Details of the Drug

General Information of Drug (ID: DM83WVF)

Drug Name
Apicidin
Synonyms
CHEMBL430060; OSI-2040; (3S,6S,9S,12R)-3-[(2S)-butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone; Acipidin; AC1OCFAM; Apicidin _120249; SCHEMBL147997; ChEMBL_275631; GTPL7495; DTXSID40274182; MolPort-005-944-562; BDBM50238632; ZINC17654900; AKOS030622920; MCULE-8969470747; NCGC00165733-01
Indication
Disease Entry ICD 11 Status REF
Solid tumour/cancer 2A00-2F9Z Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 2 Molecular Weight (mw) 623.8
Logarithm of the Partition Coefficient (xlogp) 4.4
Rotatable Bond Count (rotbonds) 12
Hydrogen Bond Donor Count (hbonddonor) 3
Hydrogen Bond Acceptor Count (hbondacc) 6
Chemical Identifiers
Formula
C34H49N5O6
IUPAC Name
(3S,6S,9S,12R)-3-[(2S)-butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone
Canonical SMILES
CC[C@H](C)[C@H]1C(=O)N2CCCC[C@@H]2C(=O)N[C@H](C(=O)N[C@H](C(=O)N1)CC3=CN(C4=CC=CC=C43)OC)CCCCCC(=O)CC
InChI
InChI=1S/C34H49N5O6/c1-5-22(3)30-34(44)38-19-13-12-18-29(38)33(43)35-26(16-9-7-8-14-24(40)6-2)31(41)36-27(32(42)37-30)20-23-21-39(45-4)28-17-11-10-15-25(23)28/h10-11,15,17,21-22,26-27,29-30H,5-9,12-14,16,18-20H2,1-4H3,(H,35,43)(H,36,41)(H,37,42)/t22-,26-,27-,29+,30-/m0/s1
InChIKey
JWOGUUIOCYMBPV-GMFLJSBRSA-N
Cross-matching ID
PubChem CID
6918328
TTD ID
D0W1PV

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Histone deacetylase (HDAC) TTBH0VX NOUNIPROTAC Inhibitor [2]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
7SK snRNA methylphosphate capping enzyme (MEPCE) OTRBQEYP MEPCE_HUMAN Gene/Protein Processing [3]
A-kinase anchor protein 8 (AKAP8) OTK3EQAI AKAP8_HUMAN Gene/Protein Processing [3]
Apoptosis regulator BAX (BAX) OTAW0V4V BAX_HUMAN Gene/Protein Processing [4]
Apoptosis regulator Bcl-2 (BCL2) OT9DVHC0 BCL2_HUMAN Gene/Protein Processing [4]
ATP-dependent translocase ABCB1 (ABCB1) OTEJROBO MDR1_HUMAN Drug Response [5]
Caspase-3 (CASP3) OTIJRBE7 CASP3_HUMAN Gene/Protein Processing [4]
Caspase-6 (CASP6) OTXLD3EC CASP6_HUMAN Gene/Protein Processing [4]
Caspase-8 (CASP8) OTA8TVI8 CASP8_HUMAN Gene/Protein Processing [6]
Caspase-9 (CASP9) OTD4RFFG CASP9_HUMAN Gene/Protein Processing [4]
Cellular tumor antigen p53 (TP53) OTIE1VH3 P53_HUMAN Gene/Protein Processing [6]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 149 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 -2.4737 2.359 -2.6134 50.0813
MEC1 CTRP2 -2.0309 2.2044 -2.1267 47.2521
JM1 CTRP2 -4.0153 -0.1077 -4.037 60.0193
DoHH2 CTRP2 -7.641 -3.0164 -7.6511 80.5325
KMS-26 CTRP2 -7.5856 -4.9024 -7.5857 83.06
EoL-1 CTRP2 -7.2982 -5.7468 -7.2982 82.1218
SEM CTRP2 -6.223 -2.3653 -6.2287 73.7727
GA-10 CTRP2 -5.9386 -1.908 -5.9478 71.9111
Ri-1 CTRP2 -5.7978 -1.1591 -5.8225 70.4858
OCI-AML-3 CTRP2 -5.7626 -3.3854 -5.7627 71.8512
A4/Fukuda CTRP2 -5.321 -1.4101 -5.3315 68.249
CA46 CTRP2 -5.1027 -0.9746 -5.1196 66.7508
MOLP-8 CTRP2 -4.8792 -0.4719 -4.9075 65.1884
KMS-12-BM CTRP2 -4.8768 -1.9067 -4.8785 65.8959
HH [Human lymphoma] CTRP2 -4.8282 -0.3274 -4.8609 64.8139
JVM-2 CTRP2 -4.805 6.2389 -6.053 59.7816
MOLT-13 CTRP2 -4.739 -1.6915 -4.7413 64.9752
MOLM-16 CTRP2 -4.5279 -2.9707 -4.5279 63.7699
MV4-11 CTRP2 -4.4908 -1.9951 -4.4913 63.4659
697 CTRP2 -4.3665 -2.1703 -4.3666 62.6725
Mino CTRP2 -4.3315 -1.1396 -4.3361 62.2806
RCH-ACV CTRP2 -4.1716 -0.7741 -4.1796 61.1847
ST486 CTRP2 -4.1193 -0.5819 -4.1301 60.8056
TALL-1 [Human adult T-ALL] CTRP2 -4.0844 -1.091 -4.0877 60.7082
SUP-T1 CTRP2 -4.0419 -0.6634 -4.0503 60.3471
OPM-2 CTRP2 -4.0191 -1.5429 -4.0198 60.3463
Peer CTRP2 -3.9582 -2.6218 -3.9582 59.9763
Daudi CTRP2 -3.9574 1.1793 -4.0548 59.1506
HuT 78 CTRP2 -3.9043 -1.4496 -3.905 59.5873
SU-DHL-6 CTRP2 -3.8526 0.5085 -3.897 58.8275
KMS-11 CTRP2 -3.8485 -0.7589 -3.8536 59.1426
Karpas-299 CTRP2 -3.708 -1.189 -3.7091 58.2807
RPMI-8226 CTRP2 -3.6956 -0.4682 -3.7033 58.1168
NU-DUL-1 CTRP2 -3.6587 -1.483 -3.659 57.9713
MHH-CALL-4 CTRP2 -3.6371 -0.508 -3.6435 57.7482
RPMI-8402 CTRP2 -3.5303 -1.4509 -3.5305 57.1197
JVM-3 CTRP2 -3.5016 -1.761 -3.5016 56.933
M-07e CTRP2 -3.4437 -2.3921 -3.4437 56.5487
PL21 CTRP2 -3.3527 -0.5382 -3.3563 55.9061
NOMO-1 CTRP2 -3.3482 0.2132 -3.3664 55.793
SUP-M2 CTRP2 -3.3363 0.622 -3.3704 55.6486
CML-T1 CTRP2 -3.3099 -1.0851 -3.3105 55.6502
WSU-DLCL2 CTRP2 -3.292 -1.5879 -3.2921 55.5377
SK-MM-2 CTRP2 -3.2614 2.864 -3.5312 54.6497
HPB-ALL CTRP2 -3.2201 0.3841 -3.2413 54.9527
F-36P CTRP2 -3.2074 -1.2453 -3.2076 54.9724
KE-97 CTRP2 -3.1977 -0.9089 -3.1984 54.902
THP-1 CTRP2 -3.1847 -0.0147 -3.1943 54.7682
Kasumi-2 CTRP2 -3.1001 -2.0933 -3.1001 54.2599
Mono-Mac-1 CTRP2 -3.0738 1.2481 -3.1363 53.9059
KE-37 CTRP2 -3.0425 -1.3085 -3.0425 53.8751
KMS-34 CTRP2 -3.0271 0.2286 -3.0398 53.7248
SET-2 CTRP2 -3.0201 0.6386 -3.0461 53.6439
NCO2 CTRP2 -3.0093 1.9197 -3.1298 53.4037
AML-193 CTRP2 -3.0018 -1.1298 -3.0019 53.6036
SU-DHL-8 CTRP2 -2.9949 0.27 -3.0081 53.5126
Granta-519 CTRP2 -2.9855 3.4301 -3.3368 52.9972
Ki-JK CTRP2 -2.9398 -0.4421 -2.9418 53.1829
BL-70 CTRP2 -2.909 -0.3701 -2.9114 52.9774
Kasumi-1 CTRP2 -2.8937 -0.2849 -2.8967 52.8745
RS4;11 CTRP2 -2.8869 0.0849 -2.9024 49.6323
