Details of the Drug

General Information of Drug (ID: DMJAGXQ)

Drug Name
Niclosamide
Synonyms
niclosamide; 50-65-7; Niclocide; 5-Chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxybenzamide; Tredemine; Bayluscid; Phenasal; Yomesan; Fenasal; Dichlosale; Helmiantin; Sagimid; Iomezan; Devermine; Atenase; Vermitid; Radeverm; Mansonil; Iomesan; Devermin; Cestocid; Sulqui; Lintex; Nasemo; Mato; Fedal-Telmin; Bayer 73; Radewerm; Zestocarp; Bayer 2353; 2',5-Dichloro-4'-nitrosalicylanilide; Chemagro 2353; BAY 2353; Benzamide, 5-chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxy-; 5-Chloro-2'-chloro-4'-nitrosalicylanilide; nicolsamide; HL 2447; Niclosamidum [I
Indication
Disease Entry ICD 11 Status REF
Cestodes infection 1F70-1F76 Approved [1]
Haemophilus influenza 1G40 Approved [2]
Taeniasis N.A. Approved [2]
Affected Organisms
Helminthic Microorganisms
ATC Code
P02DA01: Niclosamide
P02DA: Salicylic acid derivatives
P02D: ANTICESTODALS
P02: ANTHELMINTICS
P: ANTIPARASITIC PRODUCTS, INSECTICIDES AND REPELLENTS
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 327.12
Logarithm of the Partition Coefficient (xlogp) 4
Rotatable Bond Count (rotbonds) 2
Hydrogen Bond Donor Count (hbonddonor) 2
Hydrogen Bond Acceptor Count (hbondacc) 4
ADMET Property
BDDCS Class
Biopharmaceutics Drug Disposition Classification System (BDDCS) Class 4: low solubility and low permeability [3]
MRTD
The Maximum Recommended Therapeutic Dose (MRTD) of drug that ensured maximising efficacy and moderate side effect is 87.34 micromolar/kg/day [4]
Water Solubility
The ability of drug to dissolve in water is measured as 0.013 mg/mL [3]
Chemical Identifiers
Formula
C13H8Cl2N2O4
IUPAC Name
5-chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxybenzamide
Canonical SMILES
C1=CC(=C(C=C1[N+](=O)[O-])Cl)NC(=O)C2=C(C=CC(=C2)Cl)O
InChI
InChI=1S/C13H8Cl2N2O4/c14-7-1-4-12(18)9(5-7)13(19)16-11-3-2-8(17(20)21)6-10(11)15/h1-6,18H,(H,16,19)
InChIKey
RJMUSRYZPJIFPJ-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
4477
ChEBI ID
CHEBI:7553
CAS Number
50-65-7
UNII
8KK8CQ2K8G
DrugBank ID
DB06803
TTD ID
D0J9ZR
INTEDE ID
DR1146
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug
Repurposed Drugs (RPD) Click to Jump to the Detailed RPD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug-Metabolizing Enzyme (DME)
DME Name DME ID UniProt ID MOA REF
Cytochrome P450 2C9 (CYP2C9) DE5IED8 CP2C9_HUMAN Substrate [5]
Nitroreductase (NTR) DE0K82S A0A5K1UB29_SALTM Substrate [6]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
17-beta-hydroxysteroid dehydrogenase 14 (HSD17B14) OT0ETO72 DHB14_HUMAN Gene/Protein Processing [7]
2'-5'-oligoadenylate synthase 1 (OAS1) OT8ZLOCY OAS1_HUMAN Gene/Protein Processing [7]
2,4-dienoyl-CoA reductase , mitochondrial (DECR1) OTCDIR6X DECR_HUMAN Gene/Protein Processing [8]
24-hydroxycholesterol 7-alpha-hydroxylase (CYP39A1) OTBAJT4I CP39A_HUMAN Gene/Protein Processing [9]
3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 (HSD3B1) OTNAZVKB 3BHS1_HUMAN Gene/Protein Processing [7]
3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2 (HSD3B2) OT02MSKN 3BHS2_HUMAN Gene/Protein Processing [7]
3',5'-cyclic-AMP phosphodiesterase 4B (PDE4B) OTOA8WU2 PDE4B_HUMAN Gene/Protein Processing [7]
3'-5' exoribonuclease HELZ2 (HELZ2) OTM6HVO6 HELZ2_HUMAN Gene/Protein Processing [7]
4-hydroxy-2-oxoglutarate aldolase, mitochondrial (HOGA1) OT7XETW4 HOGA1_HUMAN Gene/Protein Processing [7]
5'(3')-deoxyribonucleotidase, mitochondrial (NT5M) OTJF73BA NT5M_HUMAN Gene/Protein Processing [7]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 144 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 0.0807 2.7454 0.0408 33.2008
JK1 CTRP2 3.0547 7.6754 1.8463 17.8227
JM1 CTRP2 1.077 4.061 0.9381 26.9033
Mino CTRP2 -10.0428 22.9131 -18.2765 62.1384
KMS-34 CTRP2 -2.564 0.6382 -2.5797 50.6802
SUP-M2 CTRP2 -1.2055 1.9073 -1.2395 41.732
KM-H2 CTRP2 -0.954 1.4604 -0.9633 39.9915
Daudi CTRP2 -0.9373 1.6813 -0.953 39.8994
CML-T1 CTRP2 -0.9304 1.5026 -0.9404 39.8361
SU-DHL-1 CTRP2 -0.9113 1.3774 -0.9181 39.6994
RPMI-8402 CTRP2 -0.7938 1.4012 -0.7996 38.9133
WSU-DLCL2 CTRP2 -0.7913 0.9688 -0.7924 38.882
Pfeiffer CTRP2 -0.7588 1.8078 -0.7749 38.7126
KMS-18 CTRP2 -0.6277 2.9726 -0.7275 38.0894
TF-1 CTRP2 -0.6229 1.663 -0.6318 37.7853
KCL-22 CTRP2 -0.6064 2.2451 -0.6394 37.7508
CA46 CTRP2 -0.5658 2.3036 -0.6009 37.4869
RPMI-8226 CTRP2 -0.5649 3.1517 -0.6834 37.7283
Jurkat CTRP2 -0.5227 1.7685 -0.5327 37.1215
DB CTRP2 -0.4963 2.5492 -0.5462 37.0707
KMS-20 CTRP2 -0.4921 1.164 -0.4931 36.8884
P12-Ichikawa CTRP2 -0.4786 2.266 -0.5083 36.8904
Namalwa CTRP2 -0.4775 2.1716 -0.502 36.8667
JURL-MK1 CTRP2 -0.4681 2.1147 -0.4895 36.7943
BL-70 CTRP2 -0.4449 2.1802 -0.4688 36.6478
KMS-21-BM CTRP2 -0.3946 2.1087 -0.4136 36.2972
EB1 CTRP2 -0.3923 2.024 -0.4079 36.2708
F-36P CTRP2 -0.3314 1.2834 -0.3324 35.8175
DEL CTRP2 -0.2493 1.5466 -0.2518 35.2755
NALM-6 CTRP2 -0.1825 2.4693 -0.2138 34.9248
HD-MY-Z CTRP2 -0.1681 2.7772 -0.2219 34.9014
LAMA-84 CTRP2 -0.1489 4.2048 -0.418 35.4327
KE-37 CTRP2 -0.0681 1.9064 -0.0742 34.0806
Ki-JK CTRP2 -0.0023 1.2614 -0.0025 33.6226
