Details of the Drug

General Information of Drug (ID: DMYA50U)

Drug Name
phloretin
Synonyms
phloretin; 60-82-2; 3-(4-Hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one; Dihydronaringenin; Phloretol; 3-(4-Hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)-1-propanone; NSC 407292; UNII-S5J5OE47MK; 1-Propanone, 3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)-; CCRIS 7459; beta-(p-Hydroxyphenyl)phloropropiophenone; 2',4',6'-Trihydroxy-3-(p-hydroxyphenyl)propiophenone; 2',4',6'-Trihydroxy-3-(4-Hydroxyphenyl)propiophenone; EINECS 200-488-7; NSC407292; S5J5OE47MK; beta-(p-Hydroxyphenyl)-2,4,6-trihydroxypropiophenone
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Drug Type
Small molecular drug
Structure
3D MOL is unavailable 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 274.27
Logarithm of the Partition Coefficient (xlogp) 2.6
Rotatable Bond Count (rotbonds) 4
Hydrogen Bond Donor Count (hbonddonor) 4
Hydrogen Bond Acceptor Count (hbondacc) 5
Chemical Identifiers
Formula
C15H14O5
IUPAC Name
3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
Canonical SMILES
C1=CC(=CC=C1CCC(=O)C2=C(C=C(C=C2O)O)O)O
InChI
InChI=1S/C15H14O5/c16-10-4-1-9(2-5-10)3-6-12(18)15-13(19)7-11(17)8-14(15)20/h1-2,4-5,7-8,16-17,19-20H,3,6H2
InChIKey
VGEREEWJJVICBM-UHFFFAOYSA-N
Cross-matching ID
PubChem CID
4788
ChEBI ID
CHEBI:17276
CAS Number
60-82-2
UNII
S5J5OE47MK
DrugBank ID
DB07810
TTD ID
D0HD2G
VARIDT ID
DR00911
INTEDE ID
DR1943

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Aquaporin-9 (AQP9) TTQEI32 AQP9_HUMAN Inhibitor [2]
Chloride channel protein 3 (CLC-3) TT8XNZ7 CLCN3_HUMAN Blocker (channel blocker) [3]
Solute carrier family 23 member 1 (SLC23A1) TT6XAGK S23A1_HUMAN Inhibitor [4]

Drug-Metabolizing Enzyme (DME)
DME Name DME ID UniProt ID MOA REF
UDP-glucuronosyltransferase 1A1 (UGT1A1) DEYGVN4 UD11_HUMAN Substrate [5]
UDP-glucuronosyltransferase 1A9 (UGT1A9) DE85D2P UD19_HUMAN Substrate [5]
UDP-glucuronosyltransferase 1A8 (UGT1A8) DE2GB8N UD18_HUMAN Substrate [5]
UDP-glucuronosyltransferase 1A7 (UGT1A7) DEZO4N3 UD17_HUMAN Substrate [5]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Estrogen receptor beta (ESR2) OTXNR2WQ ESR2_HUMAN Protein Interaction/Cellular Processes [6]
Glycogen synthase kinase-3 beta (GSK3B) OTL3L14B GSK3B_HUMAN Gene/Protein Processing [7]
Nitric oxide synthase 3 (NOS3) OTLDT7NR NOS3_HUMAN Gene/Protein Processing [8]
Sex hormone-binding globulin (SHBG) OTPWU5IW SHBG_HUMAN Protein Interaction/Cellular Processes [9]
Sodium/hydrogen exchanger 1 (SLC9A1) OT6HNHFV SL9A1_HUMAN Gene/Protein Processing [10]
Sodium/hydrogen exchanger 9B2 (SLC9B2) OTZVOY8T SL9B2_HUMAN Gene/Protein Processing [11]
Solute carrier family 2, facilitated glucose transporter member 1 (SLC2A1) OTA675TJ GTR1_HUMAN Gene/Protein Processing [12]
Solute carrier family 2, facilitated glucose transporter member 2 (SLC2A2) OTBL2W7R GTR2_HUMAN Gene/Protein Processing [13]
UDP-glucuronosyltransferase 1-6 OTGTQ2C9 UD16_HUMAN Gene/Protein Processing [14]
UDP-glucuronosyltransferase 1A1 OTH1C8OJ UD11_HUMAN Gene/Protein Processing [14]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 145 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JK1 CTRP2 6.4746 12.4389 4.9842 23.6446
MEC1 CTRP2 7.429 10.1163 6.9592 13.5523
JM1 CTRP2 8.317 9.6177 8.0984 6.7124
EoL-1 CTRP2 3.0188 6.7606 2.9311 41.4694
MV4-11 CTRP2 3.8959 9.4125 3.3529 36.9488
LP-1 CTRP2; CTRP1 4.6976 10.2492 3.9669 32.416
P12-Ichikawa CTRP2 4.9876 6.3081 4.9865 28.1158
697 CTRP2 5.0655 7.7528 4.9852 27.864
Pfeiffer CTRP2 5.0962 7.9684 4.988 27.7542
KMS-28BM CTRP2 5.1178 7.1789 5.094 27.3243
Peer CTRP2 5.2012 7.2191 5.178 26.7662
BL-70 CTRP2; CTRP1 5.2668 5.9469 5.2668 26.2512
JVM-2 CTRP2 5.4237 7.8588 5.3529 25.4448
KMS-34 CTRP2 5.4686 6.9771 5.4627 24.9257
KMS-20 CTRP2 5.4934 6.2589 5.4934 24.7405
EM-2 CTRP2 5.5969 6.292 5.5969 24.0502
KMS-26 CTRP2 5.6026 9.8659 5.075 25.8537
KMS-21-BM CTRP2 5.6299 7.9683 5.5584 24.0726
MOLT-3 CTRP2 5.6338 8.7781 5.4153 24.5572
MOLT-13 CTRP2 5.6695 7.8846 5.6107 23.7651
M-07e CTRP2 5.7412 7.5138 5.7195 23.1614
Ku812 CTRP2; CTRP1 5.8066 8.4349 5.6745 23.1043
KMS-18 CTRP2 5.8533 7.3526 5.8433 22.3748
TALL-1 [Human adult T-ALL] CTRP2 5.9031 9.1998 5.6029 23.0554