NALM-6 CTRP2 -2.8362 -0.8112 -2.8365 52.5001
MM1.S CTRP2 -2.8327 0.2419 -2.8427 52.455
NU-DHL-1 CTRP2 -2.7948 -1.7429 -2.7948 52.2259
KMS-21-BM CTRP2 -2.7702 -0.6812 -2.7707 52.0602
MOLT-16 CTRP2 -2.7665 0.1136 -2.7732 52.0236
BV-173 CTRP2 -2.7626 0.2152 -2.7711 51.9955
DB CTRP2 -2.7256 0.3801 -2.7372 51.7475
OCI-AML-5 CTRP2 -2.7059 -1.9979 -2.7059 51.6333
KMS-28BM CTRP2 -2.6963 3.7354 -3.0852 51.3447
RL CTRP2 -2.6073 1.6514 -2.6807 50.9368
P12-Ichikawa CTRP2 -2.5975 -1.4093 -2.5975 50.9112
JJN-3 CTRP2 -2.5326 0.0462 -2.5362 50.4772
MOTN-1 CTRP2 -2.4746 0.2396 -2.4802 50.0924
ALL-SIL CTRP2 -2.4586 -0.9433 -2.4587 49.9863
MOLT-3 CTRP2 -2.4548 0.7098 -2.4705 49.961
Namalwa CTRP2 -2.4092 1.7433 -2.4811 49.6697
HEL 92.1.7 CTRP2 -2.4064 1.5536 -2.4632 49.6494
PF-382 CTRP2 -2.3297 0.3432 -2.3353 49.1309
MOLM-13 CTRP2 -2.272 -0.9106 -2.272 48.7427
P31/FUJ CTRP2 -2.1676 -0.1244 -2.1683 48.0483
LP-1 CTRP2 -2.0326 1.5531 -2.0747 47.2055
EM-2 CTRP2 -1.9381 -0.1845 -1.9383 46.5188
NCI-H929 CTRP2 -1.934 0.5346 -1.9385 46.5001
Ku812 CTRP2 -1.9129 0.945 -1.9252 46.3739
Hs 611.T CTRP2 -1.8418 5.3077 -2.5442 46.6271
U266B1 CTRP2 -1.8355 1.1648 -1.8531 45.87
KMS-27 CTRP2 -1.8041 1.1079 -1.8191 45.657
OCI-Ly3 CTRP2 -1.6929 1.3257 -1.7131 44.9301
KMS-20 CTRP2 -1.6471 0.8939 -1.6542 44.5975
SKM-1 CTRP2 -1.634 -0.2816 -1.634 44.4926
JURL-MK1 CTRP2 -1.6121 -0.653 -1.6121 44.3464
OCI-Ly10 CTRP2 -1.5671 3.8028 -1.8738 44.5849
Raji CTRP2 -1.5165 1.751 -1.5521 43.7951
HT CTRP2 -1.4739 0.5197 -1.4753 43.43
Karpas-422 CTRP2 -1.4581 2.1109 -1.5163 43.4587
Reh CTRP2 -1.4322 1.5561 -1.4553 43.2082
OCI-AML-2 CTRP2 -1.3728 -0.6804 -1.3728 42.7522
NB4 CTRP2 -1.3661 -0.5081 -1.3661 42.7075
KM-H2 CTRP2 -1.3511 1.5662 -1.3724 42.6653
HEL CTRP2 -1.348 1.3514 -1.3615 42.6247
SUP-B15 CTRP2 -1.2456 1.9705 -1.2849 42.0114
HDLM-2 CTRP2 -1.216 3.0051 -1.3582 42.0562
KO52 CTRP2 -1.2047 0.9773 -1.2083 41.6434
KHM-1B CTRP2 -1.1955 1.4353 -1.2085 41.6095
EHEB CTRP2 -1.1836 1.8131 -1.2117 41.5716
LAMA-84 CTRP2 -1.1435 5.049 -1.7099 42.403
MOLM-6 CTRP2 -1.0905 0.3113 -1.0906 40.8716
EB1 CTRP2 -1.0764 1.8795 -1.1046 40.8599
KCL-22 CTRP2 -1.0653 1.0857 -1.0691 40.7159
JeKo-1 CTRP2 -1.0635 0.9851 -1.0661 40.6998
AMO1 CTRP2 -1.0462 1.0892 -1.0499 40.5882
K-562 CTRP2 -1.0233 1.6925 -1.0415 40.4788
EJM CTRP2 -0.9825 2.859 -1.0904 40.4486
A3/Kawakami CTRP2 -0.9709 -0.0216 -0.9709 40.0751
L-428 CTRP2 -0.9374 1.0004 -0.9394 39.8582
L-363 CTRP2 -0.8923 2.9504 -1.0059 39.8706
KMS-18 CTRP2 -0.8777 1.5696 -0.8886 39.4881
SUP-HD1 CTRP2 -0.8749 3.0655 -1.0024 39.7924
MC116 CTRP2 -0.829 1.3039 -0.8336 39.1442
HL-60 CTRP2 -0.8252 0.9233 -0.8262 39.1075
MOLP-2 CTRP2 -0.8111 1.768 -0.827 39.0601
U-937 CTRP2 -0.7537 0.5697 -0.7538 38.6281
SU-DHL-1 CTRP2 -0.7129 1.4659 -0.7189 38.3753
Jurkat CTRP2 -0.7009 3.3657 -0.86 38.7351
GDM-1 CTRP2 -0.6483 1.9151 -0.6659 37.9818
OCI-M1 CTRP2 -0.6058 0.211 -0.6058 37.6421
SU-DHL-4 CTRP2 -0.5973 1.2051 -0.599 37.5912
SR CTRP2 -0.5692 2.5447 -0.6221 37.564
L-540 CTRP2 -0.5677 1.5275 -0.573 37.4062
SIG-M5 CTRP2 -0.559 0.1815 -0.559 37.3307
CMK CTRP2 -0.5546 1.513 -0.5595 37.3175
SU-DHL-10 CTRP2 -0.5428 0.1743 -0.5428 37.223
DEL CTRP2 -0.5225 0.2162 -0.5225 37.0876
ME1 CTRP2 -0.4624 4.0007 -0.716 37.433
KYO-1 CTRP2 -0.437 0.5509 -0.437 36.5181
RPMI-6666 CTRP2 -0.2196 1.956 -0.2293 35.1016
SUP-T11 CTRP2 -0.1135 3.4734 -0.2465 34.7886
OCI-Ly19 CTRP2 0.0351 1.772 0.0324 33.3816
HD-MY-Z CTRP2 0.2055 3.0958 0.1407 32.4522
L-1236 CTRP2 0.478 10.8411 -2.187 37.2798
Mono-Mac-6 CTRP2 1.008 15.0769 -3.6343 38.0319
MJ CTRP2 1.1732 24.9566 -8.2971 41.9947
Toledo CTRP2 2.082 16.5855 -3.349 34.8757
MHH-CALL-3 CTRP2 2.2018 27.614 -8.6889 40.3783
P3HR-1 CTRP2 3.9104 10.5312 1.3068 17.8456
REC-1 CTRP2 5.8077 7.8173 4.2308 2.1965
Karpas-620 CTRP2 6.935 8.6716 4.4612 0.4608
KMM-1 CTRP2 8.1338 22.2192 -1.1242 18.0755
⏷ Show the Full List of 149 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 -1.3041 3.0976 -1.4658 42.6685
TE15 CTRP2 -0.4034 4.1354 -0.6797 37.1115
TE-5 CTRP2 -2.2195 4.4918 -2.7391 48.6468
OE21 CTRP2 -1.1049 4.2751 -1.4732 41.8089
OE33 CTRP2 -1.0076 2.9889 -1.1337 40.6588
TE-14 CTRP2 -1.0055 4.7467 -1.4792 41.3946
TE-1 CTRP2 -0.6192 1.4999 -0.6247 37.7497
KYSE-410 CTRP2 -0.1087 1.8823 -0.1149 34.3513
TE-6 CTRP2 0.0082 4.225 -0.2517 34.3763
COLO 680N CTRP2 0.3439 4.0825 0.1416 31.9829
KYSE-70 CTRP2 0.523 3.2594 0.4586 30.3376
EC-GI-10 CTRP2 0.59 2.269 0.5855 29.6906
KYSE-510 CTRP2 0.6171 2.3395 0.6116 29.5136
KYSE-30 CTRP2 0.6424 4.5061 0.3759 30.2198
TE-4 CTRP2 0.7334 3.1006 0.6947 28.8499
KYSE-150 CTRP2 0.8026 1.9255 0.8023 28.2606
TE-9 CTRP2 1.151 3.0904 1.1298 26.0095
OE19 CTRP2 1.2816 2.4339 1.2808 25.0707
KYSE-520 CTRP2 1.3997 7.4181 0.2373 28.2755
KYSE-180 CTRP2 1.6309 5.7443 1.107 24.5828
TE-11 CTRP2 1.7359 3.8989 1.6699 22.2652
TE-10 CTRP2 1.7607 4.909 1.4969 22.793
KYSE-450 CTRP2 2.2776 4.612 2.131 18.938
KYSE-140 CTRP2 2.3814 7.3058 1.3147 21.6532
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 1.0297 7.1621 -0.0542 30.3472
HuP-T4 CTRP2 -2.1632 3.169 -2.4003 48.1906
PaTu 8988s CTRP2 -1.8916 5.8659 -2.7644 47.0197
