General Information of Drug (ID: DMCRXAM)

Drug Name
PF3845
Synonyms PF-3845; PF 3845
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 456.5
Logarithm of the Partition Coefficient (xlogp) 4.4
Rotatable Bond Count (rotbonds) 5
Hydrogen Bond Donor Count (hbonddonor) 1
Hydrogen Bond Acceptor Count (hbondacc) 7
Chemical Identifiers
Formula
C24H23F3N4O2
IUPAC Name
N-pyridin-3-yl-4-[[3-[5-(trifluoromethyl)pyridin-2-yl]oxyphenyl]methyl]piperidine-1-carboxamide
Canonical SMILES
C1CN(CCC1CC2=CC(=CC=C2)OC3=NC=C(C=C3)C(F)(F)F)C(=O)NC4=CN=CC=C4
InChI
InChI=1S/C24H23F3N4O2/c25-24(26,27)19-6-7-22(29-15-19)33-21-5-1-3-18(14-21)13-17-8-11-31(12-9-17)23(32)30-20-4-2-10-28-16-20/h1-7,10,14-17H,8-9,11-13H2,(H,30,32)
InChIKey
NBOJHRYUGLRASX-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
25154867
ChEBI ID
CHEBI:95030
CAS Number
1196109-52-0
TTD ID
D0E9UX
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Fatty acid amide hydrolase (FAAH) TTDP1UC NOUNIPROTAC Inhibitor [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Discovery agent
ICD Disease Classification N.A.
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Fatty acid amide hydrolase (FAAH) DTT NO-GeName 2.65E-01 0.02 0.1
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U2OS CTRP1 6.4605 8.7521 4.2081 3.4485
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MCF-7 CTRP1 5.4104 8.39 3.6764 10.9944
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LN-229 CTRP1 4.1749 7.9968 2.8009 23.6047
SF295 CTRP1 5.6549 8.4401 3.8357 8.7441
GaMG CTRP1 6.0927 8.1603 4.2616 3.8643
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-151 CTRP1 3.0576 6.1291 2.5117 32.3162
HEC-59 CTRP1 4.5195 6.24 3.975 12.254
HEC-265 CTRP1 5.4144 7.8741 3.9355 8.7233
HEC-6 CTRP1 5.6931 7.1402 4.4873 3.0417
MFE-319 CTRP1 5.7267 10.4123 2.9163 15.8925
JHUEM-2 CTRP1 5.9412 9.9508 3.3036 12.1779
HEC-108 CTRP1 6.1076 11.2616 2.7822 15.4993
HEC-251 CTRP1 6.2619 8.4281 4.2398 3.6392
KLE CTRP1 6.2849 9.0785 3.9557 5.8384
Ishikawa (Heraklio) 02 ER- CTRP1 6.0329 9.304 3.683 8.8022
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NU-DUL-1 CTRP1 1.0032 51.9505 -21.8469 50.598
LP-1 CTRP1 3.35 10.1669 0.9708 37.1884
SU-DHL-5 CTRP1 3.3576 4.0003 3.3558 24.3172
Ku812 CTRP1 3.3733 5.7916 2.9778 27.0306
PL21 CTRP1 3.5739 6.2534 3.007 25.5412
U-937 CTRP1 3.6795 6.078 3.1904 23.497
THP-1 CTRP1 3.7193 6.0156 3.2578 22.7278
KE-97 CTRP1 3.9365 5.0476 3.8371 16.7776
BL-70 CTRP1 4.1135 5.5444 3.8633 15.4614
WSU-DLCL2 CTRP1 4.331 5.0126 4.2767 10.8029
OCI-AML-3 CTRP1 4.4479 6.1097 3.9658 12.7096
SKM-1 CTRP1 4.461 8.6519 2.7427 22.5572