EB1 CTRP2 5.9569 9.0692 5.6963 22.5569
Kasumi-1 CTRP2 6.0996 13.5959 4.0849 27.7065
KMS-12-BM CTRP2 6.1053 8.7861 5.9267 21.2779
BV-173 CTRP2 6.204 10.9223 5.3411 23.1131
MOLM-13 CTRP2 6.4234 9.3708 6.1225 19.5987
MHH-CALL-4 CTRP2 6.4318 10.2203 5.851 20.5732
RL CTRP2 6.4573 8.4374 6.3756 18.593
SUP-B15 CTRP2 6.5606 9.5301 6.2241 18.8163
NALM-6 CTRP2 6.5801 8.8021 6.4395 17.9809
SUP-M2 CTRP2 6.6775 10.0069 6.1923 18.5902
Ri-1 CTRP2 6.6825 9.8124 6.2651 18.3048
ST486 CTRP2 6.713 9.3521 6.4438 17.5573
KMS-11 CTRP2; CTRP1 6.7462 9.5544 6.4197 17.5725
KM-H2 CTRP2 6.7669 8.7506 6.6531 16.6419
F-36P CTRP2 6.7802 8.6297 6.6907 16.4684
RS4;11 CTRP2 6.8116 10.5035 6.1512 18.3626
OCI-AML-3 CTRP2; CTRP1 6.832 9.6268 6.49 17.0599
KHM-1B CTRP2 6.9128 11.2577 5.9495 18.8547
RPMI-8226 CTRP2; CTRP1 6.9194 9.6212 6.5868 16.4443
RPMI-8402 CTRP2 6.9404 8.891 6.8117 15.5386
K-562 CTRP2 6.9589 8.7836 6.8545 15.3297
Reh CTRP2 6.9591 9.353 6.7119 15.84
MOLT-16 CTRP2 6.963 9.1458 6.7741 15.6027
NCO2 CTRP2 7.0593 9.0297 6.9087 14.8242
RCH-ACV CTRP2 7.0763 10.4512 6.4532 16.4718
CML-T1 CTRP2 7.0934 9.755 6.7298 15.3764
Daudi CTRP2 7.1325 10.1652 6.6237 15.664
ALL-SIL CTRP2 7.1495 9.5967 6.8437 14.7892
KE-37 CTRP2 7.1589 9.6507 6.8361 14.7897
DND-41 CTRP2 7.1612 9.4138 6.9141 14.495
OCI-Ly3 CTRP2 7.2068 10.5155 6.5657 15.679
L-428 CTRP2 7.2107 9.2791 7.0078 14.0048
SKM-1 CTRP2; CTRP1 7.2173 10.282 6.671 15.2728
A4/Fukuda CTRP2 7.2613 9.5291 6.9871 13.9292
JVM-3 CTRP2 7.2782 9.8869 6.8832 14.2677
DEL CTRP2 7.2881 8.7432 7.2185 13.0141
JeKo-1 CTRP2 7.2928 9.2779 7.0977 13.4301
Mono-Mac-1 CTRP2 7.2978 10.4331 6.6951 14.9299
KE-97 CTRP2; CTRP1 7.3409 9.9865 6.914 13.9724
DB CTRP2 7.3441 10.5839 6.6825 14.852
HEL CTRP2 7.3466 9.9458 6.9353 13.8757
MOLM-16 CTRP2; CTRP1 7.3777 9.7034 7.0566 13.358
HT CTRP2; CTRP1 7.4596 9.5206 7.2054 12.5374
TF-1 CTRP2 7.4965 9.6066 7.2171 12.3858
LAMA-84 CTRP2 7.507 10.6801 6.8127 13.9054
CA46 CTRP2 7.5179 18.7942 2.9406 27.3315
SU-DHL-6 CTRP2 7.5234 9.8902 7.1457 12.5762
PF-382 CTRP2 7.5419 9.707 7.2317 12.1992
Jurkat CTRP2 7.5534 10.2011 7.0583 12.8259
OPM-2 CTRP2 7.5566 9.6255 7.2758 11.9919
AML-193 CTRP2 7.5572 9.1246 7.428 11.4323
MOLM-6 CTRP2 7.5585 10.9486 6.7505 14.0135
Ki-JK CTRP2 7.6063 9.8821 7.2377 11.992
JURL-MK1 CTRP2 7.6136 10.0086 7.1976 12.1244
SU-DHL-4 CTRP2; CTRP1 7.6208 9.8319 7.2733 11.8444
U266B1 CTRP2 7.6331 9.2885 7.4659 11.0644
NU-DUL-1 CTRP2; CTRP1 7.6524 12.1453 6.3037 15.5798
NOMO-1 CTRP2; CTRP1 7.6743 10.2863 7.1535 12.1546
Raji CTRP2 7.6933 9.3302 7.5193 10.6887
KCL-22 CTRP2 7.7079 10.5583 7.0733 12.3488
P31/FUJ CTRP2 7.71 11.2483 6.7718 13.5375
OCI-AML-2 CTRP2 7.7349 9.3553 7.5571 10.426
HPB-ALL CTRP2 7.7423 10.1287 7.2873 11.4227
GDM-1 CTRP2; CTRP1 7.778 8.9798 7.7034 9.7968
SU-DHL-1 CTRP2 7.7945 12.0345 6.4929 14.4458
OCI-M1 CTRP2 7.8113 9.9404 7.4348 10.6645
SU-DHL-8 CTRP2 7.8389 10.0705 7.4128 10.6726
U-937 CTRP2; CTRP1 7.8397 10.5463 7.217 11.4626
MM1.S CTRP2 7.8635 11.2484 6.9263 12.5308
L-540 CTRP2 7.8847 9.7402 7.5892 9.8695
HuT 78 CTRP2 7.907 9.8111 7.5866 9.8163
HD-MY-Z CTRP2 7.9288 10.4681 7.3409 10.7111
MOLP-8 CTRP2 7.9392 10.1252 7.4964 10.0743
GA-10 CTRP2 7.9773 11.0134 7.1477 11.3554
OCI-Ly19 CTRP2 8.0064 12.1221 6.6572 13.2697
WSU-DLCL2 CTRP2; CTRP1 8.0227 9.119 7.9378 8.2038
SR CTRP2 8.0335 10.4543 7.4548 9.9865
SUP-T11 CTRP2 8.0992 9.3674 7.9502 7.8975
JJN-3 CTRP2 8.1299 9.6541 7.8843 8.055
HDLM-2 CTRP2 8.1488 10.5033 7.5512 9.3043
NB4 CTRP2 8.1544 9.0833 8.0892 7.2265
Kasumi-2 CTRP2 8.1593 9.6429 7.92 7.8364
Karpas-299 CTRP2 8.1666 10.7029 7.4793 9.5464
KMS-27 CTRP2 8.1835 11.7811 6.9907 11.4896
PL21 CTRP2; CTRP1 8.2046 9.5139 8.0169 7.3711
A3/Kawakami CTRP2 8.2424 10.3547 7.7126 8.4207
HEL 92.1.7 CTRP2 8.2475 12.6017 6.6547 12.7177
THP-1 CTRP2; CTRP1 8.2834 9.4556 8.1223 6.7484
L-363 CTRP2 8.2874 9.1588 8.2158 6.3636
MOTN-1 CTRP2 8.3246 12.2799 6.8835 11.6017
EJM CTRP2; CTRP1 8.3413 12.3221 6.8814 11.6
MC116 CTRP2; CTRP1 8.3647 12.3936 6.8655 11.5848
SUP-HD1 CTRP2 8.3688 14.5112 5.8261 15.7942
EHEB CTRP2 8.4024 11.1093 7.5223 8.7941
OCI-Ly10 CTRP2; CTRP1 8.4077 13.0538 6.5841 12.6738
SET-2 CTRP2 8.4133 10.2433 7.9361 7.0902
NU-DHL-1 CTRP2 8.4223 9.3382 8.311 5.6105
SU-DHL-5 CTRP1 8.4466 9.0182 8.4203 11.091
