General Information of Drug (ID: DMI7A6R)

Drug Name
Narciclasine
Synonyms
Narciclasine; Lycoricidinol; 29477-83-6; Lycoricidin-A; Narciclasina; NSC 266535; BRN 1087400; NSC266535; Lycorcidinol; Nacriclasine; C14H13NO7; CHEMBL98745; 3,4,4a,5-Tetrahydro-2,3,4,7-tetrahydroxy-(1,3)dioxolo(4,5-j)phenanthridin-6(2H)-one; CHEBI:70169; (2s,3r,4s,4ar)-2,3,4,7-tetrahydroxy-3,4,4a,5-tetrahydro[1,3]dioxolo[4,5-j]phenanthridin-6(2h)-one; (2S,3R,4S,4aR)-2,3,4,7-Tetrahydroxy-3,4,4a,5-tetrahydro-2H-[1,3]dioxolo[4,5-j]phenanthridin-6-one
Indication
Disease Entry ICD 11 Status REF
Melanoma 2C30 Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 307.25
Logarithm of the Partition Coefficient (xlogp) -1.2
Rotatable Bond Count (rotbonds) 0
Hydrogen Bond Donor Count (hbonddonor) 5
Hydrogen Bond Acceptor Count (hbondacc) 7
Chemical Identifiers
Formula
C14H13NO7
IUPAC Name
(2S,3R,4S,4aR)-2,3,4,7-tetrahydroxy-3,4,4a,5-tetrahydro-2H-[1,3]dioxolo[4,5-j]phenanthridin-6-one
Canonical SMILES
C1OC2=C(O1)C(=C3C(=C2)C4=C[C@@H]([C@H]([C@H]([C@@H]4NC3=O)O)O)O)O
InChI
InChI=1S/C14H13NO7/c16-6-1-5-4-2-7-13(22-3-21-7)11(18)8(4)14(20)15-9(5)12(19)10(6)17/h1-2,6,9-10,12,16-19H,3H2,(H,15,20)/t6-,9+,10+,12-/m0/s1
InChIKey
LZAZURSABQIKGB-AEKGRLRDSA-N
Cross-matching ID
PubChem CID
72376
ChEBI ID
CHEBI:70169
CAS Number
29477-83-6
TTD ID
D0OQ1I

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Elongation factor 1A (EF1A) TT8R0BZ EF1A1_HUMAN ; EF1A2_HUMAN Inhibitor [1]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 148 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 -5.1117 -0.8239 -5.133 66.6944
MEC1 CTRP2 -4.5077 -2.7797 -4.5077 63.6326
JM1 CTRP2 -5.0218 -2.1234 -5.0231 66.862
NU-DUL-1 CTRP2; CTRP1 -7.4777 -6.755 -7.4777 83.4385
SKM-1 CTRP2; CTRP1 -7.4299 -6.8767 -7.4299 83.1221
EoL-1 CTRP2 -7.2959 -6.6401 -7.2959 82.2123
MOLM-6 CTRP2 -7.2813 -3.6558 -7.2831 80.1492
MOLM-16 CTRP2; CTRP1 -7.2749 -4.839 -7.275 81.4663
Daudi CTRP2 -7.02 -6.153 -7.02 80.3731
Pfeiffer CTRP2 -6.9965 -6.0934 -6.9965 80.2164
GA-10 CTRP2 -6.9935 -6.0973 -6.9935 80.1966
KMS-34 CTRP2 -6.9007 -4.2067 -6.9009 78.9361
MOLT-16 CTRP2 -6.8799 -3.9944 -6.8802 78.6452
697 CTRP2 -6.862 -4.526 -6.862 78.95
BCP-1 CTRP2 -6.8372 -4.7474 -6.8372 78.9251
Ri-1 CTRP2 -6.775 1.2528 -7.0519 71.1888
KMS-12-BM CTRP2 -6.7498 -3.929 -6.75 77.9038
OCI-AML-2 CTRP2 -6.6957 -5.9807 -6.6957 78.2143
SUP-M2 CTRP2 -6.6955 -4.6235 -6.6955 78.0203
SU-DHL-6 CTRP2 -6.689 -4.4184 -6.689 77.8867
SU-DHL-10 CTRP2 -6.5986 -4.3884 -6.5986 77.3359
SU-DHL-4 CTRP2; CTRP1 -6.58 -3.9429 -6.5801 77.0034
OCI-Ly3 CTRP2 -6.5799 -4.4935 -6.5799 77.2665
MHH-CALL-4 CTRP2 -6.5159 -4.1435 -6.516 76.728
SU-DHL-8 CTRP2 -6.4075 -3.1045 -6.409 75.4015
BV-173 CTRP2 -6.3127 -3.4446 -6.3132 75.1501
NOMO-1 CTRP2; CTRP1 -6.3086 -3.9338 -6.3086 75.4188
L-540 CTRP2 -6.1217 -3.5803 -6.1219 74.1182
MOLT-13 CTRP2 -5.938 -3.0203 -5.9387 72.7524
EB1 CTRP2 -5.8942 -2.4294 -5.8972 72.1188
MV4-11 CTRP2 -5.8329 -4.1129 -5.8329 72.4394
NU-DHL-1 CTRP2 -5.7195 -3.8351 -5.7195 71.6706
NALM-6 CTRP2 -5.6662 -3.9286 -5.6662 71.3325
OCI-AML-5 CTRP2 -5.6616 -3.5784 -5.6616 71.2579
Reh CTRP2 -5.5326 -2.4499 -5.5341 70.0821
Kasumi-1 CTRP2 -5.316 -3.2985 -5.316 68.9837
JVM-2 CTRP2 -5.3035 -3.2776 -5.3035 68.9002
NCO2 CTRP2 -5.2973 -3.2745 -5.2973 68.8597
RCH-ACV CTRP2 -5.2697 -1.1521 -5.2849 67.7854
SEM CTRP2 -5.2402 -3.7125 -5.2402 68.5122
RS4;11 CTRP2 -5.2018 -1.5353 -5.2089 76.7083
MOLM-13 CTRP2 -5.1975 -3.223 -5.1976 68.2036
SUP-T1 CTRP2 -5.1954 -2.6553 -5.1957 68.0969
BL-70 CTRP2 -5.1863 -3.243 -5.1863 68.1317
RPMI-8402 CTRP2 -5.1404 -3.5064 -5.1404 67.8454
Kasumi-2 CTRP2 -5.1084 -1.7899 -5.112 67.2558
THP-1 CTRP2; CTRP1 -5.0905 -2.7706 -5.0907 67.4831
DB CTRP2 -5.0674 -2.5375 -5.0678 67.2593
SIG-M5 CTRP2 -5.0657 -3.7644 -5.0657 67.3542
DND-41 CTRP2 -5.0489 -1.8581 -5.0517 66.9305
KYO-1 CTRP2 -5.044 -1.4333 -5.051 66.6993
MOLT-3 CTRP2 -4.9874 -2.8713 -4.9875 66.7971
ST486 CTRP2 -4.9546 -3.181 -4.9546 66.6042
SUP-T11 CTRP2 -4.9482 -1.2561 -4.957 66.0501
HT CTRP2 -4.9148 -3.2032 -4.9148 66.3414
Raji CTRP2 -4.9015 -1.985 -4.903 66.0731
Peer CTRP2 -4.8895 -2.5772 -4.8897 66.1257
MOLP-8 CTRP2 -4.8849 -1.7719 -4.8875 65.9013
AML-193 CTRP2 -4.8817 -2.1059 -4.8827 65.9833
PL21 CTRP2; CTRP1 -4.8789 -2.0739 -4.88 65.9902
KE-37 CTRP2 -4.8783 -3.4237 -4.8783 66.1046
CML-T1 CTRP2 -4.8746 -2.55 -4.8748 66.0252
OCI-Ly19 CTRP2 -4.867 -2.0651 -4.868 65.88
OCI-AML-3 CTRP2; CTRP1 -4.862 -3.1572 -4.862 66.0234
SU-DHL-1 CTRP2 -4.8479 -3.4833 -4.8479 65.9029
Jurkat CTRP2 -4.7845 -3.1631 -4.7845 65.4774
PF-382 CTRP2 -4.7659 -2.2524 -4.7663 65.2784
JURL-MK1 CTRP2 -4.7608 -3.4886 -4.7608 65.323
P31/FUJ CTRP2 -4.7314 -2.4281 -4.7316 65.0815
SR CTRP2 -4.7125 -2.4241 -4.7127 64.958
JVM-3 CTRP2 -4.7112 -1.631 -4.7138 64.7844
NB4 CTRP2 -4.703 -4.0352 -4.703 64.9389
TALL-1 [Human adult T-ALL] CTRP2 -4.697 2.2854 -4.9804 62.1715
KMS-26 CTRP2 -4.6701 -3.5525 -4.6701 64.7194
Karpas-299 CTRP2 -4.6548 -2.0891 -4.6554 64.5374
EM-2 CTRP2 -4.6319 -3.5148 -4.6319 64.465
Mono-Mac-1 CTRP2 -4.5828 -0.4128 -4.6064 63.4963
F-36P CTRP2 -4.577 -2.1056 -4.5775 64.0389
