General Information of Drug (ID: DMBO28J)

Drug Name
CI-976
Synonyms
CI 976; 114289-47-3; 2,2-Dimethyl-N-(2,4,6-trimethoxyphenyl)dodecanamide; CI-976; PD 128042; BRN 5831010; CHEMBL22373; UNII-8653IQ20EA; 8653IQ20EA; Dodecanamide,2,2-dimethyl-N-(2,4,6-trimethoxyphenyl)-; Dodecanamide, 2,2-dimethyl-N-(2,4,6-trimethoxyphenyl)-; 2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phenyl)-amide; C23H39NO4; ACMC-1CUXF; AC1L3UE4; SCHEMBL691688; CTK4A8660; CHEBI:95040; DTXSID00150690; MolPort-002-018-232; HMS3268D10; HMS3262L19; ZINC8022586; Tox21_500859; BN0150; BDBM50005944; AKOS022180044; LP00859; CCG-222163
Indication
Disease Entry ICD 11 Status REF
Hyperlipidaemia 5C80 Discontinued in Phase 2 [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 2 Molecular Weight (mw) 393.6
Logarithm of the Partition Coefficient (xlogp) 7.1
Rotatable Bond Count (rotbonds) 14
Hydrogen Bond Donor Count (hbonddonor) 1
Hydrogen Bond Acceptor Count (hbondacc) 4
Chemical Identifiers
Formula
C23H39NO4
IUPAC Name
2,2-dimethyl-N-(2,4,6-trimethoxyphenyl)dodecanamide
Canonical SMILES
CCCCCCCCCCC(C)(C)C(=O)NC1=C(C=C(C=C1OC)OC)OC
InChI
InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25)
InChIKey
WAFNZAURAWBNDZ-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
122327
ChEBI ID
CHEBI:95040
CAS Number
114289-47-3
TTD ID
D0D1XG

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Liver carboxylesterase (CES1) TTMF541 EST1_HUMAN Inhibitor [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Hyperlipidaemia
ICD Disease Classification 5C80
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Liver carboxylesterase (CES1) DTT CES1 3.82E-08 1.86 1.9
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 138 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 9.7936 10.8337 7.7425 0.0827
JK1 CTRP2 11.0588 13.2807 7.3497 0.3437
EB1 CTRP2 4.7463 7.1807 4.6417 22.5229
EoL-1 CTRP2 4.8477 6.5299 4.8255 21.5665
OCI-AML-3 CTRP2; CTRP1 5.0261 6.0526 5.0248 20.3089
GDM-1 CTRP2; CTRP1 5.1165 6.1015 5.1153 19.707
PL21 CTRP2; CTRP1 5.1916 6.5221 5.1813 19.2377
Pfeiffer CTRP2 5.2976 6.1917 5.2968 18.5004
SUP-M2 CTRP2 5.2996 6.0666 5.2993 18.4853
OPM-2 CTRP2 5.3019 6.4954 5.2954 18.4908
697 CTRP2 5.371 6.6531 5.3598 18.0465
GA-10 CTRP2 5.4459 6.2003 5.4456 17.5118
NOMO-1 CTRP2; CTRP1 5.6023 6.7348 5.5939 16.4979
RPMI-8226 CTRP2; CTRP1 5.6025 6.6372 5.5976 16.4845
MOLT-3 CTRP2 5.6495 7.4021 5.5768 16.4029
HH [Human lymphoma] CTRP2 5.6746 6.997 5.6528 16.0616
Toledo CTRP2 5.7067 6.6754 5.7026 15.7884
KMS-11 CTRP2; CTRP1 5.7291 7.2391 5.6854 15.7732
WSU-DLCL2 CTRP2; CTRP1 5.7348 6.4931 5.734 15.5904
CA46 CTRP2 5.7493 7.674 5.6343 15.8866
SU-DHL-5 CTRP1 5.7534 6.5063 5.7526 32.9412
THP-1 CTRP2; CTRP1 5.7719 6.5843 5.7705 15.3456
HD-MY-Z CTRP2 5.7773 6.6652 5.7746 15.3138
SET-2 CTRP2 5.8499 6.9778 5.8367 14.866
LP-1 CTRP2; CTRP1 5.851 7.1252 5.8265 14.897
A3/Kawakami CTRP2 5.8728 6.5021 5.8725 14.6705
Namalwa CTRP2 5.9786 7.0951 5.9625 14.0192
EJM CTRP2; CTRP1 6.2464 8.0471 6.0872 12.7381
DEL CTRP2 6.2467 6.8154 6.2463 12.1822
SKM-1 CTRP2; CTRP1 6.2973 7.094 6.2919 11.862
NU-DUL-1 CTRP2; CTRP1 6.311 8.7694 5.9245 13.1496
RS4;11 CTRP2 6.4177 8.543 6.1204 12.1079
NALM-6 CTRP2 6.4581 7.8696 6.3623 11.1045
Karpas-620 CTRP2 6.6116 7.2765 6.6068 9.768
JVM-2 CTRP2 6.753 11.8832 4.9827 15.7495
AML-193 CTRP2 6.8274 7.3921 6.8234 8.3292
SEM CTRP2 7.2861 8.1424 7.1951 5.5834
KMS-20 CTRP2 7.2868 9.2688 6.7402 7.3484
AMO1 CTRP2; CTRP1 7.502 8.979 7.0883 5.411
HuT 78 CTRP2 7.7264 9.5108 7.0503 5.0377
Mino CTRP2 8.0214 8.7737 7.6811 1.7717
KE-97 CTRP2; CTRP1 8.0704 9.1947 7.5125 2.3821
MOTN-1 CTRP2 8.2185 9.8172 7.3217 2.9079
U-937 CTRP2; CTRP1 8.2707 12.0749 6.237 7.3586
JeKo-1 CTRP2 8.4564 9.9318 7.4434 2.011
KYO-1 CTRP2 8.4938 9.7552 7.5545 1.5074
KMS-12-BM CTRP2 8.5538 10.2884 7.3389 2.2908
Granta-519 CTRP2 8.5803 12.5744 5.4126 4.6005
NCO2 CTRP2 8.8767 14.0512 5.7272 8.4089
OCI-AML-2 CTRP2 8.8891 11.1742 7.1415 2.6097
KM-H2 CTRP2 8.9984 11.1259 7.2348 2.1038
OCI-AML-5 CTRP2 9.045 10.5493 7.5237 0.9918
MC116 CTRP2; CTRP1 9.0946 9.9376 7.7976 0.1738
HPB-ALL CTRP2 9.1531 10.9635 7.401 1.3144
SU-DHL-4 CTRP2; CTRP1 9.1533 10.6882 7.5215 0.9023
Raji CTRP2 9.2042 11.511 7.1835 2.054
RL CTRP2 9.235 11.6127 7.1555 2.1235
Ci-1 CTRP2 9.3026 10.1741 7.793 0.1174
SIG-M5 CTRP2 9.3259 10.2192 7.7857 0.1225
Jurkat CTRP2 9.3627 11.1376 7.4386 0.9962
Reh CTRP2 9.3747 15.0917 5.5834 8.1851
BL-70 CTRP2; CTRP1 9.4044 14.2627 6.0082 6.4272
NB4 CTRP2 9.4134 10.669 7.6538 0.3501
P31/FUJ CTRP2 9.4217 10.4864 7.7261 0.1949
JVM-3 CTRP2 9.4237 12.7401 6.7493 3.4493
MOLP-2 CTRP2 9.4457 11.0632 7.5113 0.7093
SU-DHL-10 CTRP2 9.4508 10.3699 7.7791 0.1024
SU-DHL-1 CTRP2 9.4951 12.4484 6.9295 2.6723
RPMI-6666 CTRP2 9.5227 11.7564 7.2564 1.4619
SU-DHL-8 CTRP2 9.5319 10.8153 7.6482 0.3094
OCI-M1 CTRP2 9.536 10.5694 7.7404 0.1376
EM-2 CTRP2 9.5607 11.3495 7.4493 0.8116
KMS-26 CTRP2 9.6284 10.6319 7.7527 0.1001
MOLM-13 CTRP2 9.6325 11.6283 7.3688 1.0026
TF-1 CTRP2 9.647 11.451 7.4492 0.753
HT CTRP2; CTRP1 9.658 11.134 7.58 0.4058
Karpas-422 CTRP2 9.6714 10.9457 7.6566 0.2393
HEL 92.1.7 CTRP2 9.6743 10.5616 7.7931 0.051