Panc 08.13 CTRP2 -1.8914 3.1029 -2.0969 46.4794
HuP-T3 CTRP2 -0.6491 9.3495 -2.7085 41.8803
MIA PaCa-2 CTRP2 -0.389 1.5333 -0.3925 36.2096
BxPC-3 CTRP2 -0.2191 2.1156 -0.234 35.1151
Capan-1 CTRP2 -0.2179 3.1771 -0.3172 35.3754
AsPC-1 CTRP2 -0.1303 4.8328 -0.5466 35.7329
Panc 05.04 CTRP2 -0.0726 2.6414 -0.1112 34.217
Hs 766T CTRP2 -0.0334 2.7539 -0.0789 33.9785
SU.86.86 CTRP2 0.0976 1.5468 0.0969 32.9586
PaTu 8902 CTRP2 0.1452 1.6273 0.1442 32.6425
PK-59 CTRP2 0.2383 2.254 0.2286 32.0514
DAN-G CTRP2 0.3754 1.609 0.3752 31.1061
Panc 10.05 CTRP2 0.4381 3.7063 0.3094 31.1167
SNU-213 CTRP2 0.5143 5.9934 -0.1877 32.436
TCC-Pan2 CTRP2 0.5799 2.0594 0.5781 29.7493
HPAC CTRP2 0.653 3.1361 0.6075 29.4088
PSN1 CTRP2 0.7269 4.6479 0.4346 29.7474
PK-45H CTRP2 0.8992 4.9435 0.5478 28.8089
L3.3 CTRP2 0.9592 3.8856 0.8407 27.6172
QGP-1 CTRP2 1.0431 5.4476 0.5612 28.3036
Panc 04.03 CTRP2 1.0615 3.3159 1.02 26.674
SW1990 CTRP2 1.2857 5.4576 0.8225 26.6439
Panc 03.27 CTRP2 1.3365 3.5818 1.2836 24.8807
Capan-2 CTRP2 1.4228 5.736 0.8837 26.0068
KP-3 CTRP2 1.624 4.2125 1.5014 23.2059
Panc 02.03 CTRP2 1.9713 4.8242 1.7481 21.248
KP-2 CTRP2 2.1913 5.2026 1.8861 20.0798
YAPC CTRP2 2.2403 6.4372 1.5165 21.298
KP-4 CTRP2 2.4185 4.8587 2.2271 18.159
CFPAC-1 CTRP2 2.6861 5.5745 2.3086 17.0582
HPAF-II CTRP2 2.9411 5.5388 2.5972 15.2408
SNU-410 CTRP2 3.1192 10.9203 0.3802 23.0812
PaTu 8988t CTRP2 3.2764 5.7873 2.8711 13.248
SUIT-2 CTRP2 4.5685 7.2918 3.503 7.46
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 0.1017 8.644 -1.6294 37.4576
LOX-IMVI CTRP2 -3.5472 2.9159 -3.8483 56.1726
IGR-1 CTRP2 -1.4396 1.5623 -1.4632 43.2584
UACC-257 CTRP2 -1.2542 4.0602 -1.5879 42.6787
Mel Ho CTRP2 -1.0135 1.9604 -1.044 40.4488
Malme-3M CTRP2 -0.7349 5.2122 -1.3093 39.9311
MeWo CTRP2 -0.7271 2.6181 -0.7943 38.6533
WM88 CTRP2 -0.6342 4.2308 -0.9511 38.7084
G-361 CTRP2 -0.5782 1.9759 -0.5965 37.5171
RPMI-7951 CTRP2 -0.4408 0.8024 -0.4409 36.5434
Hs 852.T CTRP2 -0.3261 7.719 -1.7151 39.1487
SK-MEL-5 CTRP2 -0.2474 1.6617 -0.2514 35.268
Hs 944.T CTRP2 -0.1872 3.4201 -0.3176 35.2684
HT-144 CTRP2 -0.1471 4.2318 -0.4218 35.437
UACC-62 CTRP2 -0.1221 1.5559 -0.1239 34.4261
SK-MEL-1 CTRP2 -0.06 1.4992 -0.0611 34.0098
IGR-37 CTRP2 -0.023 3.1378 -0.1055 34.0291
COLO 829 CTRP2 0.1188 4.4356 -0.1779 33.7635
COLO 741 CTRP2 0.1994 13.0622 -3.478 40.0927
Hs 936.T CTRP2 0.2315 2.2512 0.2218 32.0966
WM115 CTRP2 0.2969 2.3532 0.2852 31.6675
WM266-4 CTRP2 0.3329 1.826 0.3316 31.3928
IPC-298 CTRP2 0.4809 4.026 0.3006 31.0036
K029AX CTRP2 0.5354 2.8663 0.5056 30.1393
SK-MEL-2 CTRP2 0.5619 1.8649 0.5613 29.8652
Mel JuSo CTRP2 0.5751 2.8065 0.5505 29.8576
Hs 294T CTRP2 0.6642 2.3244 0.6596 29.1967
COLO 792 CTRP2 0.6718 3.1177 0.6288 29.2749
COLO 800 CTRP2 0.7883 3.2858 0.7358 28.5309
A2058 CTRP2 0.7996 1.8578 0.7995 28.2797
SK-MEL-30 CTRP2 0.8115 3.7435 0.7041 28.5622
RVH-421 CTRP2 0.8532 3.3356 0.7992 28.1041
A-375 CTRP2 0.8616 2.3241 0.8591 27.8746
SK-MEL-3 CTRP2 0.9336 2.7342 0.9228 27.4227
A101D CTRP2 0.9337 1.7794 0.9337 27.3862
WM983B CTRP2 0.9499 5.0406 0.577 28.5474
SK-MEL-31 CTRP2 1.1797 3.2763 1.147 25.8568
SK-MEL-24 CTRP2 1.2702 2.7757 1.2646 25.1628
WM1799 CTRP2 1.2971 4.487 1.0925 25.6663
CJM [Human melanoma] CTRP2 1.3083 3.6687 1.2439 25.1079
Hs 940.T CTRP2 1.4095 4.0692 1.2949 24.6064
WM793 CTRP2 1.4117 4.2492 1.2653 24.702
MDA-MB-435S CTRP2 1.4204 4.0331 1.3126 24.5104
HMCB CTRP2 1.4609 4.2704 1.3145 24.374
Hs 895.T CTRP2 1.8512 6.3617 1.1283 23.8494
SK-MEL-28 CTRP2 2.3877 4.2245 2.3208 17.9266
IGR-39 CTRP2 2.5318 7.9713 1.1822 21.7347
WT2-iPS CTRP2 5.534 11.1156 2.4065 10.1403
Hs 839.T CTRP2 5.5564 8.8772 3.5362 5.417
Hs 688(A).T CTRP2 6.6379 12.1607 2.7109 7.1037
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 0.8003 4.7724 0.484 29.3434
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-DZ CTRP2 -5.6277 -1.3142 -5.6447 69.7941
CHP-212 CTRP2 -4.4676 -0.2549 -4.4943 62.7535
KP-N-SI9s CTRP2 -2.7752 1.1235 -2.8179 52.0348
NH-6 CTRP2 -2.7564 0.5278 -2.7725 51.9442
IMR-32 CTRP2 -1.7859 -0.0237 -1.7862 45.505
SK-N-BE(2) CTRP2 -1.4747 3.0881 -1.6472 43.7878
NB1 CTRP2 -1.2506 1.1721 -1.2579 41.9599
CHP-126 CTRP2 -1.2376 0.9748 -1.2415 41.8633
MHH-NB-11 CTRP2 -1.1351 1.3641 -1.145 41.1985
SiMa CTRP2 -0.6777 1.5537 -0.6849 38.1449
Kelly CTRP2 -0.6714 0.377 -0.6714 38.0793
SK-N-SH CTRP2 -0.0574 2.7281 -0.1019 34.1348
SK-N-AS CTRP2 0.4056 5.8428 -0.2566 33.0096
SK-N-FI CTRP2 0.482 1.771 0.4815 30.397
KP-N-YN CTRP2 5.5571 7.1608 4.377 1.9563
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 -4.4412 -0.0578 -4.4752 62.4998
SNU-478 CTRP2 -0.8502 1.0526 -0.8521 39.2769
HuH-28 CTRP2 -0.5457 1.5651 -0.5514 37.2605
SNU-245 CTRP2 -0.1687 2.3756 -0.1941 34.8136
SNU-1196 CTRP2 0.9136 3.2499 0.8708 27.6636
SNU-308 CTRP2 1.3109 6.5739 0.4696 27.7768
SNU-869 CTRP2 1.3309 5.8232 0.7551 26.7382
HuCC-T1 CTRP2 7.1368 8.7583 4.5115 0.2805
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-MC CTRP2 -1.6164 0.5667 -1.6189 44.382
MHH-ES-1 CTRP2 -1.1285 0.5135 -1.1289 41.1261
A-673 CTRP2 -0.6611 2.378 -0.7051 38.1477
SK-ES-1 CTRP2 -0.631 1.5495 -0.6374 37.8311