SET-2 CTRP2 -4.561 -3.0609 -4.561 63.9908
Hs 611.T CTRP2 -4.5608 -1.7091 -4.5623 63.8629
Ku812 CTRP2 -4.5605 -2.6693 -4.5606 63.9788
HuT 78 CTRP2 -4.555 -1.0911 -4.5621 63.642
M-07e CTRP2 -4.5432 -0.8121 -4.5552 63.4591
SUP-B15 CTRP2 -4.5128 -1.5919 -4.5148 63.5328
AMO1 CTRP2 -4.4781 -3.6744 -4.4781 63.4403
KE-97 CTRP2 -4.4754 -2.9707 -4.4754 63.4207
KMS-21-BM CTRP2 -4.4442 -3.477 -4.4442 63.2145
L-363 CTRP2 -4.4313 -2.3746 -4.4313 63.1116
Ki-JK CTRP2 -4.4298 -2.8902 -4.4298 63.1166
U-937 CTRP2; CTRP1 -4.4206 -3.4547 -4.4206 63.0926
LAMA-84 CTRP2 -4.4164 -2.2658 -4.4165 63.0071
HEL CTRP2 -4.3922 -2.9453 -4.3922 62.8667
P12-Ichikawa CTRP2 -4.3673 -3.445 -4.3673 62.7019
KCL-22 CTRP2 -4.3015 -1.4304 -4.3035 62.1571
RPMI-8226 CTRP2; CTRP1 -4.2906 -2.8789 -4.2906 62.227
WSU-DLCL2 CTRP2; CTRP1 -4.2891 -2.8936 -4.2891 62.2167
A4/Fukuda CTRP2 -4.2748 -2.5739 -4.2748 62.0822
KMS-27 CTRP2 -4.2662 -3.2687 -4.2662 62.0283
KMS-20 CTRP2 -4.2619 -1.6984 -4.2627 61.9444
JJN-3 CTRP2 -4.2515 -1.082 -4.2561 61.7649
KM-H2 CTRP2 -4.2129 -2.4124 -4.2129 61.6688
HL-60 CTRP2 -4.1985 -2.4185 -4.1985 61.5729
DEL CTRP2 -4.1409 -3.5788 -4.1409 61.1936
SK-MM-2 CTRP2 -4.1251 5.8224 -5.1853 62.4801
MOTN-1 CTRP2 -4.112 -2.4134 -4.112 60.9988
DoHH2 CTRP2 -4.0965 -3.2327 -4.0965 60.898
Karpas-422 CTRP2 -4.0914 -2.2322 -4.0914 60.8587
KHM-1B CTRP2 -4.0762 -2.5575 -4.0762 60.7616
CA46 CTRP2 -4.0709 -0.3892 -4.0854 60.4496
HPB-ALL CTRP2 -4.063 1.1831 -4.1661 59.7332
OPM-2 CTRP2 -3.9676 -2.1335 -3.9676 60.0351
Namalwa CTRP2 -3.9655 -1.9951 -3.9656 60.0181
CMK CTRP2 -3.9285 -3.2606 -3.9285 59.7787
OCI-Ly10 CTRP2 -3.928 -0.7227 -3.9343 59.6427
KO52 CTRP2 -3.9235 -1.981 -3.9236 59.7395
GDM-1 CTRP2; CTRP1 -3.8724 -0.6343 -3.8792 59.311
JeKo-1 CTRP2 -3.8008 -2.7718 -3.8008 58.928
U266B1 CTRP2 -3.7571 0.1167 -3.7809 58.3745
EHEB CTRP2 -3.7124 -1.6149 -3.7126 58.3304
HEL 92.1.7 CTRP2 -3.6893 -2.919 -3.6893 58.1854
Granta-519 CTRP2 -3.6826 -0.6479 -3.6875 58.06
EJM CTRP2 -3.6221 -1.9867 -3.6221 57.7366
KMS-11 CTRP2 -3.5967 0.0734 -3.6156 57.3883
A3/Kawakami CTRP2 -3.5727 -3.0329 -3.5727 57.4082
MOLP-2 CTRP2 -3.5444 -0.5783 -3.5491 57.1586
SUP-HD1 CTRP2 -3.5419 -0.8921 -3.5438 57.1705
KMS-18 CTRP2 -3.5374 -0.6605 -3.5411 57.1212
L-428 CTRP2 -3.4942 -0.6962 -3.4973 56.843
SU-DHL-5 CTRP1 -3.3571 -2.044 -3.3571 99.2367
HDLM-2 CTRP2 -3.3379 0.295 -3.3585 55.7146
RL CTRP2 -3.2602 3.6916 -3.6883 54.4099
KMS-28BM CTRP2 -3.2074 4.9378 -3.9321 53.8087
ALL-SIL CTRP2 -3.072 -0.8757 -3.0726 54.0677
NCI-H929 CTRP2 -2.9789 -1.1055 -2.9791 53.4514
TF-1 CTRP2 -2.9134 0.5442 -2.9333 52.9648
LP-1 CTRP2 -2.9015 -0.6757 -2.9023 52.933
ME1 CTRP2 -2.8094 2.4527 -2.9833 52.1286
K-562 CTRP2 -2.7589 2.2069 -2.8976 51.8478
MHH-CALL-3 CTRP2 -2.6298 21.9787 -10.4375 50.364
HD-MY-Z CTRP2 -2.495 2.7127 -2.6841 50.2098
Mono-Mac-6 CTRP2 -0.3552 36.0723 -15.1711 46.8822
P3HR-1 CTRP2 2.2326 18.6936 -4.245 35.891
MC116 CTRP2 6.003 8.2933 4.1324 2.33
Toledo CTRP2 6.6213 11.8715 2.8389 6.6171
Karpas-620 CTRP2 6.9278 10.2842 3.7777 2.6027
BL-41 CTRP2 7.6492 18.8384 0.1793 14.886
KMM-1 CTRP2 7.6505 14.8601 2.1015 8.0497
REC-1 CTRP2 10.6998 25.2096 -0.8045 13.6884
⏷ Show the Full List of 148 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 -4.0877 0.209 -4.1241 68.5485
TE15 CTRP2 -1.7372 3.1809 -1.9437 45.5109
TE-6 CTRP2 -4.6559 -0.9976 -4.6657 73.1209
OE21 CTRP2 -3.8993 -2.3463 -3.8993 59.5833
KYSE-180 CTRP2 -3.6494 -1.4391 -3.6498 57.9083
TE-4 CTRP2 -3.4143 0.7456 -3.4572 64.0756
TE-9 CTRP2 -3.4131 -2.0494 -3.4131 56.3448
TE-5 CTRP2 -3.0152 0.9575 -3.0566 53.5778
KYSE-140 CTRP2 -2.6565 2.8169 -2.8731 51.182
OE33 CTRP2 -2.5945 1.1826 -2.6344 50.8689
TE-14 CTRP2 -2.5648 2.8544 -2.7806 50.6304
TE-10 CTRP2 -2.4975 1.5286 -2.5563 50.237
KYSE-410 CTRP2 -2.4567 5.003 -3.1305 49.9786
KYSE-510 CTRP2 -1.9286 1.5468 -1.9666 46.5173
TE-11 CTRP2 -1.7113 2.3911 -1.8089 45.188
EC-GI-10 CTRP2 -1.0976 3.4084 -1.2932 41.4062
KYSE-30 CTRP2 -0.7556 4.9931 -1.2714 39.9348
COLO 680N CTRP2 -0.7238 4.6566 -1.1491 39.5363
KYSE-520 CTRP2 -0.6362 6.0694 -1.4624 39.8484
KYSE-150 CTRP2 0.1176 4.8733 -0.2866 34.0963
KYSE-450 CTRP2 0.9858 5.0682 0.6087 28.3247
OE19 CTRP2 7.3961 21.6086 -1.3688 19.8981
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 31 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 -0.411 3.8047 -0.6224 36.9808
BxPC-3 CTRP2 -4.0197 -1.3062 -4.0213 60.3253
SU.86.86 CTRP2 -3.9223 0.2975 -3.958 67.517
Panc 03.27 CTRP2 -3.6997 0.8888 -3.7622 57.7883
QGP-1 CTRP2 -3.4927 1.3291 -3.5806 56.4252
Panc 08.13 CTRP2 -3.4716 1.4357 -3.5682 56.269
KP-4 CTRP2 -2.664 0.9011 -2.6918 51.3281
MIA PaCa-2 CTRP2 -2.2947 1.4376 -2.3393 48.9208
PSN1 CTRP2 -2.2485 5.8188 -3.1388 48.9107
KP-3 CTRP2 -2.0862 3.9852 -2.4759 47.8152
Hs 766T CTRP2 -1.9576 3.1522 -2.1761 46.906
CFPAC-1 CTRP2 -1.6328 3.8706 -1.959 45.0178
Panc 10.05 CTRP2 -1.5595 9.3383 -3.6628 46.1692
DAN-G CTRP2 -1.5132 6.6194 -2.5967 45.1669
Panc 04.03 CTRP2 -1.3911 7.7691 -2.8741 44.9092
PaTu 8988s CTRP2 -1.3247 6.5553 -2.3707 44.1132
SNU-213 CTRP2 -1.3075 2.8089 -1.4297 42.6088