KO52 CTRP2 9.7085 15.7082 5.5206 7.926
KE-37 CTRP2 9.7267 10.85 7.7124 0.1324
ME1 CTRP2 9.7287 11.869 7.3161 1.092
MM1.S CTRP2 9.7422 11.008 7.6617 0.2072
HL-60 CTRP2 9.7474 10.8425 7.7227 0.1142
KHM-1B CTRP2 9.7838 11.4248 7.5221 0.4816
HEL CTRP2 9.7932 11.0791 7.6558 0.2021
MOLM-16 CTRP2; CTRP1 9.8094 11.5612 7.48 0.5721
RPMI-8402 CTRP2 9.8289 11.4567 7.5293 0.4428
Ku812 CTRP2; CTRP1 9.8358 15.1425 5.8805 6.3163
PF-382 CTRP2 9.8464 11.7909 7.4054 0.748
P12-Ichikawa CTRP2 9.8663 11.4478 7.5486 0.383
CMK CTRP2 9.878 11.0926 7.6831 0.1388
Ri-1 CTRP2 9.9392 12.8595 7.0012 1.9477
L-363 CTRP2 9.9816 11.2524 7.6653 0.1404
KMS-34 CTRP2 10.0039 11.2619 7.6702 0.1294
MV4-11 CTRP2 10.0357 11.4854 7.6027 0.22
NCI-H929 CTRP2 10.0543 11.4137 7.6354 0.1651
CML-T1 CTRP2 10.0622 11.4882 7.6119 0.1981
KMS-21-BM CTRP2 10.0774 11.5769 7.5858 0.236
Peer CTRP2 10.0827 11.6399 7.565 0.2703
MOLM-6 CTRP2 10.0971 12.2856 7.323 0.8193
REC-1 CTRP2 10.1019 12.6795 7.1637 1.2788
Ki-JK CTRP2 10.1343 11.7008 7.563 0.2577
Karpas-299 CTRP2 10.1427 11.4762 7.6461 0.1321
K-562 CTRP2 10.1532 11.4829 7.6476 0.1282
MHH-CALL-4 CTRP2 10.1773 11.7185 7.5733 0.2281
SR CTRP2 10.1859 11.5837 7.6244 0.151
KMS-27 CTRP2 10.1938 11.4686 7.6672 0.0992
L-428 CTRP2 10.1997 11.8726 7.526 0.3026
RCH-ACV CTRP2 10.226 11.8965 7.5276 0.291
U266B1 CTRP2 10.2299 11.7941 7.5663 0.2248
JURL-MK1 CTRP2 10.2331 12.0427 7.4765 0.3858
SU-DHL-6 CTRP2 10.2337 11.6743 7.6102 0.1597
MOLT-16 CTRP2 10.2429 11.834 7.5569 0.2362
NU-DHL-1 CTRP2 10.2492 11.7924 7.5742 0.2074
LAMA-84 CTRP2 10.2498 12.3392 7.3705 0.6133
M-07e CTRP2 10.2766 11.9055 7.5441 0.2475
JJN-3 CTRP2 10.2897 11.856 7.5669 0.2082
P3HR-1 CTRP2; CTRP1 10.2994 11.7629 7.6034 0.1548
TALL-1 [Human adult T-ALL] CTRP2 10.3093 12.8742 7.1845 1.0703
MOLT-13 CTRP2 10.321 11.7578 7.6131 0.1385
Kasumi-2 CTRP2 10.3277 12.004 7.5283 0.259
BV-173 CTRP2 10.3337 11.8395 7.5892 0.1663
Kasumi-1 CTRP2 10.3719 11.9707 7.5571 0.2024
L-540 CTRP2 10.3863 11.8251 7.6134 0.1263
KMS-18 CTRP2 10.4078 12.2964 7.4529 0.3679
KCL-22 CTRP2 10.4352 12.406 7.4233 0.4158
HDLM-2 CTRP2 10.4508 12.0835 7.5467 0.1986
SUP-T1 CTRP2 10.5245 12.0931 7.5705 0.1516
SUP-T11 CTRP2 10.5284 12.4366 7.4494 0.3338
EHEB CTRP2 10.5314 12.3237 7.4915 0.2614
F-36P CTRP2 10.5882 12.2114 7.5525 0.1615
SUP-HD1 CTRP2 10.6711 12.4919 7.4845 0.2359
Hs 611.T CTRP2 10.6986 12.5181 7.4855 0.2277
MHH-CALL-3 CTRP2 10.9479 12.8395 7.4649 0.2005
KMM-1 CTRP2 10.9666 12.9289 7.4404 0.2293
OCI-Ly3 CTRP2 11.4994 22.3229 3.5648 12.5097
OCI-Ly10 CTRP2; CTRP1 13.6739 27.5377 2.5218 12.9154
OCI-Ly19 CTRP2 13.6965 32.0571 0.3853 18.4223
⏷ Show the Full List of 138 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 6.3129 7.1054 6.3075 11.7584
TE-5 CTRP2 5.9467 6.9572 5.9378 14.2072
TE-6 CTRP2 6.0254 6.8696 6.0217 15.7426
KYSE-410 CTRP2; CTRP1 6.4235 7.328 6.4089 11.0532
TE-4 CTRP2 7.2243 8.3524 7.0589 6.2684
KYSE-140 CTRP2; CTRP1 7.5933 8.5157 7.3876 3.9856
COLO 680N CTRP2 9.3167 10.8937 7.5182 0.7814
OE19 CTRP2 9.6599 10.8098 7.7015 0.1652
TE-10 CTRP2 9.7332 11.6523 7.4082 0.813
KYSE-30 CTRP2 10.0887 11.322 7.68 0.1023
EC-GI-10 CTRP2 10.1098 12.292 7.3263 0.8028
KYSE-150 CTRP2 10.1275 11.3942 7.669 0.1079
TE-9 CTRP2 10.2828 11.4672 7.6987 0.0594
KYSE-450 CTRP2; CTRP1 10.3201 11.7191 7.6262 0.1232
KYSE-70 CTRP2 10.3357 11.7491 7.6214 0.1259
KYSE-180 CTRP2 10.3631 11.8376 7.6006 0.1456
TE-1 CTRP2 10.3763 11.8396 7.6047 0.1382
TE-11 CTRP2 10.5021 11.9931 7.597 0.1249
KYSE-510 CTRP2 10.5718 12.2257 7.5415 0.1788
TE-14 CTRP2 10.6133 12.3786 7.503 0.2228
OE33 CTRP2 10.7008 12.4156 7.5225 0.177
OE21 CTRP2 10.8259 12.3885 7.5764 0.0982
KYSE-520 CTRP2 10.8799 13.0376 7.3683 0.3659
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 10.5543 11.8375 7.6678 0.0555
PSN1 CTRP2 5.879 7.787 5.7508 15.0704
SU.86.86 CTRP2 6.083 6.838 6.0809 13.2774
PaTu 8988s CTRP2 6.0998 7.0448 6.0912 13.1871
KP-4 CTRP2 6.1265 6.8962 6.1238 12.9898
MIA PaCa-2 CTRP2 6.2941 7.4759 6.2563 11.9933
Hs 766T CTRP2 7.0116 14.9007 3.741 19.8867
Panc 03.27 CTRP2; CTRP1 7.0359 8.3857 6.8436 7.6179
Panc 04.03 CTRP2 7.8854 10.117 6.8931 5.3525
SW1990 CTRP2 8.3766 17.6809 3.5223 17.8101
Capan-1 CTRP2 8.6415 11.6477 6.7374 4.625
KP-2 CTRP2 8.7851 10.4651 7.4087 1.6977
Panc 02.03 CTRP2 9.0844 10.5787 7.5322 0.9272
Panc 05.04 CTRP2 9.4141 11.232 7.425 0.9977
PaTu 8902 CTRP2; CTRP1 9.4937 10.9019 7.5984 0.4437
SNU-213 CTRP2 9.5329 10.9773 7.5862 0.4532
PaTu 8988t CTRP2 9.5615 10.5455 7.7584 0.1063
SUIT-2 CTRP2; CTRP1 9.795 11.5154 7.4916 0.5506
TCC-Pan2 CTRP2 9.8116 11.3311 7.5699 0.3601
YAPC CTRP2 9.8729 10.9888 7.7175 0.097
HuP-T4 CTRP2; CTRP1 9.8835 11.7263 7.4482 0.6127
DAN-G CTRP2 9.9389 11.2096 7.6645 0.1508
SNU-410 CTRP2 9.9873 12.0703 7.3585 0.7896
KP-3 CTRP2; CTRP1 10.0923 12.3515 7.2942 0.9016
HuP-T3 CTRP2 10.1122 15.3691 5.9554 5.6505
QGP-1 CTRP2; CTRP1 10.1762 25.2256 1.183 21.5492
L3.3 CTRP2 10.1794 11.4054 7.6836 0.0848
Capan-2 CTRP2; CTRP1 10.1957 15.8715 5.7723 6.2506
CFPAC-1 CTRP2; CTRP1 10.2051 11.6619 7.604 0.1746
Panc 08.13 CTRP2 10.2883 12.14 7.4627 0.3926
HPAC CTRP2; CTRP1 10.2956 11.7391 7.6103 0.1468
