4205 18.9577 2.761 19.0994
Calu-3 CTRP2 8.4313 19.7931 2.3526 20.3627
NCI-H1435 CTRP2; CTRP1 8.4502 14.9193 4.799 11.6077
A-549 CTRP2 8.5053 11.6634 6.4546 4.6976
NCI-H1915 CTRP2; CTRP1 8.5114 13.3204 5.6412 8.0599
NCI-H2073 CTRP1 8.5414 14.9817 4.8518 21.5134
EPLC-272H CTRP2 8.5609 13.6174 5.5319 8.4268
NCI-H661 CTRP2 8.5732 13.3338 5.6817 7.7875
HCC2108 CTRP2; CTRP1 8.5906 19.009 2.884 18.4509
NCI-H841 CTRP2; CTRP1 8.6136 12.8123 5.9825 6.5679
NCI-H2228 CTRP2 8.6283 15.1304 4.8331 11.1539
NCI-H2444 CTRP2 8.6372 11.211 6.7681 3.2153
PC-14 CTRP2 8.6538 12.4986 6.1534 5.7051
HCC2935 CTRP2; CTRP1 8.6928 13.063 5.9178 6.7059
NCI-H1155 CTRP2 8.7005 15.7265 4.5929 11.9795
NCI-H446 CTRP2 8.7193 16.5572 4.1947 13.4865
NCI-H2029 CTRP2 8.7303 13.5438 5.6959 7.4674
NCI-H2126 CTRP2 8.7732 10.2976 7.279 1.0796
HCC4006 CTRP2; CTRP1 8.7845 16.7315 4.1712 13.5418
NCI-H322 CTRP2 8.8175 13.1346 5.9607 6.239
HOP-92 CTRP2 8.8298 21.3624 1.8888 20.9948
COR-L23 CTRP1 8.8636 10.8954 7.0771 3.8521
NCI-H460 CTRP2; CTRP1 8.8887 10.6181 7.217 1.2608
BEN CTRP2 8.9631 9.9665 7.5096 0.2529
DMS 114 CTRP2 9.0004 12.4754 6.4079 4.1505
NCI-H2110 CTRP2; CTRP1 9.0033 15.6265 4.8855 10.39
MOR/CPR CTRP2 9.022 9.9125 7.5536 0.1444
LK2 CTRP2 9.0481 11.4444 6.9221 2.0865
NCI-H2087 CTRP2 9.1311 16.5095 4.5326 11.4773
DMS 79 CTRP2 9.1319 16.2475 4.6625 10.9703
HCC15 CTRP2; CTRP1 9.1795 14.9425 5.3513 8.2411
NCI-H226 CTRP2 9.2276 11.6216 6.9469 1.8022
COLO 699 CTRP2; CTRP1 9.2328 14.5008 5.6047 7.1382
NCI-H1666 CTRP2 9.2382 13.2725 6.1865 4.7058
NCI-H292 CTRP2 9.2828 10.9363 7.2701 0.6936
NCI-H1651 CTRP2 9.2997 14.548 5.6152 6.9082
T3M-10 CTRP2; CTRP1 9.3153 18.5228 3.6896 14.3938
NCI-H2085 CTRP2 9.334 15.5217 5.1661 8.6552
SW1271 CTRP2 9.3656 13.7537 6.042 5.1057
NCI-H2196 CTRP2 9.3866 11.0033 7.2915 0.5701
COR-L105 CTRP2 9.4936 15.6537 5.215 8.217
NCI-H1755 CTRP2; CTRP1 9.5067 14.6412 5.7263 6.2504
COR-L95 CTRP2 9.5109 12.0529 6.914 1.6426
NCI-H2172 CTRP2; CTRP1 9.5483 17.9744 4.1336 12.3869
NCI-H2023 CTRP2; CTRP1 9.5488 12.869 6.5861 2.855
NCI-H196 CTRP2 9.5507 10.945 7.3844 0.2789
HARA [Human squamous cell lung carcinoma] CTRP2 9.5633 13.4179 6.3275 3.733
VMRC-LCD CTRP2 9.5826 12.0744 6.943 1.4812