HuP-T3 CTRP2 -1.1792 6.778 -2.2892 43.399
PaTu 8902 CTRP2 -0.7127 5.3905 -1.5571 36.6944
Capan-2 CTRP2 -0.3392 8.1672 -1.9033 39.538
SW1990 CTRP2 -0.1522 6.3637 -1.035 37.0698
HPAF-II CTRP2 0.6998 6.9086 -0.3106 32.1819
PaTu 8988t CTRP2 0.9252 7.6758 -0.3679 31.6173
Capan-1 CTRP2 1.6658 9.712 -0.4764 29.6758
KP-2 CTRP2 1.6781 8.8846 -0.0942 28.4998
AsPC-1 CTRP2 1.7462 9.3539 -0.2337 28.7283
SUIT-2 CTRP2 2.199 9.9049 -0.0308 26.8283
PANC-1 CTRP2 2.9139 9.7797 0.7302 22.3788
Panc 02.03 CTRP2 3.6354 15.8702 -1.5834 27.611
PK-45H CTRP2 4.1743 10.5326 1.5453 16.3334
SNU-410 CTRP2 4.7081 22.1636 -3.797 30.0676
⏷ Show the Full List of 31 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 43 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 -2.1167 2.7444 -2.2841 47.8579
LOX-IMVI CTRP2 -4.4189 -2.1308 -4.4191 63.0129
Mel Ho CTRP2 -3.8448 -1.768 -3.8449 59.2119
MeWo CTRP2 -3.7077 1.0581 -3.7831 57.7761
COLO 792 CTRP2 -3.6597 -0.9115 -3.6621 57.9423
Hs 294T CTRP2 -3.4158 -0.5591 -3.4196 56.3197
Mel JuSo CTRP2 -3.2703 0.9906 -3.3229 55.1673
A2058 CTRP2 -3.1783 -2.7265 -3.1783 54.7809
SK-MEL-5 CTRP1 -3.1769 1.0113 -3.2269 88.9055
A-375 CTRP2; CTRP1 -3.1423 -1.5253 -3.1423 54.5842
IGR-1 CTRP2 -3.0094 1.1496 -3.0624 53.5177
COLO 741 CTRP2 -3.0059 9.983 -5.4514 52.0378
Hs 944.T CTRP2 -2.9458 0.7017 -2.9726 53.1613
RVH-421 CTRP2 -2.7463 0.1401 -2.7533 51.8902
CJM [Human melanoma] CTRP2 -2.6317 -0.8218 -2.6318 51.1388
RPMI-7951 CTRP2 -2.4765 3.6827 -2.8357 50.0915
SK-MEL-1 CTRP2; CTRP1 -2.1953 0.8181 -2.2091 48.2965
WM88 CTRP2 -1.9569 2.0139 -2.0305 46.7489
IGR-37 CTRP2 -1.635 1.9489 -1.6885 44.6131
K029AX CTRP2 -1.5567 2.0658 -1.6158 44.1094
SK-MEL-3 CTRP2 -1.3894 2.9963 -1.5423 43.2021
A101D CTRP2 -1.3632 0.9819 -1.3684 42.7035
HT-144 CTRP2 -1.279 2.2314 -1.3389 42.2827
COLO 829 CTRP2 -1.1988 3.0026 -1.3395 41.9411
Hs 940.T CTRP2 -0.81 3.7037 -1.0349 39.6147
COLO 800 CTRP2 -0.7854 5.2941 -1.3877 40.2983
WT2-iPS CTRP2 -0.5003 5.1998 -1.0499 38.4231
HMCB CTRP2 -0.4918 1.736 -0.5004 36.9108
SK-MEL-2 CTRP2 -0.4584 1.893 -0.4709 36.7013
WM115 CTRP2 -0.0628 4.4079 -0.3692 34.9799
UACC-62 CTRP2 -0.038 2.4872 -0.0653 33.9497
Hs 688(A).T CTRP2 0.0631 4.8993 -0.353 34.4844
WM983B CTRP2 0.2511 10.5655 -2.2959 38.194
WM266-4 CTRP2 0.2685 3.0662 0.2101 32.0117
Malme-3M CTRP2 0.3631 6.0639 -0.3752 33.5014
Hs 839.T CTRP2 0.5389 4.9043 0.165 31.2536
IGR-39 CTRP2 1.2163 9.1596 -0.6885 31.6061
SK-MEL-28 CTRP1 1.2543 3.4458 1.2112 54.095
UACC-257 CTRP2 1.307 6.5914 0.4589 27.8252
SK-MEL-24 CTRP2 2.9492 8.412 1.4049 19.7973
Hs 895.T CTRP2 3.144 10.5035 0.6051 22.2428
Hs 934.T CTRP2 3.3739 7.82 2.1008 16.0075
SK-MEL-31 CTRP2 6.1425 7.6055 3.6109 0.2115
⏷ Show the Full List of 43 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 -3.1885 5.9281 -4.1964 53.4791
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Kelly CTRP2 -5.2434 -1.6557 -5.2494 67.9717
SK-N-FI CTRP2 -4.9434 -1.623 -4.9475 66.1973
MHH-NB-11 CTRP2 -4.5899 -2.4792 -4.5899 64.1613
IMR-32 CTRP2 -4.5576 -1.2471 -4.5628 63.7137
NB1 CTRP2 -4.2879 -3.2452 -4.2879 62.1731
CHP-126 CTRP2 -4.2262 -2.0172 -4.2264 61.7406
KP-N-SI9s CTRP2 -4.1933 -1.7192 -4.1939 61.5002
SiMa CTRP2 -3.6409 -0.1368 -3.6546 57.7087
SK-N-SH CTRP2 -3.1197 -0.4395 -3.1227 54.3706
SK-N-DZ CTRP2 -2.6878 3.1327 -2.9594 51.3445
SK-N-AS CTRP2 -2.611 1.5542 -2.6767 50.964
SK-N-BE(2) CTRP2 -2.3262 3.9398 -2.7269 49.2243
CHP-212 CTRP2 -2.0931 3.0518 -2.3053 47.7424
NH-6 CTRP2 -0.3767 7.8809 -1.8314 39.5482
KP-N-YN CTRP2 6.6721 11.0142 3.2826 4.787
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-478 CTRP2 -3.1136 0.8207 -3.1509 54.2176
HuCC-T1 CTRP2 -2.8423 1.6022 -2.9226 52.4199
SNU-308 CTRP2 -2.0369 1.3114 -2.0659 47.2179
HuH-28 CTRP2 -1.7652 1.344 -1.788 45.4141
SNU-1079 CTRP2 -0.9807 7.4541 -2.3168 42.6254
SNU-869 CTRP2 -0.1105 6.9733 -1.205 37.309
SNU-1196 CTRP2 0.1302 8.0629 -1.3642 36.8037
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U2OS CTRP2 -6.2317 0.583 -6.3911 70.2396
SK-ES-1 CTRP2 -5.0208 -2.0495 -5.0224 66.8315
A-673 CTRP2 -4.6427 -0.4735 -4.6656 63.871
MHH-ES-1 CTRP2 -4.2372 -1.4936 -4.2386 61.7558
SK-N-MC CTRP2 -3.8527 -0.069 -3.8722 59.014
SJSA-1 CTRP2 -3.838 5.3877 -4.7451 61.7835
Hs 888.T CTRP2 -3.1408 4.8707 -3.8415 53.5009
CAL-78 CTRP2 -2.8043 -0.2316 -2.8072 52.2815
TC71 CTRP2 -2.7946 0.4277 -2.8085 52.1975
SaOS-2 CTRP2 -2.679 2.5346 -2.8553 51.336
SW1353 CTRP2 -2.3802 1.402 -2.4257 49.4774
G-292 clone A141B1 CTRP2 -1.6227 5.6197 -2.3965 45.4646
HOS CTRP2 -0.9302 4.8681 -1.4286 40.9786
MG-63 CTRP2 2.2418 7.8141 0.9529 23.3678
Hs 822.T CTRP2 2.604 7.7536 1.352 20.9063
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 70 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 CTRP2 -6.9754 -6.0181 -6.9754 80.0745
SK-BR-3 CTRP2 -4.1684 2.376 -4.4271 59.6088
CAL-51 CTRP2 -3.9602 -1.2575 -3.9619 59.9337
HCC1954 CTRP2 -3.8159 0.9005 -3.884 58.4649
HCC1806 CTRP2 -3.6265 -1.5901 -3.6266 57.7604
HMC-1-8 CTRP2 -3.4333 -1.9171 -3.4333 56.4794
MDA-MB-157 CTRP2 -3.3302 1.761 -3.4518 55.3467
CAL-148 CTRP2 -3.2068 -0.2413 -3.2128 54.9308