TALL-1 [Human adult T-ALL] CTRP2 0.0239 3.2124 -0.0646 33.7365
EoL-1 CTRP2 0.0256 2.729 -0.0153 33.5708
RL CTRP2 0.0334 2.2902 0.0178 33.4357
U-937 CTRP2 0.0357 3.9494 -0.1664 34.0179
JeKo-1 CTRP2 0.0744 2.1045 0.0659 33.1389
A3/Kawakami CTRP2 0.0893 1.5986 0.0883 33.0149
KMS-12-BM CTRP2 0.0981 2.4462 0.0775 33.0213
ST486 CTRP2 0.1063 2.6802 0.0722 33.0113
MOLT-3 CTRP2 0.1125 1.4119 0.1123 32.8577
PF-382 CTRP2 0.114 2.8383 0.0683 32.9982
OPM-2 CTRP2 0.119 1.3304 0.1189 32.8142
LP-1 CTRP2 0.1301 2.013 0.1246 32.7578
GA-10 CTRP2 0.1384 1.5173 0.1379 32.6863
Raji CTRP2 0.1401 3.2358 0.0559 32.9505
KMS-27 CTRP2 0.1818 2.1079 0.175 32.418
HEL CTRP2 0.1905 4.6551 -0.1518 33.4344
MV4-11 CTRP2 0.2248 1.7648 0.2233 32.1139
AML-193 CTRP2 0.2363 1.1698 0.2363 32.0324
K-562 CTRP2 0.2437 4.2159 0.006 32.7586
NCO2 CTRP2 0.297 2.7039 0.2687 31.722
KHM-1B CTRP2 0.3184 4.5641 0.0095 32.4927
Peer CTRP2 0.3233 4.6876 -0.015 32.5534
HDLM-2 CTRP2 0.3551 3.022 0.3051 31.4073
DND-41 CTRP2 0.3881 2.8666 0.3523 31.1406
ALL-SIL CTRP2 0.3892 2.383 0.3785 31.0494
HEL 92.1.7 CTRP2 0.4003 2.2029 0.3946 30.9585
CMK CTRP2 0.4018 1.6121 0.4016 30.9302
697 CTRP2 0.4607 1.4099 0.4606 30.5376
OCI-Ly3 CTRP2 0.4633 3.9134 0.302 31.0573
OCI-AML-3 CTRP2 0.4872 1.3772 0.4872 30.3604
SUP-HD1 CTRP2 0.493 2.1965 0.4886 30.3369
MOTN-1 CTRP2 0.5108 3.09 0.4624 30.3653
KYO-1 CTRP2 0.5409 2.3693 0.5335 30.0275
SU-DHL-4 CTRP2 0.5411 4.8717 0.1759 31.2107
PL21 CTRP2 0.5602 4.2724 0.3378 30.6176
RS4;11 CTRP2 0.5705 2.3324 0.5645 31.9545
MOLM-13 CTRP2 0.5883 4.1711 0.3889 30.355
KMS-11 CTRP2 0.5938 4.129 0.4031 30.2895
P31/FUJ CTRP2 0.6199 3.3282 0.5536 29.6988
L-540 CTRP2 0.6672 4.9489 0.2932 30.4116
SKM-1 CTRP2 0.7073 3.4037 0.6377 29.1284
SET-2 CTRP2 0.7217 2.0745 0.7206 28.8024
A4/Fukuda CTRP2 0.7375 1.6467 0.7375 28.6934
M-07e CTRP2 0.7714 2.5551 0.7631 28.4951
NCI-H929 CTRP2 0.8236 2.454 0.8186 28.1364
THP-1 CTRP2 0.8418 5.5799 0.3013 29.816
REC-1 CTRP2 0.8605 4.9034 0.5161 29.0404
SIG-M5 CTRP2 0.8765 2.1253 0.8758 27.7696
Karpas-422 CTRP2 0.8903 2.4015 0.887 27.6863
Karpas-299 CTRP2 0.9967 4.2412 0.8175 27.5754
OCI-M1 CTRP2 1.015 2.2991 1.0139 26.8481
EJM CTRP2 1.0188 3.8939 0.9033 27.2103
MOLP-8 CTRP2 1.0226 2.0393 1.0224 26.7943
GDM-1 CTRP2 1.0316 4.2706 0.8495 27.3533
NOMO-1 CTRP2 1.0529 4.2092 0.8846 27.1644
NB4 CTRP2 1.1511 3.9448 1.0374 26.3237
OCI-AML-2 CTRP2 1.1608 4.2475 0.994 26.4418
HuNS1 CTRP2 1.2557 2.9237 1.2454 25.2751
OCI-AML-5 CTRP2 1.2818 2.2741 1.2816 25.0678
MOLT-16 CTRP2 1.2837 4.9188 0.9738 26.1227
Toledo CTRP2 1.3081 3.9487 1.2054 25.2405
HuT 78 CTRP2 1.311 2.78 1.306 24.8892
SK-MM-2 CTRP2 1.3237 2.9313 1.3147 24.8176
Ri-1 CTRP2 1.3335 6.0587 0.6784 26.9956
HL-60 CTRP2 1.3335 3.6944 1.2676 24.9449
Kasumi-2 CTRP2 1.3905 2.0941 1.3905 24.3426
NU-DUL-1 CTRP2 1.4037 6.5596 0.5746 27.1368
MM1.S CTRP2 1.4849 5.3019 1.0865 25.1012
HPB-ALL CTRP2 1.519 3.283 1.4993 23.5527
SR CTRP2 1.538 5.2524 1.159 24.6806
SUP-T11 CTRP2 1.5557 3.523 1.52 23.3623
Mono-Mac-1 CTRP2 1.5621 3.158 1.5501 23.2396
U266B1 CTRP2 1.5876 4.082 1.4843 23.3814
MOLP-2 CTRP2 1.5886 3.7287 1.5341 23.2073
SU-DHL-10 CTRP2 1.6132 5.4182 1.1914 24.335
Ci-1 CTRP2 1.6652 4.4564 1.4989 23.0838
AMO1 CTRP2 1.6699 5.5455 1.2136 24.0831
SEM CTRP2 1.6726 2.1909 1.6726 22.4635
Reh CTRP2 1.7534 4.902 1.4908 22.8372
Kasumi-1 CTRP2 1.7723 4.0652 1.6853 22.0947
Karpas-620 CTRP2 1.7802 2.7014 1.7798 21.748
SUP-T1 CTRP2 1.7876 4.1604 1.6867 22.0411
RPMI-6666 CTRP2 1.8217 4.7355 1.6067 22.2141
L-363 CTRP2 2.106 4.4587 1.9764 20.0206
KO52 CTRP2 2.1286 4.4899 1.9948 19.885
Granta-519 CTRP2 2.177 5.9277 1.636 21.038
BV-173 CTRP2 2.3035 5.6419 1.871 19.8
JJN-3 CTRP2 2.3057 5.3066 1.9801 19.3934
OCI-Ly19 CTRP2 2.4938 6.7887 1.6467 20.0951
L-1236 CTRP2 2.5573 5.3226 2.2494 17.657
EM-2 CTRP2 2.6686 7.8842 1.3605 20.7009
ME1 CTRP2 2.6687 5.2585 2.3902 16.8095
MOLM-16 CTRP2 2.7158 7.6803 1.4989 20.0515
SUP-B15 CTRP2 2.7333 6.475 2.0261 17.989
MOLM-6 CTRP2 2.8045 9.1821 0.9043 22.0339
RCH-ACV CTRP2 3.0628 7.6185 1.88 17.6701
SU-DHL-6 CTRP2 3.4145 8.4783 1.8332 16.9663
SU-DHL-8 CTRP2 4.003 8.8397 2.2217 14.0146
JVM-2 CTRP2 4.1475 10.8797 1.3493 17.1514
EHEB CTRP2 4.1567 10.1057 1.7406 15.6035
JVM-3 CTRP2 4.3096 11.7303 1.0709 17.8506
MC116 CTRP2 4.5169 9.9479 2.1403 13.218
MOLT-13 CTRP2 4.8371 9.2837 2.7496 10.0444
MJ CTRP2 4.9126 15.4027 -0.245 21.1094
Hs 611.T CTRP2 5.3237 10.1616 2.7146 9.2527
P3HR-1 CTRP2 6.0322 9.7312 3.4644 4.9587
MHH-CALL-4 CTRP2 6.5208 8.8838 4.1706 1.6183
OCI-Ly10 CTRP2 6.8103 10.5921 3.5676 3.512
KMM-1 CTRP2 7.7461 11.9003 3.52 2.7038
MHH-CALL-3 CTRP2 8.7786 10.7908 4.4019 0.1025
⏷ Show the Full List of 144 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 0.8758 3.8527 0.7563 28.1754
TE15 CTRP2 2.3165 6.8711 1.4263 21.4179
KYSE-30 CTRP2 -0.1947 1.5703 -0.197 34.9112
EC-GI-10 CTRP2 0.2082 2.3432 0.1949 32.2636
TE-10 CTRP2 0.436 3.6513 0.3156 31.1033
KYSE-510 CTRP2 0.5316 1.4343 0.5316 30.0646
TE-4 CTRP2 0.5847 3.1089 0.5383 29.8664
TE-9 CTRP2 0.5961 4.2093 0.3897 30.3268
OE21 CTRP2 0.7008 2.4464 0.6941 28.96
TE-11 CTRP2 0.7146 5.0597 0.3149 30.185