HCC1438 CTRP2 9.6015 17.1964 4.5404 10.6858
NCI-H1792 CTRP2 9.6878 14.4599 5.9188 5.1596
DMS 273 CTRP2 9.7417 16.5015 4.9778 8.7796
HCC2279 CTRP2 9.7433 17.1531 4.6628 9.997
LCLC-103H CTRP2 9.7533 19.9931 3.279 15.0214
Lu-99 CTRP2 9.7939 15.2045 5.6356 6.1266
NCI-H1568 CTRP2 9.8144 11.8017 7.1687 0.6484
RERF-LC-MS CTRP2 9.8177 12.8666 6.7255 2.0025
NCI-H1703 CTRP2 9.8592 17.1279 4.7565 9.462
LC-1/sq-SF CTRP2 9.8821 17.0968 4.7875 9.3084
HCC827 CTRP2; CTRP1 9.9018 13.7589 6.3908 3.186
NCI-H1339 CTRP2 9.9025 11.7233 7.2372 0.4438
NCI-H1869 CTRP2 9.955 13.8256 6.3768 3.1014
LOU-NH91 CTRP2 10.0062 17.2844 4.7828 9.1442
SHP-77 CTRP2 10.0122 11.374 7.4066 0.1235
HCC1588 CTRP2 10.0159 11.2148 7.4622 0.0676
NCI-H1373 CTRP2 10.0797 15.7384 5.5695 6.0055
NCI-H1299 CTRP2 10.115 11.8663 7.2702 0.2999
NCI-H1650 CTRP2 10.1621 15.247 5.851 4.8256
HCC78 CTRP2 10.2608 12.0025 7.2774 0.2455
NCI-H727 CTRP2 10.2973 17.5574 4.8496 8.4755
NCI-H650 CTRP2 10.3418 15.2712 5.9491 4.2487
RERF-LC-A1 CTRP2 10.4146 17.2582 5.0694 7.4814
LXF 289 CTRP2; CTRP1 10.4455 18.597 4.4518 9.7606
Sq-1 CTRP2; CTRP1 10.4926 25.2815 1.2361 20.0313
NCI-H2405 CTRP2 10.5009 15.0993 6.1196 3.4576
HCC1171 CTRP2 10.5682 12.0697 7.3655 0.0841
NCI-H1623 CTRP2 10.6019 21.4311 3.1903 13.9841
HCC95 CTRP2 10.6234 21.7554 3.0477 14.4223
NCI-H2286 CTRP2; CTRP1 10.6426 17.0072 5.3329 6.1954
NCI-H2030 CTRP2; CTRP1 10.7103 19.6761 4.1276 10.6464
NCI-H838 CTRP2 10.8166 18.5073 4.7407 8.1834
KNS-62 CTRP2 10.8301 19.0273 4.5035 9.039
Lu-65 CTRP2 10.8385 27.7212 0.2783 21.8061
NCI-H1092 CTRP2 10.8759 32.3127 -1.9635 26.262
LUDLU-1 CTRP2 10.8812 24.7453 1.7726 17.9114
NCI-H1793 CTRP2 11.052 22.401 3.0358 13.825
RERF-LC-Ad2 CTRP2 11.0808 17.5259 5.362 5.5713
NCI-H1395 CTRP2 11.6714 25.5495 1.9436 16.264
HOP-62 CTRP2 11.7593 26.6103 1.4909 17.3982
Calu-6 CTRP2 11.9242 21.1265 4.2181 8.6612
NCI-H441 CTRP2; CTRP1 12.0025 24.2249 2.8214 13.2458
SW1573 CTRP2 12.0675 44.6475 -7.1663 31.5536
SBC-5 CTRP2 12.1815 27.5849 1.3141 17.2811
NCI-H2081 CTRP2; CTRP1 12.3471 25.0747 2.646 13.3286
NCI-H2009 CTRP2 12.619 27.1348 1.8305 15.2875
NCI-H1563 CTRP2 12.6556 26.0476 2.3734 13.6814
NCI-H23 CTRP2 12.7329 27.1429 1.9031 14.935
