Details of the Drug-Related molecule(s) Interaction Atlas

General Information of Drug (ID: DM4XVLB)

Drug Name

RGS4 inhibitor 13 Drug Info

Synonyms

CHEMBL2037369; RGS4 inhibitor 13; GTPL8034; SCHEMBL13517588; BDBM50384771

Indication

Disease Entry	ICD 11	Status	REF
Discovery agent	N.A.	Investigative	[1]

Cross-matching ID

Molecule-Related Drug Atlas

Molecule Type:

DTT

Drug Status:

Patented Agent(s)

Investigative Drug(s)

Download the Complete Related Drug List

Drug(s) Targeting Regulator of G-protein signaling 8 (RGS8)

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
1-Benzyl-3-bromo-1H-pyrrole-2,5-dione	DML8RVS	N. A.	N. A.	Patented	[4]
1-Benzyl-3-p-tolyl-1H-pyrrole-2,5-dione	DMWY9GM	N. A.	N. A.	Patented	[4]
thiadiazolidinone (TDZD) deriv. 6	DM9CF45	Discovery agent	N.A.	Investigative	[3]
CCG-50014	DMUQJ6X	Discovery agent	N.A.	Investigative	[3]
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Drug(s) Targeting Regulator of G-protein signaling 4 (RGS4)

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
thiadiazolidinone (TDZD) deriv. 6	DM9CF45	Discovery agent	N.A.	Investigative	[2]
CCG-50014	DMUQJ6X	Discovery agent	N.A.	Investigative	[2]
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Molecular Interaction Atlas of This Drug

Molecular Interaction Atlas

Download the Complete Interaction Atlas for Visualization in Cytoscape

Drug Therapeutic Target (DTT)

DTT Name	DTT ID	UniProt ID	MOA	REF
Regulator of G-protein signaling 4 (RGS4)	TTGTKX9	RGS4_HUMAN	Inhibitor	[2]
Regulator of G-protein signaling 8 (RGS8)	TTWME23	RGS8_HUMAN	Inhibitor	[3]

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References

1	URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 8034).
2	URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Target id: 2811).
3	URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Target id: 2813).
4	Small molecule inhibitors of RGS proteins. US8865750.