MOLM-16 CTRP1 4.5076 6.5579 3.8118 13.7374
SU-DHL-4 CTRP1 4.5825 5.5187 4.3682 8.5267
MC116 CTRP1 4.7354 5.8504 4.3693 7.6974
P3HR-1 CTRP1 4.7778 5.477 4.5861 5.5876
GDM-1 CTRP1 4.934 7.7783 3.5938 13.6402
KMS-11 CTRP1 5.0764 8.3576 3.4241 14.4694
RPMI-8226 CTRP1 5.0852 9.5441 2.8381 19.0127
AMO1 CTRP1 5.1544 6.2986 4.5167 4.5052
EJM CTRP1 5.3203 8.4552 3.5734 12.2206
NOMO-1 CTRP1 5.622 8.2975 3.8815 8.4613
OCI-Ly10 CTRP1 6.2051 8.3179 4.2565 3.639
HT CTRP1 6.3373 9.2188 3.9232 5.9627
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RCC10RGB CTRP1 2.9391 5.2091 2.7028 31.9361
VMRC-RCW CTRP1 6.276 10.7406 3.1574 12.204
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW620 CTRP1 2.5201 4.1176 2.4771 36.5578
SW480 CTRP1 2.7117 5.4539 2.3795 35.6386
C2BBe1 CTRP1 3.622 5.5215 3.3439 22.6507
CW-2 CTRP1 3.8041 5.658 3.4894 20.3689
SNU-175 CTRP1 3.8845 5.432 3.659 18.5137
SW48 CTRP1 4.1974 8.0382 2.8019 23.4777
SNU-C4 CTRP1 4.3057 5.526 4.0748 12.5793
HCT 116 CTRP1 4.4653 6.2041 3.939 12.8494
LS513 CTRP1 4.6682 9.7194 2.3955 23.8693
SNU-C5 CTRP1 4.7868 7.1775 3.7651 12.8065
LS180 CTRP1 4.793 6.6382 4.038 10.3601
SW948 CTRP1 4.9841 6.9721 4.0392 9.4989
LS123 CTRP1 5.0916 7.6652 3.7829 11.3252
SNU-81 CTRP1 5.1068 6.6755 4.2902 6.732
COLO 320 CTRP1 5.1999 8.0124 2.9329 7.2511
RKO CTRP1 5.239 6.357 4.5531 3.8652
HT-55 CTRP1 5.258 7.6855 3.9076 9.5585
HCT 8 CTRP1 5.4023 7.8747 3.9259 8.8519
SNU-C2A CTRP1 5.5776 9.6929 3.1587 14.6176
MDST8 CTRP1 5.6171 7.6491 4.1943 5.7593
GP2d CTRP1 5.6228 7.2361 4.3968 3.9968
HT115 CTRP1 5.6545 7.1648 4.4513 3.4462
DLD-1 CTRP1 5.7342 7.2128 4.4792 3.0018
LS411N CTRP1 5.7726 7.4122 4.4105 3.4659
SW403 CTRP1 5.8234 8.986 3.6903 9.4148
SK-CO-1 CTRP1 5.8648 9.3455 3.5445 10.4901
LoVo CTRP1 5.893 9.3944 3.5408 10.4264
COLO205 CTRP1 5.922 8.6749 3.9098 7.2488
NCI-H508 CTRP1 5.934 8.327 4.0839 5.7458
SNU-61 CTRP1 6.0043 9.9542 3.3474 11.6182
COLO 678 CTRP1 6.0865 8.3106 4.1887 4.4658
KM12 CTRP1 6.4631 8.2252 4.4362 1.8336
RCM-1 [Human ESC] CTRP1 6.4876 10.3987 3.4652 9.1937
HT-29 CTRP1 6.4981 11.8024 2.7982 14.1041
CL-34 CTRP1 6.6226 16.4724 0.5972 25.3483
CL-40 CTRP1 6.7958 8.3223 4.5494 0.783
SNU-1040 CTRP1 6.9137 12.3768 2.8064 12.7922
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 4 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-449 CTRP1 5.1285 8.4578 3.4171 14.3084
Hep-G2 CTRP1 5.4384 8.3093 3.7381 10.3575
SNU-398 CTRP1 5.4766 7.2313 4.298 5.3092
JHH-6 CTRP1 6.2657 7.2353 4.7389 0.3963
Cancer Drug Sensitivity Data Curated from 91 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Lu-99 CTRP1 2.4207 4.0146 2.3835 37.9298