SUP-T1 CTRP2 8.4512 9.3185 8.3487 5.386
NCI-H929 CTRP2 8.4558 10.7505 7.7443 7.7597
REC-1 CTRP2 8.4565 9.6494 8.2349 5.8006
Karpas-422 CTRP2 8.4582 13.0029 6.6524 12.2548
AMO1 CTRP2; CTRP1 8.464 9.268 8.3792 5.2667
ME1 CTRP2 8.4729 13.6541 6.3441 13.4866
OCI-AML-5 CTRP2 8.5076 9.0892 8.472 4.7689
CMK CTRP2 8.5088 11.5059 7.4328 8.9144
HL-60 CTRP2 8.5208 9.1388 8.4752 4.7167
SK-MM-2 CTRP2 8.5294 9.3167 8.4344 4.8386
Hs 611.T CTRP2 8.5366 9.4345 8.402 4.9383
RPMI-6666 CTRP2 8.537 17.8223 4.3275 20.9079
SIG-M5 CTRP2 8.5459 9.0308 8.5246 4.4639
SU-DHL-10 CTRP2 8.5746 9.5236 8.4096 4.8016
KO52 CTRP2 8.5804 9.0358 8.561 4.2272
MOLP-2 CTRP2 8.5822 9.5787 8.3962 4.8322
KYO-1 CTRP2 8.5974 9.6449 8.3855 4.8321
Granta-519 CTRP2 8.6062 10.3999 8.0565 6.1243
Ci-1 CTRP2 8.6782 9.1337 8.6478 3.6143
MHH-CALL-3 CTRP2 8.7376 11.0566 7.8654 6.6044
P3HR-1 CTRP2; CTRP1 8.7512 10.0098 8.3816 4.4496
Namalwa CTRP2 8.826 17.3617 4.8064 18.6497
Karpas-620 CTRP2 8.9175 11.8482 7.6366 7.1712
⏷ Show the Full List of 145 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE15 CTRP2 8.4353 13.0432 6.6117 12.4729
TE8 CTRP2 8.4591 10.3437 7.9367 6.9723
EC-GI-10 CTRP2 7.2699 10.2335 6.7443 14.8184
KYSE-140 CTRP2; CTRP1 7.9379 12.3779 6.4691 14.1957
KYSE-520 CTRP2 8.1435 11.1631 7.2441 10.5529
TE-6 CTRP2 8.1625 9.9697 7.795 8.3078
TE-11 CTRP2 8.3354 13.938 6.0795 14.859
KYSE-510 CTRP2 8.4198 10.2195 7.9534 7.0045
TE-5 CTRP2 8.4367 9.3009 8.3384 5.4672
KYSE-30 CTRP2 8.4376 11.913 7.168 10.1712
TE-9 CTRP2 8.4781 12.191 7.0698 10.4855
TE-14 CTRP2 8.4865 9.7651 8.2195 5.7781
KYSE-70 CTRP2 8.5139 9.6864 8.2807 5.4658
KYSE-450 CTRP2; CTRP1 8.5224 10.7606 7.8043 7.3548
KYSE-410 CTRP2; CTRP1 8.5251 12.578 6.9228 10.9902
OE21 CTRP2 8.5284 9.9593 8.1797 5.8238
KYSE-150 CTRP2 8.5721 9.0783 8.5443 4.3119
TE-1 CTRP2 8.5808 9.8939 8.2622 5.3602
OE19 CTRP2 8.6049 19.2697 3.664 22.8652
TE-4 CTRP2 8.6722 9.6095 8.4787 4.2667
COLO 680N CTRP2 8.7361 24.0781 1.3739 28.379
OE33 CTRP2 8.7739 9.4547 8.6487 3.3302
TE-10 CTRP2 8.7816 13.6413 6.6245 11.6772
KYSE-180 CTRP2 10.2651 16.6271 6.3358 10.0914
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 38 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 8.5614 9.0676 8.5348 4.3789
PSN1 CTRP2 6.4859 13.4242 4.5509 25.1205
HPAC CTRP2; CTRP1 8.0797 13.7944 5.916 16.0865
SNU-410 CTRP2 8.1522 10.631 7.4974 9.5107
Capan-2 CTRP2; CTRP1 8.2689 9.645 8.0367 7.0829
KP-4 CTRP2 8.3271 9.8758 8.0065 7.0386
BxPC-3 CTRP2 8.3872 12.2353 6.9637 11.1289
HPAF-II CTRP2 8.4208 19.0474 3.6157 23.4046
QGP-1 CTRP2; CTRP1 8.4315 12.1758 7.034 10.7385
Panc 03.27 CTRP2; CTRP1 8.4385 12.0778 7.0884 10.4978
SW1990 CTRP2 8.4388 11.5279 7.356 9.3923
SU.86.86 CTRP2 8.4473 9.2774 8.3572 5.3665
PK-59 CTRP2 8.4537 9.9111 8.1237 6.2413
DAN-G CTRP2 8.4769 10.5675 7.8509 7.2748
HuP-T3 CTRP2 8.4785 15.8378 5.265 17.7153
Panc 10.05 CTRP2; CTRP1 8.4946 9.7596 8.2303 5.7144
HuP-T4 CTRP2; CTRP1 8.5184 12.8192 6.7977 11.5229
L3.3 CTRP2 8.5502 15.9349 5.2797 17.5058
MIA PaCa-2 CTRP2 8.5618 9.1342 8.521 4.4263
AsPC-1 CTRP2 8.6039 9.5164 8.4437 4.5896
SNU-213 CTRP2 8.6395 9.1647 8.5983 3.9105
TCC-Pan2 CTRP2 8.6475 9.0984 8.622 3.8012
YAPC CTRP2 8.6809 9.1934 8.6361 3.6476
Panc 08.13 CTRP2 8.6872 9.4283 8.5662 3.8884
Panc 02.03 CTRP2 8.7083 12.7504 7.0028 10.2618
CFPAC-1 CTRP2; CTRP1 8.7187 13.8893 6.4459 12.5441
Panc 04.03 CTRP2 8.7209 13.1952 6.7932 11.1062
PK-45H CTRP2 8.725 9.8322 8.4367 4.2937
Panc 05.04 CTRP2 8.7289 9.8315 8.4409 4.2669
SUIT-2 CTRP2; CTRP1 8.7323 9.2769 8.6678 3.3775
Capan-1 CTRP2 8.7471 9.4702 8.6141 3.5375
Hs 766T CTRP2 8.7658 9.287 8.701 3.1557
PANC-1 CTRP2 8.7755 9.391 8.6749 3.2256
PaTu 8988s CTRP2 8.786 9.2729 8.7274 2.9985
KP-3 CTRP2; CTRP1 8.925 16.3656 5.3885 16.3085
PaTu 8988t CTRP2 8.9459 9.6189 8.7559 2.4546
KP-2 CTRP2 8.948 10.9689 8.1005 5.1644
PaTu 8902 CTRP2; CTRP1 9.4336 10.4286 8.7713 1.4247
⏷ Show the Full List of 38 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 9.011 12.6376 6.6374 5.6948
COLO 741 CTRP2; CTRP1 6.609 9.5337 6.2757 18.4831
HMCB CTRP2 6.7221 11.7947 5.5211 20.9997
A2058 CTRP2 7.2002 8.7452 7.1232 13.6257
G-361 CTRP2; CTRP1 7.2317 10.9779 6.3999 16.254
IGR-37 CTRP2 7.2383 10.0057 6.7968 14.7079
COLO 792 CTRP2 7.6918 9.3749 7.5042 10.7484
