General Information of Drug (ID: DMDN12L)

Drug Name
2,6-Dihydroanthra/1,9-Cd/Pyrazol-6-One
Synonyms
Anthra[1,9-cd]pyrazol-6(2H)-one; 129-56-6; 1,9-Pyrazoloanthrone; SP600125; Pyrazolanthrone; Dibenzo[cd,g]indazol-6(2H)-one; Pyrazoleanthrone; SP 600125; Anthra-1,9-pyrazol-6-none; SP-600125; CI 70300; 2H-Dibenzo[cd,g]indazol-6-one; JNK Inhibitor II; SAPK Inhibitor II; NSC 75890; UNII-1TW30Y2766; ANTHRA(1,9-cd)PYRAZOL-6(2H)-ONE; EINECS 204-955-6; 2,6-DIHYDROANTHRA/1,9-CD/PYRAZOL-6-ONE; BRN 0746890; CHEMBL7064; MLS002693964; CHEBI:90695; ACPOUJIDANTYHO-UHFFFAOYSA-N; 1TW30Y2766
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 220.23
Logarithm of the Partition Coefficient (xlogp) 2.7
Rotatable Bond Count (rotbonds) 0
Hydrogen Bond Donor Count (hbonddonor) 1
Hydrogen Bond Acceptor Count (hbondacc) 2
Chemical Identifiers
Formula
C14H8N2O
IUPAC Name
14,15-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),2,4,6,9(16),10,12-heptaen-8-one
Canonical SMILES
C1=CC=C2C(=C1)C3=NNC4=CC=CC(=C43)C2=O
InChI
InChI=1S/C14H8N2O/c17-14-9-5-2-1-4-8(9)13-12-10(14)6-3-7-11(12)15-16-13/h1-7H,(H,15,16)
InChIKey
ACPOUJIDANTYHO-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
8515
ChEBI ID
CHEBI:90695
CAS Number
129-56-6
UNII
1TW30Y2766
DrugBank ID
DB01782
TTD ID
D02PVB

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Dual specificity protein kinase TTK (MPS1) TTP7EGM TTK_HUMAN Inhibitor [1]
Jun N terminal kinase (JNK) TTR2TXZ MK08_HUMAN ; MK09_HUMAN ; MK10_HUMAN Inhibitor [2]
Stress-activated protein kinase JNK1 (JNK1) TT0K6EO MK08_HUMAN Inhibitor [1]
Stress-activated protein kinase JNK2 (JNK2) TTHS0U8 MK09_HUMAN Inhibitor [3]
Stress-activated protein kinase JNK3 (JNK3) TT056SO MK10_HUMAN Inhibitor [1]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Apoptosis regulator BAX (BAX) OTAW0V4V BAX_HUMAN Gene/Protein Processing [4]
C-type lectin domain family 4 member K (CD207) OTI9RUDN CLC4K_HUMAN Gene/Protein Processing [5]
Cadherin-1 (CDH1) OTFJMXPM CADH1_HUMAN Gene/Protein Processing [5]
Casein kinase I isoform delta (CSNK1D) OTNF4S77 KC1D_HUMAN Gene/Protein Processing [6]
Caspase-2 (CASP2) OTUDYSPP CASP2_HUMAN Gene/Protein Processing [7]
Caspase-3 (CASP3) OTIJRBE7 CASP3_HUMAN Gene/Protein Processing [8]
Caspase-9 (CASP9) OTD4RFFG CASP9_HUMAN Gene/Protein Processing [4]
Cellular tumor antigen p53 (TP53) OTIE1VH3 P53_HUMAN Gene/Protein Processing [9]
Cyclic AMP-responsive element-binding protein 1 (CREB1) OT1MDLA1 CREB1_HUMAN Post-Translational Modifications [10]
Cyclin-dependent kinase 2 (CDK2) OTB5DYYZ CDK2_HUMAN Gene/Protein Processing [6]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Discovery agent
ICD Disease Classification N.A.
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Stress-activated protein kinase JNK1 (JNK1) DTT MAPK8 1.48E-07 1.2 2.27
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 149 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 4.1001 6.9787 3.6102 14.7361
JK1 CTRP2 6.5763 10.6823 4.1524 6.9804
JM1 CTRP2 4.721 6.5276 4.4444 9.815
MV4-11 CTRP2 0.9528 5.4639 0.6349 34.9124
MOLM-13 CTRP2 1.6561 3.6877 1.6402 29.2886
EoL-1 CTRP2 1.8489 2.7135 1.8489 27.9511
MOLM-16 CTRP2 2.1535 3.5943 2.15 25.9333
697 CTRP2 2.572 4.3792 2.5482 23.2133
Pfeiffer CTRP2 2.6791 4.7808 2.624 22.6064
KMS-26 CTRP2 2.7888 3.8077 2.788 21.692
NALM-6 CTRP2 3.3291 4.9604 3.2917 18.2158
A4/Fukuda CTRP2 3.3869 5.8564 3.1932 18.3775
Peer CTRP2 3.6552 5.1171 3.6195 16.0377
P31/FUJ CTRP2 3.6648 5.7582 3.5197 16.3548
Jurkat CTRP2 3.6842 5.4961 3.595 16.0289
F-36P CTRP2 3.7261 14.4344 -0.2106 28.8207
KE-97 CTRP2 3.7335 6.3012 3.4479 16.4047
ALL-SIL CTRP2 3.7781 7.2134 3.1765 17.291
SKM-1 CTRP2 3.8561 5.5477 3.7712 14.8696
RPMI-8402 CTRP2 4.0035 5.6641 3.9082 13.9239
OCI-AML-2 CTRP2 4.0922 6.6744 3.7138 14.3675
Ri-1 CTRP2 4.0934 7.8766 3.2373 16.1946
JVM-3 CTRP2 4.1359 7.6353 3.3839 15.5098
NCO2 CTRP2 4.1441 5.9236 4.0023 13.153
WSU-DLCL2 CTRP2 4.156 6.0425 3.984 13.1824
Ki-JK CTRP2 4.158 5.8362 4.0386 12.9804
Kasumi-1 CTRP2 4.164 6.4469 3.8698 13.5766
Mono-Mac-1 CTRP2 4.2175 9.5221 2.6196 18.2906
GA-10 CTRP2 4.2198 6.5441 3.8973 13.3116
Ku812 CTRP2 4.2538 8.003 3.348 15.3372
SUP-M2 CTRP2 4.2623 5.9566 4.1228 12.358
MOLM-6 CTRP2 4.2707 7.1664 3.7183 13.848
EM-2 CTRP2 4.2812 6.2732 4.0532 12.5538
HEL CTRP2 4.2914 5.9707 4.1509 12.1681
JURL-MK1 CTRP2 4.3095 6.184 4.1112 12.2569
SET-2 CTRP2 4.3097 5.8184 4.2078 11.9089
DEL CTRP2 4.3258 6.0851 4.1576 12.0394
A3/Kawakami CTRP2 4.337 5.8506 4.2301 11.7448
REC-1 CTRP2 4.3374 6.2528 4.1207 12.1389
NU-DUL-1 CTRP2 4.3434 5.8788 4.2305 11.7232
RS4;11 CTRP2 4.3628 7.3437 3.743 13.501
MOLT-3 CTRP2 4.3697 5.0084 4.3678 11.1635
M-07e CTRP2 4.414 8.3645 3.3496 14.9179
RCH-ACV CTRP2 4.4334 6.7136 4.0669 12.0606
LAMA-84 CTRP2 4.4541 10.1208 2.5659 17.9164
PF-382 CTRP2 4.4575 5.9165 4.3458 10.96
KE-37 CTRP2 4.4609 5.3243 4.4472 10.5956
HEL 92.1.7 CTRP2 4.4727 6.7667 4.0892 11.8647
P12-Ichikawa CTRP2 4.4986 5.2388 4.4918 10.321
OPM-2 CTRP2 4.5297 6.0851 4.38 10.6161
BDCM CTRP2 4.543 7.6141 3.8152 12.7384
JVM-2 CTRP2 4.5707 7.9107 3.7126 13.0732