SW1353 CTRP2 -0.5876 1.355 -0.5906 37.5309
TC71 CTRP2 -0.2925 1.359 -0.2937 35.5592
U2OS CTRP2 -0.2483 3.2356 -0.3571 35.6066
SaOS-2 CTRP2 0.1307 2.6799 0.0976 32.8455
CAL-78 CTRP2 0.1729 4.5851 -0.154 33.5025
G-292 clone A141B1 CTRP2 1.1588 7.3167 0.0226 29.7028
Hs 888.T CTRP2 1.5008 8.0168 0.0968 28.4239
SJSA-1 CTRP2 2.0242 5.7893 1.2189 17.8694
MG-63 CTRP2 2.5154 7.8494 1.2192 21.6416
HOS CTRP2 2.798 6.8043 1.96 18.0643
Hs 822.T CTRP2 8.3953 32.2318 -5.8677 27.5826
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 73 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-453 CTRP2 -2.9879 -1.9634 -2.9879 53.5124
MDA-MB-157 CTRP2 -2.3253 4.3334 -2.816 49.2379
MDA-MB-361 CTRP2 -2.0625 0.5733 -2.0689 47.3576
SK-BR-3 CTRP2 -1.7409 0.2603 -1.742 45.2077
AU565 CTRP2 -1.3889 0.8666 -1.3927 42.8706
DU4475 CTRP2 -1.3069 3.1084 -1.4704 42.69
CAL-85-1 CTRP2 -1.2327 5.3776 -1.8998 43.0933
MDA-MB-231 CTRP2 -0.7509 3.8611 -1.0008 39.294
HCC1954 CTRP2 -0.7363 3.8605 -0.985 39.1967
MDA-MB-415 CTRP2 -0.6427 2.4148 -0.6887 38.0312
HCC1143 CTRP2 -0.6201 4.1156 -0.9109 38.5521
CAL-148 CTRP2 -0.5055 1.6384 -0.5121 36.996
Hs 578T CTRP2 -0.4648 2.7641 -0.5324 36.9153
EFM-192A CTRP2 -0.2716 1.4787 -0.2736 35.4224
HCC202 CTRP2 -0.1551 5.0967 -0.6444 36.0923
BT-474 CTRP2 -0.141 2.7593 -0.192 34.7123
HCC1500 CTRP2 -0.1223 2.7267 -0.1696 34.5759
CAL-120 CTRP2 -0.0828 1.6147 -0.0848 34.1647
MCF-7 CTRP2 -0.0158 4.0439 -0.2405 34.4269
T-47D CTRP2 0.0122 2.1856 0.0001 33.5655
HCC1428 CTRP2 0.0354 1.6348 0.0339 33.3754
HCC1569 CTRP2 0.239 1.9812 0.2353 32.0266
HCC1419 CTRP2 0.4812 1.7126 0.4808 30.402
ZR-75-30 CTRP2 0.5419 5.6757 -0.0552 31.9396
CAL-51 CTRP2 0.8257 4.1238 0.6551 28.6825
ZR-75-1 CTRP2 0.8257 3.1266 0.7891 28.2282
HCC1806 CTRP2 0.8855 3.0281 0.8584 27.798
HCC1395 CTRP2 0.8864 4.0228 0.7391 28.1998
HCC38 CTRP2 1.0481 3.63 0.9722 26.8801
MDA-MB-468 CTRP2 1.0593 3.3857 1.0113 26.7109
BT-549 CTRP2 1.1367 3.1373 1.1121 26.1161
JIMT-1 CTRP2 1.2269 2.8562 1.2184 25.461
CAMA-1 CTRP2 1.2863 4.5396 1.0691 25.7818
HMC-1-8 CTRP2 1.3361 3.4326 1.2977 24.8343
BT-20 CTRP2 1.9749 5.7747 1.4701 22.2419
HCC1937 CTRP2 1.9996 5.3735 1.6261 21.6001
HDQ-P1 CTRP2 2.8502 6.3805 2.1876 17.0473
Hs 578Bst CTRP2 3.0057 6.0139 2.4959 15.4369
KPL-1 CTRP2 5.9249 6.7005 4.7855 0.1865
BT 145 CTRP2 -0.3391 5.9447 -1.0992 37.9188
BT 428 CTRP2 0.1298 5.9338 -0.5859 34.9056
BT 416 CTRP2 0.4891 2.0453 0.4868 30.3558
BT 179 CTRP2 0.8885 3.7894 0.7798 28.0544
BT 224 CTRP2 1.1807 4.1655 1.0311 26.2501
BT164 CTRP2 1.3882 6.8923 0.4322 27.6663
BT 245 CTRP2 1.4558 7.1371 0.4088 27.5396
BT 187 CTRP2 1.4949 5.076 1.1621 24.8026
BT 139 CTRP2 1.907 5.2882 1.5509 22.1516
BT 112 CTRP2 1.9979 8.3631 0.4629 25.7709
BT 444 CTRP2 2.0259 5.9402 1.4684 22.0974
BT 159 CTRP2 2.0394 4.7664 1.8365 20.7227
BT 498 CTRP2 2.0854 6.4344 1.352 22.3514
BT 239 CTRP2 2.4353 8.2494 0.9603 22.8096
BT 330 CTRP2 2.5071 9.0961 0.649 23.7273
BT 228 CTRP2 3.1339 9.0578 1.2859 19.7797
BT 248 CTRP2 3.2784 10.9331 0.5242 22.1951
BT 271 CTRP2 3.4007 11.5186 0.3528 22.4885
BT 216 CTRP2 3.4759 9.9344 1.1947 19.2859
BT 333 CTRP2 3.7738 9.4198 1.7248 16.5351
BT 286 CTRP2 4.1155 11.1233 1.1999 17.7915
BT 172 CTRP2 4.6498 11.3102 1.5769 15.1931
BT 131 CTRP2 4.7142 12.9195 0.8284 17.8854
BT 359 CTRP2 4.9697 10.8764 2.0659 12.5954
BT 231 CTRP2 5.2338 13.9358 0.7555 17.1032
BT147 CTRP2 5.5845 13.3522 1.3316 14.3067
BT 232 CTRP2 5.7462 12.2998 1.9837 11.4709
BT 504 CTRP2 5.809 12.2737 2.0455 11.1129
BT 482 CTRP2 5.9045 10.0188 3.2325 6.1055
BT 320 CTRP2 5.9913 9.7676 3.4178 5.2104
BT 340 CTRP2 6.4875 11.238 3.0521 5.9577
BT 422 CTRP2 6.5212 10.7732 3.2976 4.9311
BT 440 CTRP2 6.914 8.1932 4.6292 0.1533
BT 328 CTRP2 7.4223 15.155 1.8073 9.4769
⏷ Show the Full List of 73 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 0.5509 2.6782 0.5324 29.9981
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D283 Med CTRP2 -7.2209 -6.0781 -7.2209 81.6956
KNS-60 CTRP2 -1.3106 2.2706 -1.4252 38.7692
SF268 CTRP2 -0.7395 1.7985 -0.7548 38.5816
SF539 CTRP2 -0.5006 4.6626 -0.9072 38.0782
U-87MG ATCC CTRP2 -0.343 7.1109 -1.5053 38.8058
LN-18 CTRP2 -0.3203 1.0573 -0.3206 35.7412
SNU-466 CTRP2 -0.1464 0.7812 -0.1464 34.5816
SNU-1105 CTRP2 0.1508 2.4334 0.1323 32.6633
ONS-76 CTRP2 0.2286 2.6996 0.198 32.1852
SF295 CTRP2 0.3946 2.2547 0.3876 31.001
KG-1-C CTRP2 0.4339 2.5029 0.4199 30.7625
DK-MG CTRP2 0.4596 3.7317 0.3285 30.982
Daoy CTRP2 0.4815 3.1938 0.4217 30.5984
SNU-201 CTRP2 0.5191 4.7462 0.1839 31.2582
GaMG CTRP2 0.5614 2.5735 0.5478 29.9117
42-MG-BA CTRP2 0.5638 3.4664 0.4777 30.1387
M059K CTRP2 0.6806 1.4894 0.6806 29.072
A-172 CTRP2 0.6856 2.4852 0.6776 29.0656
U-251MG CTRP2 0.6899 2.4221 0.6837 29.031
Hs 683 CTRP2 0.8091 2.9057 0.7868 28.2906
LN-229 CTRP2 0.9035 4.5065 0.66 28.4142
SW1088 CTRP2 0.9357 4.4724 0.7028 28.1643
U-118MG CTRP2 0.9581 3.6166 0.8782 27.493
SNU-626 CTRP2 0.9895 3.3821 0.9381 27.1871
YH-13 CTRP2 1.0518 4.5329 0.8154 27.4061
Becker CTRP2 1.1318 3.0194 1.1139 26.1263
TM-31 CTRP2 1.2269 3.2693 1.1968 25.5338
CAS-1 CTRP2 1.3366 4.8655 1.0454 25.7066
YKG-1 CTRP2 1.3523 3.6078 1.2975 24.7819