Hs 944.T CTRP2; CTRP1 7.8998 9.4971 7.6912 9.4434
SK-MEL-5 CTRP2; CTRP1 8.0125 9.0877 7.9343 8.2479
WM115 CTRP2 8.2653 9.8996 7.9318 7.4968
CJM [Human melanoma] CTRP2 8.3367 11.9829 7.0392 10.9329
SK-MEL-1 CTRP2; CTRP1 8.3574 9.2131 8.2785 5.9545
WM88 CTRP2 8.3704 12.8269 6.6586 12.4243
WM266-4 CTRP2 8.4314 11.2752 7.4708 8.9371
WM1799 CTRP2 8.4394 16.9936 4.6554 20.0036
Hs 936.T CTRP2; CTRP1 8.4584 8.9883 8.4374 5.0458
RVH-421 CTRP2 8.491 12.6998 6.8317 11.4425
SK-MEL-24 CTRP2 8.4985 11.9052 7.2286 9.7826
MDA-MB-435S CTRP2 8.5058 15.7324 5.3415 17.3686
HT-144 CTRP2 8.5062 14.1855 6.1106 14.3605
Mel JuSo CTRP2 8.5132 9.2707 8.431 4.8994
WM983B CTRP2 8.52 13.7928 6.3177 13.492
UACC-257 CTRP2 8.5205 9.1075 8.4822 4.6926
IPC-298 CTRP2 8.5319 14.1794 6.1365 14.2008
K029AX CTRP2 8.535 9.0546 8.5087 4.5539
Hs 940.T CTRP2 8.5383 9.2888 8.4528 4.7442
SK-MEL-31 CTRP2 8.5398 9.1567 8.4915 4.5996
WM793 CTRP2 8.5653 16.1358 5.1928 17.7977
MeWo CTRP2 8.5672 12.644 6.9285 10.8743
SK-MEL-28 CTRP2; CTRP1 8.5728 8.9635 8.5631 4.2756
LOX-IMVI CTRP2 8.5784 9.2021 8.5219 4.3723
Hs 294T CTRP2 8.5953 8.9866 8.5841 4.0995
UACC-62 CTRP2 8.6215 9.071 8.5991 3.9638
A101D CTRP2 8.6278 9.0584 8.6081 3.9123
COLO 829 CTRP2 8.6332 9.376 8.527 4.1907
COLO 800 CTRP2 8.649 9.1943 8.601 3.8715
SK-MEL-30 CTRP2 8.6617 9.1338 8.6299 3.7289
Hs 839.T CTRP2 8.6634 9.0786 8.643 3.6774
Hs 895.T CTRP2 8.6734 9.1312 8.6431 3.6456
Hs 852.T CTRP2; CTRP1 8.6769 10.0376 8.2949 4.9841
WT2-iPS CTRP2 8.6838 9.118 8.6574 3.5627
A-375 CTRP2; CTRP1 8.7072 9.2228 8.6576 3.5213
SK-MEL-3 CTRP2 8.7177 9.3793 8.6171 3.609
IGR-1 CTRP2 8.7322 9.3229 8.6525 3.4341
IGR-39 CTRP2 8.8069 9.4005 8.7049 3.0229
Hs 688(A).T CTRP2 8.8362 9.2711 8.7826 2.6466
RPMI-7951 CTRP2 8.9616 10.5493 8.3203 4.2167
Mel Ho CTRP2 9.5228 16.12 6.0083 12.7202
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 CTRP2 7.53 10.6597 6.8453 13.7165
Cancer Drug Sensitivity Data Curated from 11 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-BE(2) CTRP2 5.7332 7.1792 5.7265 23.164
Kelly CTRP2 6.3529 8.6162 6.2311 19.4285
IMR-32 CTRP2 7.2605 10.7852 6.5112 15.7436
NB1 CTRP2 7.5269 8.6807 7.4856 11.3245
CHP-212 CTRP2 7.7637 10.352 7.2184 11.6315
KP-N-SI9s CTRP2 8.1713 11.28 7.2167 10.5965
NH-6 CTRP2 8.4224 11.8495 7.1846 10.1369
SK-N-FI CTRP2 8.4435 16.5946 4.8576 19.2821
SK-N-SH CTRP2 8.4993 11.9478 7.2085 9.8638
SK-N-AS CTRP2 8.5598 9.1345 8.5187 4.4407
CHP-126 CTRP2 8.6317 9.6538 8.4178 4.6133
⏷ Show the Full List of 11 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 7 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-1079 CTRP2 6.3773 8.9018 6.1961 19.4755
SNU-478 CTRP2 8.1664 10.2589 7.6767 8.7609
HuH-28 CTRP2 8.4001 9.5198 8.2241 5.9999
SNU-1196 CTRP2 8.444 14.3107 5.993 14.967
SNU-869 CTRP2 8.5551 14.6155 5.9405 14.9362
HuCC-T1 CTRP2 8.6027 10.7458 7.8889 6.8176
SNU-308 CTRP2 8.6826 9.1686 8.6443 3.6129
⏷ Show the Full List of 7 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SK-N-MC CTRP2 5.5596 7.0393 5.5536 24.319
TC71 CTRP2 5.8576 7.9266 5.8052 22.4898
U2OS CTRP2 6.646 9.4481 6.3423 18.1286
MHH-ES-1 CTRP2 7.1077 10.2181 6.5772 15.9107
SK-ES-1 CTRP2 7.1304 9.0587 6.9791 14.3532
A-673 CTRP2 8.4502 12.5606 6.8628 11.4046
MG-63 CTRP2 8.4521 13.0691 6.6142 12.4254
G-292 clone A141B1 CTRP2 8.5239 9.7153 8.2793 5.4443
SJSA-1 CTRP2 8.5308 9.9055 8.2058 5.7141
HOS CTRP2 8.619 12.7306 6.9326 10.7449
Hs 888.T CTRP2 8.7685 9.2901 8.7028 3.141
Hs 822.T CTRP2 8.783 9.091 8.7698 2.8554
CAL-78 CTRP2 8.8334 9.6043 8.6484 3.1715
SW1353 CTRP2 13.0727 23.2724 5.074 10.642
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 64 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-453 CTRP2 5.5332 7.6255 5.4937 24.6082
Hs 578T CTRP2 7.04 23.0853 0.3869 33.7471
HCC1954 CTRP2 7.4847 15.2741 4.6395 22.2515
T-47D CTRP2 7.5212 9.2312 7.3601 11.787
CAMA-1 CTRP2 7.6855 11.0572 6.8327 13.3581
BT-20 CTRP2 7.9917 10.8638 7.2301 10.9888
HMC-1-8 CTRP2 8.0274 10.2079 7.5543 9.6107
HCC1500 CTRP2 8.2599 11.1812 7.3498 9.8402
EFM-192A CTRP2 8.4167 10.2193 7.9504 7.0245
HCC202 CTRP2 8.4172 10.8921 7.6397 8.279
ZR-75-1 CTRP2 8.4329 9.5957 8.2307 5.8825
ZR-75-30 CTRP2 8.4356 10.6657 7.7643 7.7271
AU565 CTRP2 8.4438 10.1362 8.015 6.6976
SK-BR-3 CTRP2 8.4478 9.7972 8.1656 6.093