OCI-AML-5 CTRP2 4.5907 14.9573 0.3252 25.2732
EB1 CTRP2 4.5988 7.5157 3.9155 12.1964
MOLT-16 CTRP2 4.6068 6.0329 4.4786 10.0256
OCI-AML-3 CTRP2 4.6127 7.2476 4.0445 11.6529
TF-1 CTRP2 4.6238 7.0182 4.1511 11.2082
NCI-H929 CTRP2 4.669 6.8019 4.2851 10.5674
Karpas-299 CTRP2 4.6927 8.4723 3.5782 13.3045
PL21 CTRP2 4.6975 7.8857 3.8523 12.1919
KMS-11 CTRP2 4.7091 7.1177 4.1997 10.7881
SEM CTRP2 4.7158 5.6801 4.6752 8.9899
KYO-1 CTRP2 4.738 7.1247 4.227 10.604
KM-H2 CTRP2 4.7508 6.9757 4.3022 10.2766
HDLM-2 CTRP2 4.7653 9.0852 3.3603 14.0085
U-937 CTRP2 4.7793 6.5605 4.495 9.4578
NB4 CTRP2 4.7841 7.4941 4.1154 10.922
Kasumi-2 CTRP2 4.7908 6.6933 4.4571 9.5696
SU-DHL-6 CTRP2 4.8072 8.0517 3.8866 11.7785
MOLT-13 CTRP2 4.8189 8.6012 3.6418 12.7393
AML-193 CTRP2 4.8302 11.9303 2.0371 19.0451
CML-T1 CTRP2 4.8329 6.3736 4.6197 8.8352
OCI-Ly19 CTRP2 4.8352 7.4699 4.1782 10.5406
BV-173 CTRP2 4.849 8.7752 3.5887 12.8822
Daudi CTRP2 4.8616 6.9183 4.4423 9.4319
NU-DHL-1 CTRP2 4.8631 7.1531 4.3451 9.8078
KO52 CTRP2 4.9407 7.6193 4.2182 10.1113
NOMO-1 CTRP2 5.0086 14.4262 0.9618 22.3759
MHH-CALL-3 CTRP2 5.0133 7.7127 4.2482 9.8082
Mino CTRP2 5.0143 6.4549 4.7865 7.6871
KMS-20 CTRP2 5.0414 6.8314 4.6668 8.0722
KMM-1 CTRP2 5.1444 10.1754 3.188 13.8323
Namalwa CTRP2 5.1748 7.9792 4.2825 9.2747
SU-DHL-10 CTRP2 5.1928 6.4827 3.6375 0.637
RPMI-8226 CTRP2 5.2233 8.9103 3.8805 10.8129
DB CTRP2 5.2336 8.3093 4.1813 9.5502
Hs 611.T CTRP2 5.2379 7.7986 4.4294 8.5241
SIG-M5 CTRP2 5.2403 6.9495 4.8223 6.9343
KCL-22 CTRP2 5.2569 11.5095 2.6307 15.8174
JeKo-1 CTRP2 5.2597 9.6319 3.561 12.0482
HD-MY-Z CTRP2 5.2611 8.3235 4.2006 9.407
THP-1 CTRP2 5.2797 8.1087 4.3218 8.8653
L-363 CTRP2 5.2915 6.6122 5.0198 6.0222
SUP-T1 CTRP2 5.302 8.4975 4.155 9.5008
CA46 CTRP2 5.332 7.7473 4.545 7.8273
P3HR-1 CTRP2 5.3495 9.3565 2.416 5.6647
SU-DHL-1 CTRP2 5.3497 6.6616 5.0599 5.7098
SU-DHL-8 CTRP2 5.3549 7.7832 3.1585 2.3355
KMS-21-BM CTRP2 5.3565 7.0226 4.9077 6.2959
RPMI-6666 CTRP2 5.3653 7.3184 4.7801 6.7886
HT CTRP2 5.3841 7.7498 4.594 7.5033
L-540 CTRP2 5.4143 6.5075 5.1918 5.021
CMK CTRP2 5.4208 6.5282 5.1902 5.0096
DND-41 CTRP2 5.4232 7.5109 4.7457 6.7892
MOLP-8 CTRP2 5.4264 7.7091 4.6539 7.158
Granta-519 CTRP2 5.455 7.46 4.8006 6.4891
Karpas-422 CTRP2 5.4583 8.1962 4.448 7.9341
BL-70 CTRP2 5.5226 6.3734 5.3605 4.0722
HuT 78 CTRP2 5.5329 7.5171 4.8479 6.1119
HH [Human lymphoma] CTRP2 5.5618 8.9499 4.1722 8.8527
LP-1 CTRP2 5.5794 8.4337 4.443 7.6858
TALL-1 [Human adult T-ALL] CTRP2 5.6116 7.8782 4.7458 6.3553
OCI-M1 CTRP2 5.6154 6.4183 5.4395 3.514
SR CTRP2 5.6331 7.375 5.0115 5.2066
MOTN-1 CTRP2 5.7051 8.5918 4.478 7.2695
Karpas-620 CTRP2 5.7421 7.1252 5.2352 4.0335
K-562 CTRP2 5.7569 9.8431 3.9005 9.5778
SUP-HD1 CTRP2 5.7838 7.4529 5.1127 4.4499
OCI-Ly3 CTRP2 5.8232 7.3446 5.2019 3.9927
HL-60 CTRP2 5.8327 8.2855 4.7429 5.8932
HPB-ALL CTRP2 5.8593 7.2437 5.2843 3.5709
L-428 CTRP2 5.8691 13.2838 2.2776 15.8994
JJN-3 CTRP2 5.8921 7.5942 5.1392 4.1093
KMS-27 CTRP2 5.9151 7.4961 5.2082 3.7727
KMS-18 CTRP2 5.9323 9.4606 4.242 7.7943
SUP-B15 CTRP2 6.0489 8.6359 4.7524 5.4221
RL CTRP2 6.0532 6.9239 5.6119 1.801
ST486 CTRP2 6.1084 8.7499 4.7446 5.3413
SUP-T11 CTRP2 6.1628 8.8169 4.7556 5.1929
SK-MM-2 CTRP2 6.2507 7.5619 5.45 2.1275
U266B1 CTRP2 6.3002 17.5236 0.5165 21.0746
L-1236 CTRP2 6.3718 10.5788 4.0439 7.7937
EJM CTRP2 6.5978 8.1796 5.3953 1.8268
MOLP-2 CTRP2 6.6313 10.299 4.3842 5.9232
Ci-1 CTRP2 6.7205 7.5429 5.7554 0.3791
Reh CTRP2 6.7301 8.6622 5.2534 2.2111
MM1.S CTRP2 6.829 8.8199 5.2433 2.1198
OCI-Ly10 CTRP2 6.9046 9.0493 5.1841 2.2541
KHM-1B CTRP2 6.9632 10.7694 4.3969 5.3391
SU-DHL-4 CTRP2 6.9856 11.1356 4.2342 5.9706
EHEB CTRP2 7.0403 10.1626 4.7445 3.8143
MC116 CTRP2 7.1771 7.9631 5.789 0.0984
AMO1 CTRP2 7.7763 9.1169 5.6039 0.2312
ME1 CTRP2 7.8916 12.5594 4.1676 4.9494
GDM-1 CTRP2 7.9631 10.5072 5.1364 1.3463
MHH-CALL-4 CTRP2 8.0471 10.2312 5.2912 0.829
Raji CTRP2 8.0505 9.2875 5.6463 0.1048
Mono-Mac-6 CTRP2 8.3407 11.4402 4.9345 1.6848
Toledo CTRP2 8.4521 10.4499 5.3825 0.4143
⏷ Show the Full List of 149 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 4.1305 8.5715 2.9697 17.1445
TE8 CTRP2 5.2273 9.3239 3.6823 11.6211
TE-11 CTRP2 4.4078 8.5554 3.2564 15.3042
EC-GI-10 CTRP2 5.0172 8.6291 3.8207 11.5365
KYSE-410 CTRP2 5.1338 9.7744 3.3751 13.0931
TE-4 CTRP2 5.2016 10.783 2.9407 14.7054
TE-6 CTRP2 5.3167 9.8572 2.861 9.999
TE-9 CTRP2 5.319 9.0563 3.8982 10.524
OE21 CTRP2 5.877 9.2919 4.2791 7.7492
TE-14 CTRP2 6.0802 8.6985 4.747 5.3845
TE-5 CTRP2 6.1139 9.5535 4.3474 6.9991
KYSE-140 CTRP2 6.1971 11.4198 3.4828 10.4492
KYSE-180 CTRP2 6.3985 8.4537 5.1206 3.2508
TE-10 CTRP2 6.7346 11.5032 3.8667 7.8946
KYSE-70 CTRP2 6.9822 10.0151 4.7758 3.7708
TE-1 CTRP2 7.1035 11.3931 4.1931 5.9566
COLO 680N CTRP2 7.2447 11.2442 4.3641 5.0531
KYSE-510 CTRP2 7.3785 13.2797 3.4694 8.4638
KYSE-450 CTRP2 7.623 10.0543 5.152 1.5864
OE19 CTRP2 7.6984 9.3934 5.4658 0.5694
OE33 CTRP2 7.9569 9.4469 5.5544 0.2616
KYSE-520 CTRP2 7.9787 11.4535 4.7311 2.7178
KYSE-30 CTRP2 8.2238 15.5839 2.9461 9.2381