PK-45H CTRP2 10.3225 12.2853 7.4222 0.4628
PK-59 CTRP2 10.3312 11.885 7.5722 0.1903
Panc 10.05 CTRP2; CTRP1 10.3794 12.3043 7.4385 0.4064
HPAF-II CTRP2 10.5186 12.1288 7.5559 0.1712
BxPC-3 CTRP2 10.8899 12.6732 7.5017 0.1661
AsPC-1 CTRP2 11.3806 21.2137 4.0158 11.1447
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 13.5731 29.8446 1.3624 16.1998
WM115 CTRP2 5.4851 5.9541 5.4851 17.2494
WM266-4 CTRP2 5.5924 6.121 5.5924 16.5357
UACC-62 CTRP2 5.8825 6.848 5.8766 14.6243
A-375 CTRP2; CTRP1 5.913 6.7868 5.9095 14.4134
COLO 741 CTRP1 6.0531 8.2597 4.1916 4.5276
HT-144 CTRP2 6.1252 7.3824 6.0886 13.113
MeWo CTRP2 6.1518 7.0851 6.1427 12.8428
WT2-iPS CTRP2 6.249 6.887 6.248 12.1688
SK-MEL-5 CTRP2; CTRP1 6.3408 7.5564 6.2948 11.7108
RVH-421 CTRP2 6.3929 6.9216 6.3925 11.2089
UACC-257 CTRP2 6.4237 7.695 6.3608 11.2177
RPMI-7951 CTRP2 6.569 7.1783 6.5666 10.0436
SK-MEL-24 CTRP2 7.4171 8.5453 7.191 5.2256
Hs 688(A).T CTRP2 7.8926 8.5084 7.6932 2.0052
A2058 CTRP2 7.9878 9.0669 7.5058 2.5754
Hs 940.T CTRP2 8.0081 9.1705 7.4718 2.6764
WM88 CTRP2 8.2227 9.5619 7.4521 2.3553
COLO 792 CTRP2 8.4341 9.9948 7.3968 2.2359
IGR-39 CTRP2 8.5271 9.8408 7.536 1.5355
WM983B CTRP2 8.5549 16.4233 4.295 14.671
Hs 895.T CTRP2 8.5561 11.2084 6.8903 4.1312
A101D CTRP2 8.6078 11.2861 6.8904 4.0471
SK-MEL-3 CTRP2 8.6536 9.9961 7.5447 1.3362
SK-MEL-28 CTRP2; CTRP1 9.0125 9.9766 7.7474 0.3272
IGR-37 CTRP2 9.1073 10.2184 7.6944 0.4123
SK-MEL-2 CTRP2 9.1468 10.1019 7.7574 0.2368
SK-MEL-30 CTRP2 9.2732 10.8671 7.5074 0.8488
Mel Ho CTRP2 9.3257 11.3344 7.3334 1.3827
Hs 839.T CTRP2 9.3667 10.3656 7.7486 0.1723
Hs 936.T CTRP2; CTRP1 9.4378 10.6144 7.685 0.2702
Hs 294T CTRP2 9.494 10.7687 7.65 0.3219
WM1799 CTRP2 9.5692 11.3971 7.4337 0.8519
SK-MEL-31 CTRP2 9.6322 11.0175 7.6136 0.3418
WM793 CTRP2 9.7459 11.1776 7.6005 0.3225
HMCB CTRP2 9.8122 10.7432 7.7796 0.0466
MDA-MB-435S CTRP2 9.9448 11.1668 7.6817 0.1266
K029AX CTRP2 9.9888 11.2543 7.6673 0.1362
IPC-298 CTRP2 10.0568 11.0917 7.7468 0.0465
COLO 800 CTRP2 10.1209 11.638 7.5806 0.232
COLO 829 CTRP2 10.1385 11.9638 7.467 0.4439
Mel JuSo CTRP2 10.1749 11.4301 7.6736 0.0954
Hs 944.T CTRP2; CTRP1 10.2482 11.7236 7.5983 0.1728
G-361 CTRP2; CTRP1 10.2735 11.7646 7.5932 0.174
LOX-IMVI CTRP2 10.3711 11.6678 7.6618 0.0797
SK-MEL-1 CTRP2; CTRP1 10.3938 16.1867 5.7519 6.0705
Hs 852.T CTRP2; CTRP1 10.4067 12.1996 7.4881 0.3038
IGR-1 CTRP2 11.196 23.1668 2.9468 14.9453
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-BE(2) CTRP2 7.5206 8.2702 7.4078 4.1084
SK-N-AS CTRP2 8.3028 10.3499 7.1227 3.5917
KP-N-YN CTRP2 8.745 15.3381 4.9869 11.6363
SK-N-SH CTRP2 8.9674 15.2547 5.2004 10.3939
SiMa CTRP2 9.0575 12.8161 6.4664 5.0888
CHP-126 CTRP2 9.1959 11.9671 6.9665 2.8949
Kelly CTRP2 9.6632 11.1578 7.5731 0.4195
KP-N-SI9s CTRP2 9.76 11.2036 7.5965 0.325
MHH-NB-11 CTRP2 9.84 11.3484 7.5752 0.3375
NH-6 CTRP2 9.878 12.3344 7.1955 1.3545
NB1 CTRP2 10.0609 11.1506 7.7285 0.0599
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-245 CTRP2 7.8042 9.6745 7.0408 4.9066
SNU-869 CTRP2 8.3464 9.9174 7.3704 2.4853
HuCC-T1 CTRP2 9.582 11.286 7.4855 0.6925
SNU-478 CTRP2 9.7344 11.0545 7.6416 0.2457
SNU-308 CTRP2 10.0391 11.9848 7.416 0.61
HuH-28 CTRP2 10.058 11.2597 7.6905 0.096
SNU-1079 CTRP2 10.1378 11.8702 7.5019 0.371
SNU-1196 CTRP2 10.6081 11.9524 7.6478 0.0645
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-673 CTRP2 5.7074 6.7625 5.7006 15.7928
SaOS-2 CTRP2 7.4962 8.026 7.4564 4.0024
Hs 888.T CTRP2 7.5275 8.1997 7.4398 3.969
SJSA-1 CTRP2 7.6622 8.3729 7.5194 3.2871
Hs 822.T CTRP2 7.6689 8.1123 7.6215 2.8818
SK-ES-1 CTRP2 7.7505 9.7069 6.9761 5.2926
TC71 CTRP2 8.0684 8.8598 7.6783 1.69
MG-63 CTRP2 8.4016 17.5647 3.6007 17.4885
HOS CTRP2 8.8879 10.2109 7.5859 0.9263
SK-N-MC CTRP2 9.3627 10.3934 7.7368 0.1952
SW1353 CTRP2 10.0389 11.4646 7.6115 0.205
U2OS CTRP2 10.5577 12.4497 7.4562 0.3126
MHH-ES-1 CTRP2 10.7319 12.3798 7.5461 0.1428
CAL-78 CTRP2 10.8158 12.5839 7.5057 0.1752
G-292 clone A141B1 CTRP2 11.7958 21.8196 4.0027 10.6308
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 69 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-361 CTRP2 2.6239 9.1531 -2.6182 13.1288
DU4475 CTRP2 5.4367 6.0242 5.4366 17.5722
MCF-7 CTRP2; CTRP1 5.8907 7.4107 5.8343 14.7417
CAL-85-1 CTRP2 6.0176 7.1741 5.9969 13.7752
KPL-1 CTRP2 6.1315 6.7086 6.1312 12.9487
CAL-120 CTRP2 6.5035 7.144 6.5009 10.4803
BT-20 CTRP2 6.7708 10.0943 5.8456 12.234
MDA-MB-453 CTRP2 7.2057 8.9586 6.796 7.3346
Hs 578Bst CTRP2 7.7254 8.3219 7.6067 2.7768
HDQ-P1 CTRP2 7.8533 8.6255 7.5995 2.4813
MDA-MB-157 CTRP2 7.9561 9.1076 7.4577 2.8425
HMC-1-8 CTRP2 8.9304 10.3879 7.5312 1.0766
AU565 CTRP2 9.441 14.4822 5.9275 6.698
HCC38 CTRP2 9.4723 12.178 7.0395 2.2877
ZR-75-1 CTRP2 9.6903 10.9326 7.6689 0.2108
CAMA-1 CTRP2 9.724 11.227 7.5726 0.3923
HCC1428 CTRP2 9.7378 11.2886 7.5548 0.4265
HCC1937 CTRP2 9.8443 11.5579 7.4968 0.512
MDA-MB-231 CTRP2 9.9732 11.7405 7.4821 0.4841
HCC1419 CTRP2 10.0817 11.3472 7.6688 0.1162
SK-BR-3 CTRP2 10.1194 12.8221 7.1126 1.4244
BT-474 CTRP2 10.1224 11.4595 7.6445 0.1381
MDA-MB-415 CTRP2 10.1229 14.1255 6.5396 3.4133