Calu-1 CTRP2 12.8001 24.2253 3.3244 10.577
HCC366 CTRP2 13.1815 32.2199 -0.2322 19.6842
Hs 888.Lu CTRP2 10.4701 16.9066 5.2709 6.6447
⏷ Show the Full List of 151 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 8.9017 10.9326 7.068 1.7079
COV434 CTRP2; CTRP1 5.9339 9.7728 5.0452 16.1869
RMUG-S CTRP1 6.6032 10.8565 5.2199 28.2135
JHOS-4 CTRP1 6.9256 13.5431 2.8685 20.0361
OVMANA CTRP1 7.1232 10.5183 4.4831 7.98
TOV-112D CTRP2 7.1494 11.5401 5.3902 11.7579
OVCAR-8 CTRP2; CTRP1 7.1675 12.4126 4.9853 13.4765
OVCAR-4 CTRP2; CTRP1 7.4324 10.0493 6.393 7.0665
OVKATE CTRP1 7.5282 12.284 5.3675 22.5245
A2780 CTRP2; CTRP1 7.6361 13.2983 4.9539 12.6241
OV-90 CTRP2; CTRP1 7.6482 10.8484 6.1876 7.4711
OVK18 CTRP2; CTRP1 7.8559 12.4085 5.5842 9.5869
TYK-nu CTRP2; CTRP1 7.9076 11.6123 6.0252 7.6412
IGROV-1 CTRP2; CTRP1 8.1851 13.3877 5.3641 9.8787
COV318 CTRP1 8.3334 12.9047 4.1254 7.6
MCAS CTRP2 8.4056 11.2266 6.596 4.2724
RMG-I CTRP2; CTRP1 8.6266 11.5695 6.6009 4.0012
OVISE CTRP2 8.8295 13.6051 5.7389 7.1303
COV362 CTRP2; CTRP1 8.9555 16.9759 4.1817 13.202
SNU-119 CTRP2 8.96 12.779 6.2344 4.9069
OAW42 CTRP2; CTRP1 9.2179 12.4857 6.5595 3.3503
EFO-27 CTRP2; CTRP1 9.2485 14.4497 5.6405 6.97
OV56 CTRP2 9.3192 13.141 6.3021 4.1397
SNU-840 CTRP2; CTRP1 9.3476 13.148 6.3314 4.0734
COV644 CTRP2; CTRP1 9.3908 20.38 2.8275 17.2027
DOV13 CTRP2 9.4168 23.0706 1.4995 21.0411
JHOC-5 CTRP2; CTRP1 9.5011 14.526 5.7778 6.0538
SNU-8 CTRP2 9.6823 10.6767 7.5279 0.0517
FU-OV-1 CTRP2 9.8223 34.7899 -4.0169 30.8791
JHOS-2 CTRP2 9.8945 13.1828 6.629 2.2633
EFO-21 CTRP2 9.9454 14.5894 6.0215 4.4391
JHOM-1 CTRP2; CTRP1 10.058 15.253 5.7976 5.2378
OVSAHO CTRP2 10.1654 11.5143 7.413 0.0926
OAW28 CTRP2 10.1768 14.6506 6.1335 3.752
Caov-3 CTRP2; CTRP1 10.224 14.7258 6.1422 3.7462
Kuramochi CTRP2 10.5598 19.437 4.1261 10.7908
OVCAR-5 CTRP2 10.736 19.7321 4.1044 10.6181
HEY A8 CTRP2 10.8247 15.6832 6.0426 3.4056
OC 314 CTRP2 11.0736 18.9317 4.7063 7.9785
OVTOKO CTRP2 11.3176 25.5185 1.7089 17.4375
ONCO-DG-1 CTRP2 11.6291 31.4036 -0.9483 23.2893
SK-OV-3 CTRP2 12.1027 21.0713 4.3538 7.9807
ES2 CTRP2 12.8535 30.8921 0.1819 19.1766
OV7 CTRP2; CTRP1 14.9237 28.7797 2.5384 10.6214