KYSE-150 CTRP2 11.0257 20.1059 2.6031 6.9972
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 37 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 7.5156 11.3813 4.4799 4.2187
HuP-T4 CTRP2 3.7261 8.2181 2.7104 19.2166
KP-3 CTRP2 4.9469 9.2234 3.4679 13.1422
SNU-410 CTRP2 4.9848 13.1838 1.5573 20.4265
KP-4 CTRP2 5.4078 8.24 4.3795 8.3323
PSN1 CTRP2 5.6629 7.4939 4.9815 5.2632
PK-59 CTRP2 5.8521 10.2578 3.7754 9.9068
Hs 766T CTRP2 6.0476 7.7854 5.1766 3.6415
MIA PaCa-2 CTRP2 6.0989 7.8809 5.1712 3.5665
L3.3 CTRP2 6.117 8.3123 4.9704 4.3763
SU.86.86 CTRP2 6.2669 9.4018 4.5473 5.8758
SW1990 CTRP2 6.2923 9.4872 4.525 5.9236
Panc 08.13 CTRP2 6.3256 8.5364 5.0242 3.7752
BxPC-3 CTRP2 6.3302 12.0045 3.2991 10.9537
Panc 03.27 CTRP2 6.3386 9.7876 4.4119 6.3141
HPAC CTRP2 6.4379 9.6874 4.5396 5.6052
AsPC-1 CTRP2 6.5563 9.2858 4.828 4.2058
Panc 05.04 CTRP2 6.5709 11.1051 3.9383 7.8799
PaTu 8902 CTRP2 6.5823 7.8602 5.536 1.2943
Panc 10.05 CTRP2 6.6095 9.526 4.7491 4.446
Panc 04.03 CTRP2 6.617 8.5294 5.2406 2.4203
PaTu 8988t CTRP2 6.7079 8.1649 5.4729 1.3831
Capan-1 CTRP2 6.7433 11.5686 3.8409 7.986
SUIT-2 CTRP2 6.789 8.7115 5.2687 2.0724
TCC-Pan2 CTRP2 6.9067 10.2992 4.5857 4.6532
HuP-T3 CTRP2 6.9219 11.3135 4.1006 6.6203
CFPAC-1 CTRP2 7.0015 10.7238 4.4464 5.0784
Capan-2 CTRP2 7.0388 12.7634 3.4733 8.9959
KP-2 CTRP2 7.1359 9.7795 4.9892 2.7179
YAPC CTRP2 7.3299 11.027 4.5258 4.2862
Panc 02.03 CTRP2 7.34 10.3729 4.841 3.0361
DAN-G CTRP2 7.7166 16.0551 2.3551 12.2534
QGP-1 CTRP2 7.7306 9.3918 5.4808 0.5142
PK-45H CTRP2 7.7633 11.4685 4.5958 3.4608
SNU-213 CTRP2 7.7844 17.6032 1.6433 14.7072
HPAF-II CTRP2 7.8239 13.8264 3.518 7.5975
PaTu 8988s CTRP2 7.9899 12.134 4.4277 3.8294
⏷ Show the Full List of 37 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 51 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 7.1515 13.719 3.0862 10.3638
IGR-37 CTRP2 5.0959 7.6185 4.3739 9.0961
SK-MEL-1 CTRP2 5.2749 7.3445 4.6785 7.4226
Hs 934.T CTRP2 5.4165 10.5283 3.2598 12.9439
COLO 792 CTRP2 5.5712 7.9323 4.682 6.7104
Hs 940.T CTRP2 5.5863 7.1825 5.0597 5.1171
HMCB CTRP2 5.6142 9.3097 4.0407 9.289
RPMI-7951 CTRP2 5.6944 8.4178 4.5547 6.9716
LOX-IMVI CTRP2 5.7198 8.4859 4.5436 6.9641
SK-MEL-5 CTRP2 5.8088 6.7898 5.4609 2.9485
A-375 CTRP2 5.8479 8.1491 4.8241 5.5214
G-361 CTRP2 5.8664 9.5308 4.1507 8.3085
WM115 CTRP2 5.9482 8.1514 4.9097 4.9584
A2058 CTRP2 5.9593 6.8158 5.5857 2.0986
IGR-1 CTRP2 5.9714 6.993 5.508 2.3998
SK-MEL-3 CTRP2 6.0155 8.796 4.6445 5.9401
WM1799 CTRP2 6.0904 8.98 4.6147 5.9211
WM88 CTRP2 6.1134 7.4146 5.4159 2.5113
Hs 895.T CTRP2 6.137 9.6744 4.306 7.1297
Mel Ho CTRP2 6.2174 8.334 5.0404 3.8978
Mel JuSo CTRP2 6.2772 7.8683 5.3185 2.6304
CJM [Human melanoma] CTRP2 6.2966 8.5195 5.0102 3.8838
WT2-iPS CTRP2 6.3325 7.9661 5.3118 2.566
IPC-298 CTRP2 6.3581 8.324 5.1543 3.1777
Hs 852.T CTRP2 6.4461 11.7556 3.5163 9.849
Hs 839.T CTRP2 6.4547 12.2873 3.258 10.891
WM266-4 CTRP2 6.525 8.587 5.148 2.9353
RVH-421 CTRP2 6.546 8.0791 5.4086 1.8452
Hs 944.T CTRP2 6.5793 12.8075 3.0977 11.3134
SK-MEL-30 CTRP2 6.6102 8.2341 5.3776 1.8804
UACC-257 CTRP2 6.7401 8.0702 5.5358 1.1101
WM793 CTRP2 6.7476 9.1362 5.0381 3.0499
HT-144 CTRP2 6.7993 8.6838 5.2883 1.9823
A101D CTRP2 6.8035 8.0152 5.5966 0.827
IGR-39 CTRP2 6.8204 9.5001 4.9127 3.4515
MeWo CTRP2 6.9345 12.0119 3.7661 7.974
MDA-MB-435S CTRP2 6.9489 9.6757 4.916 3.2553
SK-MEL-28 CTRP2 6.949 7.9237 5.7089 0.3615
Hs 294T CTRP2 6.9673 8.8437 5.3186 1.6623
COLO 800 CTRP2 7.0295 10.4539 4.5969 4.4251
SK-MEL-24 CTRP2 7.1757 11.167 4.3537 5.1956
COLO 741 CTRP2 7.2578 22.2574 -1.0744 23.6226
SK-MEL-2 CTRP2 7.4084 8.4974 5.6853 0.2042
SK-MEL-31 CTRP2 7.4385 9.8752 5.1282 1.8496
Malme-3M CTRP2 7.4848 14.5671 2.9158 10.4881
Hs 936.T CTRP2 7.5744 9.594 5.3241 1.0616
K029AX CTRP2 7.5961 11.1213 4.6531 3.4437
UACC-62 CTRP2 7.9143 11.7138 4.5749 3.3636
WM983B CTRP2 8.0304 12.9833 4.0575 5.1981
Hs 688(A).T CTRP2 8.1229 22.8108 -0.6759 21.1539
COLO 829 CTRP2 9.2384 21.0464 1.0097 14.5454
⏷ Show the Full List of 51 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 6.9615 17.2631 1.1798 17.7165
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IMR-32 CTRP2 2.7813 4.4344 2.7618 21.8045
CHP-212 CTRP2 2.8041 4.5652 2.7765 21.6799
MHH-NB-11 CTRP2 3.826 6.1923 3.5815 15.6399
SK-N-BE(2) CTRP2 4.0972 7.0326 3.5864 14.8351
SK-N-SH CTRP2 4.743 6.7925 4.3676 10.0454
KP-N-SI9s CTRP2 5.2487 8.7839 3.9658 10.4031
CHP-126 CTRP2 5.2802 6.9329 4.8705 6.6395
SK-N-DZ CTRP2 5.3197 11.8516 2.5167 16.1275
Kelly CTRP2 5.3633 6.9733 4.9368 6.1621
NB1 CTRP2 5.3777 6.5208 5.148 5.2907
NH-6 CTRP2 5.7473 8.1997 4.7102 6.2093
SK-N-AS CTRP2 6.1024 8.9753 4.627 5.8466
SK-N-FI CTRP2 6.2197 9.3996 4.5106 6.1165
KP-N-YN CTRP2 6.6896 9.0975 5.0164 3.2231
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 4.4497 6.3409 4.2149 11.4595
HuCC-T1 CTRP2 4.7329 8.4792 3.6147 13.0585
SNU-478 CTRP2 4.9355 8.5283 3.7898 11.8571
HuH-28 CTRP2 6.3002 8.4748 5.0353 3.7728
SNU-308 CTRP2 6.5318 9.7143 4.5981 5.201
SNU-1196 CTRP2 6.6818 8.9233 5.0953 2.9143
SNU-869 CTRP2 7.1425 9.406 5.1667 2.0312