NCI-H2029 CTRP1 3.0815 5.1793 2.8669 29.7941
VMRC-LCD CTRP1 3.12 5.3676 2.8512 29.639
Lu-65 CTRP1 3.1303 4.2733 3.1054 27.7283
NCI-H1105 CTRP1 3.3099 11.4512 0.3093 39.155
SCLC-21H CTRP1 3.3592 6.0036 2.8815 27.8207
NCI-H1963 CTRP1 3.4667 7.9235 2.1517 31.6868
NCI-H82 CTRP1 3.5815 6.1856 3.0431 25.2225
COR-L51 CTRP1 3.6294 7.9744 2.2878 29.9586
NCI-H460 CTRP1 3.6425 4.3981 3.6315 20.3133
NCI-H2342 CTRP1 3.6623 5.6332 3.3467 22.3779
CAL-12T CTRP1 3.9105 5.6096 3.6216 18.6548
NCI-H1373 CTRP1 3.9408 6.5009 3.278 21.2632
NCI-H1568 CTRP1 4.2519 6.1037 3.7718 15.4312
HCC44 CTRP1 4.3221 8.1444 2.866 22.3705
SHP-77 CTRP1 4.4098 8.8255 2.6106 23.7152
NCI-H2030 CTRP1 4.4593 5.2331 4.3499 9.4074
Calu-3 CTRP1 4.507 7.3483 3.427 17.0372
HCC2108 CTRP1 4.5352 7.0524 3.5979 15.452
NCI-H1930 CTRP1 4.6716 8.6504 2.931 20.1811
NCI-H23 CTRP1 4.681 7.3322 3.5938 14.7855
NCI-H1836 CTRP1 4.6983 8.3883 3.0849 18.8873
NCI-H841 CTRP1 4.7661 8.7071 2.9854 19.3355
NCI-H1299 CTRP1 4.8099 7.0636 3.8421 12.0217
SK-LU-1 CTRP1 4.8153 6.994 3.8816 11.6491
COR-L279 CTRP1 4.8796 7.4044 3.7336 12.6643
NCI-H1944 CTRP1 4.9082 8.1254 3.3983 15.4076
NCI-H1755 CTRP1 4.9307 7.319 3.8204 11.6773
COLO 668 CTRP1 4.9679 8.1595 3.4321 14.865
NCI-H3255 CTRP1 5.0119 8.182 3.458 14.4596
NCI-H2141 CTRP1 5.0515 11.3672 1.8986 25.0596
HCC15 CTRP1 5.0784 7.8318 3.6887 12.2036
BEN CTRP1 5.0816 7.4428 3.8858 10.4568
NCI-H596 CTRP1 5.2146 7.6227 3.9043 9.7569
Calu-6 CTRP1 5.2856 7.2648 4.1387 7.3974
NCI-H810 CTRP1 5.2971 7.8567 3.8532 9.8869
DMS 273 CTRP1 5.3122 8.0339 3.7769 10.4971
A-549 CTRP1 5.3135 7.5219 4.0326 8.2375
COR-L88 CTRP1 5.3165 7.33 4.1302 7.3581
NCI-H2172 CTRP1 5.3211 8.0974 3.7523 10.678
NCI-H2122 CTRP1 5.3261 6.6358 4.4805 4.2063
NCI-H1694 CTRP1 5.3743 10.0384 2.8268 17.8989
T3M-10 CTRP1 5.3788 8.1406 3.7758 10.2537
HCC33 CTRP1 5.3977 7.5732 4.0717 7.5811
HCC4006 CTRP1 5.3994 8.0604 3.8316 9.6899
LXF 289 CTRP1 5.4115 7.4942 4.1212 7.0938
NCI-H1048 CTRP1 5.4664 7.7425 4.0397 7.6189
NCI-H2110 CTRP1 5.4797 8.2013 3.8231 9.4694
NCI-H2286 CTRP1 5.4924 7.6781 4.0906 7.08
NCI-H1793 CTRP1 5.4989 9.0681 3.4081 12.9169
HCC1833 CTRP1 5.5049 7.6979 4.0901 7.0422
NCI-H2081 CTRP1 5.5054 9.2626 3.3165 13.6391
NCI-H2009 CTRP1 5.5831 8.8938 3.5589 11.3534
HCC78 CTRP1 5.586 7.8534 4.0728 6.9185
HCC2935 CTRP1 5.5992 7.8085 4.1042 6.6016
NCI-H2126 CTRP1 5.6294 7.1083 4.4616 3.4288
NCI-H727 CTRP1 5.6369 10.4853 2.811 16.9897
COLO 699 CTRP1 5.6546 9.9625 3.0841 14.9051
NCI-H1792 CTRP1 5.6658 8.3102 3.907 8.0921