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Aska-SS CTRP2 9.0374 10.6536 7.2663 0.8861
Yamato-SS CTRP2 9.4206 10.7634 7.3991 0.2987
TE 617.T CTRP2 6.5981 11.5048 4.8949 15.0355
G-402 CTRP2 7.049 11.6411 5.2489 12.5622
RKN CTRP2; CTRP1 7.8326 9.5549 6.9914 3.7234
Rh41 CTRP2 7.8489 12.3447 5.5987 9.4452
TE 441.T CTRP2 7.9026 10.3665 6.6323 4.9992
HT-1080 CTRP2; CTRP1 8.0087 11.6293 6.0997 7.1375
A-204 CTRP2 8.042 14.3944 4.7333 12.6289
SK-LMS-1 CTRP2 8.4421 14.3029 5.0995 10.4079
Hs 729.T CTRP2 8.6355 13.8243 5.4862 8.4883
MES-SA CTRP2 8.7172 12.4933 6.2019 5.4054
BT-16 CTRP2 8.7375 11.2162 6.833 2.8158
TTC-709 CTRP2 8.8376 10.6006 7.1805 1.3655
SW982 CTRP2 9.1659 10.4733 7.4016 0.4098
G-401 CTRP2 9.2489 15.8749 4.9318 9.7198
Tm87-16 CTRP2 9.3459 14.0448 5.8895 5.7407
KYM-1 CTRP2 9.3644 15.5992 5.15 8.6723
Rh18 CTRP2 9.5181 14.283 5.8913 5.4944
GCT CTRP2 10.058 16.2874 5.2955 7.0935
BT-12 CTRP2 10.7484 21.1754 3.4174 13.0026
SK-UT-1 CTRP2 14.8952 33.5605 0.2816 16.4331
RD CTRP2 15.14 30.5727 1.8325 12.28
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 9.2871 10.8866 7.2923 0.6281
P-STS CTRP2 9.8342 16.8627 4.8674 9.0712
H-STS CTRP2 10.2264 22.8525 2.222 17.6311
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 9.5402 11.3002 7.2434 0.6086
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2 8.285 14.7368 4.7589 12.0695
ACC-MESO-1 CTRP2 8.3527 16.2884 4.039 14.7462
NCI-H2452 CTRP2 8.4308 12.2077 6.1309 6.1629
NCI-H28 CTRP2 8.7547 13.548 5.7119 7.3619
MPP 89 CTRP2 9.4899 12.8512 6.5441 2.9981
JL-1 CTRP2 9.8296 21.0947 2.793 16.5056
IST-Mes1 CTRP2 10.9758 22.1716 3.0937 13.7471
NCI-H2052 CTRP2 11.8968 22.1995 3.6987 10.4704
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PaCa-3 CTRP2; CTRP1 8.0011 12.126 5.8335 8.1722
DU145 CTRP2 8.1912 13.244 5.4286 9.5085
LNCaP clone FGC CTRP2 8.2167 11.4059 6.3644 5.5548
NCI-H660 CTRP2 8.3339 17.9362 3.2011 17.7987
22Rv1 CTRP2 9.3018 13.0508 6.3334 4.0399
VCaP CTRP2 9.7481 14.8824 5.7583 5.7075
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 CTRP2 7.6365 12.4655 5.3591 10.8632
YD-15 CTRP2 8.3053 9.2799 6.5901 0.1322
Cancer Drug Sensitivity Data Curated from 34 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