CAL-148 CTRP2 10.1354 11.5442 7.6196 0.1687
Hs 578T CTRP2 10.1571 12.07 7.4343 0.5083
HCC1954 CTRP2 10.1719 11.8997 7.5048 0.3525
BT-549 CTRP2 10.2016 11.8195 7.5462 0.2662
CAL-51 CTRP2 10.2288 11.854 7.5442 0.2613
T-47D CTRP2 10.2874 12.2021 7.439 0.4416
HCC1500 CTRP2 10.3609 11.7463 7.6314 0.1106
HCC1806 CTRP2 10.3835 11.9104 7.5827 0.1644
MDA-MB-468 CTRP2 10.4086 12.542 7.3608 0.5602
HCC1395 CTRP2 10.5519 12.5591 7.4137 0.3919
HCC202 CTRP2 10.7417 12.5765 7.481 0.224
HCC1143 CTRP2 10.8879 12.908 7.4182 0.2811
BT 248 CTRP2 7.3427 8.3048 7.2036 5.3857
BT 498 CTRP2 7.7045 8.1437 7.6505 2.6699
BT 428 CTRP2 7.7238 18.8132 2.4116 22.6923
BT 444 CTRP2 8.2742 10.3496 7.1004 3.7352
BT 320 CTRP2 9.1321 10.2429 7.696 0.3932
BT 286 CTRP2 9.2341 11.1088 7.382 1.3016
BT164 CTRP2 9.3876 10.7473 7.6118 0.4677
BT 172 CTRP2 9.4026 11.1873 7.4381 0.9653
BT 228 CTRP2 9.427 11.8257 7.1721 1.852
BT 328 CTRP2 9.4339 10.8979 7.5728 0.5438
BT 340 CTRP2 9.4586 10.5963 7.7002 0.2311
BT 422 CTRP2 9.4834 10.8946 7.5967 0.4534
BT 482 CTRP2 9.5596 10.8252 7.656 0.2816
BT 271 CTRP2 9.5644 11.0032 7.59 0.4278
BT 359 CTRP2 9.5761 10.998 7.5971 0.4051
BT 179 CTRP2 9.6307 10.5785 7.772 0.0772
BT147 CTRP2 9.6596 11.2212 7.5468 0.4845
BT 112 CTRP2 9.6778 10.7229 7.739 0.1075
BT 239 CTRP2 9.683 10.97 7.6522 0.2434
BT 145 CTRP2 9.7185 11.1481 7.6002 0.3341
BT 232 CTRP2 9.7238 10.913 7.6889 0.1678
BT 504 CTRP2 9.7272 10.9079 7.692 0.1621
BT 216 CTRP2 9.7379 12.2701 7.1491 1.6289
BT 245 CTRP2 9.7487 11.3415 7.5391 0.4583
BT 330 CTRP2 9.7828 10.9396 7.7017 0.1346
BT 159 CTRP2 9.8184 11.0638 7.671 0.1707
BT 139 CTRP2 9.8244 11.1113 7.6562 0.1925
BT 224 CTRP2 9.8366 11.2499 7.6105 0.2689
BT 333 CTRP2 9.8858 11.0308 7.7076 0.1061
BT 131 CTRP2 9.8955 11.4666 7.5536 0.3601
BT 440 CTRP2 10.1366 12.3678 7.3083 0.8352
BT 187 CTRP2 10.3522 12.1515 7.4842 0.3285
BT 231 CTRP2 10.7772 12.8385 7.4005 0.3415
BT 416 CTRP2 11.9589 42.8768 -6.2033 31.1746
⏷ Show the Full List of 69 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 9.9193 10.9751 7.7386 0.0684
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LN-229 CTRP2; CTRP1 5.0823 5.7678 5.0822 19.931
KNS-60 CTRP2 5.6039 5.9723 5.6039 16.4588
GB-1 CTRP2 5.9013 6.5837 5.9007 14.4817
Hs 683 CTRP2 6.038 6.9341 6.0326 13.5879
SW1088 CTRP2 6.3211 7.0197 6.3186 11.694
GaMG CTRP2; CTRP1 6.3821 6.9062 6.3817 11.2808
Daoy CTRP2 6.4329 6.962 6.4324 10.9432
KALS-1 CTRP2 6.4974 7.3691 6.4828 10.5613
LN-18 CTRP2 6.787 7.5143 6.7738 8.629
KNS-81 CTRP2 6.8162 7.4714 6.8076 8.4189
SF268 CTRP2 7.0612 9.1431 6.567 8.6166
SF539 CTRP2 7.2763 8.4579 7.0759 6.0566
SF126 CTRP2 7.4428 7.9768 7.4094 4.335
U-251MG CTRP2 7.6701 8.2126 7.5897 2.9962
TM-31 CTRP2 8.4324 9.495 7.6377 1.2605
KNS-42 CTRP2 8.5141 9.9757 7.4625 1.8485
SNU-738 CTRP2 8.6681 10.1148 7.4983 1.4977
YKG-1 CTRP2 8.7028 10.8256 7.1826 2.7058
GOS-3 CTRP2 8.8823 11.4827 6.9894 3.2269
SNU-201 CTRP2 9.1986 10.7799 7.506 0.9146
SF295 CTRP2; CTRP1 9.1998 10.6462 7.5633 0.7311
SNU-489 CTRP2 9.2887 10.2763 7.7503 0.1953
SNU-626 CTRP2 9.4421 10.7777 7.6241 0.407
CCF-STTG1 CTRP2 9.5298 10.481 7.7693 0.0987
SNU-1105 CTRP2 9.543 10.5706 7.7426 0.1326
U-87MG ATCC CTRP2 9.6189 10.9243 7.6432 0.2846
KG-1-C CTRP2 9.6252 10.728 7.7176 0.1493
NMC-G1 CTRP2 9.6438 11.0023 7.6242 0.3141
M059K CTRP2 9.8017 11.1108 7.6476 0.2134
SNU-466 CTRP2 9.8409 10.7002 7.8036 0.0284
D283 Med CTRP2 9.8675 11.922 7.3622 0.8554
U-118MG CTRP2 9.8708 11.0937 7.68 0.1447
GMS-10 CTRP2 9.9386 10.9426 7.7562 0.0513
8-MG-BA CTRP2 9.9838 11.4054 7.6116 0.2203
Becker CTRP2 10.0057 11.4316 7.6106 0.2156
YH-13 CTRP2 10.038 11.5793 7.5695 0.2767
42-MG-BA CTRP2 10.0661 11.6316 7.5614 0.2822
DK-MG CTRP2 10.1004 11.5288 7.6119 0.1883
DBTRG-05MG CTRP2 10.3261 11.5607 7.6822 0.0677
ONS-76 CTRP2 10.5376 11.7498 7.6912 0.0422
SW1783 CTRP2 10.6585 13.2024 7.2137 0.787
SNB-75 CTRP2 10.9821 12.9422 7.4414 0.2244
A-172 CTRP2 12.9839 27.519 2.0784 15.0378
T98G CTRP2 14.7773 30.4601 1.8546 13.47
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-151 CTRP2; CTRP1 5.4773 6.5937 5.4713 17.3216
JHUEM-1 CTRP2 5.9897 7.1026 5.9735 13.9454
JHUEM-2 CTRP2; CTRP1 6.1404 7.0353 6.1334 12.9115
EFE-184 CTRP2 6.3752 6.8863 6.3749 11.3266
HEC-265 CTRP2; CTRP1 7.2773 9.5047 6.6219 7.8488
MFE-296 CTRP2 7.6448 11.652 5.9176 9.9319
HEC-1-A CTRP2 7.8514 9.304 7.2666 3.8637
HEC-108 CTRP2; CTRP1 9.6665 10.8338 7.6954 0.1731
HEC-251 CTRP2; CTRP1 9.7489 11.1335 7.6182 0.2854
JHUEM-7 CTRP2 9.7577 11.118 7.6275 0.2641
EN CTRP2 9.8604 10.8918 7.7462 0.0692
HEC-1-B CTRP2 10.0224 11.4097 7.6248 0.1886
HEC-6 CTRP2; CTRP1 10.1077 11.1963 7.7293 0.0542
ESS-1 CTRP2 10.1556 11.6019 7.6067 0.1824
MFE-319 CTRP2; CTRP1 10.2666 20.8407 3.4151 14.8534
JHUEM-3 CTRP2 10.3014 12.2017 7.4449 0.4236
RL95-2 CTRP2 10.3754 11.5631 7.6983 0.0508
HEC-50B CTRP2 10.4479 12.0683 7.551 0.1932
KLE CTRP2; CTRP1 10.4526 12.4638 7.4088 0.4383
HEC-59 CTRP2; CTRP1 10.5198 11.9588 7.6151 0.1033
AN3-CA CTRP2 10.6144 12.1107 7.5966 0.1079
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 9.4322 10.3326 7.7853 0.098
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RCC10RGB CTRP2; CTRP1 6.0506 7.2843 6.021 13.5859