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U2OS CTRP2 3.781 13.877 0.1122 27.8241
SK-ES-1 CTRP2 3.9864 6.2444 3.7408 14.5777
MHH-ES-1 CTRP2 4.4838 6.1067 4.3239 10.9582
SK-N-MC CTRP2 4.5545 6.3308 4.3321 10.7176
A-673 CTRP2 4.9173 7.1932 4.3838 9.5122
TC71 CTRP2 5.5 7.4023 4.8716 6.0917
CAL-78 CTRP2 5.7691 9.9684 3.8485 9.7702
G-292 clone A141B1 CTRP2 5.9613 9.439 4.2774 7.5886
Hs 888.T CTRP2 6.0209 9.6703 4.2118 7.7472
SJSA-1 CTRP2 6.0902 8.9468 4.6312 5.8521
Hs 822.T CTRP2 6.3643 7.4591 5.5827 1.4033
MG-63 CTRP2 6.5342 10.0253 4.4459 5.8303
SaOS-2 CTRP2 6.574 9.6146 4.6792 4.7936
HOS CTRP2 6.6869 9.0759 5.025 3.1924
SW1353 CTRP2 7.8407 10.814 4.938 2.1202
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 71 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HCC2218 CTRP2 2.8616 8.7112 1.6018 25.6851
Hs 578Bst CTRP2 4.752 14.2247 0.8329 23.3669
CAL-51 CTRP2 5.5416 7.9852 4.6286 6.9984
MDA-MB-157 CTRP2 5.5785 24.3362 -3.4925 31.4849
MDA-MB-468 CTRP2 5.842 8.8344 4.4774 6.9878
UACC-812 CTRP2 6.2917 10.1592 4.1893 7.3314
MDA-MB-453 CTRP2 6.3885 17.1306 0.7854 20.0709
MDA-MB-231 CTRP2 6.4938 10.1736 4.3413 6.3357
HMC-1-8 CTRP2 6.5164 9.4236 4.7302 4.6771
KPL-1 CTRP2 6.5299 8.0494 5.412 1.8543
HCC1395 CTRP2 6.6068 11.7248 3.6582 8.9764
HCC1428 CTRP2 6.6265 8.0601 5.4705 1.493
SK-BR-3 CTRP2 6.8125 11.2583 4.0466 7.0209
T-47D CTRP2 6.8493 10.0424 4.67 4.396
CAL-148 CTRP2 6.8722 10.6715 4.3792 5.553
BT-549 CTRP2 6.9911 12.6952 3.4713 9.0834
CAL-120 CTRP2 7.1639 8.7915 5.4534 0.9839
HDQ-P1 CTRP2 7.1668 11.5256 4.1735 5.9401
CAL-85-1 CTRP2 7.2291 12.1508 3.9134 6.9023
HCC38 CTRP2 7.24 11.6399 4.1695 5.8465
ZR-75-30 CTRP2 7.2738 9.7109 5.1062 2.1077
HCC1954 CTRP2 7.4655 12.6462 3.8397 6.8424
HCC202 CTRP2 7.4766 10.1355 5.0333 2.1533
ZR-75-1 CTRP2 7.4925 11.1039 4.5957 3.7954
BT-20 CTRP2 7.6661 9.5719 5.3787 0.8286
Hs 578T CTRP2 7.7201 16.341 2.2171 12.7586
MCF-7 CTRP2 7.7421 12.5347 4.0817 5.4841
HCC1143 CTRP2 7.7748 11.324 4.6694 3.1699
HCC1937 CTRP2 7.8403 10.4517 5.0962 1.5789
HCC1806 CTRP2 7.899 11.6065 4.6148 3.232
MDA-MB-361 CTRP2 7.9071 13.8613 3.5582 7.3191
HCC1419 CTRP2 8.0843 9.3972 5.6205 0.1289
BT-474 CTRP2 8.097 9.6363 5.5403 0.2428
JIMT-1 CTRP2 8.7793 16.3935 2.9332 8.5076
HCC1500 CTRP2 9.1711 22.3934 0.3065 16.7902
AU565 CTRP2 9.1874 19.2181 1.8571 11.8142
CAMA-1 CTRP2 10.8101 27.4568 -0.9973 17.9867
BT 416 CTRP2 2.3975 6.9209 1.7948 26.3954
BT 239 CTRP2 5.1742 6.2954 5.016 6.3651
BT 172 CTRP2 5.2412 7.1965 4.7127 7.3693
BT147 CTRP2 5.6143 7.716 4.8278 6.0095
BT 248 CTRP2 5.7655 8.3427 4.6553 6.4006
BT 504 CTRP2 5.8032 7.3571 5.1776 4.1372
BT 231 CTRP2 5.8312 8.8864 4.4421 7.1581
BT 228 CTRP2 5.9332 7.7612 5.0916 4.2248
BT 286 CTRP2 6.0231 7.6243 5.2367 3.4365
BT 145 CTRP2 6.0258 7.1658 5.4681 2.4583
BT 330 CTRP2 6.0885 8.4743 4.866 4.8687
BT 428 CTRP2 6.0962 8.588 4.8155 5.0665
BT 440 CTRP2 6.1254 8.4965 4.8851 4.7187
BT 131 CTRP2 6.1384 8.3272 4.9804 4.2944
BT 271 CTRP2 6.2442 8.1586 5.1489 3.3957
BT 112 CTRP2 6.5445 9.6465 4.6413 5
BT 444 CTRP2 6.6121 8.7874 5.1124 2.9483
BT 139 CTRP2 6.6168 10.1492 4.4473 5.6852
BT164 CTRP2 6.8226 9.3565 4.9835 3.1622
BT 482 CTRP2 6.8433 10.0301 4.6717 4.3983
BT 216 CTRP2 6.8609 8.7566 5.2933 1.8852
BT 245 CTRP2 6.8675 9.8694 4.7668 3.9739
BT 187 CTRP2 6.9224 11.8418 3.8409 7.687
BT 422 CTRP2 7.0141 11.0702 4.2867 5.7115
BT 328 CTRP2 7.0599 10.2953 4.6941 3.9889
BT 320 CTRP2 7.1515 11.6554 4.0994 6.2648
BT 179 CTRP2 7.1876 10.087 4.8779 3.0856
BT 498 CTRP2 7.2476 14.8494 2.6 12.1039
BT 224 CTRP2 7.7715 10.4685 5.0519 1.7909
BT 359 CTRP2 7.7746 9.7848 5.3437 0.8566
BT 159 CTRP2 8.5787 15.109 3.4101 6.9763
BT 232 CTRP2 9.1294 19.4154 1.7225 12.3579
BT 340 CTRP2 9.4289 19.0834 2.0839 10.6945
BT 333 CTRP2 10.6444 21.1441 1.8971 9.7758
⏷ Show the Full List of 71 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 5.0771 9.1917 3.6065 12.2742
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
GB-1 CTRP2 3.9012 8.3351 2.8405 18.2476
D283 Med CTRP2 4.7426 7.5584 4.0445 11.3106
DBTRG-05MG CTRP2 4.9499 8.3696 3.8789 11.4599
SW1783 CTRP2 4.9873 8.3788 3.911 11.239
NMC-G1 CTRP2 5.0383 11.3219 2.5265 16.709
SF268 CTRP2 5.5038 10.1337 3.5334 11.6318
LN-229 CTRP2 5.8063 10.0342 3.8477 9.6976
42-MG-BA CTRP2 5.8125 11.533 3.1045 12.7531
SF539 CTRP2 5.8345 10.2844 3.747 10.0608
YH-13 CTRP2 5.8728 7.2943 5.2713 3.5966
ONS-76 CTRP2 5.9366 8.8567 4.5474 6.5033
SNU-466 CTRP2 5.969 9.3882 4.3093 7.4393
A-172 CTRP2 6.1921 7.816 5.2785 2.9453
Hs 683 CTRP2 6.2074 8.8515 4.7743 5.0321
SW1088 CTRP2 6.2094 8.8993 4.752 5.1219
KG-1-C CTRP2 6.2336 8.1327 5.1534 3.3956
TM-31 CTRP2 6.298 9.0001 4.7722 4.8777
YKG-1 CTRP2 6.3494 8.7391 4.942 4.0773
GOS-3 CTRP2 6.4376 8.619 5.0683 3.4036
T98G CTRP2 6.4485 8.4938 5.138 3.0972
SNB-75 CTRP2 6.4824 9.2358 4.7974 4.4547
GaMG CTRP2 6.4927 8.193 5.3169 2.2934
KNS-60 CTRP2 6.5474 11.0053 3.9697 7.7906
M059K CTRP2 6.5494 7.8126 5.5374 1.3307
Becker CTRP2 6.5607 10.8852 4.0397 7.4764
SF126 CTRP2 6.6346 9.4789 4.7907 4.2339
LN-18 CTRP2 6.638 9.4571 4.8039 4.1742
8-MG-BA CTRP2 6.6923 9.8799 4.6362 4.7797