TE-14 CTRP2 0.8874 3.1041 0.8552 27.8024
COLO 680N CTRP2 0.9796 5.1362 0.583 28.4317
KYSE-520 CTRP2 0.9876 5.8559 0.3715 29.1165
TE-6 CTRP2 1.3113 2.6818 1.3082 26.6566
KYSE-180 CTRP2 1.4312 6.0745 0.7785 26.3491
KYSE-450 CTRP2 1.5917 3.6951 1.5411 23.173
TE-5 CTRP2 1.7768 4.0322 1.6951 22.0467
KYSE-70 CTRP2 1.9447 5.7595 1.4424 22.4322
KYSE-140 CTRP2 2.422 9.7335 0.2697 25.2505
KYSE-150 CTRP2 2.8508 10.8982 0.1355 24.5717
KYSE-410 CTRP2 3.1739 5.7241 2.7841 13.8682
TE-1 CTRP2 4.4036 10.067 1.981 14.1042
OE33 CTRP2 5.7302 9.9186 3.1526 6.7192
OE19 CTRP2 7.0392 8.5692 4.5422 0.2571
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 38 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 7.5712 9.2011 4.518 0.1612
KP-4 CTRP2 -0.9483 1.3811 -0.9557 39.9472
QGP-1 CTRP2 0.3531 3.4319 0.2579 31.5708
MIA PaCa-2 CTRP2 0.423 2.7475 0.3966 30.8766
DAN-G CTRP2 0.8799 7.0022 -0.1529 31.1269
PSN1 CTRP2 0.9652 4.1763 0.796 27.7506
Panc 03.27 CTRP2 1.1658 4.033 1.0386 26.2719
SU.86.86 CTRP2 1.6082 3.5878 1.5693 23.0235
KP-3 CTRP2 1.8599 10.367 -0.5815 29.421
SW1990 CTRP2 1.9856 6.5177 1.2136 23.1469
HuP-T3 CTRP2 2.1305 7.433 0.9994 23.5116
PANC-1 CTRP2 2.283 5.2971 1.9581 19.5418
Panc 02.03 CTRP2 2.5265 6.5225 1.788 19.4703
SNU-410 CTRP2 2.5589 5.0486 2.3308 17.3565
Capan-2 CTRP2 2.5783 8.1039 1.1708 21.652
Panc 04.03 CTRP2 2.6253 7.5435 1.4658 20.4198
PK-59 CTRP2 2.6923 7.8482 1.4006 20.4865
YAPC CTRP2 2.8884 5.316 2.612 15.3416
Panc 10.05 CTRP2 2.9343 6.8127 2.099 17.1584
PaTu 8988t CTRP2 2.9486 7.2995 1.9049 17.8727
PaTu 8988s CTRP2 3.9953 6.6999 3.2362 9.9017
Panc 08.13 CTRP2 4.5116 9.1863 2.5142 11.6945
AsPC-1 CTRP2 4.5754 8.3111 3.0054 9.5186
CFPAC-1 CTRP2 5.2967 10.9031 2.3226 10.9202
PaTu 8902 CTRP2 5.4436 12.9237 1.4323 14.1856
SUIT-2 CTRP2 6.5916 8.0475 4.5538 0.4079
SNU-213 CTRP2 6.7288 7.9724 4.6378 0.1875
Capan-1 CTRP2 6.7418 9.2335 4.1381 1.526
Panc 05.04 CTRP2 6.9244 11.1242 3.3919 4.0437
TCC-Pan2 CTRP2 6.9419 8.5234 4.5202 0.3317
KP-2 CTRP2 6.9458 8.3288 4.5929 0.1997
HuP-T4 CTRP2 6.9808 9.3845 4.1967 1.1462
HPAF-II CTRP2 7.089 9.6825 4.1262 1.2807
L3.3 CTRP2 7.3084 8.6645 4.6087 0.1036
HPAC CTRP2 7.4318 8.7835 4.6116 0.0837
BxPC-3 CTRP2 7.5325 14.144 2.3635 7.2141
Hs 766T CTRP2 7.5961 8.9004 4.6289 0.0534
PK-45H CTRP2 8.1981 10.0274 4.4579 0.1242
⏷ Show the Full List of 38 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 1.9718 8.5542 0.3522 26.2178
SK-MEL-1 CTRP2 -0.6947 0.8534 -0.6951 38.2361
WM115 CTRP2 -0.4226 1.4853 -0.4258 36.4326
COLO 741 CTRP2 -0.3711 3.7461 -0.5686 36.6797
UACC-62 CTRP2 -0.2689 2.0174 -0.2815 35.4395
CJM [Human melanoma] CTRP2 -0.2276 1.9697 -0.2378 35.1564
RVH-421 CTRP2 -0.2188 1.8617 -0.2261 35.0884
HT-144 CTRP2 -0.196 2.2153 -0.2144 34.9727
WT2-iPS CTRP2 -0.1129 1.5961 -0.1149 34.3652
G-361 CTRP2 -0.1096 3.4141 -0.2337 34.7351
MeWo CTRP2 0.0039 3.0986 -0.0726 33.8309
WM266-4 CTRP2 0.029 2.0338 0.0216 33.4378
COLO 792 CTRP2 0.0391 1.8493 0.0353 33.3587
HMCB CTRP2 0.1109 1.896 0.1072 32.8798
Hs 944.T CTRP2 0.1212 5.4081 -0.4321 34.5073
WM88 CTRP2 0.2573 1.9968 0.2536 31.9045
SK-MEL-24 CTRP2 0.3558 2.5659 0.337 31.2989
SK-MEL-3 CTRP2 0.5282 3.317 0.4579 30.3226
Mel Ho CTRP2 0.5526 3.6033 0.4474 30.2775
RPMI-7951 CTRP2 0.5955 2.8942 0.5661 29.7376
UACC-257 CTRP2 0.8283 3.7438 0.722 28.4468
SK-MEL-2 CTRP2 0.8392 1.665 0.8391 28.0159
COLO 829 CTRP2 0.8663 6.4798 0.0254 30.6221
A101D CTRP2 0.9132 3.8197 0.8016 27.8999
Hs 294T CTRP2 1.0278 2.5158 1.0242 26.771
SK-MEL-5 CTRP2 1.0363 6.8403 0.0757 29.9205
WM983B CTRP2 1.1631 4.5093 0.9418 26.615
IGR-37 CTRP2 1.3506 6.7951 0.4291 27.7913
SK-MEL-30 CTRP2 1.546 4.8184 1.2858 24.2069
SK-MEL-28 CTRP2 1.5882 2.064 1.5882 23.026
Mel JuSo CTRP2 1.6285 7.1078 0.6036 26.3615
LOX-IMVI CTRP2 1.7101 5.7571 1.1886 24.0516
IGR-1 CTRP2 1.9635 7.5317 0.7835 24.7578
Hs 895.T CTRP2 2.1498 4.693 1.9739 19.8921
K029AX CTRP2 2.4355 6.1001 1.8525 19.4852
Hs 688(A).T CTRP2 2.5312 3.8282 2.5147 16.7984
A2058 CTRP2 2.5619 6.2028 1.9495 18.7604
WM1799 CTRP2 2.6304 7.2869 1.5817 19.9665
IPC-298 CTRP2 2.6592 8.3039 1.163 21.4647
COLO 800 CTRP2 2.777 8.5202 1.1832 21.0795
A-375 CTRP2 3.3893 7.651 2.1941 15.5986
Hs 934.T CTRP2 3.4186 5.4694 3.1383 11.8348
SK-MEL-31 CTRP2 3.7067 10.6452 1.0637 19.2313
Hs 839.T CTRP2 4.2596 8.9425 2.408 12.6776
Hs 936.T CTRP2 4.8061 10.7156 2.0078 13.1578
Hs 940.T CTRP2 4.8385 8.3424 3.2208 8.0711
IGR-39 CTRP2 5.5373 10.0617 2.9337 7.9576
MDA-MB-435S CTRP2 5.6526 13.5341 1.2952 14.3188
Hs 852.T CTRP2 6.3747 11.7475 2.7264 7.4355
WM793 CTRP2 7.1649 15.5303 1.4463 11.2086
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 0.4257 3.5093 0.3249 31.1066
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NB1 CTRP2 0.4465 2.8725 0.4127 30.7445
MHH-NB-11 CTRP2 0.6138 2.2125 0.6105 29.5284
Kelly CTRP2 0.6426 4.4617 0.3863 30.1847
SiMa CTRP2 0.6578 2.4004 0.6516 29.2447
SK-N-BE(2) CTRP2 0.7045 2.4228 0.6984 28.9334
CHP-212 CTRP2 0.8076 2.2592 0.8054 28.2335
IMR-32 CTRP2 0.9048 2.0045 0.9046 27.5793
SK-N-SH CTRP2 0.9797 2.6495 0.9725 27.1037
NH-6 CTRP2 1.3316 2.8304 1.3257 24.7547
SK-N-DZ CTRP2 1.6111 2.092 1.6111 22.8734