GSS CTRP2 2.8333 10.3212 1.5448 36.9676
SNU-16 CTRP2 4.4228 6.1658 4.4018 22.9137
NCC-StC-K140 CTRP2 5.5541 9.8371 4.617 18.7727
SNU-5 CTRP2 7.4656 10.4652 5.5692 4.9504
SNU-620 CTRP2 7.7006 9.9435 6.6734 5.2228
KE-39 CTRP2 7.8828 10.9729 6.3128 6.382
NUGC-4 CTRP2 8.065 9.4653 7.2104 2.2786
ECC10 CTRP2 8.1815 11.3589 6.3603 5.6334
HGC-27 CTRP2 8.2219 13.0259 5.5619 8.8995
SNU-668 CTRP2 8.4975 13.1469 4.9922 5.8111
SNU-1 CTRP2 8.5184 13.3121 5.6507 8.0087
AGS CTRP2; CTRP1 8.8551 11.097 6.9788 2.1814
NCI-N87 CTRP2 8.862 11.6439 6.712 3.1281
Hs 746.T CTRP2 8.884 14.789 5.1967 9.2535
GSU CTRP2 8.9827 9.5628 7.6607 0.0236
SNU-216 CTRP2 8.9964 14.0222 5.6559 7.2056
Fu97 CTRP2 9.0248 13.0857 6.1312 5.2298
NUGC-3 CTRP2 9.0651 13.5452 5.937 5.9575
MKN45 CTRP2 9.1353 10.1152 7.5242 0.1607
MKN7 CTRP2 9.2519 14.0364 5.8293 6.1172
KATO III CTRP2 9.2707 12.3756 6.6293 2.9325
OCUM-1 CTRP2 9.2795 15.3393 5.216 8.5408
SNU-719 CTRP2 9.5186 12.7187 6.6217 2.6767
SH-10-TC CTRP2 9.59 15.5765 5.3196 7.6599
HuG1-N CTRP2 10.0964 13.796 6.4706 2.6205
SNU-601 CTRP2 10.4196 16.7138 5.3291 6.4885
IM95 CTRP2 11.0996 22.8858 2.8343 14.4029
MKN74 CTRP2; CTRP1 11.133 18.3733 5.0038 6.8175
ECC12 CTRP2 11.9384 23.9303 2.9052 13.0041
LMSU CTRP2 12.0365 21.6169 4.0603 9.0682
MKN1 CTRP2 12.2199 28.5433 0.8767 18.3557
SNG-M CTRP2; CTRP1 9.3368 14.3403 5.7412 6.3477
SNU-1077 CTRP2 10.2774 11.8548 7.3359 0.1592
SNU-685 CTRP2 10.3582 16.1998 5.5305 5.8011
⏷ Show the Full List of 34 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW579 CTRP2 7.4237 10.4038 6.1998 7.7908
TT2609-C02 CTRP2 8.1934 13.0477 5.5283 9.0908
TT CTRP2 8.7621 11.3147 6.8025 2.9037
BHT-101 CTRP2 9.3815 16.6705 3.9015 9.0067
B-CPAP CTRP2 9.3845 23.3929 1.3142 21.5936
FTC-133 CTRP2 9.576 15.2692 5.458 7.1316
8305C CTRP2 9.6692 11.1015 7.3741 0.2575
ML-1 [Human leukemia] CTRP2 9.6894 11.3741 7.2802 0.4423
8505C CTRP2 10.0872 18.1277 4.4316 10.3565
FTC-238 CTRP2 12.7123 23.7138 3.5074 10.6567
CGTH-W-1 CTRP2 13.4384 29.5795 1.2118 15.8985
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 29 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-2 CTRP2 6.765 10.4223 5.5742 11.8782
YD-10B CTRP2 7.0118 8.2078 6.3417 2.3307