SNU-626 CTRP2 6.6971 9.1762 4.9835 3.3459
SNU-201 CTRP2 6.7001 9.2556 4.947 3.4903
KNS-81 CTRP2 6.8302 9.2185 5.0549 2.8648
DK-MG CTRP2 6.8473 10.5746 4.4086 5.4718
SNU-738 CTRP2 6.8561 9.9624 4.7137 4.2075
SNU-489 CTRP2 6.9438 8.7698 5.3383 1.6157
KALS-1 CTRP2 6.9577 11.4329 4.0682 6.696
GMS-10 CTRP2 7.0196 10.007 4.805 3.6006
SF295 CTRP2 7.0206 10.0934 4.7644 3.7623
SNU-1105 CTRP2 7.0259 12.1456 3.7681 7.8162
U-251MG CTRP2 7.443 12.5082 3.8909 6.67
CCF-STTG1 CTRP2 7.4984 11.0528 4.6234 3.68
U-118MG CTRP2 7.6717 17.113 1.8008 14.3424
CAS-1 CTRP2 7.7303 9.3429 5.4996 0.4686
U-87MG ATCC CTRP2 7.7934 9.3972 5.506 0.4237
KNS-42 CTRP2 7.8383 12.921 3.9617 5.8261
Daoy CTRP2 8.6034 16.6793 2.6788 9.6986
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-2 CTRP2 2.9478 6.2521 2.6061 21.8291
JHUEM-1 CTRP2 3.5373 5.2228 3.481 16.8936
RL95-2 CTRP2 4.0233 6.5401 3.6859 14.6712
AN3-CA CTRP2 5.0059 7.6788 4.2564 9.7935
HEC-151 CTRP2 6.0646 8.0426 5.0621 4.0903
JHUEM-7 CTRP2 6.0654 8.9142 4.627 5.9172
HEC-1-A CTRP2 6.0945 9.5451 4.3356 7.0856
JHUEM-3 CTRP2 6.2178 9.4398 4.489 6.2106
MFE-296 CTRP2 6.2549 10.2322 4.1232 7.6754
ESS-1 CTRP2 6.6095 8.1692 5.408 1.7608
EN CTRP2 6.7374 8.4415 5.3624 1.7725
HEC-59 CTRP2 6.7764 9.995 4.641 4.6273
HEC-108 CTRP2 6.9484 9.554 4.9737 3.0254
HEC-265 CTRP2 7.1143 8.8813 5.3871 1.2569
EFE-184 CTRP2 7.1823 11.1696 4.3569 5.1728
MFE-319 CTRP2 7.3325 9.059 5.4269 0.9288
HEC-6 CTRP2 7.6673 11.7031 4.4262 4.2317
HEC-251 CTRP2 7.8547 11.4032 4.6811 3.0354
KLE CTRP2 8.0497 11.8442 4.5962 3.1335
HEC-50B CTRP2 8.2042 11.981 4.6242 2.8679
HEC-1-B CTRP2 8.695 17.7823 2.2106 11.2778
Ishikawa (Heraklio) 02 ER- CTRP2 6.8272 11.4865 3.945 7.4156
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UO-31 CTRP2 3.6619 10.839 1.4564 23.9855
CAL-54 CTRP2 5.2822 7.7571 4.4922 8.1617
TUHR14TKB CTRP2 5.4338 14.1607 1.4668 33.5352
ACHN CTRP2 5.7186 7.9582 4.804 5.8789
OS-RC-2 CTRP2 5.8487 10.1685 3.8171 9.74
BFTC-909 CTRP2 6.1688 9.5751 4.3816 6.7523
786-O CTRP2 6.6036 9.8465 4.5869 5.1279
TUHR10TKB CTRP2 6.6591 11.2793 3.9199 7.8035
KMRC-1 CTRP2 6.6974 10.8632 4.1552 6.7629
KMRC-2 CTRP2 6.768 9.8304 4.7153 4.3349
TUHR4TKB CTRP2 6.7886 12.3647 3.481 9.3874
KMRC-3 CTRP2 6.8986 11.7817 3.8528 7.6772
VMRC-RCZ CTRP2 6.9357 9.8955 4.8015 3.734
Caki-1 CTRP2 6.9651 10.9929 4.2892 5.7773
Caki-2 CTRP2 7.1158 10.3805 4.6911 3.9222
VMRC-RCW CTRP2 7.1234 10.4081 4.6831 3.9436
SNU-1272 CTRP2 7.147 10.5684 4.6222 4.1545
RCC10RGB CTRP2 7.3608 10.1726 4.947 2.6055
A-498 CTRP2 7.5141 19.3312 0.5826 18.6383
769-P CTRP2 7.8089 11.1006 4.7915 2.6792
KMRC-20 CTRP2 8.2838 13.5513 3.9527 5.2811
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 47 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-175 CTRP2 3.3401 10.9786 1.0746 26.109
NCI-H716 CTRP2 3.6001 6.5922 3.2095 17.6776
SW48 CTRP2 3.8844 4.9568 3.8729 14.4288
KM12 CTRP2 4.2111 8.4232 3.1181 16.3536
HCT 15 CTRP2 4.4274 7.0862 3.9162 12.6537
COLO205 CTRP2 4.6293 10.2385 2.6764 17.065
SNU-81 CTRP2 4.724 8.9453 3.3867 14.0008
LoVo CTRP2 4.8874 7.7588 4.1011 10.715
HT115 CTRP2 4.8952 7.2987 4.3151 9.8414
SNU-C1 CTRP2 4.9724 9.1985 3.5042 12.9349
GP2d CTRP2 5.1053 8.2469 4.0881 10.2347
LS513 CTRP2 5.1957 6.9461 4.7781 7.2257
SW620 CTRP2 5.2219 7.5131 4.5478 8.0815
SNU-407 CTRP2 5.3538 7.783 4.5489 7.7596
SW948 CTRP2 5.414 7.5491 4.7186 6.922
COLO 320 CTRP2 5.4147 10.9228 3.0624 13.7511
CW-2 CTRP2 5.525 8.4308 2.9647 2.944
CL-11 CTRP2 5.6456 9.762 3.8436 10.0451
COLO 678 CTRP2 5.6469 9.1966 4.1259 8.8642
SW1417 CTRP2 5.8726 7.8326 5.0034 4.7188
T84 CTRP2 5.9636 8.9496 4.5239 6.5488
NCI-H508 CTRP2 5.9725 7.1107 5.4502 2.64
SNU-C5 CTRP2 5.9777 9.3957 4.3128 7.4074
LS1034 CTRP2 5.9996 6.8611 5.5981 1.9641
HCC-56 CTRP2 6.1474 7.0257 5.6367 1.5247
SNU-1033 CTRP2 6.2363 8.5184 4.9634 4.1866
LS180 CTRP2 6.239 9.2116 4.6199 5.6223
RKO CTRP2 6.358 14.3649 2.1425 15.4464
NCI-H747 CTRP2 6.4022 9.3495 4.6797 5.0817
SNU-61 CTRP2 6.4684 9.8279 4.4934 5.7451
SK-CO-1 CTRP2 6.4799 8.7019 5.0588 3.3744
HCT 116 CTRP2 6.5915 8.1206 5.4192 1.7407
SNU-C4 CTRP2 6.5942 8.3417 5.3153 2.1517
DLD-1 CTRP2 6.6417 8.2984 5.3679 1.8763
HCT 8 CTRP2 6.6831 9.0608 5.0296 3.1791
C2BBe1 CTRP2 6.7769 9.1348 5.0588 2.9243
MDST8 CTRP2 6.7883 8.9038 5.177 2.4352
COLO201 CTRP2 6.8234 15.8469 1.7763 15.9132
SNU-503 CTRP2 7.0162 10.407 4.6103 4.3903
HT-55 CTRP2 7.1683 8.622 5.5279 0.7405
LS411N CTRP2 7.2783 8.6369 5.5751 0.5251
SNU-C2A CTRP2 7.4178 12.7247 3.7681 7.202
OUMS-23 CTRP2 7.4349 13.04 3.6268 7.7441
LS123 CTRP2 7.5339 9.8977 5.1718 1.6019
HT-29 CTRP2 7.7489 9.0544 5.6159 0.2186
RCM-1 [Human ESC] CTRP2 7.7999 9.2413 5.5675 0.291
CCK-81 CTRP2 7.9544 10.7962 5.0081 1.7723
⏷ Show the Full List of 47 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Li-7 CTRP2 4.5509 8.5467 3.4031 14.3598
SNU-886 CTRP2 5.2879 10.7083 3.0555 14.0535
SNU-761 CTRP2 5.4116 9.0936 3.3171 7.6101
SNU-449 CTRP2 5.479 8.2389 4.4464 7.894
SNU-878 CTRP2 5.515 7.3843 4.8946 5.9622
SNU-387 CTRP2 5.7238 9.0069 4.2882 8.0243
SNU-182 CTRP2 5.7974 13.0148 2.3513 15.7636