VMRC-RCZ CTRP2 6.2286 8.3897 5.9664 13.2316
BFTC-909 CTRP2 6.5558 7.1366 6.5541 10.1291
TUHR14TKB CTRP2 6.6315 12.3866 4.6243 17.4515
UO-31 CTRP2 7.3284 8.3118 7.1856 5.4942
KMRC-2 CTRP2 7.6149 8.5082 7.4132 3.8279
TUHR4TKB CTRP2 8.9371 10.5573 7.459 1.3304
TUHR10TKB CTRP2 9.0996 10.276 7.6675 0.4919
OS-RC-2 CTRP2 9.4462 12.66 6.8011 3.2204
CAL-54 CTRP2 9.4713 15.6747 5.368 8.8958
Caki-1 CTRP2 9.5776 11.7012 7.3097 1.2348
Caki-2 CTRP2 9.6391 12.0763 7.18 1.6151
KMRC-20 CTRP2 9.7091 11.0718 7.625 0.2868
SNU-1272 CTRP2 9.7283 11.0053 7.6573 0.2193
A-498 CTRP2 9.9247 11.5989 7.5157 0.4299
KMRC-1 CTRP2 9.9512 11.2224 7.6646 0.1479
VMRC-RCW CTRP2; CTRP1 10.2897 16.5269 5.5231 7.0886
769-P CTRP2 10.3943 12.0253 7.5461 0.213
786-O CTRP2 10.4571 12.1112 7.5392 0.2078
ACHN CTRP2 10.5449 12.1593 7.5548 0.1672
KMRC-3 CTRP2 12.7931 31.7563 -0.0997 20.6837
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 52 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW480 CTRP1 5.0171 6.1611 5.0141 43.4715
SW620 CTRP2; CTRP1 5.6741 6.9202 5.6579 16.046
CW-2 CTRP2; CTRP1 5.7161 12.594 3.6404 23.383
C2BBe1 CTRP2; CTRP1 5.7683 7.0993 5.7421 15.4527
SNU-C5 CTRP2; CTRP1 5.7806 6.8281 5.773 15.3085
LS180 CTRP2; CTRP1 5.9452 6.7973 5.942 14.1983
SNU-C4 CTRP2; CTRP1 6.081 6.9096 6.0773 13.2959
SW948 CTRP2; CTRP1 6.0884 7.3117 6.057 13.237
HT115 CTRP2; CTRP1 6.156 7.6696 6.0761 13.0579
SNU-81 CTRP1 6.4114 7.6338 6.3567 23.9356
SW403 CTRP1 6.5611 9.1946 4.0681 4.2867
KM12 CTRP2; CTRP1 6.5932 7.5373 6.5669 9.9633
SNU-61 CTRP2; CTRP1 6.8634 11.9932 5.0339 15.286
CL-34 CTRP1 7.198 9.1684 6.6881 16.4376
COLO 320 CTRP2; CTRP1 7.2387 11.9611 5.3986 12.955
CL-40 CTRP1 7.2955 9.1727 6.7846 15.0843
NCI-H747 CTRP2 7.4143 8.4363 7.2316 5.0769
NCI-H508 CTRP2; CTRP1 7.6906 9.3101 7.1147 4.8521
COLO 678 CTRP2; CTRP1 7.9437 11.1904 6.4077 7.2698
RKO CTRP2; CTRP1 8.0911 9.6024 7.3259 3.126
SNU-503 CTRP2 8.4889 17.6689 3.6197 17.2545
SW1417 CTRP2 8.9988 11.3042 7.1516 2.4256
SNU-C1 CTRP2 9.0647 10.7738 7.4354 1.2814
MDST8 CTRP2; CTRP1 9.1253 10.4379 7.6132 0.6341
HCC-56 CTRP2 9.1839 10.2573 7.7135 0.3209
SNU-1040 CTRP1 9.2397 12.6564 6.6541 8.4129
SNU-175 CTRP2; CTRP1 9.2783 15.7571 5.1862 9.9297
HT-55 CTRP2; CTRP1 9.399 11.1492 7.4524 0.9229
DLD-1 CTRP2; CTRP1 9.4004 10.3402 7.7708 0.1261
SW1116 CTRP2 9.4279 11.0894 7.4919 0.8978
HT-29 CTRP2; CTRP1 9.5311 10.7853 7.6593 0.2862
CL-11 CTRP2 9.5491 11.6765 7.3053 1.2739
SNU-1033 CTRP2 9.5607 14.4482 6.0269 6.1237
LS1034 CTRP2 9.5836 11.427 7.4284 0.8574
HCT 116 CTRP2; CTRP1 9.6191 11.2699 7.5093 0.604
LoVo CTRP2; CTRP1 9.6323 13.1791 6.6761 3.4717
COLO205 CTRP2; CTRP1 9.6451 11.0422 7.6097 0.3448
HCT 15 CTRP2 9.6646 12.3573 7.0702 1.9735
HCT 8 CTRP2; CTRP1 9.6914 14.2387 6.2153 5.1924
COLO201 CTRP2 9.7033 11.0418 7.6338 0.2715
LS411N CTRP2; CTRP1 9.7117 10.919 7.6821 0.1821
GP2d CTRP2; CTRP1 9.7794 11.9607 7.3031 1.0935
OUMS-23 CTRP2 9.9381 10.9976 7.7375 0.0669
LS513 CTRP2; CTRP1 9.9833 11.4279 7.6032 0.2344
SK-CO-1 CTRP2; CTRP1 10.0106 11.6342 7.5381 0.3466
RCM-1 [Human ESC] CTRP2; CTRP1 10.0224 11.4485 7.6109 0.2104
SW48 CTRP2; CTRP1 10.0337 11.4989 7.5971 0.2299
LS123 CTRP2; CTRP1 10.1519 12.2071 7.3789 0.6428
SNU-407 CTRP2 10.2553 12.0359 7.488 0.3549
NCI-H716 CTRP2 10.2693 11.8973 7.5443 0.2493
CCK-81 CTRP2 10.3786 12.3532 7.4199 0.4448
SNU-C2A CTRP2; CTRP1 10.808 12.8895 7.394 0.3433
⏷ Show the Full List of 52 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHH-5 CTRP2 5.4903 6.9479 5.4639 17.3037
SNU-761 CTRP2 5.5481 6.8382 5.5325 19.4483
HuH-6 CTRP2 5.6785 7.6057 5.5714 16.3298
SNU-182 CTRP2 6.1093 7.0858 6.0989 13.13
HuH-1 CTRP2 7.9692 8.6957 7.6737 1.9126
Hep-G2 CTRP2; CTRP1 8.2269 10.0142 7.2302 3.2761
SNU-423 CTRP2 8.3022 10.0361 7.2781 2.9439
SNU-878 CTRP2 8.4919 10.1145 7.3797 2.2173
JHH-4 CTRP2 8.6151 15.7701 4.669 13.1242
JHH-1 CTRP2 8.7657 9.9458 7.6348 0.8751
HLF CTRP2 9.0175 10.3876 7.5791 0.8296
SNU-398 CTRP2; CTRP1 9.293 11.5111 7.2361 1.7617
JHH-6 CTRP2; CTRP1 9.3445 10.2055 7.7975 0.1007
SNU-886 CTRP2 9.508 12.2517 7.0271 2.2937
SNU-475 CTRP2 9.7408 11.0017 7.6635 0.2047
Hep 3B2.1-7 CTRP2 9.8254 10.9926 7.6988 0.1291
PLC/PRF/5 CTRP2 9.8554 17.6154 4.6963 10.9111
SK-HEP-1 CTRP2 9.8913 11.007 7.7178 0.0936
SNU-387 CTRP2 10.2603 19.7984 3.9211 13.1211
JHH-2 CTRP2 10.3457 14.786 6.3714 3.7865
SNU-449 CTRP2; CTRP1 10.6157 12.4478 7.4792 0.2581
Li-7 CTRP2 11.099 13.0524 7.4459 0.1944
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 154 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LC-1F CTRP2 -0.5411 19.5444 -10.2267 42.1394
NCI-H1048 CTRP1 4.3168 5.1238 4.2304 11.2533
NCI-H810 CTRP2; CTRP1 4.4524 5.7249 4.4502 24.1302
NCI-H1573 CTRP1 4.5597 5.3141 4.4281 8.1599
NCI-H1105 CTRP1 4.6668 6.1489 4.658 48.4756
VMRC-LCD CTRP1 4.6839 5.7633 4.3604 8.0406
NCI-H1666 CTRP2; CTRP1 4.6949 6.4825 4.6698 22.5933
NCI-H2342 CTRP2; CTRP1 4.7057 5.9018 4.7035 22.4444
SCLC-21H CTRP1 4.7825 5.8443 4.7814 46.811
NCI-H1963 CTRP1 4.9357 7.1264 4.8523 44.9361
NCI-H82 CTRP1 4.952 5.8812 4.5556 4.9989
NCI-H2141 CTRP1 5.0018 6.7502 4.9683 43.8347
COR-L279 CTRP1 5.0633 6.4237 4.3802 6.0986