Hs 578T CTRP2 -3.0271 -1.7011 -3.0271 53.7736
AU565 CTRP2 -2.7635 0.8572 -2.7922 51.9754
MDA-MB-231 CTRP2 -2.2737 3.1613 -2.518 48.8689
MDA-MB-468 CTRP2 -2.2681 2.081 -2.3642 48.7739
HCC2218 CTRP2 -2.1856 3.3172 -2.4503 48.3419
CAL-85-1 CTRP2 -1.9249 3.7044 -2.2419 46.795
HCC38 CTRP2 -1.5089 2.4524 -1.6016 43.862
MCF-7 CTRP2 -1.052 5.101 -1.6244 41.8612
HCC1500 CTRP2 -1.047 4.5649 -1.4788 41.5707
HCC1395 CTRP2 -0.9703 3.1994 -1.1235 40.4815
MDA-MB-453 CTRP2 -0.8712 5.5529 -1.5572 40.9799
EFM-192A CTRP2 -0.6642 3.2801 -0.8076 38.4519
BT-549 CTRP2 -0.4137 5.0409 -0.9113 37.7541
BT-20 CTRP2 -0.1764 4.0144 -0.4087 35.5044
HDQ-P1 CTRP2 -0.0377 6.6146 -0.998 36.5635
CAL-120 CTRP2 0.104 4.616 -0.2365 33.9938
CAMA-1 CTRP2 0.2588 4.2075 0.0241 32.6491
MDA-MB-361 CTRP2 1.0031 10.3887 -1.4515 34.1561
HCC202 CTRP2 1.358 5.6817 0.8308 26.391
JIMT-1 CTRP2 1.7097 7.9306 0.351 26.9772
HCC1428 CTRP2 1.8197 4.3314 1.691 21.9238
T-47D CTRP2 1.908 11.3141 -0.9755 30.3609
BT-474 CTRP2 2.0847 8.1879 0.6287 24.9563
HCC1937 CTRP2 2.365 12.0796 -0.8964 28.9166
ZR-75-30 CTRP2 2.4495 13.7226 -1.6099 30.5053
HCC1419 CTRP2 3.053 9.2086 1.1358 20.5472
Hs 578Bst CTRP2 4.7511 13.8973 0.3712 19.4201
KPL-1 CTRP2 5.9826 6.6235 4.8365 0.1145
BT 239 CTRP2 -5.0616 -2.8153 -5.0617 67.2719
BT 286 CTRP2 -4.5856 1.5405 -4.7566 62.2164
BT 245 CTRP2 -4.5225 0.0906 -4.5662 62.8731
BT 504 CTRP2 -4.5087 -1.7432 -4.51 63.5392
BT 428 CTRP2 -4.5085 1.3033 -4.6477 62.0049
BT 482 CTRP2 -3.9875 1.0049 -4.0712 59.4008
BT 145 CTRP2 -3.9788 -1.9476 -3.9789 60.1049
BT 172 CTRP2 -3.7639 -0.2784 -3.7761 58.513
BT 416 CTRP2 -3.7038 -1.8714 -3.7039 58.279
BT 112 CTRP2 -3.6977 -1.506 -3.6981 58.2301
BT164 CTRP2 -3.6832 -1.2889 -3.6839 58.1241
BT 131 CTRP2 -3.4397 1.3671 -3.5284 56.1006
BT 231 CTRP2 -3.3072 1.2748 -3.3818 55.3314
BT147 CTRP2 -3.2374 2.7922 -3.4935 54.5369
BT 330 CTRP2 -3.2323 1.9464 -3.369 54.7253
BT 228 CTRP2 -2.87 1.1739 -2.9192 52.6351
BT 271 CTRP2 -2.6239 0.7797 -2.6457 51.0701
BT 333 CTRP2 -2.4804 2.9213 -2.7006 50.1194
BT 440 CTRP2 -2.3337 3.9871 -2.7455 49.2702
BT 159 CTRP2 -2.0472 1.6189 -2.0942 47.3068
BT 187 CTRP2 -1.7279 5.3602 -2.4351 45.9923
BT 444 CTRP2 -1.6728 8.3951 -3.4122 46.4643
BT 359 CTRP2 -1.3791 2.3198 -1.4517 42.9708
BT 139 CTRP2 -1.1724 2.5899 -1.2608 41.6483
BT 422 CTRP2 -1.1493 2.4736 -1.2246 41.4648
BT 498 CTRP2 -1.0337 6.58 -2.0637 42.4882
BT 179 CTRP2 -0.8772 3.4233 -1.0586 39.9439
BT 232 CTRP2 -0.8112 8.2277 -2.4289 42.1143
BT 224 CTRP2 -0.4432 3.975 -0.69 37.2893
BT 248 CTRP2 -0.1318 6.8335 -1.1774 37.3249
BT 216 CTRP2 0.2954 12.2484 -3.0082 39.1715
BT 328 CTRP2 0.526 8.6664 -1.1938 35.0772
BT 340 CTRP2 1.8318 15.0953 -2.8577 34.6566
BT 320 CTRP2 5.3857 16.4659 -0.3845 20.606
⏷ Show the Full List of 70 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 -3.8085 -1.8167 -3.8086 58.9726
Cancer Drug Sensitivity Data Curated from 46 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KNS-60 CTRP2 -4.2124 -1.7349 -4.2131 71.0328
AM-38 CTRP2 -4.0666 -0.6426 -4.0756 60.4959
SF539 CTRP2 -3.8243 -1.2355 -3.8255 59.046
D283 Med CTRP2 -3.776 -2.3505 -3.776 58.7625
M059K CTRP2 -3.5335 -2.8108 -3.5335 57.1475
LN-229 CTRP2; CTRP1 -3.5118 -0.3179 -3.5198 56.9574
ONS-76 CTRP2 -3.2191 1.331 -3.2943 54.7847
LN-18 CTRP2 -3.12 -1.6926 -3.12 54.3925
SNU-466 CTRP2 -2.9109 -1.9549 -2.9109 52.9994
SF268 CTRP2 -2.4869 2.1107 -2.5983 50.1649
KALS-1 CTRP2 -1.9378 5.2241 -2.6253 47.1517
Hs 683 CTRP2 -1.8984 2.5229 -2.0222 46.4314
U-118MG CTRP2 -1.7232 6.2281 -2.6954 46.1892
Daoy CTRP2 -1.6321 2.8969 -1.7877 44.769
42-MG-BA CTRP2 -1.4621 3.4268 -1.6891 43.8014
DK-MG CTRP2 -1.3388 2.0123 -1.3845 42.6437
YH-13 CTRP2 -1.2932 5.0115 -1.8631 43.3056
SNU-626 CTRP2 -1.1918 2.3717 -1.2597 41.7265
SNU-1105 CTRP2 -1.1709 3.0172 -1.3118 41.7601
SNU-738 CTRP2 -0.9258 3.8301 -1.1842 40.4408
CAS-1 CTRP2 -0.9133 9.5927 -3.0863 54.5591
SF126 CTRP2 -0.8853 3.0677 -1.0138 39.8634
SW1088 CTRP2 -0.21 8.6463 -2.3218 36.6241
DBTRG-05MG CTRP2 -0.1714 8.6695 -1.9272 38.9776
SNB-75 CTRP2 -0.1459 3.6467 -0.3086 35.0943
GB-1 CTRP2 0.0809 7.2414 -1.0985 36.377
TM-31 CTRP2 0.131 6.8103 -0.8859 35.6847
GaMG CTRP2 0.5061 7.4495 -1.0647 30.9569
SF295 CTRP2 0.7222 6.1865 -0.0273 31.2554
GOS-3 CTRP2 0.7505 11.1022 -2.0289 36.1388
8-MG-BA CTRP2 0.9028 5.5262 0.3843 29.3455
GMS-10 CTRP2 1.0506 7.3296 -0.0974 30.4137
Becker CTRP2 1.143 6.8314 0.1933 29.2093
SNU-489 CTRP2 1.2793 3.039 1.2649 25.1319
CCF-STTG1 CTRP2 1.3094 6.4327 0.5197 27.6124
YKG-1 CTRP2 1.3575 9.8458 -0.8486 31.6089
A-172 CTRP2 2.7945 15.0865 -1.9561 30.4507
NMC-G1 CTRP2 2.7982 10.6586 0.1999 24.4944
U-251MG CTRP2 2.8762 13.0492 -0.8828 27.5727
U-87MG ATCC CTRP2 3.2258 10.3086 0.7769 21.4311
KG-1-C CTRP2 3.2482 11.5989 0.1717 23.4633
KNS-81 CTRP2 3.2532 10.9865 0.4746 25.4662
T98G CTRP2 3.7513 12.6915 0.0961 22.5221
SNU-201 CTRP2 4.4565 6.3982 3.8316 6.3589
KNS-42 CTRP2 5.1152 14.5816 0.3346 18.8069
SW1783 CTRP2 7.2827 13.5395 2.4861 7.0784
⏷ Show the Full List of 46 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-151 CTRP2 -4.7902 -2.2873 -4.7911 63.089
RL95-2 CTRP2 -4.3951 -1.8698 -4.3957 62.8296