JHH-1 CTRP2 5.815 7.5219 5.1067 4.4076
JHH-4 CTRP2 6.0688 8.9002 4.6368 5.8698
Hep 3B2.1-7 CTRP2 6.1848 13.9487 2.2086 15.533
HLF CTRP2 6.2132 12.7638 2.8244 13.0908
Hep-G2 CTRP2 6.2705 9.4305 4.5359 5.9175
JHH-5 CTRP2 6.2747 9.9813 4.2644 7.0478
SK-HEP-1 CTRP2 6.4319 9.1648 4.7942 4.5528
HuH-6 CTRP2 6.4798 10.6963 4.0706 7.4895
HuH-1 CTRP2 6.5487 10.7972 4.0741 7.3538
SNU-423 CTRP2 6.5732 9.7251 4.624 5.0238
JHH-6 CTRP2 7.0165 8.0257 5.6992 0.3481
SNU-475 CTRP2 7.2461 11.4698 4.2562 5.4866
JHH-2 CTRP2 7.3303 11.905 4.1043 5.9765
PLC/PRF/5 CTRP2 7.5217 9.7955 5.2099 1.4824
SNU-398 CTRP2 8.0785 12.4785 4.3231 4.1204
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 142 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1734 CTRP2 3.1882 7.0861 2.5916 21.1693
HCC44 CTRP2 3.359 7.2559 2.7123 20.2287
COR-L51 CTRP2 3.3823 5.5395 3.2598 18.1561
NCI-H1975 CTRP2 3.5155 6.9036 3.01 18.6659
NCI-H1563 CTRP2 3.5544 5.6812 3.4168 17.0631
EPLC-272H CTRP2 3.9061 7.6857 3.1225 17.1443
NCI-H358 CTRP2 3.9196 9.9396 2.1311 20.9042
NCI-H2087 CTRP2 4.1352 12.8403 0.9485 24.4642
DV-90 CTRP2 4.2453 7.3605 3.6127 14.3253
HCC15 CTRP2 4.2776 8.0143 3.3675 15.1984
LCLC-97TM1 CTRP2 4.3742 8.9068 3.061 16.1646
NCI-H1568 CTRP2 4.4087 7.2516 3.8293 13.0411
NCI-H1755 CTRP2 4.493 7.5659 3.7845 12.9908
NCI-H1581 CTRP2 4.4943 8.1268 3.5381 13.963
Lu-99 CTRP2 4.5458 9.1275 3.1269 15.4781
NCI-H1666 CTRP2 4.585 10.5228 2.4971 17.8699
HCC2108 CTRP2 4.6967 9.7547 2.9737 15.727
NCI-H2081 CTRP2 4.72 7.7285 3.9458 11.7618
EKVX CTRP2 4.7984 8.271 3.7764 12.2445
HARA [Human squamous cell lung carcinoma] CTRP2 4.808 6.8742 4.4037 9.7273
NCI-H2122 CTRP2 4.8412 6.2898 4.657 8.6723
HCC1588 CTRP2 4.8913 6.5973 4.6012 8.7383
NCI-H2110 CTRP2 4.9541 7.8975 4.104 10.5368
NCI-H1355 CTRP2 4.97 11.7267 2.2647 17.871
NCI-H2405 CTRP2 4.9755 9.214 3.4997 12.9461
NCI-H2085 CTRP2 4.9755 9.8758 1.896 8.7445
HCC827 CTRP2 5.0182 9.7039 3.3021 13.6535
LXF 289 CTRP2 5.1691 8.8068 3.8798 10.9398
Lu-65 CTRP2 5.199 7.6754 4.4495 8.5366
HOP-62 CTRP2 5.2057 11.1047 2.7853 15.318
A-549 CTRP2 5.253 7.8549 4.4174 8.5372
RERF-LC-MS CTRP2 5.2727 7.5329 4.5886 7.7918
PC-14 CTRP2 5.2856 8.3789 4.1971 9.3649
NCI-H1184 CTRP2 5.3142 10.3354 3.2636 13.1493
SK-MES-1 CTRP2 5.3144 8.1793 4.3209 8.7884
NCI-H810 CTRP2 5.3164 8.1128 4.3548 8.6439
VMRC-LCD CTRP2 5.3333 7.8004 4.5209 7.9228
HCC4006 CTRP2 5.3499 9.2296 3.8416 10.6895
NCI-H647 CTRP2 5.3852 10.03 3.4787 12.1125
NCI-H1341 CTRP2 5.3992 8.5684 4.2113 9.0476
NCI-H1155 CTRP2 5.4059 8.1945 4.3999 8.252
NCI-H1944 CTRP2 5.4377 8.4902 4.2852 8.6548
NCI-H211 CTRP2 5.4384 8.5495 4.2568 8.7713
COR-L279 CTRP2 5.4558 7.2781 4.8878 6.1314
DMS 53 CTRP2 5.4587 8.1319 4.4798 7.8019
NCI-H1703 CTRP2 5.475 7.8995 4.6081 7.2343
NCI-H841 CTRP2 5.5024 11.0994 3.0522 13.6063
NCI-H69 CTRP2 5.5296 7.2609 4.9676 5.6287
Calu-3 CTRP2 5.538 11.4283 2.9196 14.066
NCI-H446 CTRP2 5.6743 7.9199 4.7828 6.0636
NCI-H1373 CTRP2 5.6745 9.2899 4.1039 8.8982
HCC95 CTRP2 5.7217 8.3477 4.6138 6.6664
HOP-92 CTRP2 5.7742 18.1917 -0.2559 24.3321
CAL-12T CTRP2 5.778 11.1886 3.2471 12.2414
NCI-H2009 CTRP2 5.787 9.6092 4.0432 8.9199
HCC1171 CTRP2 5.8856 12.2589 2.8038 13.8159
NCI-H1694 CTRP2 5.9124 7.5639 5.1721 3.9296
NCI-H2444 CTRP2 5.9227 7.8763 4.2763 2.169
NCI-H526 CTRP2 5.923 8.2261 4.8508 5.2564
SHP-77 CTRP2 5.9381 7.7125 5.1202 4.0946
NCI-H1915 CTRP2 6.0115 9.0924 4.4929 6.5851
HCC1438 CTRP2 6.0171 10.2248 3.9315 8.929
SK-LU-1 CTRP2 6.0408 9.801 4.1631 7.9126
NCI-H2106 CTRP2 6.0511 10.0395 4.0524 8.3568
NCI-H2286 CTRP2 6.0552 11.0894 3.5309 10.5223
LK2 CTRP2 6.0689 6.7915 5.6911 1.4385
NCI-H2228 CTRP2 6.0981 10.8474 3.6875 9.7899
Calu-6 CTRP2 6.116 8.4628 4.8944 4.6975
EBC-1 CTRP2 6.1279 8.5949 4.8381 4.9118
HCC1195 CTRP2 6.1504 9.7851 4.2616 7.2903
DMS 454 CTRP2 6.1685 9.3925 4.4726 6.3706
NCI-H23 CTRP2 6.1903 8.9082 4.7321 5.2408
NCI-H889 CTRP2 6.1948 9.2834 4.5485 6.0035
MOR/CPR CTRP2 6.2614 8.081 5.2008 3.1489
LUDLU-1 CTRP2 6.302 8.4961 5.026 3.8085
NCI-H460 CTRP2 6.3341 7.5712 5.5069 1.7579
NCI-H292 CTRP2 6.3502 10.3683 4.1317 7.4658
COR-L105 CTRP2 6.3723 8.4963 5.0798 3.4638
NCI-H650 CTRP2 6.3732 11.0925 3.7889 8.8537
NCI-H661 CTRP2 6.3854 11.2834 2.9594 6.936
NCI-H2141 CTRP2 6.3901 8.4459 5.1181 3.2749
NCI-H226 CTRP2 6.3925 8.9457 4.8727 4.2927
NCI-H2030 CTRP2 6.4111 11.7305 3.5009 9.9763
NCI-H727 CTRP2 6.4202 9.688 4.5255 5.6945
NCI-H838 CTRP2 6.4254 10.0437 4.3527 6.4077
NCI-H522 CTRP2 6.4434 8.0703 5.3416 2.2671
NCI-H1395 CTRP2 6.4491 9.0922 4.8433 4.3195
NCI-H1105 CTRP2 6.4596 8.324 5.2294 2.7027
NCI-H1339 CTRP2 6.4628 9.0606 4.8692 4.1886
DMS 273 CTRP2 6.4734 7.9657 5.4135 1.9292
COR-L95 CTRP2 6.4861 8.2083 5.3048 2.3528
NCI-H1435 CTRP2 6.5106 10.4015 4.2411 6.7245
DMS 114 CTRP2 6.5357 9.3007 4.8054 4.3331
NCI-H1838 CTRP2 6.5359 10.7373 4.0939 7.2938
NCI-H2291 CTRP2 6.6156 9.0818 4.9714 3.5198
SW1271 CTRP2 6.664 10.2572 4.4294 5.6812
NCI-H1623 CTRP2 6.6816 10.1204 4.51 5.3188
RERF-LC-A1 CTRP2 6.6897 11.3644 3.9012 7.8286
DMS 79 CTRP2 6.7185 8.2926 5.4201 1.5727
HCC2279 CTRP2 6.7595 10.7411 4.2621 6.2174