T98G CTRP2 1.3791 3.4686 1.3396 24.5516
SNU-738 CTRP2 1.3994 3.328 1.3722 24.3746
SF126 CTRP2 1.4522 3.2194 1.434 23.9928
GOS-3 CTRP2 1.5913 4.2822 1.4533 23.4768
SNU-489 CTRP2 1.7011 4.8692 1.4421 23.1721
KNS-81 CTRP2 1.7516 4.8957 1.4904 22.844
GMS-10 CTRP2 1.7882 4.235 1.6745 22.0814
KALS-1 CTRP2 1.9119 5.586 1.4639 22.4522
GB-1 CTRP2 1.9701 4.7304 1.7696 21.1754
SNB-75 CTRP2 2.088 7.472 0.9387 23.8505
DBTRG-05MG CTRP2 2.0918 5.2036 1.7773 20.7744
8-MG-BA CTRP2 2.1818 4.0718 2.1222 19.2731
CCF-STTG1 CTRP2 2.6438 5.4139 2.3151 17.1588
KNS-42 CTRP2 2.9648 5.265 2.711 14.7511
SW1783 CTRP2 4.1996 13.3018 0.1922 21.1981
NMC-G1 CTRP2 6.7371 8.1107 4.5906 0.2689
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RL95-2 CTRP2 -1.9888 0.7772 -1.9982 46.8728
JHUEM-3 CTRP2 -1.3308 5.7136 -2.1067 43.8145
HEC-6 CTRP2 -1.1562 1.8967 -1.1879 41.3991
HEC-1-A CTRP2 -1.1172 1.9433 -1.1502 41.1437
HEC-151 CTRP2 -0.4614 2.3601 -0.4962 36.792
KLE CTRP2 -0.3211 4.323 -0.6311 36.6703
HEC-1-B CTRP2 -0.1935 2.3822 -0.2201 34.9829
ESS-1 CTRP2 -0.0628 4.1156 -0.3059 34.7914
JHUEM-1 CTRP2 0.2161 3.2797 0.1313 32.4474
HEC-59 CTRP2 0.5889 2.8825 0.5601 29.7794
JHUEM-7 CTRP2 0.752 6.5284 -0.1152 31.4279
MFE-319 CTRP2 0.8419 2.0587 0.8413 27.9996
MFE-296 CTRP2 0.8515 5.6532 0.2889 29.8255
AN3-CA CTRP2 1.5709 6.6216 0.7305 26.094
HEC-251 CTRP2 1.6852 4.6587 1.476 23.1016
HEC-108 CTRP2 1.6983 4.1294 1.5957 22.6417
EFE-184 CTRP2 2.1275 4.8397 1.9145 20.1724
EN CTRP2 2.3952 10.1886 0.0307 26.1014
HEC-50B CTRP2 3.587 8.7591 1.8667 16.4149
JHUEM-2 CTRP2 3.7406 17.7594 -2.4298 29.3362
Ishikawa (Heraklio) 02 ER- CTRP2 1.3546 2.3685 1.3543 24.5831
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UO-31 CTRP2 -1.8779 4.1994 -2.2973 46.6033
CAL-54 CTRP2 -0.2293 3.865 -0.4372 35.7792
TUHR14TKB CTRP2 0.1801 3.0241 -3.8973 1.5733
769-P CTRP2 0.3867 2.649 0.3646 31.1037
Caki-1 CTRP2 0.5715 4.1316 0.3785 30.4452
VMRC-RCZ CTRP2 0.9196 2.7107 0.9093 27.5144
KMRC-3 CTRP2 1.059 4.5797 0.8126 27.3926
ACHN CTRP2 1.12 2.8183 1.1104 26.177
BFTC-909 CTRP2 1.1328 4.9046 0.8129 27.1573
TUHR4TKB CTRP2 1.2619 4.0424 1.1405 25.6125
VMRC-RCW CTRP2 1.3002 3.9755 1.1926 25.3097
KMRC-1 CTRP2 1.3839 3.5858 1.3333 24.5572
TUHR10TKB CTRP2 1.3841 2.8052 1.3796 24.4005
OS-RC-2 CTRP2 1.3928 6.5028 0.5838 27.1389
A-498 CTRP2 1.6226 3.4752 1.594 22.8925
RCC10RGB CTRP2 1.8337 4.2505 1.7209 21.7755
Caki-2 CTRP2 1.896 4.4605 1.7484 21.4819
SNU-1272 CTRP2 1.9865 7.6848 0.7432 24.8338
786-O CTRP2 2.005 4.1514 1.9216 20.5327
KMRC-2 CTRP2 2.2727 10.5455 -0.257 27.3278
KMRC-20 CTRP2 2.663 5.1706 2.41 16.7546
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 46 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
GP2d CTRP2 -2.2502 4.3695 -2.7428 48.8124
LS123 CTRP2 -0.9361 0.4332 -0.9362 39.8433
CCK-81 CTRP2 -0.8958 2.492 -0.9598 39.7612
T84 CTRP2 -0.7039 3.0653 -0.8202 38.6383
SNU-C5 CTRP2 -0.5281 2.6691 -0.5899 37.318
HT115 CTRP2 -0.5235 1.1195 -0.5243 37.0968
MDST8 CTRP2 -0.4425 0.7006 -0.4425 36.5547
SW48 CTRP2 -0.4219 1.4425 -0.4246 36.4264
COLO205 CTRP2 -0.4161 1.2433 -0.4172 36.3824
OUMS-23 CTRP2 -0.4114 0.0521 -0.4114 36.3473
LoVo CTRP2 -0.3915 3.9236 -0.6238 36.9117
SNU-1033 CTRP2 -0.2603 2.4668 -0.2944 35.4515
COLO201 CTRP2 -0.1937 0.3533 -0.1937 34.8969
LS411N CTRP2 -0.1686 0.9326 -0.1686 34.7299
SNU-C1 CTRP2 -0.1067 1.4558 -0.1077 34.3206
SW620 CTRP2 0.0474 1.583 0.0464 33.294
LS180 CTRP2 0.1488 2.6292 0.1197 32.7117
SNU-C2A CTRP2 0.2652 4.8872 -0.1292 33.1072
SW948 CTRP2 0.3056 1.6978 0.3049 31.5729
SNU-81 CTRP2 0.3699 1.9651 0.3676 31.1499
SNU-407 CTRP2 0.4318 4.5286 0.1414 31.6878
RCM-1 [Human ESC] CTRP2 0.4372 1.9637 0.4354 30.6997
COLO 678 CTRP2 0.4945 5.1593 0.0471 31.7783
NCI-H508 CTRP2 0.4996 2.3318 0.4925 30.3019
SNU-61 CTRP2 0.6045 3.455 0.5225 29.8543
KM12 CTRP2 0.6557 2.9532 0.6247 29.3419
C2BBe1 CTRP2 0.6829 3.9745 0.5282 29.5774
COLO 320 CTRP2 0.7063 3.8905 0.5679 29.3671
SK-CO-1 CTRP2 0.8534 2.6039 0.8452 27.9482
HCT 116 CTRP2 0.859 3.5975 0.7752 28.1661
SNU-503 CTRP2 0.9304 6.01 0.2582 29.6717
RKO CTRP2 1.1163 4.8923 0.7981 27.2603
CL-11 CTRP2 1.1955 3.6152 1.1306 25.8611
SW1417 CTRP2 1.1993 2.7431 1.1935 25.6359
HCT 8 CTRP2 1.2018 1.9877 1.2017 25.6002
SW1116 CTRP2 1.3182 2.5838 1.3165 24.8301
CW-2 CTRP2 1.4828 3.2266 1.4652 23.7869
LS513 CTRP2 1.544 2.7749 1.5419 23.3272
HT-29 CTRP2 1.5782 3.1068 1.5688 23.1237
HT-55 CTRP2 1.7205 3.4005 1.701 22.2096
DLD-1 CTRP2 1.8576 3.0683 1.8542 21.242
HCC-56 CTRP2 1.9835 3.5989 1.961 20.4676
NCI-H716 CTRP2 2.0256 7.2789 0.9535 23.9746
HCT 15 CTRP2 2.4309 3.9971 2.3954 17.5314
SNU-C4 CTRP2 2.638 4.5915 2.5265 16.4148
LS1034 CTRP2 2.8206 4.9374 2.6459 15.4235
⏷ Show the Full List of 46 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHH-1 CTRP2 -2.2291 0.8726 -2.2454 48.4724
SNU-182 CTRP2 -1.9648 3.0766 -2.1715 46.9395
HuH-6 CTRP2 -0.969 0.3223 -0.969 40.0619
Hep-G2 CTRP2 -0.4983 3.3941 -0.6469 37.3755
SNU-886 CTRP2 -0.0877 3.1949 -0.181 34.4929
JHH-2 CTRP2 0.0557 2.705 0.0178 33.3606
SNU-387 CTRP2 0.119 5.9653 -0.6079 35.004
JHH-4 CTRP2 0.2921 2.6762 0.2653 31.7497
Hep 3B2.1-7 CTRP2 0.4083 3.6945 0.2793 31.3157