SK-N-AS CTRP2 2.0278 5.6031 1.5843 21.6679
KP-N-YN CTRP2 2.5004 8.1004 1.093 22.1486
SK-N-FI CTRP2 3.0569 9.0491 1.2147 20.2421
KP-N-SI9s CTRP2 3.4149 6.7093 2.6419 13.7576
CHP-126 CTRP2 6.7986 13.0198 2.4071 8.0721
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 6 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 0.6098 1.8137 0.6094 29.5452
SNU-478 CTRP2 0.808 3.3598 0.749 28.4218
HuCC-T1 CTRP2 2.1002 5.7897 1.6008 21.393
SNU-869 CTRP2 2.2863 7.5667 1.1051 22.6909
SNU-1196 CTRP2 5.6899 10.0039 3.0799 7.0877
SNU-308 CTRP2 7.6386 9.1648 4.5547 0.1092
⏷ Show the Full List of 6 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 15 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HOS CTRP2 0.3883 3.6083 0.2709 31.4099
SK-N-MC CTRP2 0.5074 0.9288 0.5074 30.2258
SJSA-1 CTRP2 0.7372 4.0719 0.5691 31.3416
SaOS-2 CTRP2 0.8515 2.5748 0.8441 27.9583
MG-63 CTRP2 0.9053 3.3512 0.8525 27.7526
SK-ES-1 CTRP2 1.0135 2.5269 1.0096 26.8674
TC71 CTRP2 1.3992 4.3706 1.2279 24.8715
A-673 CTRP2 1.499 2.0066 1.499 23.62
G-292 clone A141B1 CTRP2 2.9632 7.1858 1.9694 17.5838
MHH-ES-1 CTRP2 4.087 11.1929 1.1398 18.0813
CAL-78 CTRP2 4.5596 8.2662 3.0135 9.5188
U2OS CTRP2 4.6328 18.2079 -1.8834 26.2207
Hs 822.T CTRP2 4.7962 8.9271 2.8925 9.5309
Hs 888.T CTRP2 4.9219 8.7001 3.1135 8.3539
SW1353 CTRP2 7.453 16.4696 1.1933 11.6983
⏷ Show the Full List of 15 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 65 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU4475 CTRP2 0.1486 1.6995 0.1472 32.621
BT-20 CTRP2 0.2392 3.9083 0.0611 32.5971
Hs 578Bst CTRP2 0.396 13.3509 -3.4167 39.4365
HCC1500 CTRP2 0.4764 3.9427 0.311 30.9838
ZR-75-30 CTRP2 0.5095 2.2566 0.5043 30.2294
BT-549 CTRP2 0.6293 4.1784 0.4319 30.0763
HCC1428 CTRP2 0.7286 4.7487 0.4118 29.8182
CAMA-1 CTRP2 0.8168 4.7209 0.5148 29.1861
HCC1419 CTRP2 0.834 2.2442 0.8322 28.0564
MDA-MB-361 CTRP2 0.8584 2.445 0.854 27.9023
EFM-192A CTRP2 1.1398 4.7385 0.8626 26.9629
MDA-MB-453 CTRP2 1.1678 4.6291 0.9195 26.6771
SK-BR-3 CTRP2 1.1722 3.2662 1.14 25.905
T-47D CTRP2 1.1753 5.3819 0.7252 27.326
CAL-85-1 CTRP2 1.2214 3.3667 1.1832 25.5978
JIMT-1 CTRP2 1.3154 6.1914 0.6126 27.2773
MDA-MB-468 CTRP2 1.3902 3.2813 1.3659 24.4261
MDA-MB-231 CTRP2 2.5606 8.2065 1.1069 21.9354
AU565 CTRP2 2.5927 5.8928 2.0971 18.1174
HCC1143 CTRP2 3.2575 9.31 1.2862 19.4712
BT-474 CTRP2 3.3057 7.633 2.1186 16.1094
MCF-7 CTRP2 3.552 9.4183 1.5162 17.8742
HDQ-P1 CTRP2 3.6555 9.0417 1.7963 16.5301
HCC1937 CTRP2 4.3392 13.3786 0.276 20.6133
HCC1395 CTRP2 4.3867 8.8379 2.575 11.7117
HCC1806 CTRP2 5.0272 8.7411 3.1817 7.8611
HCC202 CTRP2 5.232 10.321 2.5607 10.0613
HCC38 CTRP2 5.5638 8.8193 3.5704 5.2622
CAL-51 CTRP2 5.6415 10.9668 2.5649 9.2994
CAL-148 CTRP2 5.8152 9.8812 3.2344 6.2409
ZR-75-1 CTRP2 6.486 9.014 4.0933 1.9259
HCC1954 CTRP2 7.5534 16.6027 1.1992 11.5273
BT 172 CTRP2 -0.4102 1.1749 -0.4109 36.3415
BT 416 CTRP2 -0.2199 1.5005 -0.2218 35.0781
BT147 CTRP2 -0.0123 3.1449 -0.0951 33.9588
BT 232 CTRP2 0.1045 3.0519 0.0387 33.1271
BT 231 CTRP2 0.3733 1.8465 0.3721 31.1234
BT 145 CTRP2 0.3747 1.9381 0.3727 31.1168
BT 428 CTRP2 0.7585 2.5315 0.7506 28.5796
BT 159 CTRP2 0.7678 2.5471 0.7596 28.5186
BT 286 CTRP2 0.7882 2.2315 0.7862 28.3623
BT164 CTRP2 0.8597 2.7794 0.8453 27.9269
BT 131 CTRP2 0.9368 2.4839 0.9327 27.3794
BT 248 CTRP2 0.9396 3.5592 0.8658 27.5955
BT 112 CTRP2 0.9799 3.2447 0.9407 27.2098
BT 216 CTRP2 0.9869 4.3855 0.7773 27.7446
BT 245 CTRP2 1.0433 8.891 -0.7505 32.307
BT 271 CTRP2 1.0659 3.105 1.0407 26.59
BT 139 CTRP2 1.1312 2.3807 1.13 26.0741
BT 228 CTRP2 1.2087 2.8711 1.1993 25.5852
BT 444 CTRP2 1.3896 4.6213 1.1629 25.1288
BT 359 CTRP2 1.4691 4.6591 1.2406 24.6066
BT 422 CTRP2 1.5316 4.5571 1.332 24.0895
BT 187 CTRP2 1.6823 5.5002 1.2413 23.9465
BT 498 CTRP2 2.0009 6.5388 1.2219 23.0723
BT 179 CTRP2 2.0279 6.3705 1.3145 22.6555
BT 340 CTRP2 2.2187 6.984 1.2774 22.246
BT 224 CTRP2 2.274 5.8888 1.7545 20.3168
BT 482 CTRP2 2.41 9.3945 0.4148 24.7959
BT 320 CTRP2 3.1336 12.0113 -0.1363 24.7364
BT 440 CTRP2 4.7557 13.0139 0.8165 17.8429
BT 328 CTRP2 4.8414 15.4791 -0.3431 21.5603
BT 333 CTRP2 5.1599 13.1378 1.0935 16.0127
BT 504 CTRP2 6.1427 16.3672 0.2702 17.0877
BT 330 CTRP2 8.1262 22.2066 -1.1235 18.0851
⏷ Show the Full List of 65 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 0.6705 3.4156 0.5973 29.3853
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-466 CTRP2 -1.2254 -0.2397 -1.2254 41.77
SF126 CTRP2 -0.6898 1.2198 -0.6921 38.2096
GB-1 CTRP2 -0.4705 2.8242 -0.5445 36.9729
SF539 CTRP2 -0.4511 2.5323 -0.4978 36.7604
D283 Med CTRP2 -0.1534 1.7748 -0.158 34.6438
T98G CTRP2 0.0724 3.4697 -0.047 33.5137
U-251MG CTRP2 0.1813 1.7353 0.1799 32.4033
8-MG-BA CTRP2 0.3749 1.4212 0.3749 31.1087
TM-31 CTRP2 0.4469 2.637 0.4273 30.6949
Daoy CTRP2 0.4519 2.2364 0.4462 30.6148
SNU-201 CTRP2 0.623 2.8782 0.5957 29.547
SF268 CTRP2 0.6489 4.2808 0.4323 30.0106
SNU-738 CTRP2 0.8056 4.4047 0.5762 29.0151
LN-18 CTRP2 0.9503 4.731 0.6579 28.2705
KNS-42 CTRP2 1.2125 2.4953 1.2108 25.5342
A-172 CTRP2 1.2573 4.4862 1.0494 25.9424
KG-1-C CTRP2 1.2711 4.4143 1.0799 25.7926