HEC-265 CTRP2 -3.8304 -2.5415 -3.8304 59.1253
ESS-1 CTRP2 -3.5419 0.5631 -3.5792 56.9344
JHUEM-7 CTRP2 -3.5181 -1.9992 -3.5181 57.0444
JHUEM-1 CTRP2 -3.4041 -2.6297 -3.4041 56.2851
HEC-6 CTRP2 -3.3729 -0.8814 -3.3743 56.0592
HEC-108 CTRP2 -3.3261 -2.2225 -3.3261 55.7655
AN3-CA CTRP2 -2.8983 0.0066 -2.9048 52.8951
JHUEM-2 CTRP2; CTRP1 -2.7828 2.3057 -2.9345 52.0269
HEC-1-B CTRP2 -2.3694 1.9389 -2.4568 49.4176
EN CTRP2 -2.2828 1.0827 -2.3082 48.8323
MFE-296 CTRP2 -1.9326 3.3106 -2.1762 46.7746
HEC-59 CTRP2 -1.4379 3.4351 -1.6645 43.6476
KLE CTRP2 -0.9724 9.1109 -2.951 43.3507
HEC-1-A CTRP2 -0.7435 8.0701 -2.2956 41.6717
HEC-251 CTRP2 -0.5872 6.8263 -1.6661 40.045
MFE-319 CTRP2 -0.1114 3.7526 -0.2895 34.9138
JHUEM-3 CTRP2 0.1292 6.4034 -0.7439 35.3289
EFE-184 CTRP2 0.6225 9.2158 -1.7295 32.4665
HEC-50B CTRP2 3.1061 19.3007 -3.7572 33.2175
Ishikawa (Heraklio) 02 ER- CTRP2 -2.5924 0.7372 -2.6119 50.8654
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CAL-54 CTRP2 -4.3874 -0.0912 -4.4186 62.2099
UO-31 CTRP2 -2.8645 2.9323 -3.1155 52.3938
TUHR10TKB CTRP2 -2.4106 5.3584 -3.1794 49.7378
BFTC-909 CTRP2 -2.3043 3.9627 -2.7081 49.098
KMRC-3 CTRP2 -1.8572 3.7656 -2.1809 46.3893
KMRC-20 CTRP2 -1.1772 2.7963 -1.2896 41.7364
KMRC-1 CTRP2 -1.0876 1.4911 -1.1001 40.8899
769-P CTRP2 -1.0538 2.6277 -1.1396 40.8618
786-O CTRP2 -0.3946 2.7382 -0.4561 36.431
TUHR4TKB CTRP2 -0.1214 2.6582 -0.1633 34.5524
TUHR14TKB CTRP2 0.2496 2.6369 -3.7249 0.7967
ACHN CTRP2 1.7932 11.2512 -1.0588 30.897
OS-RC-2 CTRP2 1.9512 9.5454 -0.1133 27.7755
VMRC-RCZ CTRP2 2.2769 8.5065 0.6845 24.227
SNU-1272 CTRP2 2.4775 6.8007 1.6247 20.2236
KMRC-2 CTRP2 3.1641 6.4242 2.5013 14.9777
RCC10RGB CTRP2 4.1786 11.3544 1.1417 17.8716
Caki-2 CTRP2 4.8492 12.4985 1.1535 16.4088
Caki-1 CTRP2 9.39 17.0303 2.1685 5.7492
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW620 CTRP1 -7.3686 11.4846 -10.6738 73.6408
CW-2 CTRP2 -6.4038 -1.5164 -6.4295 73.6336
SNU-81 CTRP2 -5.9204 -2.7279 -5.922 72.474
HT-55 CTRP1 -5.5182 7.0166 -7.0725 76.9761
CCK-81 CTRP2 -5.3471 -1.1171 -5.3645 68.1731
SW1463 CTRP2 -5.1769 1.5597 -5.3881 64.9223
SK-CO-1 CTRP2 -4.6186 -0.095 -4.656 63.5161
LoVo CTRP1 -4.5569 2.8139 -4.9184 84.5651
HT115 CTRP2; CTRP1 -4.4765 -1.2906 -4.4805 63.2616
NCI-H508 CTRP2; CTRP1 -4.466 1.0275 -4.5744 62.0107
SNU-C5 CTRP2 -4.4295 0.8774 -4.5676 59.4488
T84 CTRP2 -4.3956 0.966 -4.4955 61.6478
SW48 CTRP2 -4.3736 -1.8441 -4.3742 62.6868
LS513 CTRP2 -4.1927 -2.7925 -4.1927 61.5383
SNU-175 CTRP2 -4.0081 -2.1977 -4.0081 60.3053
LS180 CTRP2 -3.8753 -1.6307 -3.8756 59.4078
COLO201 CTRP2 -3.8127 -0.3665 -3.8237 58.8393
COLO 320 CTRP2 -3.7969 -0.0459 -3.816 58.6634
NCI-H747 CTRP2 -3.637 2.7476 -3.9161 56.7115
RKO CTRP2; CTRP1 -3.6311 -1.5366 -3.6313 57.8305
SNU-C1 CTRP2 -3.6135 -1.1786 -3.6144 57.6595
SNU-C2A CTRP2 -3.5632 0.4564 -3.596 57.0922
KM12 CTRP2 -3.4352 0.3635 -3.4606 56.3165
COLO205 CTRP2 -3.4032 -1.6897 -3.4032 56.2782
NCI-H716 CTRP2 -3.3929 -2.3696 -3.3929 56.2102
CL-11 CTRP2 -3.2343 4.8263 -3.9317 53.9677
GP2d CTRP2 -3.1242 1.4287 -3.2031 54.1868
MDST8 CTRP1 -3.0862 1.1181 -3.1397 88.4109
CL-34 CTRP1 -3.08 0.2301 -3.0936 91.8121
SNU-1040 CTRP1 -3.0454 2.8883 -3.3015 82.2187
SNU-1033 CTRP2 -2.9822 2.8351 -3.226 53.0865
HCT 116 CTRP2; CTRP1 -2.903 -1.8037 -2.903 52.9921
CL-40 CTRP1 -2.7872 2.6082 -2.9805 82.6184
HCT 15 CTRP2 -2.6936 3.389 -3.0128 51.3583
SW480 CTRP1 -2.5034 20.216 -9.4749 59.6091
SNU-C4 CTRP2 -2.3402 2.7552 -2.5247 49.2577
LS123 CTRP1 -1.9072 6.4988 -2.9802 70.0748
DLD-1 CTRP2 -1.5618 4.2984 -1.976 44.6998
LS1034 CTRP2 -1.471 4.8505 -2.014 44.3251
HCT 8 CTRP2; CTRP1 -1.1831 2.1447 -1.2315 41.6767
SW948 CTRP2 -0.8606 5.2089 -1.4455 40.7223
LS411N CTRP2 -0.7044 6.1495 -1.5626 40.3134
COLO 678 CTRP2; CTRP1 -0.2 8.7963 -2.004 39.2609
RCM-1 [Human ESC] CTRP2; CTRP1 -0.178 5.7113 -0.847 36.7631
SW1417 CTRP2 0.8826 8.4614 -0.7352 32.7728
OUMS-23 CTRP2 1.3673 5.818 0.7964 26.4824
C2BBe1 CTRP2 1.5243 14.536 -2.88 35.4935
SNU-503 CTRP2 2.9434 8.4066 1.4016 19.8248
HT-29 CTRP2; CTRP1 3.4182 16.3335 -1.998 29.1362
HCC-56 CTRP2 4.3971 9.9556 2.0305 13.9184
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-182 CTRP2 -4.7618 -1.1692 -4.7699 64.9146
SNU-886 CTRP2 -4.1902 -1.464 -4.1916 61.4486
HuH-6 CTRP2 -3.6465 1.2817 -3.7848 54.6065
SNU-398 CTRP2 -3.4221 0.4533 -3.4509 56.2173
SNU-878 CTRP2 -3.2743 -1.9409 -3.2743 55.42
Li-7 CTRP2 -2.0793 4.7821 -2.6599 47.8812
HLF CTRP2 -1.5681 3.2057 -1.7659 44.4271
JHH-1 CTRP2 -1.4287 0.832 -1.4325 43.1355
SNU-761 CTRP2 -1.2806 6.2549 -2.2231 49.0774
SNU-423 CTRP2 -0.7928 3.0805 -0.9169 39.2445
SK-HEP-1 CTRP2 -0.5014 3.6947 -0.7001 37.5367
JHH-2 CTRP2 -0.02 4.6648 -0.3836 34.8693
JHH-4 CTRP2 0.1137 8.7365 -1.6548 37.4672
PLC/PRF/5 CTRP2 0.2702 6.5375 -0.6383 34.5545
Hep 3B2.1-7 CTRP2 0.5565 7.8883 -0.8431 34.117
SNU-387 CTRP2 0.6172 2.309 0.6123 29.511
SNU-475 CTRP2 1.1541 3.1823 1.1272 26.0078
JHH-6 CTRP2 1.3729 3.6826 1.3109 24.6695
HuH-1 CTRP2 1.3781 8.1766 -0.0984 29.4046
SNU-449 CTRP2 1.9508 10.9498 -0.7627 29.6714
Hep-G2 CTRP2 6.2326 7.5379 3.6677 0.1127