NCI-H522 CTRP2; CTRP1 5.0832 6.743 5.0551 20.0191
COLO 668 CTRP2; CTRP1 5.1888 7.4533 5.0708 19.6256
NCI-H1836 CTRP1 5.3914 6.7946 5.3721 38.2351
NCI-H1944 CTRP2; CTRP1 5.3965 7.1164 5.3471 18.0063
NCI-H1876 CTRP1 5.4027 6.6304 5.3932 38.0105
LUDLU-1 CTRP2 5.4149 8.7821 4.9526 19.3677
ChaGo-K-1 CTRP2; CTRP1 5.4258 7.3082 5.3514 17.8973
NCI-H841 CTRP2; CTRP1 5.4313 6.3149 5.4302 17.6115
HCC44 CTRP2; CTRP1 5.5459 6.7235 5.5364 16.877
NCI-H1581 CTRP2 5.5666 6.8926 5.548 16.7697
NCI-H2087 CTRP2 5.5951 6.3992 5.5943 16.5201
NCI-H647 CTRP2 5.6307 6.4583 5.6296 16.2843
NCI-H1975 CTRP1 5.6374 7.4001 4.3282 4.5402
NCI-H2081 CTRP2; CTRP1 5.6375 7.0373 5.6096 16.2294
NCI-H211 CTRP2 5.736 7.656 5.6236 15.9657
NCI-H1155 CTRP2 5.8174 7.7634 5.689 15.4807
NCI-H2122 CTRP2; CTRP1 5.8346 7.2828 5.792 15.0676
NCI-H1355 CTRP2; CTRP1 5.835 7.2091 5.8013 15.0345
NCI-H1437 CTRP1 5.8496 8.1122 4.1303 5.5993
NCI-H1915 CTRP2; CTRP1 5.8616 6.5471 5.8611 14.7455
NCI-H2106 CTRP2 5.8663 8.1451 5.6454 15.487
NCI-H1694 CTRP2; CTRP1 5.9079 6.9213 5.8997 14.4631
NCI-H2023 CTRP2; CTRP1 5.9487 7.0306 5.9358 14.2071
NCI-H2444 CTRP2 6.0336 6.63 6.0333 15.6669
NCI-H596 CTRP1 6.0413 6.9113 6.0364 28.8579
NCI-H3255 CTRP1 6.0712 7.892 5.9329 29.3964
RERF-LC-KJ CTRP1 6.077 8.1482 4.2577 3.934
NCI-H1781 CTRP1 6.0905 7.1417 6.0751 28.2311
NCI-H1930 CTRP1 6.1238 8.4057 4.1677 4.5409
CAL-12T CTRP2; CTRP1 6.1377 7.1149 6.1264 12.9441
SK-MES-1 CTRP2 6.2043 7.4373 6.1658 12.5932
NCI-H441 CTRP2; CTRP1 6.247 7.5344 6.1976 12.3467
T3M-10 CTRP2; CTRP1 6.2519 7.0748 6.2462 12.1652
NCI-H2170 CTRP2 6.2533 7.1814 6.2422 12.1738
HCC1359 CTRP1 6.2713 7.0877 6.2653 25.5802
RERF-LC-A1 CTRP2 6.2936 6.8772 6.293 11.8707
NCI-H2228 CTRP2 6.3288 7.1962 6.3195 11.6654
SK-LU-1 CTRP2; CTRP1 6.3774 7.4411 6.3493 11.4056
Calu-3 CTRP2; CTRP1 6.388 7.2762 6.3757 11.2815
HCC33 CTRP1 6.3995 8.0036 4.4969 1.5421
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 6.4307 9.7121 5.67 13.8051
SW1271 CTRP2 6.4488 7.1185 6.4459 10.8453
NCI-H226 CTRP2 6.4744 6.9422 6.4742 10.6659
NCI-H2030 CTRP2; CTRP1 6.4779 7.7371 6.4115 10.8691
SBC-5 CTRP2 6.4894 6.8933 6.4893 10.5657
COLO 699 CTRP2; CTRP1 6.527 7.8135 6.4494 10.5819
NCI-H358 CTRP2; CTRP1 6.5349 9.6741 5.7939 13.044
NCI-H2073 CTRP1 6.5449 7.5317 6.5151 21.8452
Lu-99 CTRP2; CTRP1 6.571 6.9536 6.571 10.0223
HCC4006 CTRP1 6.6 7.6002 6.5645 21.1005
NCI-H2172 CTRP2; CTRP1 6.6729 7.4915 6.6561 9.4004
DMS 454 CTRP2 6.6991 9.1534 6.1863 11.0702
NCI-H460 CTRP2; CTRP1 6.7227 7.6094 6.6955 9.1046
HCC2935 CTRP2; CTRP1 6.731 8.2721 6.5504 9.597
DMS 53 CTRP2 6.7345 9.2509 6.1824 10.9907
COR-L23 CTRP1 6.9069 7.8053 6.8607 16.7964
HCC1195 CTRP2; CTRP1 6.9378 7.7366 6.9074 7.6841
HCC15 CTRP2; CTRP1 7.0176 8.6327 6.7327 8.089
COR-L51 CTRP2; CTRP1 7.0728 7.9882 7.004 6.9209
PC-14 CTRP2 7.1982 8.6924 6.9005 6.9462
NCI-H1793 CTRP2; CTRP1 7.3017 8.0671 7.2336 5.3966
Sq-1 CTRP2; CTRP1 7.3222 9.5766 6.6325 7.6963
HOP-62 CTRP2 7.4914 8.1578 7.4141 4.1697
HCC1171 CTRP2 7.5302 8.0889 7.4769 3.8248
DV-90 CTRP1 7.6168 9.4097 4.4757 0.4964
NCI-H1650 CTRP2 7.7212 8.6133 7.4752 3.3076
NCI-H446 CTRP2 7.7583 8.4621 7.5809 2.7911
NCI-H520 CTRP2 7.7771 10.9078 6.4044 7.623
DMS 273 CTRP2; CTRP1 7.8595 9.019 7.4143 3.2317
NCI-H1563 CTRP2 7.9966 9.8498 7.1226 4.1645
NCI-H1755 CTRP2; CTRP1 8.165 11.0252 6.6755 5.7167
NCI-H2110 CTRP2; CTRP1 8.1925 13.0988 5.6616 9.9045
NCI-H2029 CTRP2; CTRP1 8.4096 16.1299 4.3241 14.835
NCI-H1339 CTRP2 8.5208 9.9417 7.4834 1.7546
HCC827 CTRP2; CTRP1 8.8045 10.6662 7.3267 1.9921
A-549 CTRP2; CTRP1 8.811 11.6624 6.853 3.8845
KNS-62 CTRP2; CTRP1 9.0169 11.0751 7.2699 1.9471
BEN CTRP2; CTRP1 9.0824 9.9023 7.8058 0.1624
LK2 CTRP2 9.2356 9.9173 7.8581 0.0487
RERF-LC-Ad1 CTRP2 9.3259 10.0445 7.8466 0.0472
NCI-H650 CTRP2; CTRP1 9.3982 11.6299 7.2432 1.6279
NCI-H196 CTRP2 9.4446 10.7683 7.6289 0.3941
NCI-H2291 CTRP2 9.4606 11.6938 7.2498 1.5433
NCI-H69 CTRP2 9.534 11.7064 7.2843 1.3571
MOR/CPR CTRP2 9.5583 10.3502 7.8241 0.039
LC-1/sq-SF CTRP2; CTRP1 9.658 10.8572 7.6837 0.1951
NCI-H1341 CTRP2 9.7651 11.4199 7.5158 0.5063
RERF-LC-Ad2 CTRP2 9.7694 11.3465 7.5461 0.4318
NCI-H1395 CTRP2 9.7748 14.3217 6.2307 5.0202
NCI-H2009 CTRP2; CTRP1 9.8208 12.1488 7.2449 1.2434
NCI-H1435 CTRP2; CTRP1 9.8349 11.4534 7.5332 0.4311
IA-LM CTRP2 9.8421 11.0874 7.6715 0.1639
COR-L95 CTRP2 9.8647 11.2374 7.6262 0.2311
Calu-1 CTRP2 9.8809 11.6648 7.4712 0.5561
NCI-H526 CTRP2 9.8823 11.0051 7.7152 0.0979
NCI-H2286 CTRP2; CTRP1 9.887 11.5113 7.5331 0.4079
NCI-H838 CTRP2 9.898 11.3224 7.6082 0.2524
HCC1438 CTRP2 9.9414 11.4853 7.5655 0.3182
LCLC-103H CTRP2; CTRP1 9.966 11.1464 7.6965 0.1047
NCI-H2126 CTRP2; CTRP1 9.9722 11.4006 7.6088 0.2283
NCI-H1568 CTRP2; CTRP1 10.0048 12.7094 7.1014 1.5536
LCLC-97TM1 CTRP2; CTRP1 10.0097 11.9093 7.4326 0.5844
NCI-H292 CTRP2 10.0248 11.3371 7.6515 0.1495
NCI-H2196 CTRP2 10.1095 11.6687 7.565 0.2619
LOU-NH91 CTRP2 10.1104 11.6231 7.5819 0.2329
NCI-H2405 CTRP2; CTRP1 10.1124 12.2067 7.3614 0.7087
Calu-6 CTRP2; CTRP1 10.1149 11.5196 7.6206 0.172
HCC1833 CTRP2; CTRP1 10.1453 12.3227 7.3303 0.7712
NCI-H322 CTRP2 10.2088 15.6097 5.9044 5.7222