HCC1428 CTRP2 8.5014 9.6157 8.2958 5.4417
HCC1419 CTRP2 8.553 9.8836 8.2382 5.5279
HCC1806 CTRP2 8.5692 15.9545 5.2865 17.4395
BT-549 CTRP2 8.5752 9.4709 8.4303 4.7214
JIMT-1 CTRP2 8.591 9.1321 8.5533 4.2208
HCC1937 CTRP2 8.6039 12.0072 7.2758 9.3516
CAL-85-1 CTRP2 8.6432 12.3844 7.1256 9.8901
HCC38 CTRP2 8.6458 9.9566 8.3005 5.0401
MCF-7 CTRP2; CTRP1 8.6632 9.2751 8.5941 3.8849
MDA-MB-231 CTRP2 8.6807 9.8824 8.3692 4.6766
BT-474 CTRP2 8.6913 9.2728 8.6244 3.6588
CAL-51 CTRP2 8.7242 10.2758 8.2301 5.1316
HCC1143 CTRP2 9.1823 18.948 4.3143 19.61
CAL-120 CTRP2 9.2117 10.1174 8.7541 1.8813
HCC1395 CTRP2 9.2238 15.3948 6.1255 12.8251
MDA-MB-468 CTRP2 9.2459 13.7079 6.9873 9.2382
HDQ-P1 CTRP2 9.6445 11.3669 8.4645 2.3589
BT 239 CTRP2 5.5905 8.2479 5.4744 24.4888
BT 416 CTRP2 6.1035 9.5174 5.7299 21.9883
BT 428 CTRP2 6.2161 10.8617 5.3778 22.944
BT 145 CTRP2 7.1427 9.7054 6.8001 14.9707
BT 231 CTRP2 7.3209 9.7119 6.991 13.7402
BT 248 CTRP2 7.3245 9.0093 7.2026 12.956
BT 112 CTRP2 7.7367 11.0012 6.9098 12.9196
BT 245 CTRP2 7.8617 10.7786 7.1361 11.6972
BT 232 CTRP2 7.9082 12.1363 6.5556 13.9169
BT 187 CTRP2 7.9224 9.5602 7.6942 9.3664
BT 482 CTRP2 8.0442 11.7747 6.8591 12.3584
BT 172 CTRP2 8.1293 11.4903 7.0764 11.2689
BT164 CTRP2 8.1699 11.8409 6.949 11.6923
BT 286 CTRP2 8.2017 13.3635 6.2398 14.5118
BT147 CTRP2 8.2215 10.7717 7.5028 9.314
BT 228 CTRP2 8.2798 9.3939 8.1379 6.671
BT 159 CTRP2 8.3074 9.5024 8.1305 6.6183
BT 359 CTRP2 8.3362 9.7187 8.0797 6.7304
BT 422 CTRP2 8.3377 11.0772 7.4748 9.1431
BT 216 CTRP2 8.3784 12.1328 7.0055 10.9763
BT 498 CTRP2 8.4193 15.8315 5.2159 18.0273
BT 504 CTRP2 8.4287 14.0902 6.0885 14.6175
BT 224 CTRP2 8.4339 11.6819 7.2769 9.7296
BT 131 CTRP2 8.4755 14.6855 5.8351 15.5261
BT 271 CTRP2 8.4821 9.5014 8.319 5.4075
BT 444 CTRP2 8.5522 9.119 8.514 4.481
BT 179 CTRP2 8.5562 9.1179 8.5187 4.4519
BT 333 CTRP2 8.6071 9.1729 8.5609 4.1439
BT 328 CTRP2 8.6093 9.181 8.5612 4.1362
BT 320 CTRP2 8.6166 10.9714 7.7935 7.1778
BT 340 CTRP2 8.6715 9.1397 8.6392 3.6655
BT 440 CTRP2 8.711 9.1619 8.6769 3.4086
BT 330 CTRP2 9.6713 16.8232 5.7769 13.354
⏷ Show the Full List of 64 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 8.5202 9.0273 8.4975 4.6399
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D283 Med CTRP2 6.6035 8.7793 6.4697 17.8009
GB-1 CTRP2 6.875 12.0106 5.5828 20.3563
SF539 CTRP2 7.6348 9.4602 7.4154 11.2444
SNU-466 CTRP2 7.849 9.1997 7.7266 9.4651
SF268 CTRP2 7.9224 9.5846 7.6858 9.3976
SW1783 CTRP2 7.9727 11.1366 7.0867 11.6122
U-251MG CTRP2 8.2906 9.6682 8.051 6.9672
LN-18 CTRP2 8.3345 9.5624 8.1379 6.513
DK-MG CTRP2 8.349 11.3878 7.3379 9.6766
U-87MG ATCC CTRP2 8.3953 15.8191 5.2008 18.1363
8-MG-BA CTRP2 8.4091 11.5163 7.3335 9.5538
ONS-76 CTRP2 8.45 12.2315 7.0239 10.7387
TM-31 CTRP2 8.468 10.1668 8.0259 6.5918
Becker CTRP2 8.4699 13.2269 6.5525 12.6398
KNS-60 CTRP2 8.4732 9.0773 8.4373 4.9993
YH-13 CTRP2 8.4895 9.21 8.4228 5.0006
GMS-10 CTRP2 8.4947 8.9627 8.48 4.7823
42-MG-BA CTRP2 8.5005 10.3477 7.9762 6.7093
SW1088 CTRP2 8.509 13.2501 6.5765 12.4561
SNU-201 CTRP2 8.5093 9.0928 8.4731 4.7596
M059K CTRP2 8.524 9.0492 8.4978 4.6267
SNB-75 CTRP2 8.5524 9.6207 8.3479 5.1006
SF295 CTRP2; CTRP1 8.5618 9.2351 8.4945 4.5218
KNS-42 CTRP2 8.5964 9.0353 8.5782 4.1165
Daoy CTRP2 8.6041 14.3712 6.1053 14.1716
KNS-81 CTRP2 8.6333 9.0951 8.6072 3.8981
LN-229 CTRP2; CTRP1 8.6413 9.2009 8.5918 3.9593
A-172 CTRP2 8.6449 9.278 8.5723 3.9881
Hs 683 CTRP2 8.6701 9.1519 8.6347 3.6858
KG-1-C CTRP2 8.6835 9.1266 8.6552 3.5713
KALS-1 CTRP2 8.7285 15.405 5.6992 15.5204
SNU-626 CTRP2 8.7485 9.2327 8.6989 3.2149
CCF-STTG1 CTRP2 8.7905 9.1865 8.7575 2.8754
SNU-738 CTRP2 8.81 10.035 8.4277 4.1191
GOS-3 CTRP2 8.8128 13.4937 6.7254 11.1947
U-118MG CTRP2 8.8255 9.4325 8.7122 2.943
GaMG CTRP2; CTRP1 8.8796 10.2271 8.4024 4.0589
T98G CTRP2 8.9958 16.2317 5.5156 15.6796
SNU-489 CTRP2 9.1056 9.7607 8.8403 1.7347
YKG-1 CTRP2 9.1407 9.9028 8.8009 1.8256
SF126 CTRP2 9.5726 14.2574 6.9779 8.6678
NMC-G1 CTRP2 9.7506 11.6053 8.4232 2.3696
DBTRG-05MG CTRP2 10.0495 16.175 6.3961 10.2151
SNU-1105 CTRP2 13.3771 27.5292 3.2434 15.9343
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 22 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JHUEM-1 CTRP2 6.5613 8.641 6.4519 17.9968