NCI-H2196 CTRP2 6.7639 11.5187 3.8813 7.7846
IA-LM CTRP2 6.765 10.603 4.3342 5.9104
NCI-H1693 CTRP2 6.8004 10.3713 4.4741 5.276
NCI-H1092 CTRP2 6.8049 8.5945 5.3337 1.799
NCI-H2126 CTRP2 6.8706 10.8843 4.2737 5.9898
LOU-NH91 CTRP2 6.8759 12.5548 3.4536 9.3495
COLO 668 CTRP2 6.9002 10.4509 4.5072 4.9843
NCI-H322 CTRP2 6.9187 9.405 5.025 2.8622
NCI-H520 CTRP2 6.9225 9.6995 4.8867 3.4096
NCI-H1573 CTRP2 6.9256 16.795 1.3847 17.093
T3M-10 CTRP2 6.9629 9.1708 5.1643 2.2569
HCC366 CTRP2 7.0245 10.5016 4.5703 4.5402
NCI-H2170 CTRP2 7.0389 9.2397 5.1799 2.1031
NCI-H2029 CTRP2 7.0398 8.3588 5.5737 0.6972
RERF-LC-Ad1 CTRP2 7.1555 8.1506 5.7114 0.2489
NCI-H2342 CTRP2 7.1733 11.2364 4.3184 5.3421
NCI-H1869 CTRP2 7.1863 12.2445 3.8368 7.28
NCI-H196 CTRP2 7.1974 10.407 4.7329 3.6438
HCC1833 CTRP2 7.2375 13.0645 3.4722 8.6763
KNS-62 CTRP2 7.2487 11.1962 4.3899 4.9434
BEN CTRP2 7.3499 8.2008 5.7693 0.0872
COLO 699 CTRP2 7.4323 13.9961 3.1575 9.6219
HCC2935 CTRP2 7.4644 13.118 3.6097 7.7677
NCI-H1792 CTRP2 7.5532 14.7751 2.8637 10.5809
HCC78 CTRP2 7.5732 10.4956 4.9269 2.4388
SBC-5 CTRP2 7.6198 8.4134 5.7918 0.0305
RERF-LC-Ad2 CTRP2 7.662 11.4116 4.5592 3.7233
Calu-1 CTRP2 7.7735 15.7579 2.5425 11.459
Sq-1 CTRP2 7.8096 14.0226 3.4134 8.0307
NCI-H1299 CTRP2 7.8704 11.8086 4.5046 3.6797
LCLC-103H CTRP2 8.0733 9.6966 5.5089 0.3062
COR-L88 CTRP2 8.118 10.1014 5.3744 0.5762
SW1573 CTRP2 8.1214 12.5877 4.2991 4.1603
NCI-H2023 CTRP2 8.1413 9.6906 5.5378 0.2342
LC-1/sq-SF CTRP2 8.2117 9.2936 5.7001 0.04
NCI-H441 CTRP2 8.2466 14.7404 3.3664 7.5901
ChaGo-K-1 CTRP2 8.2754 10.3272 5.3552 0.5459
NCI-H1793 CTRP2 8.4527 18.3549 1.7625 13.2254
NCI-H2172 CTRP2 8.5773 13.883 3.9809 4.8202
NCI-H1650 CTRP2 8.6446 11.6934 4.98 1.3202
NCI-H1385 CTRP2 8.8428 54.179 -15.7324 37.8944
Hs 888.Lu CTRP2 5.0557 8.058 4.1291 10.1865
⏷ Show the Full List of 142 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 4.8573 9.0224 3.4789 13.3086
A2780 CTRP2 3.5475 7.0416 2.9944 18.6326
COV434 CTRP2 4.8858 8.5639 3.7246 12.2416
IGROV-1 CTRP2 5.1675 8.4225 4.0638 10.1873
HEY A8 CTRP2 5.424 8.0291 4.4972 7.809
OVTOKO CTRP2 5.4312 9.6784 3.6941 11.1225
OVK18 CTRP2 5.9214 7.5142 5.2047 3.7743
TOV-21G CTRP2 6.1103 7.7364 5.2527 3.2028
SK-OV-3 CTRP2 6.1595 9.1396 4.5916 5.8878
EFO-21 CTRP2 6.1659 7.7819 5.2747 3.0084
MCAS CTRP2 6.2021 9.7561 4.3183 6.9558
OV-90 CTRP2 6.2388 7.7572 5.3441 2.5889
SNU-119 CTRP2 6.2857 11.1219 3.7038 9.3678
TYK-nu CTRP2 6.5184 10.4186 4.2387 6.7209
JHOS-2 CTRP2 6.526 10.3934 4.2571 6.6314
Caov-3 CTRP2 6.566 10.3734 4.2978 6.3931
OAW42 CTRP2 6.5952 8.2531 5.3585 1.9774
SNU-840 CTRP2 6.7931 11.838 3.7454 8.2954
OVCAR-5 CTRP2 6.8236 12.6888 3.3471 9.8721
JHOC-5 CTRP2 6.9854 9.4856 5.0307 2.7503
FU-OV-1 CTRP2 7.0738 12.9194 3.4225 9.1435
RMG-I CTRP2 7.1094 10.8678 4.4523 4.8937
OV7 CTRP2 7.1124 13.0836 3.3704 9.2906
SNU-8 CTRP2 7.1281 12.9904 3.4279 9.0323
TOV-112D CTRP2 7.1316 9.4543 5.1378 2.1527
OVCAR-8 CTRP2 7.1388 10.0778 4.8506 3.2571
JHOM-1 CTRP2 7.1767 11.5534 4.167 5.9514
COV644 CTRP2 7.1962 9.6914 5.068 2.3411
OAW28 CTRP2 7.247 11.3867 4.2969 5.3207
OVCAR-4 CTRP2 7.3784 11.1059 4.5204 4.2414
DOV13 CTRP2 7.4418 10.6852 4.7595 3.2244
Kuramochi CTRP2 7.523 11.8973 4.2395 5.159
COV362 CTRP2 7.6593 11.2389 4.6378 3.4253
EFO-27 CTRP2 7.6752 11.3308 4.6051 3.5312
OVISE CTRP2 7.8252 8.9461 5.6831 0.102
ONCO-DG-1 CTRP2 7.9944 11.1878 4.8585 2.2484
OC 314 CTRP2 8.0836 14.149 3.5397 7.1436
OVSAHO CTRP2 8.4683 15.7466 3.0343 8.5538
ES2 CTRP2 8.8946 13.9766 4.1264 3.9362
OV56 CTRP2 9.8971 26.8483 -1.3477 20.1035
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 6.3404 9.3259 4.6434 5.3417
Aska-SS CTRP2 6.5938 10.0136 4.497 5.5172
A-204 CTRP2 4.231 9.9831 2.4158 19.043
TTC-709 CTRP2 4.3416 7.6028 3.6119 14.0693
Rh41 CTRP2 4.7349 6.1858 4.5744 9.291
G-401 CTRP2 4.8448 7.3068 4.2598 10.192
KYM-1 CTRP2 4.8531 6.8048 4.4794 9.3115
GCT CTRP2 5.1279 8.4376 4.0186 10.4655
TE 617.T CTRP2 5.2466 7.2422 4.6973 7.4171
TE 441.T CTRP2 5.2657 7.5427 4.5771 7.856
MES-SA CTRP2 5.4578 7.9659 4.5596 7.4738
HT-1080 CTRP2 5.6063 7.9789 4.6915 6.5928
SW982 CTRP2 5.6725 9.2318 4.131 8.7891
G-402 CTRP2 5.9597 8.8717 4.5596 6.4064
SK-LMS-1 CTRP2 6.2522 9.5939 4.4397 6.3541
Rh18 CTRP2 6.2812 12.6351 2.9443 12.4823
BT-16 CTRP2 6.3334 8.0775 5.2575 2.7899
Tm87-16 CTRP2 6.4512 9.9027 4.4429 5.9856
BT-12 CTRP2 6.5095 9.3479 4.7624 4.555
SK-UT-1 CTRP2 6.764 10.7609 4.2557 6.2365
Hs 729.T CTRP2 6.8939 10.5341 4.4621 5.1791
RD CTRP2 6.9685 10.0875 4.7316 3.969
RKN CTRP2 7.1666 10.1049 4.8559 3.1992
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 6.67 11.7715 3.684 8.7594
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 7.3039 8.474 5.6508 0.3185
SYO-1 CTRP2 7.3501 10.8054 4.6443 3.7901
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2 3.5894 7.6438 2.8062 19.2255
NCI-H2452 CTRP2 4.6779 8.9075 3.3597 14.2217
IST-Mes1 CTRP2 6.156 7.8865 5.2146 3.2783
MPP 89 CTRP2 6.243 8.557 4.9495 4.2327
NCI-H2052 CTRP2 6.3583 12.2063 1.7286 7.1724
NCI-H28 CTRP2 6.385 8.2555 5.2083 2.9093
ACC-MESO-1 CTRP2 7.1016 9.4029 5.1431 2.1682