JHH-5 CTRP2 6.6777 17.9197 -0.0879 17.3259
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 138 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LCLC-97TM1 CTRP2 -6.1289 0.0089 -6.2294 70.5753
NCI-H1975 CTRP2 -5.061 -2.9346 -5.0611 67.2834
DV-90 CTRP2 -4.9394 -1.7434 -4.9425 66.2225
NCI-H209 CTRP2 -4.9016 15.9917 -9.9625 58.6712
NCI-H1341 CTRP2 -4.6993 -2.3732 -4.6996 64.8663
NCI-H1105 CTRP2 -4.6148 -1.6997 -4.6167 64.202
NCI-H1694 CTRP2 -4.5564 -1.7896 -4.5576 63.8522
COR-L51 CTRP2 -4.4781 -0.8398 -4.4886 63.0811
NCI-H2141 CTRP2 -4.4296 1.5468 -4.5917 61.4404
NCI-H520 CTRP2 -4.3614 2.5073 -4.6557 60.4589
NCI-H510A CTRP2 -4.3592 -2.14 -4.3594 62.6226
NCI-H211 CTRP2 -4.3531 -2.2807 -4.3532 62.5913
MOR/CPR CTRP2 -4.1611 -2.9806 -4.1611 61.328
DMS 53 CTRP2 -4.1334 -0.4257 -4.148 60.8433
NCI-H526 CTRP2 -4.0243 -0.6882 -4.032 60.2428
NCI-H446 CTRP2 -3.9812 -1.0266 -3.9844 60.0366
HCC44 CTRP2 -3.9746 -1.9258 -3.9747 60.0761
NCI-H1155 CTRP2 -3.9737 -1.0527 -3.9767 59.9926
NCI-H1666 CTRP2 -3.9367 0.6375 -3.9916 59.2718
NCI-H661 CTRP2 -3.9227 0.2179 -3.9547 59.349
NCI-H2171 CTRP2 -3.9077 -1.0188 -3.9106 59.5627
NCI-H889 CTRP2 -3.8093 0.5093 -3.8523 58.5698
COLO 668 CTRP2 -3.7654 -1.3077 -3.7663 58.6661
NCI-H1650 CTRP2 -3.7539 0.3597 -3.7877 58.2846
NCI-H1581 CTRP2 -3.7242 -1.4371 -3.7247 58.4022
HCC1588 CTRP2 -3.7108 -1.6573 -3.711 58.3212
NCI-H810 CTRP2 -3.6615 -0.8633 -3.6642 57.9489
NCI-H596 CTRP1 -3.6605 0.72 -3.7102 90.327
NCI-H2286 CTRP2 -3.652 5.8298 -4.6718 55.5468
NCI-H841 CTRP2 -3.6001 0.8311 -3.6548 57.214
COLO 699 CTRP2 -3.5448 -0.5525 -3.5498 57.158
Lu-99 CTRP2 -3.5327 -1.6187 -3.5328 57.1387
NCI-H1838 CTRP2 -3.468 -0.7355 -3.4707 56.6753
HCC2108 CTRP2 -3.4425 -1.2733 -3.4429 56.5332
NCI-H1573 CTRP2 -3.4419 2.3993 -3.6518 55.7896
EPLC-272H CTRP2 -3.4231 1.4645 -3.5198 55.9747
NCI-H2444 CTRP2 -3.4205 1.4706 -3.5177 63.4957
NCI-H2087 CTRP2 -3.3934 0.2409 -3.4134 56.0754
NCI-H1734 CTRP2 -3.3468 -0.9888 -3.3476 55.8911
HCC1438 CTRP2 -3.3352 -0.0816 -3.3455 55.7489
PC-14 CTRP2 -3.3226 0.4927 -3.3505 63.685
NCI-H1944 CTRP2 -3.2911 -2.0294 -3.2911 55.5319
NCI-H23 CTRP2 -3.2827 0.9423 -3.3327 55.2535
NCI-H2122 CTRP2; CTRP1 -3.249 -0.3971 -3.2533 55.2608
VMRC-LCD CTRP2 -3.2287 1.5802 -3.3264 54.7893
NCI-H358 CTRP2 -3.2253 -1.4103 -3.2253 55.0923
HARA [Human squamous cell lung carcinoma] CTRP2 -3.2242 -1.0338 -3.2247 55.0803
Sq-1 CTRP2 -3.1629 -0.4456 -3.1699 51.5809
NCI-H522 CTRP2 -3.1502 -0.1416 -3.157 54.5536
NCI-H1781 CTRP1 -3.0929 1.5574 -3.181 86.7996
NCI-H2405 CTRP2 -3.0023 -0.0371 -3.0092 53.5799
HCC827 CTRP2 -2.9191 -0.2887 -2.9222 53.0423
RERF-LC-MS CTRP2 -2.9103 0.8011 -2.9405 52.9249
NCI-H650 CTRP2 -2.8867 0.4541 -2.9031 52.7973
SHP-77 CTRP2 -2.8534 -0.6533 -2.8541 52.6131
HCC78 CTRP2 -2.8451 0.218 -2.8548 52.5371
DMS 273 CTRP2 -2.8197 0.5532 -2.8379 52.3558
NCI-H2030 CTRP2 -2.7707 1.0226 -2.8076 52.0122
NCI-H292 CTRP2 -2.7688 0.3781 -2.781 52.0308
SK-LU-1 CTRP1 -2.747 3.6655 -3.1239 79.2406
SK-MES-1 CTRP2 -2.6269 1.4801 -2.6876 51.0679
KNS-62 CTRP2 -2.5843 1.6942 -2.6602 50.7892
DMS 114 CTRP2 -2.5485 2.0155 -2.6532 50.5545
HCC1833 CTRP2 -2.3917 3.0897 -2.6329 49.5839
LK2 CTRP2 -2.3916 3.5501 -2.717 49.5935
LCLC-103H CTRP2 -2.383 0.2564 -2.3879 49.4841
NCI-H1373 CTRP2 -2.3789 1.8854 -2.4618 49.4775
NCI-H2009 CTRP2 -2.3186 1.2488 -2.3531 49.0718
NCI-H1703 CTRP2 -2.2557 0.719 -2.2679 48.6448
CAL-12T CTRP2 -2.2007 1.9132 -2.2773 48.3301
NCI-H1355 CTRP2 -2.161 3.7376 -2.5046 48.2334
RERF-LC-A1 CTRP2 -2.1518 2.2143 -2.2553 48.0346
NCI-H1568 CTRP2 -2.1383 0.5665 -2.1455 47.8622
NCI-H1339 CTRP2 -2.088 1.8139 -2.1509 47.5891
COR-L95 CTRP2 -2.0711 5.1866 -2.7603 47.8905
NCI-H1563 CTRP2 -1.8581 2.2742 -1.9515 46.1333
NCI-H69 CTRP2 -1.8561 4.8167 -2.4254 46.603
Calu-3 CTRP2 -1.6309 6.3356 -2.63 45.718
SBC-5 CTRP2 -1.6069 -0.2153 -1.6069 44.312
NCI-H2029 CTRP2 -1.6056 2.2707 -1.6852 44.4691
SW1271 CTRP2 -1.5674 7.6099 -3.0047 50.6247
NCI-H2085 CTRP2 -1.5392 7.212 -2.8305 45.4896
HCC1195 CTRP2 -1.5379 4.1648 -1.9194 44.5103
HCC95 CTRP2 -1.5378 4.089 -1.9024 44.486
HCC15 CTRP2; CTRP1 -1.4349 4.2089 -1.8153 43.9269
NCI-H2228 CTRP2 -1.3979 6.9701 -2.5925 49.7601
HCC4006 CTRP2 -1.3585 2.1681 -1.4169 42.8033
NCI-H1792 CTRP2 -1.3366 2.334 -1.4084 42.6895
NCI-H2196 CTRP2 -1.3359 2.285 -1.4031 42.6743
A-549 CTRP2 -1.3318 3.1811 -1.5082 42.8766
ChaGo-K-1 CTRP2 -1.2771 2.4564 -1.3575 42.3178
NCI-H838 CTRP2 -1.236 1.6342 -1.2572 41.9009
NCI-H2081 CTRP2 -1.1993 4.8094 -1.7069 42.6417
NCI-H2110 CTRP2 -1.1982 2.8146 -1.3141 41.8816
NCI-H1092 CTRP2 -1.1856 3.3832 -1.3837 41.9791
LUDLU-1 CTRP2 -1.1467 2.994 -1.2827 41.5913
NCI-H322 CTRP2 -1.0289 5.1165 -1.6034 41.725
NCI-H727 CTRP2 -1.0283 5.9712 -1.8573 42.1518
NCI-H1755 CTRP1 -0.9621 4.4647 -1.3598 70.817
HOP-62 CTRP2 -0.9387 4.7727 -1.413 40.9831
NCI-H2170 CTRP2 -0.9349 3.8904 -1.206 40.5283
LOU-NH91 CTRP2 -0.9269 3.2111 -1.0787 40.1945
NCI-H1299 CTRP2 -0.9254 4.2867 -1.2805 40.6528
T3M-10 CTRP2; CTRP1 -0.7937 2.0545 -0.8218 39.0399
NCI-H196 CTRP2 -0.7839 3.1459 -0.9164 39.2086
RERF-LC-Ad2 CTRP2 -0.7431 13.9793 -4.8403 44.2106