DMS 114 CTRP2 10.2224 15.7552 5.8446 5.9355
NCI-H727 CTRP2; CTRP1 10.2281 12.2227 7.4061 0.5401
HCC1588 CTRP2 10.24 11.4882 7.6768 0.083
COR-L88 CTRP2; CTRP1 10.2409 16.4486 5.5281 7.1358
NCI-H1651 CTRP2 10.2665 12.3656 7.3675 0.6121
RERF-LC-MS CTRP2 10.3179 11.8292 7.587 0.1728
NCI-H1792 CTRP2; CTRP1 10.3299 11.9373 7.5531 0.2188
NCI-H1623 CTRP2 10.3815 12.0853 7.5197 0.2577
HCC2108 CTRP2; CTRP1 10.3854 12.247 7.4622 0.3581
HCC78 CTRP2; CTRP1 10.3972 11.8857 7.5963 0.1444
NCI-H1092 CTRP2 10.4022 22.3748 2.7611 16.7474
Lu-65 CTRP2; CTRP1 10.4053 19.6807 3.2418 10.7094
HCC366 CTRP2 10.4099 12.043 7.5457 0.2098
NCI-H1734 CTRP2 10.4478 12.1063 7.5375 0.2126
NCI-H1838 CTRP2 10.4806 12.3425 7.4649 0.3213
SHP-77 CTRP2; CTRP1 10.4949 11.7624 7.6726 0.0576
NCI-H2085 CTRP2 10.5102 12.2566 7.5075 0.242
EBC-1 CTRP2; CTRP1 10.5127 12.2977 7.4937 0.2631
NCI-H1184 CTRP2 10.5146 12.151 7.5466 0.1843
EPLC-272H CTRP2; CTRP1 10.5362 12.2372 7.5242 0.2106
COR-L105 CTRP2 10.6203 12.7917 7.3548 0.4833
NCI-H1703 CTRP2 10.7005 12.3052 7.5606 0.132
NCI-H1869 CTRP2 10.7274 12.33 7.5617 0.1265
HOP-92 CTRP2 10.7417 18.0768 5.0852 8.1467
NCI-H1373 CTRP2; CTRP1 10.7808 12.2073 7.6218 0.0666
NCI-H1299 CTRP2; CTRP1 10.7913 12.3444 7.5793 0.1
NCI-H661 CTRP2; CTRP1 10.8296 12.6347 7.4931 0.1884
LXF 289 CTRP2; CTRP1 10.8391 12.7027 7.4727 0.2134
EKVX CTRP2 11.0753 13.0093 7.4522 0.1911
NCI-H23 CTRP2; CTRP1 11.3975 20.5805 4.3287 10.027
COR-L47 CTRP2 11.4015 27.8377 0.8116 20.5562
Hs 888.Lu CTRP2 8.5102 10.1477 7.3765 2.2028
⏷ Show the Full List of 154 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 9.2034 10.4862 7.6312 0.5268
P-STS CTRP2 9.4706 16.1976 5.1113 9.9142
SYO-1 CTRP2 10.1722 11.6024 7.6128 0.1699
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 9.7814 10.8796 7.7222 0.108
TE 441.T CTRP2 5.4356 6.967 5.4047 17.6831
G-401 CTRP1 5.7946 10.5308 2.9093 15.6951
Hs 729.T CTRP2 5.9483 7.0976 5.9307 14.226
MES-SA CTRP2 6.1706 6.7707 6.1701 12.6888
HT-1080 CTRP2; CTRP1 6.2538 7.0912 6.2475 12.1547
RKN CTRP2; CTRP1 6.541 8.0695 6.4028 10.7046
A-204 CTRP2 7.3891 11.3153 5.8539 10.7472
GCT CTRP2 7.7452 8.6576 7.4787 3.2342
G-402 CTRP2 7.7633 9.6058 7.0376 5.0089
BT-12 CTRP2 9.0523 9.9047 7.7925 0.2009
TTC-709 CTRP2 9.8622 11.4218 7.5567 0.3673
Tm87-16 CTRP2 9.872 11.36 7.5839 0.3075
BT-16 CTRP2 9.9506 11.1808 7.679 0.1289
Rh18 CTRP2 9.9903 11.4902 7.5833 0.2674
KYM-1 CTRP2 10.0448 11.4488 7.6194 0.1912
SW982 CTRP2 10.0984 11.3473 7.6748 0.1064
SK-LMS-1 CTRP2 10.1164 11.8934 7.4844 0.4158
Rh41 CTRP2 10.3125 11.7785 7.6027 0.153
RD CTRP2 13.477 24.8621 3.6437 9.7552
SK-UT-1 CTRP2 13.6011 25.5361 3.4088 10.3475
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 9.9429 11.2598 7.6482 0.1735
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 10.0369 11.7699 7.4979 0.42
COV434 CTRP2; CTRP1 4.7438 7.1152 4.6497 22.5036
COV318 CTRP1 5.3561 6.4444 4.5955 3.0952
RMUG-S CTRP1 5.3954 7.3412 5.3119 38.5661
OVCAR-4 CTRP2; CTRP1 5.6202 6.774 5.6105 16.383
OVCAR-8 CTRP2; CTRP1 5.6234 7.0944 5.59 16.442
A2780 CTRP2; CTRP1 5.7647 6.6782 5.7615 15.3993
RMG-I CTRP2; CTRP1 5.9276 7.5754 5.8467 14.581
JHOS-4 CTRP1 5.958 7.9101 4.2947 3.9333
SNU-119 CTRP2 5.9907 6.8309 5.9874 13.8958
Caov-3 CTRP2; CTRP1 5.9929 7.2624 5.9624 13.9728
TYK-nu CTRP2; CTRP1 6.096 6.8303 6.0942 13.19
OVKATE CTRP1 6.1887 7.0235 6.1832 26.7572
OVK18 CTRP2; CTRP1 6.3378 7.6206 6.2812 11.7675
COV362 CTRP2; CTRP1 6.3753 7.3479 6.3568 11.3871
TOV-112D CTRP2 6.4049 7.2776 6.3933 11.1666
OAW42 CTRP2; CTRP1 6.4274 6.9348 6.427 10.9795
OVMANA CTRP1 6.5495 8.3932 4.4091 1.8734
IGROV-1 CTRP2; CTRP1 6.8246 7.7625 6.7814 8.4819
EFO-27 CTRP2; CTRP1 7.0091 9.8774 6.1832 10.2824
JHOC-5 CTRP2; CTRP1 7.0251 7.7137 7.004 7.0713
OVCAR-5 CTRP2 7.3033 8.0177 7.248 5.3403
OV7 CTRP2; CTRP1 7.9559 9.8141 7.1055 4.3183
OC 314 CTRP2 8.0075 9.3577 7.3777 3.0722
SNU-840 CTRP2; CTRP1 8.679 10.6954 7.2291 2.5526
TOV-21G CTRP2 8.757 10.0702 7.5737 1.1057
SNU-8 CTRP2 9.5333 10.6149 7.723 0.1657
ES2 CTRP2 9.592 10.6403 7.7362 0.13
DOV13 CTRP2 9.6265 11.6816 7.3433 1.0868
OV56 CTRP2 9.6966 10.8834 7.6891 0.1749
JHOM-1 CTRP2; CTRP1 9.802 12.5609 7.0568 1.8856
FU-OV-1 CTRP2 9.8552 11.6911 7.4493 0.6255
SK-OV-3 CTRP2; CTRP1 9.8694 11.6784 7.4607 0.5884
OVISE CTRP2 9.937 11.1837 7.6729 0.1397
ONCO-DG-1 CTRP2 10.0744 11.4596 7.6267 0.1729
HEY A8 CTRP2; CTRP1 10.092 11.2548 7.7042 0.0773
JHOS-2 CTRP2 10.1734 11.7874 7.5468 0.2738
EFO-21 CTRP2; CTRP1 10.2533 11.6807 7.6152 0.149
MCAS CTRP2 10.3716 11.8689 7.5928 0.1538
OV-90 CTRP2; CTRP1 10.4321 12.3099 7.4577 0.3505
OAW28 CTRP2 10.5362 12.7901 7.3202 0.5943
OVSAHO CTRP2 10.5462 12.0568 7.5909 0.1244
Kuramochi CTRP2 10.5629 12.3203 7.5047 0.2327
OVTOKO CTRP2 10.7023 12.4874 7.4978 0.2095
COV644 CTRP2; CTRP1 12.714 23.0705 4.002 9.4842
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H2452 CTRP2 6.6464 8.2222 6.4738 10.1292
MPP 89 CTRP2 7.9767 10.2566 6.9024 5.1279
NCI-H2052 CTRP2; CTRP1 10.3607 12.0275 7.5325 0.2428
MSTO-211H CTRP2; CTRP1 10.542 12.3159 7.4984 0.2478
JL-1 CTRP2 10.543 11.7095 7.7063 0.0338
IST-Mes1 CTRP2 10.5927 12.2455 7.5423 0.1736