SNU-423 CTRP2 0.5568 2.7928 0.5323 29.9788
Li-7 CTRP2 0.7271 4.0757 0.5576 29.3337
HLF CTRP2 0.8153 2.0127 0.8148 28.1763
JHH-5 CTRP2 0.8592 3.6189 0.7725 28.1748
HuH-1 CTRP2 1.0915 2.9446 1.0761 26.3864
PLC/PRF/5 CTRP2 1.1672 2.1548 1.1671 25.8309
SNU-398 CTRP2 1.2551 4.3187 1.0822 25.8357
SK-HEP-1 CTRP2 1.3085 3.6484 1.2465 25.0985
SNU-761 CTRP2 1.8231 3.9941 1.75 21.7085
SNU-878 CTRP2 2.4416 4.354 2.3582 17.6245
SNU-449 CTRP2 2.8771 4.8409 2.7314 14.9439
SNU-475 CTRP2 4.2234 13.7092 0.0102 21.745
JHH-6 CTRP2 4.385 6.1932 3.8579 6.4253
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 141 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H146 CTRP2 -7.5324 -1.2973 -7.5991 77.3266
COR-L279 CTRP2 -4.7469 2.7918 -5.1211 61.9949
NCI-H1341 CTRP2 -4.6664 -0.8999 -4.6782 64.2266
NCI-H810 CTRP2 -4.5044 0.4081 -4.566 62.5807
NCI-H2171 CTRP2 -4.0225 -2.2028 -4.0226 60.4012
DV-90 CTRP2 -4.0153 2.0717 -4.2182 59.0078
COR-L88 CTRP2 -3.8306 4.0339 -4.3851 57.0959
NCI-H211 CTRP2 -3.646 -2.1172 -3.646 57.8962
NCI-H1694 CTRP2 -2.8507 0.1171 -2.8585 52.5781
NCI-H1568 CTRP2 -2.7033 3.9427 -3.1376 51.3667
COR-L51 CTRP2 -2.5807 1.8602 -2.6716 50.7615
NCI-H2081 CTRP2 -2.5669 2.2755 -2.7021 50.6621
DMS 273 CTRP2 -2.5248 4.5579 -3.0885 50.3511
NCI-H1734 CTRP2 -2.0303 1.2753 -2.0573 47.1718
HOP-62 CTRP2 -1.9671 1.5151 -2.0047 46.7699
NCI-H2126 CTRP2 -1.9555 1.2523 -1.9794 46.6742
VMRC-LCD CTRP2 -1.8706 3.2891 -2.1056 46.3809
NCI-H1105 CTRP2 -1.8602 1.7543 -1.909 46.084
NCI-H1666 CTRP2 -1.755 3.3799 -1.9968 45.668
NCI-H522 CTRP2 -1.5252 3.8995 -1.8481 44.3483
HOP-92 CTRP2 -1.5025 1.3271 -1.5184 43.6574
HCC44 CTRP2 -1.4975 1.3795 -1.5151 43.6286
NCI-H1755 CTRP2 -1.4757 2.2395 -1.5457 43.5994
NCI-H2009 CTRP2 -1.4618 0.7314 -1.4648 43.354
NCI-H446 CTRP2 -1.4454 3.4292 -1.6715 43.6941
NCI-H2029 CTRP2 -1.443 3.1473 -1.6224 43.5969
Calu-3 CTRP2 -1.4402 3.2858 -1.6415 43.6181
NCI-H1915 CTRP2 -1.4336 3.0647 -1.5996 43.512
NCI-H23 CTRP2 -1.319 3.7947 -1.6032 42.9966
DMS 454 CTRP2 -1.2581 1.7512 -1.2854 42.0637
MOR/CPR CTRP2 -1.201 0.5654 -1.2017 41.6099
NCI-H1693 CTRP2 -1.1172 3.3477 -1.3043 41.514
Sq-1 CTRP2 -1.113 2.3636 -1.1763 41.1954
NCI-H1184 CTRP2 -1.101 1.43 -1.1121 40.975
RERF-LC-A1 CTRP2 -1.0491 4.6972 -1.5142 41.6471
NCI-H69 CTRP2 -0.9709 0.6661 -0.9713 40.076
NCI-H1155 CTRP2 -0.9244 1.9089 -0.9493 39.8406
NCI-H2106 CTRP2 -0.8728 0.7718 -0.8733 39.4227
HCC1833 CTRP2 -0.7203 1.6696 -0.7311 38.4399
NCI-H526 CTRP2 -0.6934 1.1074 -0.6949 38.2307
NCI-H1435 CTRP2 -0.6923 0.946 -0.693 38.2211
NCI-H1651 CTRP2 -0.6567 3.7162 -0.8716 38.5938
PC-14 CTRP2 -0.6313 0.7516 -0.6314 37.8125
NCI-H1838 CTRP2 -0.6203 3.5623 -0.8052 38.2764
NCI-H2087 CTRP2 -0.6091 3.36 -0.7605 38.1118
COLO 699 CTRP2 -0.4849 5.1748 -1.026 38.3065
HCC78 CTRP2 -0.4635 1.6086 -0.469 36.7124
LXF 289 CTRP2 -0.4229 2.5304 -0.4682 36.5687
NCI-H1581 CTRP2 -0.4135 0.9047 -0.4137 36.362
NCI-H889 CTRP2 -0.275 1.4279 -0.2766 35.444
LCLC-103H CTRP2 -0.2298 0.3049 -0.2298 35.1377
HCC827 CTRP2 -0.2262 1.5373 -0.2285 35.121
NCI-H1573 CTRP2 -0.1639 2.2951 -0.1851 34.7682
NCI-H2141 CTRP2 -0.1391 3.389 -0.2616 34.9255
HCC2108 CTRP2 -0.1227 2.4693 -0.1519 34.52
NCI-H661 CTRP2 -0.1195 1.898 -0.1261 34.4247
SBC-5 CTRP2 -0.1105 0.7598 -0.1105 34.3427
EBC-1 CTRP2 -0.1071 1.3265 -0.1076 34.3217
HCC15 CTRP2 -0.0904 2.5293 -0.1221 34.3128
NCI-H358 CTRP2 -0.0728 2.2445 -0.0891 34.1455
NCI-H2110 CTRP2 -0.0205 2.7451 -0.0648 33.8888
NCI-H520 CTRP2 0.0136 4.7038 -0.3567 34.6709
NCI-H1092 CTRP2 0.1281 3.1123 0.0572 32.9869
DMS 53 CTRP2 0.1397 1.9824 0.1349 32.6918
HCC366 CTRP2 0.1918 2.1246 0.1848 32.352
LOU-NH91 CTRP2 0.1938 2.6476 0.1652 32.4104
EPLC-272H CTRP2 0.1963 5.1994 -0.2895 33.8292
NCI-H196 CTRP2 0.2309 2.1029 0.2249 32.0884
Calu-6 CTRP2 0.2409 2.5324 0.2203 32.0702
COLO 668 CTRP2 0.274 5.1154 -0.1812 33.2354
LK2 CTRP2 0.2752 0.9835 0.2752 31.773
NCI-H1944 CTRP2 0.3067 2.1753 0.3003 31.5844
NCI-H2286 CTRP2 0.3219 5.3149 -0.1857 33.0841
SK-MES-1 CTRP2 0.3455 3.3947 0.2546 31.6072
HCC2279 CTRP2 0.3745 2.4805 0.3599 31.16
HCC1438 CTRP2 0.4251 2.8353 0.393 30.8816
HCC1195 CTRP2 0.4256 2.4141 0.4147 30.8072
NCI-H2170 CTRP2 0.4711 1.9632 0.4695 30.4732
COR-L95 CTRP2 0.4724 1.5565 0.4723 30.4599
NCI-H1623 CTRP2 0.5493 3.3827 0.4726 30.204
NCI-H2228 CTRP2 0.5806 4.8877 0.2148 30.9538
NCI-H2122 CTRP2 0.6004 3.3459 0.5311 29.8389
ChaGo-K-1 CTRP2 0.6031 4.9786 0.2153 30.8776
Lu-99 CTRP2 0.6065 3.4247 0.5283 29.8282
T3M-10 CTRP2 0.6454 4.5687 0.3647 30.2474
RERF-LC-MS CTRP2 0.6728 2.7887 0.6525 29.192
LC-1/sq-SF CTRP2 0.7142 4.5201 0.4509 29.7343
NCI-H650 CTRP2 0.7178 4.0713 0.5483 29.3956
NCI-H322 CTRP2 0.7714 6.4229 -0.0567 31.1852
IA-LM CTRP2 0.7988 3.2699 0.7484 28.454
NCI-H292 CTRP2 0.822 2.8494 0.8032 28.193
NCI-H647 CTRP2 0.8234 3.1817 0.7822 28.2591
HCC4006 CTRP2 0.8454 2.4347 0.841 27.9889
SW1271 CTRP2 0.8494 5.0872 0.4545 29.283
NCI-H1869 CTRP2 0.8597 3.7287 0.7578 28.223
LCLC-97TM1 CTRP2 0.8743 3.3913 0.8157 27.9787
NCI-H1793 CTRP2 0.8749 4.199 0.694 28.3906
HCC2935 CTRP2 0.8816 3.2699 0.8354 27.8883
HCC1171 CTRP2 0.8928 5.4791 0.3878 29.3659
A-549 CTRP2 0.8939 3.3543 0.8402 27.8316