NCI-H226 CTRP2 -0.6915 3.3324 -0.8447 44.5433
NCI-H441 CTRP2; CTRP1 -0.6663 4.5389 -1.0553 39.1447
NCI-H1623 CTRP2 -0.5435 3.3124 -0.6832 37.6475
NCI-H1395 CTRP2 -0.5035 2.6377 -0.5613 37.1428
NCI-H647 CTRP2 -0.4447 5.8114 -1.1718 38.4874
NCI-H460 CTRP2; CTRP1 -0.3681 4.3201 -0.6796 37.0377
NCI-H1915 CTRP2 -0.3139 6.3565 -1.2078 38.069
NCI-H1385 CTRP2 -0.302 22.8377 -8.6237 45.097
NCI-H1869 CTRP2 -0.2583 4.2505 -0.5468 36.202
Lu-65 CTRP2 -0.211 7.0338 -1.3352 37.9633
NCI-H1693 CTRP2 -0.1141 7.9493 -1.5785 38.1138
COR-L105 CTRP2 -0.1108 7.2464 -1.306 37.5336
NCI-H2106 CTRP2 -0.056 7.9232 -1.5065 37.7603
HCC366 CTRP2 0.1136 5.1418 -0.3637 34.3372
LC-1/sq-SF CTRP2 0.1369 4.825 -0.253 33.9284
LC-1F CTRP2 0.1836 8.9283 -1.6612 37.2412
RERF-LC-Ad1 CTRP2 0.3239 7.0373 -0.7618 34.6947
HCC2279 CTRP2 0.4178 3.8469 0.2646 31.3324
EKVX CTRP2 0.4943 6.1112 -0.2487 32.6853
HCC2935 CTRP2 0.8443 8.1586 -0.6495 32.6654
HOP-92 CTRP2 0.9491 8.4492 -0.6606 32.3611
DMS 454 CTRP2 1.0848 14.3539 -3.2153 37.2148
NCI-H2342 CTRP2 1.2231 7.9621 -0.1708 30.0989
Calu-1 CTRP2 1.6135 10.1934 -0.7478 30.587
NCI-H2172 CTRP2 1.8669 6.7094 1.0133 24.2175
BEN CTRP2 2.5171 9.9551 0.2599 25.0294
NCI-H1793 CTRP2 2.8468 8.7799 1.1332 21.084
IA-LM CTRP2 4.6877 10.9008 1.8139 14.1779
NCI-H2126 CTRP2 6.0292 7.4235 3.6329 0.2069
HCC1171 CTRP2 6.1515 20.446 -1.7543 23.0167
NCI-H2291 CTRP2 6.3399 20.5612 -1.6626 22.4496
Hs 888.Lu CTRP2 -0.7595 6.2735 -1.6633 40.7199
⏷ Show the Full List of 138 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 38 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 -5.0334 -1.2797 -5.0427 66.5533
TYK-nu CTRP2; CTRP1 -5.4204 3.9505 -6.095 63.6788
MCAS CTRP2 -4.7551 -0.64 -4.775 64.6026
A2780 CTRP2 -4.5901 -1.6641 -4.5921 64.0378
COV434 CTRP2 -4.1971 -0.4485 -4.2122 61.2384
RMUG-S CTRP1 -4.0416 6.2378 -5.2181 75.938
OVCAR-4 CTRP2 -3.5903 2.999 -3.9096 56.3655
SNU-119 CTRP2 -3.5882 0.1354 -3.6089 57.3218
OVTOKO CTRP2 -3.5504 -1.4897 -3.5506 57.2537
COV644 CTRP2; CTRP1 -3.5216 1.4463 -3.621 56.5976
DOV13 CTRP2 -3.1479 0.6066 -3.176 54.4635
SNU-8 CTRP2 -3.0387 -0.7528 -3.0395 53.8446
JHOC-5 CTRP2 -2.9424 -0.3466 -2.9451 53.1977
OVCAR-8 CTRP2 -2.9307 4.1978 -3.4434 52.5661
IGROV-1 CTRP2 -2.4074 3.5834 -2.7408 49.6877
SNU-840 CTRP2; CTRP1 -2.3124 4.4455 -2.8268 49.2115
Caov-3 CTRP2; CTRP1 -2.2553 0.9139 -2.2733 48.6957
TOV-112D CTRP2 -2.2376 2.9488 -2.4442 48.6326
OC 314 CTRP2 -1.9948 0.4506 -1.9987 46.9034
OVSAHO CTRP2 -1.9118 3.565 -2.2004 46.6891
FU-OV-1 CTRP2 -1.2345 10.5959 -3.8423 45.092
ONCO-DG-1 CTRP2 -0.981 6.0512 -1.8315 41.913
ES2 CTRP2 -0.8962 2.9405 -1.0088 39.8941
TOV-21G CTRP2 -0.722 3.3269 -0.8766 38.8614
COV362 CTRP2 -0.6899 4.0659 -0.9761 38.9904
OAW28 CTRP2 -0.4451 2.8712 -0.5225 36.8146
JHOM-1 CTRP2 -0.4007 3.29 -0.5272 36.6679
OAW42 CTRP2 -0.2669 3.3434 -0.3917 35.7782
EFO-21 CTRP2 -0.1661 7.9617 -1.6387 38.4197
SK-OV-3 CTRP2 0.1895 6.391 -0.9598 31.697
OVISE CTRP2 0.2167 3.769 0.0612 32.6733
EFO-27 CTRP2 0.4086 9.3718 -1.6143 36.3929
JHOS-2 CTRP2 0.7691 7.1893 -0.3426 32.0482
Kuramochi CTRP2 1.0415 10.4912 -1.4589 34.056
OVCAR-5 CTRP2 1.1351 9.5183 -0.9293 32.4913
OV56 CTRP2 1.1766 7.6829 -0.1053 30.0437
OV-90 CTRP2; CTRP1 1.2183 11.1623 -1.5805 33.8508
OV7 CTRP2; CTRP1 1.5786 8.9345 -0.212 29.2128
⏷ Show the Full List of 38 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Aska-SS CTRP2 -3.7272 1.817 -3.8786 57.5878
Yamato-SS CTRP2 -1.696 -0.187 -1.696 44.9055
A-204 CTRP2 -4.6597 -1.012 -4.6692 64.2382
TTC-709 CTRP2 -4.1442 1.284 -4.2612 60.1203
TE 617.T CTRP2 -4.1356 -0.9537 -4.1407 61.0045
Rh41 CTRP2 -4.031 -1.8194 -4.0312 60.4437
G-402 CTRP2 -3.978 -1.398 -3.9791 60.0647
Tm87-16 CTRP2 -3.6259 -0.187 -3.6381 57.6235
KYM-1 CTRP2 -3.5131 -1.1631 -3.5138 56.9968
BT-16 CTRP2 -3.5058 -1.6105 -3.5059 56.9595
G-401 CTRP2 -3.5017 -0.7793 -3.5042 56.8993
TE 441.T CTRP2 -3.1736 1.6303 -3.2733 54.4476
SW982 CTRP2 -3.1598 3.0709 -3.4578 54.0361
GCT CTRP2 -3.1028 -0.2668 -3.1075 54.2512
BT-12 CTRP2 -2.9965 -0.8792 -2.997 53.5665
HT-1080 CTRP2; CTRP1 -2.7052 1.5384 -2.7734 51.6084
Rh18 CTRP2 -2.6845 1.3705 -2.7397 51.441
MES-SA CTRP2 -2.6168 1.552 -2.6825 51.0007
RD CTRP2 -2.5395 1.9552 -2.6375 50.4989
Hs 729.T CTRP2 -0.9959 2.6453 -1.0803 40.4767
SK-UT-1 CTRP2 -0.1904 5.0819 -0.6787 36.3145
SK-LMS-1 CTRP2 1.3586 9.6036 -0.7391 31.3131
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 -3.104 -2.5643 -3.104 54.2859
SYO-1 CTRP2 -1.6381 5.7022 -2.4381 45.5758
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 -0.2723 3.0261 -4.1055 3.2997
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2 -5.5425 0.3531 -5.6444 67.7295
NCI-H2452 CTRP2 -4.7115 4.2381 -5.3937 66.1857
NCI-H28 CTRP2 -3.7348 -0.1932 -3.7486 58.3119
NCI-H2052 CTRP2 -2.3689 5.7009 -3.2343 49.5285
MPP 89 CTRP2 -0.954 3.7549 -1.2003 40.5947
ACC-MESO-1 CTRP2 -0.3479 2.6207 -0.3969 36.0815
IST-Mes1 CTRP2 0.6837 4.7508 0.3623 30.1297
JL-1 CTRP2 1.0827 3.1731 1.0536 26.4911
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
22Rv1 CTRP2 -3.5667 2.7247 -3.8366 56.3492
VCaP CTRP2 -2.8223 -0.8072 -2.8227 52.408