JHUEM-2 CTRP2; CTRP1 6.7602 10.6282 6.0494 18.9193
HEC-1-B CTRP2 6.7934 11.204 5.8478 19.5687
HEC-151 CTRP2; CTRP1 7.4689 8.5656 7.4393 11.6996
HEC-50B CTRP2 7.5791 10.1387 7.1103 12.555
MFE-296 CTRP2 7.5924 9.2654 7.4281 11.3246
KLE CTRP2; CTRP1 7.7546 11.4723 6.7148 13.6527
HEC-1-A CTRP2 8.0655 9.7553 7.7773 8.6438
HEC-251 CTRP2; CTRP1 8.2448 11.1016 7.3726 9.7841
HEC-265 CTRP2; CTRP1 8.3396 9.7266 8.0803 6.7189
MFE-319 CTRP2; CTRP1 8.4257 10.9 7.6443 8.2401
AN3-CA CTRP2 8.4262 13.367 6.4437 13.1819
HEC-59 CTRP2; CTRP1 8.4326 12.4879 6.8823 11.3632
ESS-1 CTRP2 8.4352 12.1953 7.028 10.7551
EFE-184 CTRP2 8.4974 13.061 6.6594 12.1403
RL95-2 CTRP2 8.5172 16.5608 4.9391 18.83
HEC-6 CTRP2; CTRP1 8.5258 9.9995 8.1594 5.9112
JHUEM-7 CTRP2 8.5899 11.1971 7.659 7.7942
JHUEM-3 CTRP2 8.6626 10.0779 8.2621 5.1522
EN CTRP2 8.7004 9.2083 8.6534 3.5257
HEC-108 CTRP2; CTRP1 11.1678 17.9863 6.3226 8.7266
Ishikawa (Heraklio) 02 ER- CTRP2; CTRP1 8.615 9.2749 8.5407 4.1933
⏷ Show the Full List of 22 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 19 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
UO-31 CTRP2 7.1029 8.4381 7.0658 14.1365
OS-RC-2 CTRP2 8.0667 11.2564 7.1248 11.2251
TUHR10TKB CTRP2 8.3681 9.2358 8.283 5.8754
TUHR14TKB CTRP2 8.4188 11.0287 7.5766 8.5331
VMRC-RCZ CTRP2 8.4843 12.2288 7.057 10.5248
VMRC-RCW CTRP2; CTRP1 8.522 14.1384 6.1481 14.1751
769-P CTRP2 8.5343 15.4495 5.5073 16.676
KMRC-1 CTRP2 8.5454 9.1269 8.5048 4.535
Caki-2 CTRP2 8.5826 9.0413 8.5624 4.2155
CAL-54 CTRP2 8.613 11.9784 7.2983 9.2381
KMRC-20 CTRP2 8.6433 9.6251 8.4419 4.4882
SNU-1272 CTRP2 8.7506 9.1788 8.7159 3.1471
KMRC-2 CTRP2 8.8196 9.6166 8.6288 3.2852
BFTC-909 CTRP2 8.8309 9.4798 8.6987 2.9805
RCC10RGB CTRP2; CTRP1 8.8783 9.34 8.8056 2.47
786-O CTRP2 8.9993 12.9723 7.147 9.0556
ACHN CTRP2 9.1307 12.9024 7.2938 8.179
TUHR4TKB CTRP2 9.2961 10.3982 8.6822 2.0264
Caki-1 CTRP2 10.6989 16.5845 6.6736 8.0449
⏷ Show the Full List of 19 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SW403 CTRP1 4.3978 6.5848 3.7669 16.4251
SW620 CTRP2; CTRP1 6.2341 9.5033 5.8776 21.0843
SW480 CTRP1 6.2627 13.28 4.3945 46.0639
NCI-H747 CTRP2 6.2849 9.4212 5.9566 20.619
COLO 320 CTRP2; CTRP1 6.5106 8.5253 6.4187 18.3
GP2d CTRP2; CTRP1 6.9069 9.3752 6.6485 16.2282
LoVo CTRP2; CTRP1 7.5197 9.6901 7.2149 12.3547
SNU-407 CTRP2 7.6509 9.084 7.5403 10.7418
CCK-81 CTRP2 7.6618 9.7278 7.3537 11.3955
SNU-C1 CTRP2 7.7287 16.1818 4.4208 22.4138
LS180 CTRP2; CTRP1 8.2406 9.1455 8.1689 6.706
RKO CTRP2; CTRP1 8.2896 9.1301 8.2261 6.3503
SNU-C5 CTRP2; CTRP1 8.324 9.5966 8.1154 6.6582
HT-55 CTRP2; CTRP1 8.3514 9.4665 8.1921 6.2904
KM12 CTRP2; CTRP1 8.3788 9.2239 8.299 5.8155
CW-2 CTRP2; CTRP1 8.4211 9.1696 8.3597 5.4678
OUMS-23 CTRP2 8.4324 14.8169 5.7315 16.0268
HT115 CTRP2; CTRP1 8.4467 9.066 8.4113 5.2048
SNU-1040 CTRP1 8.4524 9.5133 8.2841 12.1212
SK-CO-1 CTRP2; CTRP1 8.454 9.3335 8.3469 5.3843
COLO201 CTRP2 8.4627 9.1338 8.4132 5.1173
NCI-H716 CTRP2 8.4773 12.3315 7.0002 10.7755
SNU-175 CTRP1 8.4802 9.5001 8.3188 11.6704
SW48 CTRP2; CTRP1 8.4974 9.4116 8.3678 5.1798
SNU-C4 CTRP2; CTRP1 8.5005 9.0235 8.4775 4.8033
MDST8 CTRP2; CTRP1 8.5063 8.9845 8.4897 4.7423
LS513 CTRP2; CTRP1 8.5435 14.9955 5.7413 15.7483
HCT 8 CTRP2; CTRP1 8.5768 9.033 8.5579 4.2806
HCT 15 CTRP2 8.5846 17.0671 4.7454 19.3751
SNU-61 CTRP2; CTRP1 8.6081 9.1681 8.564 4.1607
LS123 CTRP2; CTRP1 8.6199 9.4938 8.4709 4.4717
SNU-81 CTRP1 8.6296 9.3898 8.5196 9.131
COLO205 CTRP2; CTRP1 8.6602 9.0608 8.6426 3.6891
HCT 116 CTRP2; CTRP1 8.666 9.3478 8.5736 3.9523
CL-34 CTRP1 8.6913 9.327 8.608 8.0404
LS411N CTRP2; CTRP1 8.7234 9.1722 8.6879 3.3311
COLO 678 CTRP2; CTRP1 8.7259 9.5286 8.57 3.7972
SNU-503 CTRP2 8.7263 9.3227 8.6462 3.475
LS1034 CTRP2 8.7437 9.3479 8.6563 3.387
SW948 CTRP2; CTRP1 8.7478 9.1797 8.7135 3.1959
RCM-1 [Human ESC] CTRP2; CTRP1 8.7636 9.6067 8.5771 3.6675
NCI-H508 CTRP2; CTRP1 8.8107 9.2931 8.7489 2.8778
SW1417 CTRP2 8.8258 9.7174 8.5904 3.422
DLD-1 CTRP2; CTRP1 8.9706 9.4541 8.855 1.995
HCC-56 CTRP2 8.9819 9.4448 8.8707 1.9033
HT-29 CTRP2; CTRP1 9.0398 9.529 8.893 1.6988
CL-11 CTRP2 9.2676 11.3247 8.1966 4.1197
CL-40 CTRP1 9.3474 11.3856 8.2341 8.2305
C2BBe1 CTRP2; CTRP1 9.4605 15.0319 6.5013 10.8444
