General Information of Drug (ID: DM6LP0R)

Drug Name
Dianicline+rimonabant
Synonyms [3H]nemonapride; (2R,3R)-nemonapride; 75272-39-8; CHEBI:64219; C21H26ClN3O2; 93664-94-9
Indication
Disease Entry ICD 11 Status REF
Tobacco dependence 6C4A.2 Terminated [1]
Drug Type
Combination drug (Antibody)
Cross-matching ID
TTD ID
D0N5UA

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Cannabinoid receptor 1 (CB1) TT6OEDT CNR1_HUMAN Agonist [2]
Dopamine D2 receptor (D2R) TTEX248 DRD2_HUMAN Antagonist [3]
Dopamine D3 receptor (D3R) TT4C8EA DRD3_HUMAN Antagonist [3]
Nicotinic acetylcholine receptor (nAChR) TTJSZTB NOUNIPROTAC Agonist [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Tobacco dependence
ICD Disease Classification 6C4A.2
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Dopamine D2 receptor (D2R) DTT DRD2 2.50E-02 -0.08 -0.49
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

References

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