Details of the Drug

General Information of Drug (ID: DMDSL4E)

Drug Name
Azapropazone
Synonyms
Azapropazone; APAZONE; Cinnopropazone; Prolixan; Azapropazonum; Azapropazona; Cinnamin; Rheumox; Sinnamin; Mitrolan; Azapropazon; Prolix; Xani; Azapropazone (anhydrous); 13539-59-8; AHR-3018; Prolixan 300; MI 85; AHR 3018; Apazone [USAN]; Azapropazon [German]; Mi-85; NSC-102824; Azapropazonum [INN-Latin]; Azapropazona [INN-Spanish]; NSC 102824; 5-(Dimethylamino)-9-methyl-2-propyl-1H-pyrazolo(1,2-a)(1,2,4)benzotriazine-1,3(2H)-dione; C16H20N4O2; 3-Dimethylamino-7-methyl-1,2-(n-propylmalonyl)-1,2-dihydro-1,2,4-benzotriazine; EINECS 236-9
Indication
Disease Entry ICD 11 Status REF
Inflammation 1A00-CA43.1 Withdrawn from market [1]
ATC Code
M01AX04: Azapropazone
M01AX: Other antiinflammatory and antirheumatic agents, non-steroids
M01A: ANTIINFLAMMATORY AND ANTIRHEUMATIC PRODUCTS, NON-STEROIDS
M01: ANTIINFLAMMATORY AND ANTIRHEUMATIC PRODUCTS
M: MUSCULO-SKELETAL SYSTEM
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
Chemical Identifiers
Formula
C16H20N4O2
Canonical SMILES
CCCC1C(=O)N2C3=C(C=CC(=C3)C)N=C(N2C1=O)N(C)C
InChI
InChI=1S/C16H20N4O2/c1-5-6-11-14(21)19-13-9-10(2)7-8-12(13)17-16(18(3)4)20(19)15(11)22/h7-9,11H,5-6H2,1-4H3
InChIKey
MPHPHYZQRGLTBO-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
26098
ChEBI ID
CHEMBL38010
CAS Number
13539-59-8
UNII
K2VOT966ZI
DrugBank ID
DB07402
TTD ID
D01EQG
Drug Pharmacogenomic Perturbation (DPP)NEW Click to Jump to the Detailed DPP Information of This Drug
Drug ADMET Endpoint Profile (DAE)NEW Click to Jump to the Detailed DAE Information of This Drug

References

1 Drugs@FDA. U.S. Food and Drug Administration. U.S. Department of Health & Human Services. 2015