JL-1 CTRP2 7.6684 10.9871 4.7596 2.9539
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
VCaP CTRP2 4.6777 7.4513 4.0247 11.5583
LNCaP clone FGC CTRP2 5.8668 8.2074 4.8115 5.5355
PaCa-3 CTRP2 6.7559 8.0746 5.5431 1.0662
22Rv1 CTRP2 7.2305 13.9066 3.0526 10.3656
DU145 CTRP2 7.2396 11.5138 4.2304 5.6005
NCI-H660 CTRP2 9.5699 36.3947 -6.302 29.365
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 4.0062 7.1724 3.4353 15.6664
A-253 CTRP2 7.4524 10.6531 4.781 3.1285
Cancer Drug Sensitivity Data Curated from 34 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OCUM-1 CTRP2 3.72 7.9364 2.8233 18.8011
SNU-16 CTRP2 3.7787 6.0218 3.5779 15.7959
HGC-27 CTRP2 3.8233 5.3849 3.7635 15.0007
Fu97 CTRP2 3.9179 6.3933 3.6198 15.2255
ECC10 CTRP2 4.5019 7.1684 3.9614 12.2754
GSS CTRP2 4.585 6.6583 4.2501 10.9368
SNU-719 CTRP2 5.0263 8.4576 3.9114 11.1445
KATO III CTRP2 5.0335 9.0541 3.6319 12.2709
SNU-620 CTRP2 5.0759 7.6447 4.3419 9.2748
SNU-668 CTRP2 5.1219 9.0148 3.7345 11.6458
SNU-1 CTRP2 5.2406 7.2441 4.6904 7.4601
SNU-5 CTRP2 5.5448 8.9759 4.144 9.0066
NUGC-4 CTRP2 5.6375 8.2222 4.6002 6.9041
SNU-216 CTRP2 5.9943 12.2643 2.8926 13.2448
LMSU CTRP2 6.0017 8.3205 4.8705 5.0172
NCI-N87 CTRP2 6.0728 8.5077 4.8363 5.0235
GSU CTRP2 6.1361 6.9066 5.6871 1.3338
SNU-601 CTRP2 6.1394 7.9799 5.1547 3.5604
23132/87 CTRP2 6.22 9.9745 4.2237 7.3195
ECC12 CTRP2 6.3366 7.7905 5.4013 2.1889
KE-39 CTRP2 6.3419 11.2017 3.7093 9.2415
IM95 CTRP2 6.367 8.5766 5.0361 3.655
AGS CTRP2 6.4868 8.6652 5.0819 3.2678
Hs 746.T CTRP2 6.5026 8.374 5.2359 2.6095
HuG1-N CTRP2 6.6355 9.1833 4.9362 3.6337
MKN1 CTRP2 6.9365 9.1974 5.135 2.4047
MKN74 CTRP2 7.0019 12.1107 3.7676 7.8572
SH-10-TC CTRP2 7.162 9.2099 5.2675 1.6361
NUGC-3 CTRP2 7.2231 10.5606 4.6769 3.8311
MKN45 CTRP2 7.2743 8.2589 5.7196 0.1859
MKN7 CTRP2 7.7523 11.7957 4.4369 4.0827
SNG-M CTRP2 5.8488 7.9463 4.9258 5.0934
SNU-1077 CTRP2 6.481 9.9174 4.4586 5.8686
SNU-685 CTRP2 7.0694 10.2477 4.7234 3.8579
⏷ Show the Full List of 34 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ML-1 [Human leukemia] CTRP2 4.4561 8.2505 3.4437 14.4362
8305C CTRP2 4.4575 8.1319 3.4986 14.2142
B-CPAP CTRP2 4.7996 7.0628 4.3172 10.0862
CGTH-W-1 CTRP2 4.9257 6.5856 4.6424 8.4844
SW579 CTRP2 5.0803 7.9627 4.1981 9.8463
8505C CTRP2 5.7331 9.8336 3.8845 9.6933
TT2609-C02 CTRP2 5.8384 8.4096 4.6861 6.1199
FTC-238 CTRP2 5.8399 8.0554 4.8637 5.3722
CAL-62 CTRP2 6.4413 8.4376 5.1603 3.0165
BHT-101 CTRP2 6.7552 10.0139 4.6163 4.7617
TT CTRP2 6.7666 10.831 4.2231 6.3671
FTC-133 CTRP2 7.7854 9.9749 5.2704 1.0665
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 29 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 1.9048 5.7537 1.6026 28.6051
SCC-25 CTRP2 4.2563 8.0516 3.3293 15.4046
HSC-3 CTRP2 4.7191 7.6751 3.9687 11.673
CAL-27 CTRP2 4.7385 7.9751 3.853 12.0853
SNU-1214 CTRP2 4.7459 9.234 3.2706 14.4174
PE/CA-PJ34 (clone C12) CTRP2 4.9239 8.1101 3.9753 11.1321
SNU-899 CTRP2 4.964 8.0466 4.0445 10.7532
PE/CA-PJ15 CTRP2 5.0166 8.5367 3.8643 11.3598
SNU-1041 CTRP2 5.1084 9.3841 3.5422 12.4661
Detroit 562 CTRP2 5.2391 14.4013 1.1773 21.1615
HSC-2 CTRP2 5.4494 8.254 4.4116 8.1049
CAL-33 CTRP2 5.4645 9.4847 3.8199 10.5288
SNU-1076 CTRP2 5.4768 13.9903 1.589 19.239
BICR 56 CTRP2 5.5392 12.1488 2.5616 15.4839
YD-8 CTRP2 5.622 8.0344 4.6786 6.6118
BICR 31 CTRP2 5.8543 8.3925 4.7084 5.9938
BHY CTRP2 5.8942 12.5867 2.6473 14.4179
SCC-9 CTRP2 5.931 10.264 3.8393 9.4829
PE/CA-PJ49 CTRP2 5.9457 9.7303 4.1185 8.2857
SNU-46 CTRP2 5.9554 13.9824 2.001 16.7623
BICR 22 CTRP2 6.0396 8.7719 4.6766 5.7585
BICR 18 CTRP2 6.0877 8.5002 4.8524 4.9276
BICR 6 CTRP2 6.1275 10.2854 3.9927 8.4606
BICR 16 CTRP2 6.4874 8.9349 4.9497 3.8139
FaDu CTRP2 6.5869 10.0453 4.4761 5.6156
HSC-4 CTRP2 6.6874 11.2219 3.97 7.5475
PE/CA-PJ41 (clone D2) CTRP2 6.8174 9.6427 4.8416 3.7442
SNU-1066 CTRP2 7.0779 12.047 3.8548 7.3783
SCC-4 CTRP2 7.8071 18.0943 1.418 15.4426
⏷ Show the Full List of 29 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JMSU-1 CTRP2 3.7766 6.3436 3.4817 16.1525
5637 CTRP2 4.1157 7.2619 3.5161 15.053
U-BLC1 CTRP2 4.8717 11.3459 2.3625 17.7206
SCaBER CTRP2 4.9168 9.4998 3.3059 13.8716
RT-112 CTRP2 5.0309 9.0097 3.6509 12.1992
VM-CUB-1 CTRP2 5.0623 8.8542 3.7557 11.6968
BC-3C CTRP2 5.2731 9.5593 3.609 11.8212
UM-UC-1 CTRP2 5.5503 9.2797 3.9985 9.6011
T24 CTRP2 5.7263 10.5257 3.5334 11.1677
HT-1197 CTRP2 5.9111 9.2358 4.3363 15.7515
KU-19-19 CTRP2 6.1295 8.5399 4.8668 4.7878
SW1710 CTRP2 6.1447 9.2507 4.5241 6.1994
253J-BV CTRP2 6.3517 8.1127 5.2538 2.7751
647V CTRP2 6.4545 9.3655 4.712 4.857
KMBC-2 CTRP2 6.4621 9.4738 4.6642 5.0436
CAL-29 CTRP2 6.5895 9.5398 4.7275 4.5678
RT-4 CTRP2 6.702 10.2795 4.4468 5.5471
639V CTRP2 7.203 8.3141 5.6689 0.3247
HT-1376 CTRP2 7.2194 13.8897 3.0527 10.3837
UM-UC-3 CTRP2 7.4234 12.4512 3.9048 6.6432
J82 CTRP2 7.5495 12.014 4.2016 5.2733
BFTC-905 CTRP2 7.7742 8.869 5.6913 0.1016
TCCSUP CTRP2 7.7754 16.7627 2.0505 13.2769
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 2.9248 4.3137 2.9158 20.8132

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