NCI-H2342 CTRP2 0.895 2.8171 0.8799 27.6942
NCI-H841 CTRP2 0.9033 2.201 0.9022 27.5924
NCI-H2196 CTRP2 0.9821 3.7571 0.8847 27.3928
NCI-H1650 CTRP2 0.9839 3.7601 0.8862 27.3817
NCI-H1563 CTRP2 0.9985 7.0728 -0.053 30.4424
NCI-H2291 CTRP2 1.0454 6.0547 0.3677 28.9457
LUDLU-1 CTRP2 1.0532 3.1521 1.0244 26.6863
NCI-H441 CTRP2 1.0583 4.3727 0.8575 27.2403
COR-L105 CTRP2 1.1576 5.0887 0.7904 27.1564
NCI-H2023 CTRP2 1.2309 3.5283 1.1778 25.5851
NCI-H1373 CTRP2 1.2374 4.6033 1.0013 26.1729
SW1573 CTRP2 1.2952 5.5454 0.8058 26.6725
NCI-H2405 CTRP2 1.297 6.0737 0.6337 27.2618
CAL-12T CTRP2 1.3627 3.7807 1.2878 24.7814
NCI-H1339 CTRP2 1.3937 2.5651 1.3926 24.3249
DMS 114 CTRP2 1.3965 4.7075 1.15 25.1524
NCI-H838 CTRP2 1.4376 3.3093 1.4133 24.1105
HCC95 CTRP2 1.4437 3.2938 1.4206 24.0661
NCI-H2085 CTRP2 1.4461 3.9978 1.3457 24.3136
Lu-65 CTRP2 1.4696 4.8138 1.2036 24.735
NCI-H2444 CTRP2 1.4831 3.5903 1.4374 23.88
SHP-77 CTRP2 1.5155 3.8993 1.4347 23.7841
NCI-H1703 CTRP2 1.5536 4.0731 1.4493 23.6113
KNS-62 CTRP2 1.6037 5.1178 1.2691 24.0876
Calu-1 CTRP2 1.6185 4.9782 1.3235 23.8485
EKVX CTRP2 1.7543 6.7577 0.8746 25.0426
BEN CTRP2 1.8006 2.2472 1.8006 21.6109
NCI-H1355 CTRP2 1.8676 6.9309 0.9273 24.5238
NCI-H226 CTRP2 2.0483 4.082 1.9783 20.1977
RERF-LC-Ad2 CTRP2 2.1159 8.5086 0.5195 25.2457
SK-LU-1 CTRP2 2.1465 4.9752 1.9004 20.1644
NCI-H1395 CTRP2 2.2863 7.5011 1.1331 22.5882
NCI-H460 CTRP2 2.4378 5.4699 2.0731 18.6592
NCI-H1792 CTRP2 2.5445 6.5764 1.7857 19.4285
HARA [Human squamous cell lung carcinoma] CTRP2 2.8567 5.1277 2.6336 15.3581
NCI-H727 CTRP2 3.2818 7.0749 2.3452 15.2754
NCI-H2172 CTRP2 3.8089 11.2883 0.8412 19.8132
NCI-H1299 CTRP2 5.0255 9.7091 2.6963 9.8939
NCI-H2030 CTRP2 5.3377 13.0797 1.2685 15.0114
RERF-LC-Ad1 CTRP2 5.4698 20.0227 -2.0933 25.0962
Hs 888.Lu CTRP2 0.4644 7.0247 -0.6064 33.802
⏷ Show the Full List of 141 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 -2.256 0.1857 -2.2591 48.6396
P-STS CTRP2 -2.1236 1.1357 -2.147 47.7826
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 -0.1986 3.2765 -0.3095 35.2836
Rh18 CTRP2 -5.3001 -0.559 -5.3356 67.4695
KYM-1 CTRP2 -3.4612 -1.2813 -3.4616 56.6575
G-401 CTRP2 -2.4149 2.3474 -2.5494 49.7132
Rh41 CTRP2 -1.7143 0.8506 -1.7214 45.0444
HT-1080 CTRP2 -1.0981 4.2521 -1.4606 41.7551
GCT CTRP2 -0.654 2.5954 -0.7154 38.1522
A-204 CTRP2 -0.2935 3.8843 -0.5103 36.2266
RD CTRP2 0.2342 2.5436 0.2128 32.1176
TE 441.T CTRP2 0.6339 1.7416 0.6337 29.3841
TE 617.T CTRP2 0.8063 3.1726 0.765 28.3733
SK-LMS-1 CTRP2 0.8609 3.1116 0.827 27.9849
RKN CTRP2 0.9761 3.0592 0.9505 27.1896
G-402 CTRP2 1.1766 4.8444 0.8763 26.7989
TTC-709 CTRP2 1.9998 8.2497 0.5143 25.5904
Hs 729.T CTRP2 2.7959 11.2457 -0.0839 25.4169
SK-UT-1 CTRP2 2.8755 7.4798 1.7508 18.6623
BT-16 CTRP2 3.6559 12.5444 0.0826 22.787
BT-12 CTRP2 4.189 11.1914 1.2318 17.5083
Tm87-16 CTRP2 4.8029 11.0292 1.8485 13.8044
SW982 CTRP2 5.5374 8.8009 3.5595 5.3521
MES-SA CTRP2 6.3042 7.8202 4.5127 0.6864
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 0.6572 3.1714 0.6088 29.3903
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 2.8185 11.3796 -0.1269 25.4943
OVCAR-5 CTRP2 -2.4625 1.7284 -2.5355 50.0113
OV7 CTRP2 -2.2828 11.4175 -5.2815 49.362
A2780 CTRP2 -1.7991 2.0824 -1.871 45.7191
COV644 CTRP2 -1.545 5.1653 -2.1802 44.8732
COV434 CTRP2 -1.1937 1.5221 -1.2095 41.6048
OAW28 CTRP2 -1.1457 3.1971 -1.3111 41.6508
EFO-27 CTRP2 -0.9959 4.173 -1.3317 41.0576
RMG-I CTRP2 -0.7238 2.9179 -0.8228 38.7215
TOV-112D CTRP2 -0.6921 5.203 -1.26 39.6541
SNU-840 CTRP2 -0.4263 6.895 -1.517 39.1431
OC 314 CTRP2 -0.3558 1.4516 -0.3581 35.9847
TYK-nu CTRP2 -0.2664 2.4958 -0.3027 35.4994
SNU-8 CTRP2 -0.2411 2.1491 -0.2578 35.2676
IGROV-1 CTRP2 -0.1873 2.3407 -0.2114 34.9334
OVK18 CTRP2 -0.1311 2.2457 -0.149 34.5388
JHOM-1 CTRP2 0.004 2.717 -0.037 33.7149
HEY A8 CTRP2 0.2884 2.819 0.2519 31.8067
ONCO-DG-1 CTRP2 0.5324 2.4104 0.5238 30.0883
OV-90 CTRP2 0.601 3.0153 0.5631 29.7295
OVCAR-8 CTRP2 0.621 4.9913 0.2315 30.7657
JHOC-5 CTRP2 0.708 2.7908 0.6886 28.9545
MCAS CTRP2 0.726 2.5293 0.7175 28.7981
Caov-3 CTRP2 0.7429 7.7451 -0.5885 32.8274
FU-OV-1 CTRP2 0.7464 7.0022 -0.2957 31.9856
SK-OV-3 CTRP2 0.7961 2.9839 0.7685 28.3951
OVCAR-4 CTRP2 0.8649 7.7046 -0.4432 32.0265
ES2 CTRP2 1.1299 2.6317 1.1254 26.0941
OVTOKO CTRP2 1.422 3.3677 1.3928 24.2309
TOV-21G CTRP2 1.6557 4.4857 1.4824 23.1717
OAW42 CTRP2 1.8315 3.8153 1.7815 21.5737
OVISE CTRP2 2.0551 3.3274 2.0485 19.9372
EFO-21 CTRP2 2.0846 5.5877 1.6511 21.255
SNU-119 CTRP2 2.1 6.9297 1.1739 22.9629
Kuramochi CTRP2 2.1622 5.9626 1.6078 21.1856
JHOS-2 CTRP2 2.6632 6.1352 2.0835 17.9672
DOV13 CTRP2 2.9291 7.0855 1.9775 17.6428
OV56 CTRP2 3.1676 6.0786 2.6436 14.42
OVSAHO CTRP2 3.6053 8.3213 2.0931 15.4687
COV362 CTRP2 4.1666 6.7626 3.3768 8.9107
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2 -0.9653 4.9729 -1.4948 41.2544
NCI-H28 CTRP2 -0.6516 2.0539 -0.6755 38.0233
NCI-H2452 CTRP2 0.5035 3.7006 0.3804 30.6634
JL-1 CTRP2 1.0861 2.5803 1.0821 26.384
MPP 89 CTRP2 1.1414 4.4493 0.9314 26.72
IST-Mes1 CTRP2 1.1835 2.837 1.1747 25.7511
ACC-MESO-1 CTRP2 1.2267 3.8752 1.1292 25.7648