NCI-H1876 CTRP1 5.6684 7.6389 4.2347 5.2501
NCI-H2073 CTRP1 5.674 8.6824 3.7306 9.579
RERF-LC-KJ CTRP1 5.8182 8.6866 3.8323 8.2311
EPLC-272H CTRP1 5.8247 8.6166 3.8708 7.8827
NCI-H1355 CTRP1 5.8842 8.9252 3.7629 8.6056
ChaGo-K-1 CTRP1 5.9225 8.2869 4.0954 5.6821
HCC1195 CTRP1 5.9501 7.3585 4.5393 2.0361
NCI-H1975 CTRP1 5.9928 8.1905 4.1861 4.7318
NCI-H1573 CTRP1 5.9979 8.0434 4.2576 4.1326
HCC1359 CTRP1 6.0268 10.5831 3.056 13.7911
NCI-H1781 CTRP1 6.0338 8.9494 3.8539 7.3806
NCI-H522 CTRP1 6.0518 9.1022 3.7929 7.8336
NCI-H2023 CTRP1 6.0587 8.4329 4.1145 5.1448
NCI-H358 CTRP1 6.089 8.4118 4.1434 4.8277
KNS-62 CTRP1 6.1241 8.7264 4.0187 5.7557
NCI-H1435 CTRP1 6.1685 10.0037 3.439 10.3578
NCI-H441 CTRP1 6.2721 9.9974 3.5129 9.4506
NCI-H1437 CTRP1 6.3021 9.4049 3.814 6.9386
LC-1/sq-SF CTRP1 6.3582 10.1936 3.477 9.4779
LCLC-103H CTRP1 6.3645 9.9127 3.6148 8.3654
LCLC-97TM1 CTRP1 6.5157 9.0641 4.1005 4.1406
EBC-1 CTRP1 6.5269 13.0046 2.2331 17.6805
HARA [Human squamous cell lung carcinoma] CTRP1 6.5506 10.6211 3.4011 9.5092
NCI-H2405 CTRP1 6.5793 9.4984 3.9417 5.2151
Sq-1 CTRP1 6.6475 8.058 4.5874 0.7413
NCI-H661 CTRP1 6.7341 15.3585 1.2298 22.3315
HCC827 CTRP1 6.8286 9.8391 3.9328 4.72
NCI-H1915 CTRP1 7.1357 8.7457 4.5298 0.5976
COR-L23 CTRP1 7.1779 8.9538 4.4698 0.8099
NCI-H1666 CTRP1 7.5455 15.7755 1.6046 18.1322
DV-90 CTRP1 7.5817 9.2246 4.5279 0.3596
NCI-H650 CTRP1 7.8086 9.2023 4.6151 0.1179
⏷ Show the Full List of 91 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KYSE-140 CTRP1 5.2973 7.6056 3.9784 8.7796
KYSE-410 CTRP1 5.7167 8.1443 4.0241 6.9149
KYSE-450 CTRP1 6.1571 10.5389 3.1714 12.4821
Cancer Drug Sensitivity Data Curated from 26 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TYK-nu CTRP1 3.5969 5.3202 3.3851 22.4907
COV434 CTRP1 4.2914 6.9072 3.437 18.0483
OVCAR-8 CTRP1 4.6201 8.3494 3.035 19.6404
OV-90 CTRP1 4.7765 8.1463 3.2739 17.0239
RMUG-S CTRP1 4.8767 10.368 2.251 23.8128
COV644 CTRP1 4.9749 7.0157 4.0096 9.803
A2780 CTRP1 5.0554 10.342 2.4144 22.0227
OVCAR-4 CTRP1 5.2059 8.8638 3.2775 15.135
OVK18 CTRP1 5.287 9.83 2.8606 18.0071
HEY A8 CTRP1 5.3944 10.5995 2.563 19.6484
IGROV-1 CTRP1 5.7319 9.5002 3.3711 12.3662
RMG-I CTRP1 5.7565 9.8243 3.2296 13.4053
OVKATE CTRP1 5.7801 10.059 3.1315 14.0833
JHOC-5 CTRP1 5.846 8.4593 3.9615 7.0443
JHOS-4 CTRP1 6.1242 8.3559 4.1909 4.3524
EFO-27 CTRP1 6.1969 9.1482 3.867 6.8
COV362 CTRP1 6.2142 8.4618 4.1966 4.088
EFO-21 CTRP1 6.3116 8.5333 4.2213 3.6701
JHOM-1 CTRP1 6.4894 10.3432 3.4927 8.9738
OAW42 CTRP1 6.6188 7.8403 4.657 0.4661
SNU-840 CTRP1 6.6598 10.3731 3.588 7.7635