SNU-C2A CTRP2; CTRP1 9.7599 17.5457 5.4873 14.304
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 21 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SNU-886 CTRP2 6.0632 12.3319 2.3323 13.9767
HLF CTRP2 6.8033 10.9804 5.9511 19.1476
Hep 3B2.1-7 CTRP2 7.2992 9.1806 7.1316 13.288
PLC/PRF/5 CTRP2 7.9725 10.7748 7.2506 10.9556
SNU-398 CTRP2; CTRP1 7.9934 9.2957 7.8578 8.582
Li-7 CTRP2 8.0218 10.0611 7.6096 9.4101
JHH-2 CTRP2 8.227 10.8585 7.4683 9.4399
SNU-182 CTRP2 8.3593 11.4901 7.2986 9.8132
SNU-761 CTRP2 8.3674 9.8708 8.0508 6.7572
JHH-4 CTRP2 8.3776 11.9701 7.084 10.6543
JHH-1 CTRP2 8.3842 11.9559 7.097 10.5857
SK-HEP-1 CTRP2 8.4334 11.1161 7.549 8.6113
SNU-423 CTRP2 8.4519 11.7347 7.2682 9.7243
SNU-387 CTRP2 8.4649 11.4787 7.4045 9.132
JHH-5 CTRP2 8.5704 9.1362 8.5298 4.3682
SNU-878 CTRP2 8.6333 10.0874 8.2284 5.3612
HuH-1 CTRP2 8.6932 9.1374 8.6633 3.5123
Hep-G2 CTRP2; CTRP1 8.7799 9.6058 8.5945 3.5559
JHH-6 CTRP2; CTRP1 8.7894 9.0729 8.7795 2.8015
SNU-475 CTRP2 8.8114 12.4468 7.2452 9.0319
SNU-449 CTRP2; CTRP1 10.0298 15.5497 6.6907 9.0521
⏷ Show the Full List of 21 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 157 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1930 CTRP1 1.563 5.5043 1.1457 50.7538
HCC33 CTRP1 2.546 4.1082 2.5132 37.4594
NCI-H82 CTRP1 3.6652 5.1043 3.5517 22.4211
RERF-LC-KJ CTRP1 4.7729 5.9814 4.4186 8.9741
NCI-H1975 CTRP2; CTRP1 5.208 6.3072 5.2077 26.6442
NCI-H1341 CTRP2 5.6437 7.1784 5.6352 23.7669
COR-L51 CTRP2; CTRP1 5.8402 9.3171 5.5025 23.6324
RERF-LC-MS CTRP2 6.2064 8.2766 6.1313 20.2427
LC-1F CTRP2 6.3344 9.6879 5.9281 20.5746
SW1573 CTRP2 6.3812 9.6958 5.9765 20.2581
COR-L279 CTRP1 6.3935 12.1022 2.6932 16.3997
NCI-H1048 CTRP1 6.4246 8.3427 4.5021 2.7096
NCI-H1734 CTRP2 6.7242 10.0456 6.229 18.3178
HCC44 CTRP2; CTRP1 6.9203 11.0251 6.0554 18.428
NCI-H1581 CTRP2 6.9492 8.8589 6.8283 15.4524
NCI-H211 CTRP2 6.9942 10.1557 6.4791 16.6038
NCI-H2122 CTRP2; CTRP1 7.018 9.5027 6.7317 15.6187
NCI-H1437 CTRP1 7.0368 9.0796 4.5021 1.7039
NCI-H1092 CTRP2 7.1647 9.8947 6.758 15.0644
NCI-H1694 CTRP2; CTRP1 7.1942 9.3391 6.9734 14.2073
NCI-H661 CTRP2; CTRP1 7.2212 10.8164 6.4572 16.0597
COLO 668 CTRP2; CTRP1 7.3194 10.8751 6.5348 15.4936
NCI-H1155 CTRP2 7.35 8.8658 7.2621 12.6659
NCI-H1435 CTRP2; CTRP1 7.3795 11.0525 6.521 15.3874
NCI-H1573 CTRP2; CTRP1 7.3854 12.3197 5.9562 17.5947
Calu-3 CTRP2; CTRP1 7.3917 11.232 6.4552 15.6143
NCI-H1703 CTRP2 7.4161 10.7869 6.6728 14.6956
NCI-H446 CTRP2 7.4491 9.6438 7.153 12.7626
NCI-H2286 CTRP2; CTRP1 7.4565 10.0346 7.0198 13.2436
NCI-H2106 CTRP2 7.5132 9.3531 7.3162 11.9706
NCI-H1563 CTRP2 7.5176 9.2084 7.3624 11.7895
NCI-H2029 CTRP2; CTRP1 7.559 10.3057 7.0223 12.9494
DMS 79 CTRP2 7.573 11.942 6.3174 15.6961
HCC827 CTRP2; CTRP1 7.5772 10.0488 7.1449 12.456
NCI-H1184 CTRP2 7.6135 13.3615 5.6868 18.0826
NCI-H1793 CTRP2; CTRP1 7.6676 9.7241 7.3613 11.3502
NCI-H2141 CTRP2; CTRP1 7.7175 10.2999 7.1933 11.8826
VMRC-LCD CTRP2; CTRP1 7.7423 10.4059 7.1735 11.8644
PC-14 CTRP2 7.764 9.8503 7.4186 10.8591
SHP-77 CTRP2; CTRP1 7.8 13.5075 5.7939 17.2184
EKVX CTRP2 7.8146 18.522 3.3423 25.5492
NCI-H838 CTRP2 7.8217 10.1367 7.3679 10.8931
NCI-H1666 CTRP2; CTRP1 7.8627 10.5297 7.246 11.2596
HCC78 CTRP2; CTRP1 7.8729 12.286 6.4503 14.4274
NCI-H889 CTRP2 7.9083 12.796 6.2402 15.1892
SBC-5 CTRP2 7.9129 9.1037 7.8211 8.9298
LXF 289 CTRP2; CTRP1 7.9155 10.9256 7.1251 11.6025
Lu-65 CTRP2; CTRP1 7.9206 11.3214 6.9498 12.2934
NCI-H810 CTRP2; CTRP1 7.9304 10.1114 7.4928 10.1124
NCI-H2196 CTRP2 7.9414 10.8664 7.178 11.3254
NCI-H1963 CTRP1 7.9528 10.8083 7.2177 23.7135
HOP-62 CTRP2 7.9895 9.0894 7.9082 8.3823
EPLC-272H CTRP2; CTRP1 8.0189 11.8912 6.7793 12.7437
NCI-H2087 CTRP2 8.0305 9.8926 7.6866 9.0886
RERF-LC-A1 CTRP2 8.0312 13.1819 6.1698 15.1846
NCI-H1755 CTRP2; CTRP1 8.1039 9.1815 8.0104 7.6942
NCI-H2023 CTRP2; CTRP1 8.1509 10.1709 7.7004 8.7379
NCI-H1355 CTRP2; CTRP1 8.2151 12.38 6.7321 12.4749
COR-L88 CTRP2; CTRP1 8.2369 10.99 7.4169 9.6235
NCI-H647 CTRP2 8.2415 11.5016 7.18 10.5777
NCI-H1373 CTRP2; CTRP1 8.2489 11.109 7.3731 9.7721
LK2 CTRP2 8.2591 9.5604 8.0576 7.0317
SK-MES-1 CTRP2 8.2636 10.3208 7.7493 8.2198
NCI-H441 CTRP2; CTRP1 8.2827 9.332 8.1621 6.6033
NCI-H727 CTRP2; CTRP1 8.2904 14.5345 5.744 16.2901