NCI-H2052 CTRP2 1.3645 4.3382 1.1968 25.0896
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H660 CTRP2 -2.7541 0.4221 -2.7672 51.9331
VCaP CTRP2 -1.1005 1.9708 -1.1345 41.0356
LNCaP clone FGC CTRP2 -0.9769 3.2938 -1.1449 40.5598
22Rv1 CTRP2 -0.842 2.0757 -0.8732 39.3111
DU145 CTRP2 0.5748 6.607 -0.3345 32.6666
PaCa-3 CTRP2 2.9003 11.1727 0.0507 24.722
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 0.6412 2.9103 0.6125 29.4307
A-253 CTRP2 4.7456 8.8792 2.2156 7.1356
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ECC10 CTRP2 -3.9346 -1.1601 -3.9367 59.7558
SNU-16 CTRP2 -3.5668 0.5547 -3.6044 57.0893
GSS CTRP2 -3.3816 -1.6368 -3.3816 56.134
Fu97 CTRP2 -3.1896 -0.2535 -3.1952 54.8192
NUGC-4 CTRP2 -3.0004 0.6182 -3.0251 53.5193
SNU-216 CTRP2 -2.2363 1.1194 -2.2621 48.5269
SNU-620 CTRP2 -0.7491 0.7726 -0.7494 38.5979
NCI-N87 CTRP2 -0.6703 0.9891 -0.6711 38.0747
SNU-1 CTRP2 -0.6365 3.7208 -0.8506 38.4604
23132/87 CTRP2 -0.5426 1.7749 -0.5531 37.2555
NUGC-3 CTRP2 -0.5316 2.2987 -0.5651 37.2545
HGC-27 CTRP2 -0.1875 3.7128 -0.3646 35.4125
SNU-5 CTRP2 -0.0996 2.2416 -0.1165 34.3259
KE-39 CTRP2 -0.0549 2.4504 -0.0806 34.0571
SNU-601 CTRP2 -0.0465 2.6546 -0.085 34.0432
GSU CTRP2 0.0103 1.4475 0.0098 33.5395
Hs 746.T CTRP2 0.3693 3.0248 0.3198 31.3111
MKN74 CTRP2 0.3801 4.5992 0.0684 32.0965
AGS CTRP2 0.3921 1.7606 0.3914 30.9966
SH-10-TC CTRP2 0.5232 2.9488 0.4871 30.2417
IM95 CTRP2 0.6323 2.3093 0.6276 29.4096
MKN7 CTRP2 0.8564 4.1161 0.6898 28.4646
KATO III CTRP2 1.1112 2.2613 1.1106 26.2055
SNU-719 CTRP2 1.2345 6.1752 0.5308 27.8061
MKN1 CTRP2 1.3211 2.6889 1.318 24.8153
ECC12 CTRP2 1.5768 3.55 1.5398 23.2261
LMSU CTRP2 1.6836 7.4664 0.517 26.4947
SNU-668 CTRP2 1.7301 5.1245 1.4052 23.2139
HuG1-N CTRP2 2.4856 6.2086 1.8656 19.2929
MKN45 CTRP2 6.145 9.5447 3.6322 4.1171
SNU-685 CTRP2 -0.2124 5.6827 -0.8787 36.9132
SNG-M CTRP2 1.0554 3.4764 0.998 26.7686
SNU-1077 CTRP2 1.268 4.1427 1.1297 25.6301
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
8505C CTRP2 -0.6861 2.3756 -0.731 38.316
8305C CTRP2 -0.491 1.8545 -0.5029 36.9162
B-CPAP CTRP2 -0.1728 1.503 -0.1744 34.763
ML-1 [Human leukemia] CTRP2 -0.115 3.8492 -0.3106 34.9908
CGTH-W-1 CTRP2 -0.0346 1.6166 -0.0363 33.8426
SW579 CTRP2 0.3376 2.4792 0.3222 31.4086
FTC-238 CTRP2 0.4783 1.4413 0.4783 30.4198
FTC-133 CTRP2 1.0126 2.2444 1.0117 26.8633
BHT-101 CTRP2 1.0816 5.6728 0.5331 28.277
TT CTRP2 1.2147 5.1118 0.8463 26.7833
TT2609-C02 CTRP2 1.5522 5.4868 1.1039 24.8328
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 29 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SCC-25 CTRP2 -4.4014 4.0381 -5.0077 59.6299
BICR 16 CTRP2 -1.3141 6.4712 -2.331 44.0213
PE/CA-PJ49 CTRP2 -0.7745 1.9135 -0.7954 38.8318
BICR 56 CTRP2 -0.7007 2.0212 -0.7244 38.3493
SCC-4 CTRP2 -0.6991 1.9617 -0.72 38.3301
SNU-1214 CTRP2 -0.1269 2.3646 -0.1504 34.5291
Detroit 562 CTRP2 -0.0701 3.0542 -0.146 34.3209
PE/CA-PJ41 (clone D2) CTRP2 0.0534 4.5589 -0.278 34.2964
BICR 6 CTRP2 0.1868 3.1193 0.1185 32.5881
YD-10B CTRP2 0.1916 4.4575 -0.1037 33.2822
SNU-899 CTRP2 0.2017 3.5596 0.0783 32.6689
BICR 18 CTRP2 0.311 5.0352 -0.1188 32.9178
SNU-1076 CTRP2 0.3633 2.6307 0.3414 31.2593
YD-8 CTRP2 0.5138 2.8454 0.4845 30.2816
HSC-3 CTRP2 0.6478 3.5894 0.551 29.6157
SNU-1066 CTRP2 0.6515 5.3406 0.1663 30.8761
SNU-46 CTRP2 0.7048 4.2997 0.4891 29.6371
CAL-33 CTRP2 0.7679 2.898 0.7446 28.5685
BICR 22 CTRP2 0.7788 3.7679 0.6654 28.8003
SCC-9 CTRP2 0.8001 4.3401 0.5841 29.0062
HSC-4 CTRP2 0.8004 3.6142 0.7104 28.5773
PE/CA-PJ15 CTRP2 0.9229 5.9765 0.2613 29.6857
SNU-1041 CTRP2 1.1824 5.8658 0.5798 27.8019
FaDu CTRP2 1.2393 3.6937 1.1676 25.5925
PE/CA-PJ34 (clone C12) CTRP2 1.2417 3.5079 1.1913 25.5039
BHY CTRP2 1.2635 4.0098 1.1476 25.5829
HSC-2 CTRP2 1.5614 2.9624 1.556 23.2223
CAL-27 CTRP2 1.6326 3.5691 1.5966 22.851
BICR 31 CTRP2 1.6888 5.6619 1.1969 24.086
⏷ Show the Full List of 29 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UM-UC-1 CTRP2 -1.9748 25.9529 -11.712 49.0712
U-BLC1 CTRP2 -1.8074 1.1128 -1.8226 45.6794
SW1710 CTRP2 -1.802 6.1462 -2.7549 46.5949
5637 CTRP2 -1.3709 0.5878 -1.3723 42.7438
TCCSUP CTRP2 -0.6872 3.0014 -0.7942 38.5026
RT-112 CTRP2 -0.415 2.4767 -0.4559 36.5024
KMBC-2 CTRP2 -0.3811 3.1735 -0.4904 36.4871
KU-19-19 CTRP2 0.0032 1.8884 -0.0016 33.6011
253J CTRP2 0.0968 2.7838 0.0547 33.101
647V CTRP2 0.2069 2.2531 0.1967 32.2621
HT-1376 CTRP2 0.7215 3.084 0.6836 28.9268
VM-CUB-1 CTRP2 0.7282 3.1299 0.6868 28.894
HT-1197 CTRP2 0.8084 1.7501 0.8083 28.2212
SCaBER CTRP2 0.8686 3.4984 0.7976 28.0589
BC-3C CTRP2 1.0828 3.6016 1.0126 26.6298
JMSU-1 CTRP2 1.1212 3.12 1.0971 26.2175
RT-4 CTRP2 1.3811 3.0018 1.3709 24.4393
T24 CTRP2 1.4945 4.9704 1.1902 24.7048
CAL-29 CTRP2 1.7229 5.7177 1.2157 23.9157
UM-UC-3 CTRP2 2.3868 6.7575 1.5463 20.7721
J82 CTRP2 2.8252 8.7768 1.1131 21.2145
639V CTRP2 3.1861 4.6875 3.1015 12.6709
BFTC-905 CTRP2 4.9747 7.689 3.6635 5.9401
253J-BV CTRP2 6.7889 8.2943 4.5431 0.3445
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 0.821 2.3816 0.8173 28.1491

References

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