SNU-1214 CTRP2 7.4758 9.7388 5.9325 3.334
PE/CA-PJ49 CTRP2 8.0136 12.2272 5.7931 8.3178
SCC-25 CTRP2 8.4359 13.1828 5.6515 8.1477
SNU-899 CTRP2 8.6822 9.9854 6.4811 0.2065
PE/CA-PJ15 CTRP2 8.8236 14.4025 5.3421 8.7629
HSC-4 CTRP2 8.8304 12.6794 6.1921 5.2718
SCC-9 CTRP2; CTRP1 8.9591 12.895 6.1914 5.1721
SNU-1076 CTRP2 9.3173 10.411 7.4877 0.1683
FaDu CTRP2 9.4523 13.1456 6.3848 3.649
PE/CA-PJ34 (clone C12) CTRP2 9.4572 13.8213 6.0704 4.8692
BICR 16 CTRP2 9.4707 11.5356 7.1142 1.0243
SNU-46 CTRP2 9.619 12.7544 5.8149 1.4154
BICR 22 CTRP2 9.7057 11.5703 7.2111 0.5997
SNU-1066 CTRP2 9.71 10.9718 7.4364 0.1463
CAL-27 CTRP2 9.7462 11.1254 7.3954 0.2119
BHY CTRP2 9.8648 15.4208 5.5797 6.2498
Detroit 562 CTRP2 9.8687 21.6936 2.5267 17.2835
SCC-4 CTRP2 9.9641 11.502 7.3436 0.2211
BICR 6 CTRP2 9.9842 11.2426 7.4417 0.0903
BICR 56 CTRP2 10.064 11.1913 7.4865 0.045
YD-8 CTRP2 10.0646 19.2285 3.8806 12.416
SNU-1041 CTRP2 10.2152 11.5761 7.4095 0.0891
BICR 18 CTRP2 10.2305 12.0335 7.2546 0.2915
BICR 31 CTRP2 10.2657 13.6784 6.6134 1.9803
CAL-33 CTRP2 10.603 19.6088 4.0731 10.92
PE/CA-PJ41 (clone D2) CTRP2 10.8628 17.7861 5.1082 6.7621
HSC-3 CTRP2 12.4936 25.0374 2.7461 12.7688
⏷ Show the Full List of 29 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HT-1197 CTRP2 7.2618 13.3175 4.6091 14.7017
T24 CTRP2 7.6741 11.9318 5.6578 9.5428
BC-3C CTRP2 8.1987 14.5075 4.8041 12.0487
UM-UC-3 CTRP2 8.5054 14.3749 5.1131 10.2403
5637 CTRP2 8.5844 12.2909 6.2045 5.6048
RT-4 CTRP2 8.7183 15.0773 4.9287 10.614
253J CTRP2 8.7927 13.9704 5.5322 8.0375
U-BLC1 CTRP2 9.0652 13.3726 6.0206 5.6186
RT-112 CTRP2 9.157 12.5654 6.4686 3.6979
KU-19-19 CTRP2 9.2124 10.3454 7.4702 0.2347
JMSU-1 CTRP2 9.4378 18.8576 3.6036 14.417
SCaBER CTRP2 9.5458 11.0913 7.3272 0.429
HT-1376 CTRP2 9.6142 11.5173 7.1907 0.7053
UM-UC-1 CTRP2 9.7351 15.8842 5.271 7.6407
KMBC-2 CTRP2 9.8992 18.4241 4.1547 11.6729
647V CTRP2 10.4046 17.8192 4.7963 9.0808
TCCSUP CTRP2 10.6865 17.0502 5.3403 6.114
VM-CUB-1 CTRP2 13.0312 28.9811 1.2246 16.3831
J82 CTRP2 13.1836 25.7803 2.8405 11.6235
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 9.2939 10.3373 7.5052 0.1466

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