KNS-60 CTRP2 1.2719 5.2418 0.8718 28.3893
Hs 683 CTRP2 1.3926 3.6147 1.3394 24.5083
ONS-76 CTRP2 1.5823 7.1325 0.5448 26.7001
Becker CTRP2 1.6391 6.052 1.0113 24.8992
42-MG-BA CTRP2 1.6542 5.2216 1.2947 23.8412
DBTRG-05MG CTRP2 1.7285 3.1001 1.7224 22.1115
GOS-3 CTRP2 1.7929 3.9356 1.7258 21.8891
SNU-626 CTRP2 1.916 6.1397 1.279 23.1123
SNB-75 CTRP2 2.0606 5.4217 1.6778 21.2294
SNU-489 CTRP2 2.4138 6.6696 1.6101 20.4568
SNU-1105 CTRP2 2.5925 7.6345 1.3924 20.7851
DK-MG CTRP2 2.7728 6.4258 2.0876 17.6444
CCF-STTG1 CTRP2 2.8007 5.9036 2.3171 16.6949
YKG-1 CTRP2 3.2281 7.4009 2.1453 16.2026
NMC-G1 CTRP2 3.3522 6.7039 2.5795 14.1686
KNS-81 CTRP2 3.4874 9.1364 1.5904 17.7409
LN-229 CTRP2 3.6319 8.7591 1.9097 16.1364
KALS-1 CTRP2 3.6683 6.7737 2.873 12.1843
U-118MG CTRP2 4.0104 11.1316 1.1012 18.3971
M059K CTRP2 4.2612 9.0246 2.369 12.834
SF295 CTRP2 4.2875 9.6016 2.1078 13.8422
GMS-10 CTRP2 4.3295 8.088 2.8923 10.5247
YH-13 CTRP2 4.341 8.8092 2.5479 11.9232
AM-38 CTRP2 4.5901 10.6851 1.837 14.2881
SW1783 CTRP2 4.961 9.0244 2.9845 8.8169
U-87MG ATCC CTRP2 5.0686 6.9093 4.132 3.7885
GaMG CTRP2 6.1309 14.9413 0.9697 14.6637
SW1088 CTRP2 8.0975 15.7709 1.9621 7.9807
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HEC-6 CTRP2 -0.4873 1.8684 -0.4995 36.8927
HEC-265 CTRP2 -0.2311 1.5738 -0.2338 35.1549
JHUEM-2 CTRP2 -0.0728 3.485 -0.2046 34.5156
HEC-108 CTRP2 -0.0426 2.2629 -0.0589 33.9445
HEC-251 CTRP2 0.1407 3.7236 -0.013 33.1711
HEC-59 CTRP2 0.258 3.8332 0.0948 32.4247
MFE-319 CTRP2 0.2758 1.3786 0.2758 31.7691
AN3-CA CTRP2 0.6393 4.9193 0.2706 30.5777
MFE-296 CTRP2 0.6614 4.9227 0.2938 30.4289
JHUEM-1 CTRP2 0.8 1.7466 0.7999 28.2772
ESS-1 CTRP2 0.989 3.2596 0.9489 27.1522
KLE CTRP2 1.124 5.9108 0.5015 28.2506
HEC-1-B CTRP2 1.3371 7.6066 0.095 28.9242
JHUEM-3 CTRP2 1.4101 2.6598 1.4082 24.2188
HEC-1-A CTRP2 1.5152 6.3023 0.7886 26.0588
HEC-50B CTRP2 1.5358 4.5746 1.3327 24.074
HEC-151 CTRP2 1.6147 6.8408 0.6936 26.0916
JHUEM-7 CTRP2 1.99 6.4528 1.2429 23.0275
RL95-2 CTRP2 2.8198 8.4858 1.2417 20.749
EN CTRP2 3.5907 7.76 2.3434 14.5007
EFE-184 CTRP2 5.4463 13.0654 1.3637 14.4432
Ishikawa (Heraklio) 02 ER- CTRP2 2.2864 5.677 1.8407 19.962
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UO-31 CTRP2 0.3495 2.2083 0.3429 31.3001
ACHN CTRP2 0.3571 1.4416 0.357 31.2276
Caki-1 CTRP2 1.349 4.6781 1.1053 25.4581
TUHR4TKB CTRP2 1.3818 3.906 1.2907 24.7097
TUHR10TKB CTRP2 1.7714 4.279 1.6486 30.288
786-O CTRP2 1.9284 6.1653 1.2832 23.0606
KMRC-1 CTRP2 2.0563 5.7148 1.5784 21.6047
CAL-54 CTRP2 2.1226 4.3727 2.0108 19.8481
SNU-1272 CTRP2 2.3481 4.2262 2.2781 18.2012
VMRC-RCZ CTRP2 2.3839 3.9824 2.3472 17.8484
769-P CTRP2 2.5574 5.8837 2.0623 18.3494
KMRC-2 CTRP2 2.616 4.1352 2.576 16.3134
KMRC-3 CTRP2 3.7918 8.1417 2.3588 13.9514
RCC10RGB CTRP2 5.5714 10.5398 2.7226 8.7727
OS-RC-2 CTRP2 6.0797 11.7026 2.5338 8.6832
KMRC-20 CTRP2 6.6221 11.4041 3.0638 5.72
TUHR14TKB CTRP2 7.0488 9.9693 3.9836 1.7706
Caki-2 CTRP2 7.5926 12.8547 3.0032 4.7192
VMRC-RCW CTRP2 8.7677 18.2333 1.2347 9.723
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 46 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW620 CTRP2 -1.0373 2.7341 -1.1338 40.7804
GP2d CTRP2 -0.1767 2.2044 -0.1941 34.8412
SW48 CTRP2 0.5003 3.8967 0.3449 30.7924
COLO 320 CTRP2 0.6004 3.7463 0.4773 30.0194
HCT 116 CTRP2 0.9907 4.5551 0.7439 27.847
HCT 15 CTRP2 1.0064 6.0105 0.3405 29.1595
C2BBe1 CTRP2 1.1502 3.6045 1.0838 26.1677
LS1034 CTRP2 1.3317 3.4364 1.2928 24.8653
CL-11 CTRP2 1.4358 3.7561 1.3687 24.2681
SNU-1033 CTRP2 1.4819 4.5807 1.2726 24.4541
SW1417 CTRP2 1.4844 3.7202 1.4247 23.9188
NCI-H747 CTRP2 1.5216 4.3976 1.3551 24.0403
SNU-81 CTRP2 1.5695 3.2712 1.5522 23.2081
SNU-C1 CTRP2 1.6072 2.3844 1.6072 22.8992
COLO 678 CTRP2 1.9743 5.6522 1.5102 22.0973
T84 CTRP2 2.3745 6.2158 1.744 20.0659
RKO CTRP2 2.4173 9.3272 0.4532 24.6456
RCM-1 [Human ESC] CTRP2 2.6667 6.0071 2.1351 17.7628
SNU-503 CTRP2 2.7205 5.7488 2.2862 17.0415
KM12 CTRP2 2.7263 5.6349 2.3319 16.8541
SNU-C5 CTRP2 2.9538 11.2967 0.0417 24.6161
LS411N CTRP2 3.0492 7.5082 1.9156 17.5668
DLD-1 CTRP2 3.1008 6.9187 2.227 16.215
HT115 CTRP2 3.1009 7.0586 2.1665 16.451
NCI-H716 CTRP2 3.1527 8.1204 1.742 17.978
OUMS-23 CTRP2 4.012 7.1979 3.0206 10.7336
SNU-C2A CTRP2 4.1643 16.6853 -1.5248 26.3054
MDST8 CTRP2 4.4438 9.6559 2.2208 13.0445
SK-CO-1 CTRP2 4.766 8.5383 3.0604 8.8907
LoVo CTRP2 4.9878 10.8056 2.1165 12.3547
LS123 CTRP2 5.2334 10.8503 2.2974 11.1424
HT-55 CTRP2 5.7279 11.7369 2.2493 10.4354
CCK-81 CTRP2 6.2579 15.7688 0.6569 15.5571
SNU-C4 CTRP2 6.3393 15.676 0.7655 15.0326
SW948 CTRP2 6.4532 11.02 3.1335 5.6804
HCC-56 CTRP2 6.5595 7.4736 4.7506 0.0717
HT-29 CTRP2 6.6871 7.9431 4.6323 0.2092
SNU-407 CTRP2 6.7153 14.3231 1.7132 10.9026
LS180 CTRP2 6.8481 8.8931 4.3346 0.834
LS513 CTRP2 6.8859 10.9984 3.4263 3.959
SNU-61 CTRP2 7.0536 17.3406 0.4798 14.8276
COLO205 CTRP2 7.1659 8.3713 4.6584 0.0757
CW-2 CTRP2 7.3871 13.8472 2.4088 7.235
NCI-H508 CTRP2 7.6783 9.7471 4.3635 0.3713
COLO201 CTRP2 8.6157 15.3875 2.4589 5.5554
HCT 8 CTRP2 10.8916 30.2508 -3.0814 19.1237