NCI-H28 CTRP2; CTRP1 10.6995 12.3969 7.5285 0.1696
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PaCa-3 CTRP2; CTRP1 6.2943 8.5586 5.9815 12.9837
DU145 CTRP2 7.5441 11.0547 6.1235 9.2898
VCaP CTRP2 8.2194 9.6896 7.386 2.6376
22Rv1 CTRP2 10.7269 12.4955 7.5041 0.1955
LNCaP clone FGC CTRP2 10.9114 12.5849 7.5397 0.1212
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 CTRP2 6.173 7.1972 6.1576 12.723
YD-15 CTRP2 9.4136 10.4978 7.7186 0.2118
Cancer Drug Sensitivity Data Curated from 30 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
AGS CTRP2; CTRP1 5.7485 6.8759 5.7377 15.5328
Hs 746.T CTRP2 5.9999 6.8116 5.9972 13.8324
MKN1 CTRP2 6.4561 7.034 6.455 10.7907
HGC-27 CTRP2 7.2017 8.2213 7.0787 6.261
ECC10 CTRP2 7.5514 8.1494 7.4821 3.7424
NUGC-4 CTRP2; CTRP1 7.8935 8.9891 7.4602 2.9659
HuG1-N CTRP2 8.198 9.6692 7.3792 2.7039
LMSU CTRP2 8.7332 16.1627 4.567 13.3039
KE-39 CTRP2 8.7839 13.6938 5.8336 8.1286
KATO III CTRP2 9.0211 11.5273 7.0608 2.7523
GSU CTRP2 9.0591 9.6499 7.887 0.0458
NCI-N87 CTRP2 9.3672 12.1744 6.9775 2.6409
ECC12 CTRP2 9.4504 10.7566 7.636 0.3742
MKN45 CTRP2 9.4621 10.3052 7.8057 0.0682
SH-10-TC CTRP2; CTRP1 9.5658 11.0436 7.5748 0.4643
GSS CTRP2 9.8901 11.1859 7.6546 0.1773
SNU-620 CTRP2 9.9943 11.0926 7.725 0.071
NUGC-3 CTRP2 10.0099 11.6236 7.5418 0.3395
Fu97 CTRP2; CTRP1 10.0507 11.691 7.5333 0.3412
SNU-668 CTRP2 10.0507 10.9902 7.7783 0.028
SNU-216 CTRP2 10.2602 11.8498 7.5579 0.2299
MKN74 CTRP2; CTRP1 10.2624 12.0416 7.4888 0.3508
SNU-719 CTRP2 10.3392 12.2385 7.4467 0.4054
23132/87 CTRP2 10.3788 11.6841 7.6589 0.0812
SNU-601 CTRP2 10.6081 19.4773 4.3234 11.1531
MKN7 CTRP2; CTRP1 10.8715 17.3591 5.5065 6.3976
IM95 CTRP2 13.3627 28.8263 1.7078 15.5618
SNU-685 CTRP2 10.2198 11.4627 7.6784 0.0843
SNU-1077 CTRP2 10.2718 11.7222 7.6075 0.1552
SNG-M CTRP2; CTRP1 10.3904 11.8091 7.6204 0.1178
⏷ Show the Full List of 30 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW579 CTRP2 6.2493 6.8364 6.2487 12.1652
8505C CTRP2 6.3162 6.9945 6.3141 11.7252
ML-1 [Human leukemia] CTRP2 6.5662 7.1117 6.5651 10.0578
TT2609-C02 CTRP2 7.1105 10.0613 6.1972 9.9775
CAL-62 CTRP2 7.6723 8.3791 7.5275 3.2277
TT CTRP2 7.9316 8.8224 7.577 2.3967
CGTH-W-1 CTRP2 9.6096 11.9475 7.2202 1.5051
FTC-133 CTRP2 9.6796 11.04 7.6248 0.2984
8305C CTRP2 9.7888 11.2279 7.5993 0.3082
FTC-238 CTRP2 9.9989 11.0802 7.7307 0.0653
BHT-101 CTRP2 10.0028 11.3242 7.6479 0.1595
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-2 CTRP2; CTRP1 4.9501 5.9391 4.9492 20.8134
HSC-4 CTRP2 5.7822 6.3519 5.7821 15.2727
FaDu CTRP2 6.0127 7.2428 5.9854 13.8301
PE/CA-PJ15 CTRP2 6.0224 7.1944 6.0002 13.7485
PE/CA-PJ41 (clone D2) CTRP2 6.3471 6.879 6.3467 11.5138
SCC-9 CTRP2; CTRP1 7.0466 8.2313 6.9068 7.352
SCC-4 CTRP2 7.5826 8.0888 7.5341 3.4593
YD-8 CTRP2 7.6403 8.6082 7.3956 3.8312
BICR 22 CTRP2 8.0244 8.8012 7.67 1.812
PE/CA-PJ34 (clone C12) CTRP2 8.1408 12.4344 5.9511 8.798
CAL-27 CTRP2 8.5736 10.0704 7.4575 1.7845
BICR 18 CTRP2 8.644 10.309 7.3907 1.9535
BHY CTRP2 9.327 11.3041 7.3474 1.3327
BICR 31 CTRP2 9.418 11.706 7.2205 1.6883
BICR 56 CTRP2 9.5529 13.9802 6.2462 5.2598
SNU-1066 CTRP2 9.5702 10.9964 7.5952 0.4124
YD-10B CTRP2 9.6207 11.0214 7.6073 0.3608
BICR 6 CTRP2 9.6983 10.9804 7.6545 0.2341
SNU-46 CTRP2 9.7638 11.5096 7.4799 0.5977
SNU-1076 CTRP2 9.8383 11.0318 7.6898 0.1385
SNU-899 CTRP2 9.8726 11.1678 7.6544 0.1822
HSC-3 CTRP2 9.8784 11.3437 7.5926 0.2883
BICR 16 CTRP2 10.163 11.5216 7.6377 0.1386
CAL-33 CTRP2 10.3128 12.0423 7.5086 0.2973
SCC-25 CTRP2 10.3267 12.0831 7.4992 0.3096
SNU-1041 CTRP2 10.5688 12.2784 7.5219 0.2063
Detroit 562 CTRP2 10.6699 12.4833 7.4871 0.2323
SNU-1214 CTRP2 10.83 12.7207 7.463 0.2289
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
BC-3C CTRP2 5.9568 8.8398 5.5176 15.693
TCCSUP CTRP2 6.2538 6.8697 6.253 12.1362
T24 CTRP2 6.4449 7.6118 6.3978 11.0217
UM-UC-3 CTRP2; CTRP1 6.5549 7.8772 6.4658 10.4369
U-BLC1 CTRP2 7.4443 8.0434 7.3954 4.3799
647V CTRP2 7.8968 8.556 7.6746 2.0714
CAL-29 CTRP2 7.9165 8.7696 7.5892 2.3792
253J-BV CTRP2 8.4205 10.4206 7.1776 3.1631
KMBC-2 CTRP2; CTRP1 8.67 13.6286 5.7785 8.5517
JMSU-1 CTRP2 9.4741 10.8593 7.6064 0.4341
639V CTRP2 9.4891 10.306 7.815 0.0548
KU-19-19 CTRP2 9.5746 10.7804 7.6788 0.2309
253J CTRP2 9.5935 10.8541 7.6591 0.2623
UM-UC-1 CTRP2 9.6378 15.2914 5.6731 7.4246
SCaBER CTRP2 9.7753 11.0468 7.6606 0.1993
RT-112 CTRP2 10.1535 11.4089 7.6733 0.099
HT-1376 CTRP2; CTRP1 10.1832 11.9362 7.4959 0.3659
SW1710 CTRP2 10.258 11.8538 7.5556 0.2341
5637 CTRP2; CTRP1 10.3522 12.1644 7.4794 0.3373
RT-4 CTRP2; CTRP1 10.4483 11.9217 7.6023 0.1281
VM-CUB-1 CTRP2 11.1685 12.5735 7.6311 0.0337
J82 CTRP2 15.0782 29.7012 2.3926 11.6789
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 9.5406 10.4645 7.7789 0.0848

References

1 Trusted, scientifically sound profiles of drug programs, clinical trials, safety reports, and company deals, written by scientists. Springer. 2015. Adis Insight (drug id 800001196)
2 Acyl-coenzyme A:cholesterol-acyltransferase (ACAT) inhibitors modulate monocyte adhesion to aortic endothelial cells. Atherosclerosis. 1995 Jan 6;112(1):7-17.