COV318 CTRP1 6.6684 7.5048 4.7923 0.0787
Caov-3 CTRP1 6.7617 8.577 4.4352 1.4141
SK-OV-3 CTRP1 7.102 9.9897 4.0159 3.5793
OV7 CTRP1 7.2001 8.8043 4.5336 0.541
OVMANA CTRP1 7.7213 13.9618 2.5823 12.0792
⏷ Show the Full List of 26 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuP-T4 CTRP1 4.211 6.6053 3.5009 17.9403
CFPAC-1 CTRP1 5.1668 8.1004 3.6271 12.3718
PaTu 8902 CTRP1 5.2243 6.5741 4.4343 4.9803
SUIT-2 CTRP1 5.622 8.0938 3.9813 7.5953
Panc 03.27 CTRP1 5.7821 8.8674 3.7186 9.3138
Panc 10.05 CTRP1 5.9826 9.3595 3.6213 9.4703
HPAC CTRP1 6.0194 9.1717 3.7374 8.3931
Capan-2 CTRP1 6.1446 9.8924 3.4762 10.1363
QGP-1 CTRP1 6.3236 10.1983 3.4514 9.7827
KP-3 CTRP1 7.5761 15.9715 1.5312 18.4188
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP1 3.7494 6.2224 3.2031 22.9746
NCI-H28 CTRP1 5.6549 8.5657 3.774 9.2735
NCI-H2052 CTRP1 8.1357 14.7144 2.4906 11.6318
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PaCa-3 CTRP1 5.9827 8.3543 4.1028 5.4495
Cancer Drug Sensitivity Data Curated from 9 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-MEL-5 CTRP1 3.8372 5.8991 3.4295 20.6502
SK-MEL-28 CTRP1 3.947 4.4582 3.9431 15.9126
A-375 CTRP1 5.1149 6.5032 4.3828 5.8655
SK-MEL-1 CTRP1 5.2881 7.2594 4.1433 7.3466
G-361 CTRP1 5.6943 9.9522 3.1195 14.4861
Hs 852.T CTRP1 5.8743 7.8943 4.2495 4.527
Hs 936.T CTRP1 6.0117 7.706 4.4198 2.8097
Hs 944.T CTRP1 6.519 9.8223 3.7562 6.8181
COLO 741 CTRP1 7.3523 9.1514 4.4668 0.6897
⏷ Show the Full List of 9 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HT-1080 CTRP1 4.028 5.3187 3.8535 16.0655
G-401 CTRP1 4.0694 8.1801 2.6126 25.4611
RKN CTRP1 6.2978 10.4154 3.3296 10.8162
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH-10-TC CTRP1 4.0487 5.2451 3.9005 15.5605
Fu97 CTRP1 4.2806 7.0035 3.3805 18.5723
NUGC-4 CTRP1 5.7138 7.6194 4.2747 4.7708
MKN74 CTRP1 6.2708 10.5251 3.258 11.4536
MKN7 CTRP1 6.783 10.9037 3.418 8.7359
AGS CTRP1 6.858 8.3793 4.5537 0.7097
SNG-M CTRP1 6.5097 12.3204 2.5547 15.7107
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-2 CTRP1 2.6624 3.9098 2.6459 34.3493
SCC-9 CTRP1 6.4068 8.4928 4.2925 2.9347
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UM-UC-3 CTRP1 2.4348 3.8962 2.4096 37.6528
RT-4 CTRP1 3.1255 6.0325 2.6214 31.1535
KMBC-2 CTRP1 5.7111 9.5845 3.314 12.8986
5637 CTRP1 5.9362 9.2016 3.6653 9.2543
HT-1376 CTRP1 6.3537 11.7405 2.726 15.0657

References

1 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 5243).
2 Discovery and characterization of a highly selective FAAH inhibitor that reduces inflammatory pain. Chem Biol. 2009 Apr 24;16(4):411-20.