⏷ Show the Full List of 46 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-398 CTRP2 -13.6952 -3.7415 -13.8377 89.4942
SNU-886 CTRP2 -1.0356 4.9311 -1.5603 41.6753
SNU-182 CTRP2 -0.1242 2.833 -0.1809 34.6188
Hep 3B2.1-7 CTRP2 -0.0116 0.9643 -0.0116 33.6835
HLF CTRP2 0.484 3.2654 0.4168 30.6067
PLC/PRF/5 CTRP2 0.5224 1.0558 0.5224 30.126
SK-HEP-1 CTRP2 0.5887 2.9635 0.5542 29.8001
SNU-449 CTRP2 0.7395 4.0741 0.5713 29.2468
SNU-423 CTRP2 0.8111 4.0658 0.6502 28.7465
JHH-6 CTRP2 1.0526 2.2931 1.0516 26.5972
SNU-878 CTRP2 1.0581 2.6604 1.052 26.5775
SNU-761 CTRP2 1.0893 4.2918 0.9078 28.8878
JHH-2 CTRP2 1.3416 2.9539 1.3322 24.6999
JHH-1 CTRP2 1.3648 6.1145 0.6929 26.8495
JHH-4 CTRP2 1.4705 3.0342 1.4612 23.8407
Hep-G2 CTRP2 2.4666 4.7728 2.3004 17.7494
HuH-6 CTRP2 2.9973 8.5139 1.4057 22.6199
JHH-5 CTRP2 7.0812 11.1061 3.4958 3.4692
HuH-1 CTRP2 7.139 8.4688 4.6154 0.1247
SNU-475 CTRP2 7.5354 12.6364 3.0687 4.5414
SNU-387 CTRP2 7.6204 15.9928 1.5398 10.1884
Li-7 CTRP2 8.4536 25.6331 -2.5653 21.2589
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 140 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H510A CTRP2 -3.5626 5.6219 -4.5126 55.2356
NCI-H838 CTRP2 -2.4069 -1.0953 -2.4069 49.6415
HCC44 CTRP2 -1.2604 1.9248 -1.2974 42.1035
NCI-H1581 CTRP2 -1.0891 0.8853 -1.091 40.8683
NCI-H1155 CTRP2 -0.9085 1.4765 -0.9175 39.6874
SBC-5 CTRP2 -0.8455 0.7845 -0.846 39.2408
NCI-H211 CTRP2 -0.6104 2.1162 -0.6362 37.7549
SHP-77 CTRP2 -0.575 3.4766 -0.7423 37.9319
RERF-LC-A1 CTRP2 -0.5474 2.4425 -0.5913 37.3917
NCI-H2106 CTRP2 -0.5253 1.5022 -0.5297 37.1202
NCI-H810 CTRP2 -0.2064 2.4855 -0.2397 35.0906
HCC95 CTRP2 -0.0208 2.6591 -0.0585 33.8692
NCI-H446 CTRP2 0.0089 2.8434 -0.0421 33.7148
Lu-99 CTRP2 0.0474 2.6441 0.0134 33.4029
HCC15 CTRP2 0.0838 4.947 -0.343 34.3817
NCI-H841 CTRP2 0.1062 3.2739 0.0153 33.1974
RERF-LC-MS CTRP2 0.1702 2.7256 0.1355 32.5876
NCI-H650 CTRP2 0.1919 3.0595 0.1301 32.5327
Lu-65 CTRP2 0.203 3.2332 0.1229 32.5189
MOR/CPR CTRP2 0.2048 2.0111 0.2002 32.2573
NCI-H2141 CTRP2 0.2468 7.7893 -1.1321 35.8753
NCI-H2171 CTRP2 0.2602 3.0266 0.2051 32.0561
HOP-92 CTRP2 0.2615 2.7353 0.2298 31.9697
NCI-H1299 CTRP2 0.2675 3.6909 0.1286 32.2827
NCI-H1341 CTRP2 0.3996 2.1788 0.3944 30.9617
NCI-H23 CTRP2 0.4059 4.988 -0.0025 32.2335
PC-14 CTRP2 0.4095 4.9704 0.0063 32.1936
NCI-H1092 CTRP2 0.4117 3.8407 0.259 31.3714
NCI-H1395 CTRP2 0.4671 4.4722 0.1929 31.4027
DMS 273 CTRP2 0.4706 2.9255 0.4339 30.5937
LK2 CTRP2 0.4718 3.9236 0.3095 31.0044
NCI-H1703 CTRP2 0.4913 3.6344 0.3773 30.7144
NCI-H661 CTRP2 0.4977 4.9334 0.1123 31.5604
NCI-H1693 CTRP2 0.5163 3.3801 0.438 30.4287
T3M-10 CTRP2 0.5313 2.7186 0.5101 30.1378
NCI-H1568 CTRP2 0.5323 1.8831 0.5315 30.0626
NCI-H1355 CTRP2 0.5476 4.1822 0.3425 30.6436
NCI-H1105 CTRP2 0.56 2.622 0.5444 29.9279
HCC78 CTRP2 0.5705 3.7159 0.45 30.2096
SW1271 CTRP2 0.579 3.6624 0.4671 30.124
HCC2108 CTRP2 0.6111 5.6033 0.0428 31.4029
COR-L279 CTRP2 0.6126 2.3036 0.6077 29.5417
NCI-H2405 CTRP2 0.6322 3.4104 0.5573 29.6459
HCC1195 CTRP2 0.6495 5.8598 0.003 31.4008
NCI-H69 CTRP2 0.702 4.0242 0.5399 29.4756
NCI-H322 CTRP2 0.7166 3.3369 0.6549 29.0395
NCI-H226 CTRP2 0.73 3.2682 0.6761 28.9239
NCI-H2029 CTRP2 0.7467 3.9519 0.6009 29.1233
HOP-62 CTRP2 0.759 1.9051 0.7587 28.5509
HCC827 CTRP2 0.783 6.5722 -0.0976 31.273
VMRC-LCD CTRP2 0.7904 6.1665 0.0533 30.7807
HCC2279 CTRP2 0.8097 5.4811 0.2967 29.9349
NCI-H2228 CTRP2 0.8221 3.7699 0.7115 28.5028
NCI-H1339 CTRP2 0.8598 2.3799 0.8565 27.8893
LCLC-103H CTRP2 0.8944 3.8144 0.7823 28.0267
NCI-H292 CTRP2 0.9035 3.4752 0.8373 27.8102
NCI-H2087 CTRP2 0.9263 4.7643 0.6235 28.4651
NCI-H358 CTRP2 0.9816 5.1219 0.5891 28.4049
NCI-H647 CTRP2 0.9976 4.668 0.7249 27.8901
NCI-H522 CTRP2 1.0037 5.5431 0.489 28.673
NCI-H1373 CTRP2 1.0163 4.3483 0.8171 27.514
IA-LM CTRP2 1.0244 3.8416 0.9174 27.144
NCI-H2170 CTRP2 1.0342 3.6822 0.9506 26.999
KNS-62 CTRP2 1.0368 2.6863 1.0296 26.723
NCI-H1915 CTRP2 1.0385 3.1877 1.0065 26.7952
NCI-H2009 CTRP2 1.0386 6.8125 0.0886 29.8724
COR-L51 CTRP2 1.0797 4.2755 0.9007 27.023
NCI-H2342 CTRP2 1.0821 5.1881 0.6801 27.7747
NCI-H526 CTRP2 1.0826 6.4949 0.253 29.2051
COLO 668 CTRP2 1.0832 4.343 0.8907 27.0463
NCI-H2081 CTRP2 1.2221 5.5981 0.7096 27.2331
COR-L47 CTRP2 1.2235 8.1588 -0.2522 30.342
ChaGo-K-1 CTRP2 1.2581 5.3163 0.835 26.6864
NCI-H520 CTRP2 1.2943 5.3114 0.8759 26.4314
HCC4006 CTRP2 1.3036 4.8799 1.0056 25.9491
NCI-H2085 CTRP2 1.3344 5.106 0.9786 25.947
NCI-H1694 CTRP2 1.3472 2.7022 1.3441 24.6415
NCI-H2110 CTRP2 1.3878 4.441 1.2009 25.0016
HCC1833 CTRP2 1.3896 9.5714 -0.6932 31.0958
SK-MES-1 CTRP2 1.414 2.7169 1.4114 24.1947
DMS 114 CTRP2 1.437 4.065 1.3252 24.4135
NCI-H1944 CTRP2 1.4377 2.5592 1.4369 24.031
NCI-H2126 CTRP2 1.5052 6.4627 0.7193 26.3306
DV-90 CTRP2 1.5303 2.5796 1.5297 23.4136
EKVX CTRP2 1.5558 3.3961 1.5302 23.3272
Calu-3 CTRP2 1.5791 3.8368 1.511 23.3168
NCI-H2196 CTRP2 1.5822 5.0922 1.2528 24.2115
NCI-H1666 CTRP2 1.6182 2.9192 1.6146 22.8377
DMS 454 CTRP2 1.6197 4.9455 1.3335 23.8096
LCLC-97TM1 CTRP2 1.6637 2.8077 1.6621 22.5281
CAL-12T CTRP2 1.7527 6.4206 1.0007 24.5985
NCI-H2122 CTRP2 1.7706 3.7551 1.7237 21.9689