LNCaP clone FGC CTRP2 -2.2047 1.7552 -2.2681 48.3468
DU145 CTRP2 0.709 10.3485 -1.7323 35.6735
NCI-H660 CTRP2 2.6568 8.3461 1.1415 21.5512
PaCa-3 CTRP2 4.5655 14.2885 0.0175 20.988
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 -3.509 -2.1686 -3.509 56.9836
A-253 CTRP2 -1.729 4.2795 -2.1537 45.7201
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ECC10 CTRP2 -7.1116 -2.6319 -7.1221 78.0259
OCUM-1 CTRP2 -6.2419 1.793 -6.5615 68.7663
GSS CTRP2 -4.938 -3.2204 -4.938 66.496
Fu97 CTRP2 -4.9148 -1.8068 -4.9173 66.0964
SNU-16 CTRP2 -4.3805 -2.7475 -4.3805 62.7873
SNU-620 CTRP2 -4.3165 -2.753 -4.3165 62.3622
SNU-1 CTRP2 -4.2202 -2.1003 -4.2203 61.7058
IM95 CTRP2 -3.9853 -0.8701 -3.9901 60.035
23132/87 CTRP2 -3.9552 -2.1577 -3.9552 59.9529
HGC-27 CTRP2 -3.7454 0.5196 -3.7868 58.1833
SNU-719 CTRP2 -3.4644 0.1311 -3.4824 56.5439
NUGC-4 CTRP2 -3.4265 0.5773 -3.461 56.2189
SNU-216 CTRP2 -3.4002 2.4923 -3.621 55.5284
NCC-StC-K140 CTRP2 -3.1971 3.4247 -3.565 54.1494
ECC12 CTRP2 -3.1152 -1.5508 -3.1152 54.3603
NCI-N87 CTRP2 -2.9982 3.2836 -3.3223 53.0952
SNU-668 CTRP2 -2.7771 -0.1588 -2.7805 52.1001
SNU-5 CTRP2 -2.6018 -0.4151 -2.6027 50.9389
Hs 746.T CTRP2 -2.5496 3.6867 -2.9158 50.5134
AGS CTRP2 -2.2767 -0.1852 -2.2776 48.7753
SNU-601 CTRP2 -1.7395 4.1703 -2.14 45.7567
HuG1-N CTRP2 -1.3498 1.9259 -1.3902 42.7039
GSU CTRP2 -1.2389 2.2547 -1.2989 42.0185
MKN74 CTRP2 -0.516 8.0552 -2.0475 40.4346
MKN7 CTRP2 -0.3096 6.3164 -1.1895 38.0122
LMSU CTRP2 0.6909 7.2516 -0.4501 32.6122
SH-10-TC CTRP2 0.8678 2.9566 0.8446 27.9028
MKN1 CTRP2 1.8075 8.1755 0.3481 37.8639
KE-39 CTRP2 3.0561 14.2995 -1.3292 28.3166
MKN45 CTRP2 6.4699 15.6607 0.8724 14.4277
SNG-M CTRP2 -3.2314 2.4455 -3.4332 54.5945
SNU-685 CTRP2 0.7462 4.5793 0.4719 29.5597
SNU-1077 CTRP2 4.6427 11.9939 1.2294 16.5469
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ML-1 [Human leukemia] CTRP2 -4.3431 4.7437 -5.12 64.309
FTC-238 CTRP2 -3.6799 -0.5263 -3.6865 58.0256
8305C CTRP2 -3.3355 -1.479 -3.3356 55.8262
BHT-101 CTRP2 -2.9913 -1.7819 -2.9913 53.5348
TT CTRP2 -2.8305 0 -2.8362 52.4492
B-CPAP CTRP2 -2.527 -0.0828 -2.5295 50.4407
SW579 CTRP2 -2.2251 0.7876 -2.2387 48.4437
CAL-62 CTRP2 -2.0004 3.5232 -2.2883 47.23
CGTH-W-1 CTRP2 -1.7712 3.1232 -1.9709 45.7163
8505C CTRP2 -1.0745 4.5136 -1.4962 41.7216
FTC-133 CTRP2 -0.133 3.5279 -0.2758 34.9481
TT2609-C02 CTRP2 0.5911 12.3742 -2.7706 37.9229
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 29 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 -4.42 -1.1324 -4.4253 62.8289
HSC-2 CTRP2 -4.3566 -1.1613 -4.3611 62.4432
SCC-25 CTRP2 -4.042 -0.8914 -4.0471 60.3996
HSC-3 CTRP2 -3.5656 -1.4092 -3.5659 57.3527
SNU-1214 CTRP2 -3.5442 -0.6961 -3.5476 57.1693
BHY CTRP2 -3.3429 -0.0712 -3.3536 55.7977
BICR 22 CTRP2 -3.3349 -0.3516 -3.3406 55.775
Detroit 562 CTRP2 -3.2216 -0.7222 -3.2232 55.0546
SNU-899 CTRP2 -3.0756 -1.6128 -3.0756 54.0961
SCC-4 CTRP2 -2.9982 -0.5731 -2.9997 53.5727
CAL-33 CTRP2 -2.9305 1.0385 -2.9737 53.0321
BICR 18 CTRP2 -2.9085 0.546 -2.9283 52.9326
HSC-4 CTRP2 -2.5904 2.6272 -2.8598 47.7635
BICR 6 CTRP2 -2.5511 3.1874 -2.8217 50.538
YD-8 CTRP2 -2.5389 2.8928 -2.7589 50.4732
PE/CA-PJ34 (clone C12) CTRP2 -2.3698 1.145 -2.4006 49.4057
CAL-27 CTRP2 -2.3193 0.67 -2.3314 49.0656
BICR 16 CTRP2 -2.0843 2.4195 -2.2071 47.6186
PE/CA-PJ49 CTRP2 -1.8359 1.648 -1.8768 45.9121
SNU-1076 CTRP2 -1.6415 1.1164 -1.6537 44.5722
PE/CA-PJ15 CTRP2 -1.1809 3.3605 -1.3748 41.94
SCC-9 CTRP2 -1.1048 3.2233 -1.2712 41.3875
BICR 56 CTRP2 -1.0545 1.727 -1.0748 40.6921
FaDu CTRP2 -0.7531 3.0453 -0.8699 38.9637
BICR 31 CTRP2 -0.6384 3.4726 -0.8097 38.3584
SNU-1041 CTRP2 -0.2014 4.9292 -0.6495 36.2767
PE/CA-PJ41 (clone D2) CTRP2 0.2173 5.886 -0.4753 34.2913
SNU-1066 CTRP2 0.8957 6.5534 0.0306 30.5109
SNU-46 CTRP2 1.3403 5.0049 1.0128 25.8091
⏷ Show the Full List of 29 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
5637 CTRP2 -4.0292 0.4627 -4.0769 59.8828
RT-112 CTRP2 -3.3266 0.0443 -3.3397 55.6785
JMSU-1 CTRP2 -3.2714 -0.5688 -3.2743 55.3752
VM-CUB-1 CTRP2 -3.2622 0.3431 -3.2828 55.2264
647V CTRP2 -2.9403 1.0805 -2.9863 53.0897
BFTC-905 CTRP2 -2.8619 0.3529 -2.875 52.6409
639V CTRP2 -2.6416 -0.5634 -2.6422 51.2045
KU-19-19 CTRP2 -2.4381 -0.7676 -2.4381 49.8492
U-BLC1 CTRP2 -2.4174 4.726 -3.0142 49.7638
CAL-29 CTRP2 -2.2828 0.9176 -2.3017 48.8283
253J CTRP2 -2.1603 0.2141 -2.1631 48.0028
UM-UC-3 CTRP2 -2.0866 4.2864 -2.7058 44.9327
SW1710 CTRP2 -2.0237 3.4845 -2.3062 47.3677
BC-3C CTRP2 -1.8085 3.566 -2.0888 46.0449
UM-UC-1 CTRP2 -1.7426 3.2776 -1.9657 45.5664
TCCSUP CTRP2 -1.3522 3.7235 -1.6252 43.1858
253J-BV CTRP2 -0.9513 4.8482 -1.4464 41.1019
SCaBER CTRP2 -0.9035 3.0912 -1.0365 39.9942
HT-1197 CTRP2 0.0899 3.8141 -0.0832 33.5688
KMBC-2 CTRP2 0.1508 7.6051 -1.1625 36.2796
T24 CTRP2 0.5153 6.0832 -0.2165 32.5189
J82 CTRP2 1.1305 7.2907 0.0028 29.8531
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 -2.5942 1.5603 -2.6596 50.8563

References

1 Targeting of eEF1A with Amaryllidaceae isocarbostyrils as a strategy to combat melanomas. FASEB J. 2010 Nov;24(11):4575-84.