NCI-H1792 CTRP2 1.8333 6.5839 1.0256 24.272
LOU-NH91 CTRP2 1.837 8.7887 0.1107 27.3941
RERF-LC-Ad2 CTRP2 1.8466 6.1337 1.2063 23.5807
NCI-H1563 CTRP2 1.8617 5.0872 1.5592 22.2601
HARA [Human squamous cell lung carcinoma] CTRP2 1.8697 7.0997 0.8622 24.7493
COR-L105 CTRP2 1.884 6.0064 1.2919 23.1599
LUDLU-1 CTRP2 1.9056 6.7794 1.0273 24.0547
NCI-H2030 CTRP2 1.9949 8.9838 0.1846 26.7057
HCC366 CTRP2 2.0275 9.6117 -0.067 27.4172
NCI-H1435 CTRP2 2.0439 7.571 0.8511 24.2889
COLO 699 CTRP2 2.0836 8.1753 0.6331 24.9441
NCI-H2444 CTRP2 2.0875 7.1642 1.0657 23.3928
NCI-H727 CTRP2 2.1677 7.4314 1.039 23.2632
NCI-H1755 CTRP2 2.1817 8.136 0.7511 24.256
NCI-H1869 CTRP2 2.194 7.3795 1.0882 23.0103
COR-L95 CTRP2 2.2382 5.087 1.9702 19.6336
NCI-H1793 CTRP2 2.2555 7.8405 0.9556 23.3201
NCI-H2286 CTRP2 2.2784 6.0935 1.6859 20.5586
HCC2935 CTRP2 2.5093 5.8941 2.0067 18.6963
Calu-1 CTRP2 2.5288 6.0866 1.9576 18.8239
LC-1F CTRP2 2.5362 8.2731 1.0523 22.2017
NCI-H1734 CTRP2 2.5877 7.9764 1.237 21.3806
HCC1438 CTRP2 2.9137 8.5828 1.2908 20.3211
NCI-H1651 CTRP2 2.9423 6.436 2.2628 16.5045
NCI-H2291 CTRP2 3.1571 8.6848 1.484 18.966
NCI-H441 CTRP2 3.277 9.29 1.3146 19.3156
NCI-H1838 CTRP2 3.6071 10.892 0.8507 20.2475
HCC1171 CTRP2 3.7372 10.6502 1.0894 19.0649
A-549 CTRP2 3.7941 6.8066 2.9856 11.4139
NCI-H460 CTRP2 3.8012 9.7377 1.5954 16.9801
LXF 289 CTRP2 3.9672 11.4301 0.9147 19.1848
EBC-1 CTRP2 4.165 9.1399 2.2244 13.6381
NCI-H196 CTRP2 4.3974 12.0254 1.0011 17.9206
NCI-H2023 CTRP2 4.6483 9.7258 2.3659 12.0197
BEN CTRP2 4.8028 9.481 2.6217 10.6457
EPLC-272H CTRP2 4.8327 9.4149 2.6804 10.3415
SK-LU-1 CTRP2 5.0187 13.4689 0.8107 17.3301
NCI-H889 CTRP2 5.0438 12.4344 1.3489 15.2778
NCI-H1184 CTRP2 5.1875 8.596 3.3864 6.6973
NCI-H2172 CTRP2 5.5157 9.4203 3.2357 6.7382
Calu-6 CTRP2 5.5334 10.8927 2.5172 9.6876
NCI-H1623 CTRP2 5.5603 10.6541 2.657 9.0633
HCC1588 CTRP2 5.8837 11.3154 2.5779 8.8292
NCI-H1650 CTRP2 6.7767 16.6082 0.6351 14.7485
Sq-1 CTRP2 6.8082 8.6993 4.3941 0.6949
LC-1/sq-SF CTRP2 6.9889 8.3531 4.6006 0.1767
RERF-LC-Ad1 CTRP2 8.008 20.1803 -0.2185 15.6035
Hs 888.Lu CTRP2 2.4426 5.7214 1.995 18.9335
⏷ Show the Full List of 140 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 5.0608 11.7564 1.7021 13.8714
SYO-1 CTRP2 7.2413 19.7863 -0.5854 17.9239
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 5.9045 18.1239 -0.7931 20.8508
TOV-21G CTRP2 -1.3596 -0.3868 -1.3596 42.6645
ES2 CTRP2 -0.3217 1.4164 -0.3235 35.7559
A2780 CTRP2 -0.2811 2.8358 -0.346 35.6878
ONCO-DG-1 CTRP2 -0.267 5.9534 -1.0236 37.4697
DOV13 CTRP2 -0.0979 3.7593 -0.2762 34.8255
OC 314 CTRP2 -0.012 3.866 -0.2025 34.2965
OVSAHO CTRP2 0.048 8.4162 -1.593 37.5702
JHOM-1 CTRP2 0.1104 3.6647 -0.0359 33.348
TOV-112D CTRP2 0.1885 3.8473 0.0173 32.9105
JHOC-5 CTRP2 0.1969 3.8485 0.0262 32.8535
TYK-nu CTRP2 0.3089 4.1672 0.0867 32.2785
SNU-8 CTRP2 0.3957 2.2381 0.3891 30.9922
OV7 CTRP2 0.451 5.766 -0.1827 32.6347
SNU-119 CTRP2 0.7373 5.2647 0.282 30.2186
OAW42 CTRP2 0.8401 1.9974 0.8398 28.0107
HEY A8 CTRP2 0.9707 5.152 0.5688 28.5086
Kuramochi CTRP2 1.2682 7.6096 0.0212 29.3685
OVCAR-8 CTRP2 1.5188 5.8006 0.9666 25.4215
RMG-I CTRP2 1.5455 6.7567 0.6521 26.442
JHOS-2 CTRP2 1.6021 4.8103 1.349 23.8093
EFO-21 CTRP2 1.8452 5.8749 1.2955 23.2617
OVK18 CTRP2 2.1024 6.8778 1.1973 22.8704
IGROV-1 CTRP2 2.3689 6.1424 1.7653 20.002
OV56 CTRP2 2.4619 7.5781 1.2822 21.5528
OVTOKO CTRP2 2.6326 8.5762 1.0127 22.0893
OVCAR-4 CTRP2 2.6658 7.6348 1.4676 20.3039
OAW28 CTRP2 2.7351 6.9483 1.8341 18.7184
EFO-27 CTRP2 3.0271 7.3543 1.9612 17.447
MCAS CTRP2 3.0277 7.5852 1.8593 17.8424
COV362 CTRP2 3.3486 8.259 1.8717 16.9775
OVISE CTRP2 3.8433 9.5351 1.7335 16.3396
OVCAR-5 CTRP2 3.9081 7.6748 2.6937 12.3139
COV644 CTRP2 4.9554 12.5797 1.2023 16.0105
FU-OV-1 CTRP2 5.7548 11.4285 2.4233 9.6811
OV-90 CTRP2 6.4639 12.2867 2.5273 8.099
SK-OV-3 CTRP2 8.1862 15.8826 1.9665 7.851
Caov-3 CTRP2 9.1609 21.7216 -0.1633 13.7845
SNU-840 CTRP2 11.4385 24.3226 0.0691 10.3165
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 7.247 17.2589 0.6613 13.8962
Aska-SS CTRP2 7.6602 17.962 0.6144 13.4182
A-204 CTRP2 -0.4485 1.7209 -0.4561 36.6194
KYM-1 CTRP2 -0.2083 1.3971 -0.2094 34.9981
G-402 CTRP2 -0.0701 3.2545 -0.1698 34.3964
SK-LMS-1 CTRP2 -0.0273 2.5163 -0.0559 33.883
Rh41 CTRP2 0.0327 1.6827 0.0308 33.395
SK-UT-1 CTRP2 0.033 3.6415 -0.1154 33.8673
GCT CTRP2 0.2398 1.9398 0.2367 32.0195
HT-1080 CTRP2 0.3067 1.0348 0.3067 31.563
MES-SA CTRP2 0.3448 2.0127 0.3417 31.3198
G-401 CTRP2 0.4349 3.3888 0.3504 30.9912
TE 617.T CTRP2 0.9962 2.6508 0.9893 26.9927
TE 441.T CTRP2 1.093 2.3271 1.0921 26.3278
TTC-709 CTRP2 1.4633 8.1427 0.0047 28.8273
Rh18 CTRP2 1.6112 3.0821 1.6033 22.899
Hs 729.T CTRP2 2.0241 6.0872 1.4144 22.3005
BT-16 CTRP2 2.0373 7.7408 0.7723 24.587
Tm87-16 CTRP2 2.0672 8.1564 0.6244 25.0205
RD CTRP2 2.4041 7.852 1.1037 22.3714
BT-12 CTRP2 3.0137 8.367 1.4898 19.3074
SW982 CTRP2 8.7843 21.9668 -0.5391 15.44
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H28 CTRP2 -0.5331 2.0945 -0.5554 37.2296
ACC-MESO-1 CTRP2 0.3773 2.8771 0.3403 31.2164
NCI-H2452 CTRP2 0.5061 5.6079 -0.073 32.1145
IST-Mes1 CTRP2 1.5341 4.0062 1.4389 23.7095
MSTO-211H CTRP2 1.756 6.2555 1.0649 24.3586
MPP 89 CTRP2 2.9649 5.0691 2.7681 14.5431
JL-1 CTRP2 5.093 8.6228 3.2955 7.2568
NCI-H2052 CTRP2 7.488 16.5356 1.1859 11.6725
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
DU145 CTRP2 -0.0421 2.1194 -0.0532 33.9237
LNCaP clone FGC CTRP2 0.4852 2.6571 0.4658 30.4387
PaCa-3 CTRP2 1.8908 5.4108 1.4962 22.3984
VCaP CTRP2 6.3084 8.8572 4.06 2.2407
22Rv1 CTRP2 7.2042 17.5119 0.5062 14.4958
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 0.1234 2.7871 0.0823 32.9204
A-253 CTRP2 0.9504 5.4438 0.4614 28.9353
Cancer Drug Sensitivity Data Curated from 32 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
GSS CTRP2 -0.9296 0.9493 -0.9311 39.8045
SNU-1 CTRP2 -0.6172 1.865 -0.6322 37.7667
HGC-27 CTRP2 -0.5179 2.1858 -0.5444 37.1418
SNU-5 CTRP2 -0.2215 2.3768 -0.2487 35.1712
AGS CTRP2 0.3358 3.6363 0.2104 31.7851
ECC10 CTRP2 0.7116 2.8756 0.6877 28.9457
Hs 746.T CTRP2 0.7162 3.1584 0.6718 28.984
LMSU CTRP2 0.7163 3.8342 0.5879 29.2664
SNU-16 CTRP2 0.7165 1.26 0.7165 28.8331
SNU-668 CTRP2 0.8596 3.8956 0.732 28.3111
Fu97 CTRP2 1.0076 3.4908 0.9458 27.102
NUGC-3 CTRP2 1.2621 5.7713 0.6975 27.1507
SNU-216 CTRP2 1.3703 4.8865 1.0768 25.4908
ECC12 CTRP2 1.8264 5.9121 1.2623 23.4379
MKN74 CTRP2 2.7435 7.9839 1.3923 20.3822
MKN7 CTRP2 2.7839 11.5773 -0.2551 25.98
KATO III CTRP2 3.5108 6.7572 2.7195 13.2005
NCI-N87 CTRP2 3.5694 9.4632 1.5111 17.8527
KE-39 CTRP2 4.8121 9.9081 2.4164 11.4767
HuG1-N CTRP2 5.0476 9.1977 2.9704 8.7069
GSU CTRP2 5.6619 6.3419 4.8095 0.2629
SH-10-TC CTRP2 5.8221 10.5207 2.9243 7.5098
SNU-620 CTRP2 6.0269 7.6692 4.4321 1.1848
SNU-719 CTRP2 6.3083 15.4082 0.8745 14.6977
NUGC-4 CTRP2 6.353 11.9279 2.6229 7.8862
MKN45 CTRP2 6.6325 7.746 4.6822 0.1439
23132/87 CTRP2 6.7964 10.5931 3.5586 3.5627
IM95 CTRP2 7.3311 10.3792 3.9554 1.626
SNU-601 CTRP2 7.698 10.3895 4.1271 0.8854
SNU-1077 CTRP2 -1.3219 0.361 -1.3223 42.4145
SNU-685 CTRP2 1.847 6.3269 1.1366 23.8318
SNG-M CTRP2 2.5263 5.9861 1.9918 18.7028
⏷ Show the Full List of 32 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
8505C CTRP2 -0.807 1.5443 -0.816 39.0113
CGTH-W-1 CTRP2 -0.3555 1.3897 -0.3573 35.9809
FTC-133 CTRP2 0.5163 2.7787 0.4912 30.2507
FTC-238 CTRP2 0.8362 4.1064 0.6697 28.5988
B-CPAP CTRP2 1.1 2.0889 1.0998 26.2789
CAL-62 CTRP2 1.4389 4.2725 1.2903 24.5284
SW579 CTRP2 1.6387 3.842 1.5737 22.9092
8305C CTRP2 1.9239 5.5045 1.503 22.274
ML-1 [Human leukemia] CTRP2 2.2383 5.8532 1.7285 20.5173
TT CTRP2 2.7999 6.9015 1.9214 18.2073
TT2609-C02 CTRP2 3.7345 8.2912 2.2322 14.5995
BHT-101 CTRP2 6.69 9.6124 3.9423 2.2574
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-3 CTRP2 -0.8356 4.8675 -1.3251 40.3752
HSC-2 CTRP2 -0.5272 1.7798 -0.5376 37.1524
Detroit 562 CTRP2 -0.0936 3.9956 -0.3152 34.9287
SCC-9 CTRP2 -0.059 2.3996 -0.0822 34.0763
FaDu CTRP2 0.2855 2.095 0.2804 31.7216
PE/CA-PJ15 CTRP2 0.8877 4.4663 0.6519 28.4925
SNU-899 CTRP2 0.9342 4.4914 0.6968 28.1897
SNU-1076 CTRP2 1.24 5.0612 0.8879 26.5593
PE/CA-PJ49 CTRP2 1.3123 4.0796 1.1884 25.2855
SNU-46 CTRP2 1.4287 5.8099 0.8657 26.0519
PE/CA-PJ34 (clone C12) CTRP2 1.7407 5.8852 1.1788 23.995
YD-8 CTRP2 1.8103 3.8862 1.7506 21.7482
BHY CTRP2 1.8791 5.2325 1.5368 22.2872
CAL-33 CTRP2 2.0287 4.8588 1.8021 20.8781
SNU-1214 CTRP2 2.1481 6.3379 1.4556 21.7884
PE/CA-PJ41 (clone D2) CTRP2 2.2655 7.3181 1.1886 22.4419
CAL-27 CTRP2 2.4095 6.8276 1.542 20.7245
BICR 22 CTRP2 3.484 8.2949 1.9876 16.1845
BICR 56 CTRP2 3.545 11.1172 0.683 20.9968
HSC-4 CTRP2 3.6758 6.8287 2.856 12.2328
SCC-25 CTRP2 4.2934 8.1221 2.8422 10.8128
BICR 6 CTRP2 4.5773 8.7456 2.7914 10.4062
SCC-4 CTRP2 4.7763 13.8034 0.4395 19.1333
BICR 18 CTRP2 4.9211 11.2468 1.8399 13.601
SNU-1041 CTRP2 5.6539 13.4421 1.342 14.139
BICR 16 CTRP2 6.0005 10.6317 3.002 6.8992
BICR 31 CTRP2 6.0124 14.1393 1.2763 13.7405
SNU-1066 CTRP2 6.6947 11.246 3.1876 5.1306
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HT-1197 CTRP2 -0.1798 2.216 -0.1978 34.8636
UM-UC-3 CTRP2 -0.1699 3.6268 -0.3312 35.2485
VM-CUB-1 CTRP2 -0.0288 2.8863 -0.0855 33.9844
KU-19-19 CTRP2 -0.0288 0.7865 -0.0288 33.7987
JMSU-1 CTRP2 0.241 2.7308 0.2088 32.1082
UM-UC-1 CTRP2 0.4388 2.0516 0.436 30.6924
253J CTRP2 0.4524 3.3342 0.3756 30.8488
SCaBER CTRP2 0.7943 3.6112 0.7044 28.6177
BFTC-905 CTRP2 0.8885 3.4322 0.8263 27.8968
253J-BV CTRP2 0.961 3.4607 0.8998 27.4101
5637 CTRP2 0.9988 8.2267 -0.5156 31.8042
639V CTRP2 1.1702 5.3543 0.7279 27.3327
J82 CTRP2 1.1771 3.7804 1.0898 26.0597
TCCSUP CTRP2 1.9495 3.6329 1.923 20.7074
HT-1376 CTRP2 2.0109 6.3853 1.2908 22.7917
BC-3C CTRP2 2.088 5.0734 1.81 20.6679
KMBC-2 CTRP2 2.2148 3.7747 2.189 18.9379
U-BLC1 CTRP2 2.2596 5.4315 1.8913 19.8556
T24 CTRP2 2.3 8.2551 0.8198 23.6846
CAL-29 CTRP2 2.7882 4.4899 2.7084 15.3036
RT-112 CTRP2 2.8395 7.2623 1.8086 18.5352
SW1710 CTRP2 4.4002 8.8188 2.5967 11.5928
647V CTRP2 5.3974 9.4887 3.1091 7.4752
RT-4 CTRP2 7.1383 8.989 4.4262 0.4487
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 2.4284 7.4441 1.3049 21.56

References

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