NCI-H2009 CTRP2; CTRP1 8.2916 12.7044 6.6457 12.6545
NCI-H841 CTRP2; CTRP1 8.3115 11.2402 7.3745 9.6439
HOP-92 CTRP2 8.3155 9.7419 8.0486 6.9072
NCI-H1944 CTRP2; CTRP1 8.3293 12.0235 7.0126 11.0593
NCI-H2081 CTRP2; CTRP1 8.332 9.5118 8.1551 6.4852
HCC1438 CTRP2 8.3381 9.2613 8.2429 6.1117
NCI-H520 CTRP2 8.3427 11.8024 7.1323 10.5358
NCI-H3255 CTRP1 8.3729 10.0693 7.9738 15.162
LCLC-97TM1 CTRP2; CTRP1 8.3815 18.3389 3.9346 22.5139
DV-90 CTRP2; CTRP1 8.3859 12.0816 7.0375 10.8276
HCC95 CTRP2 8.3944 19.9596 3.1378 24.8352
HCC1588 CTRP2 8.4004 13.2182 6.4937 13.0343
NCI-H1693 CTRP2 8.4022 11.0635 7.544 8.706
DMS 454 CTRP2 8.4039 10.4602 7.8281 7.5478
NCI-H2291 CTRP2 8.4192 17.8071 4.2325 21.4763
NCI-H1105 CTRP2; CTRP1 8.4207 9.0616 8.3841 5.3822
HARA [Human squamous cell lung carcinoma] CTRP2; CTRP1 8.4257 11.0929 7.5526 8.6149
NCI-H1876 CTRP1 8.4378 9.6965 8.1979 12.9153
NCI-H1651 CTRP2 8.4378 9.818 8.1465 6.1942
NCI-H2444 CTRP2 8.4389 9.4625 8.2866 5.6534
MOR/CPR CTRP2 8.4435 8.9744 8.4236 5.1411
NCI-H596 CTRP1 8.4442 9.5366 8.2667 12.3126
KNS-62 CTRP2; CTRP1 8.4447 9.6995 8.2024 5.9585
NCI-H522 CTRP2; CTRP1 8.4459 11.3456 7.4508 8.9853
NCI-H2228 CTRP2 8.4482 10.7618 7.7315 7.8302
NCI-H1568 CTRP2; CTRP1 8.4505 13.5906 6.3553 13.4896
NCI-H1836 CTRP1 8.4548 9.6696 8.2267 12.5764
NCI-H1792 CTRP2; CTRP1 8.4697 11.562 7.3687 9.2687
NCI-H1650 CTRP2 8.475 11.231 7.5337 8.5764
NCI-H1915 CTRP2; CTRP1 8.4804 11.1081 7.5979 8.3
NCI-H2342 CTRP2; CTRP1 8.484 12.4805 6.936 11.054
A-549 CTRP2; CTRP1 8.4873 10.8303 7.7372 7.7131
NCI-H1395 CTRP2 8.4893 12.5262 6.9156 11.0993
HCC4006 CTRP2; CTRP1 8.4904 9.1372 8.4432 4.9557
SW1271 CTRP2 8.4906 9.6108 8.2863 5.5085
Lu-99 CTRP2; CTRP1 8.497 9.0929 8.4598 4.8451
HCC1833 CTRP2; CTRP1 8.5042 9.6216 8.2981 5.4559
NCI-H460 CTRP2; CTRP1 8.5046 9.0233 8.4819 4.7745
NCI-H650 CTRP2; CTRP1 8.5049 10.5739 7.8754 7.1072
HCC366 CTRP2 8.5062 11.6276 7.3711 9.1752
NCI-H2172 CTRP2; CTRP1 8.5127 9.0482 8.4862 4.7341
HCC2935 CTRP2; CTRP1 8.514 9.1248 8.4718 4.7807
LUDLU-1 CTRP2 8.5173 13.1344 6.6411 12.1719
NCI-H2170 CTRP2 8.5205 12.1663 7.121 10.1789
NCI-H2126 CTRP2; CTRP1 8.531 9.6493 8.3137 5.2915
COR-L95 CTRP2 8.5323 9.1999 8.4722 4.6918
EBC-1 CTRP2; CTRP1 8.5426 10.2566 8.0602 6.2659
LC-1/sq-SF CTRP2; CTRP1 8.5459 9.0938 8.5127 4.5055
NCI-H1781 CTRP1 8.5465 9.9935 8.1852 12.4009
DMS 114 CTRP2 8.5513 9.2628 8.4749 4.6247
NCI-H1339 CTRP2 8.5531 11.8359 7.3131 9.3098
HCC1171 CTRP2 8.5543 14.5775 5.9587 14.8655
DMS 273 CTRP2; CTRP1 8.5594 9.2895 8.4756 4.5978
NCI-H1869 CTRP2 8.5679 12.5143 6.9931 10.6049
NCI-H526 CTRP2 8.5752 9.2054 8.5175 4.3979
HCC1195 CTRP2; CTRP1 8.5765 9.0971 8.5458 4.3237
ChaGo-K-1 CTRP2; CTRP1 8.5781 13.0166 6.7542 11.573
LCLC-103H CTRP2; CTRP1 8.5879 9.084 8.5603 4.2057
NCI-H226 CTRP2 8.5954 9.0951 8.5662 4.1614
COR-L105 CTRP2 8.5958 11.7453 7.3969 8.8665
Sq-1 CTRP2; CTRP1 8.5965 9.2015 8.5427 4.2727
LOU-NH91 CTRP2 8.6033 9.3051 8.5184 4.31
NCI-H196 CTRP2 8.6104 9.799 8.3341 4.9984
NCI-H322 CTRP2 8.6159 13.9952 6.3026 13.3474
NCI-H1623 CTRP2 8.6163 12.119 7.2321 9.5057
NCI-H2085 CTRP2 8.6219 15.8688 5.3752 16.9923
Calu-6 CTRP2; CTRP1 8.6239 9.4334 8.4964 4.3329
NCI-H2073 CTRP1 8.6348 9.3686 8.5326 8.9951
SCLC-21H CTRP1 8.6388 9.2464 8.5762 8.6247
NCI-H292 CTRP2 8.6485 9.2075 8.5969 3.888
NCI-H1838 CTRP2 8.6494 9.6146 8.4527 4.4296
HCC1359 CTRP1 8.6523 9.0908 8.6292 8.1293
NCI-H358 CTRP2; CTRP1 8.6652 9.5863 8.4808 4.2775
SK-LU-1 CTRP2; CTRP1 8.6705 9.5024 8.5216 4.1363
IA-LM CTRP2 8.683 10.0114 8.313 4.8963
RERF-LC-Ad2 CTRP2 8.6902 9.2951 8.6161 3.6925
Calu-1 CTRP2 8.7446 9.1055 8.7257 3.1312
CAL-12T CTRP2; CTRP1 8.7602 9.4403 8.6413 3.4278
BEN CTRP2; CTRP1 8.8014 9.1398 8.7805 2.7598
COR-L23 CTRP1 8.8466 9.3857 8.7545 5.903
HCC15 CTRP2; CTRP1 8.8517 10.3192 8.3341 4.4351
RERF-LC-Ad1 CTRP2 9.0708 9.4948 8.937 1.4135
HCC2279 CTRP2 9.0724 17.4139 4.9893 17.4877
T3M-10 CTRP2; CTRP1 9.1036 14.2438 6.6036 11.1363
NCI-H2110 CTRP2; CTRP1 9.1747 13.5192 7.0255 9.2433
NCI-H1299 CTRP2; CTRP1 9.1769 13.8931 6.8373 9.9973
NCI-H2405 CTRP2; CTRP1 9.2629 14.6253 6.5426 11.0503
HCC2108 CTRP2; CTRP1 9.5002 15.7425 6.182 12.0927
NCI-H23 CTRP2; CTRP1 9.5918 16.2384 6.0049 12.6047
COLO 699 CTRP2; CTRP1 9.6093 18.274 5.006 16.3942
NCI-H2030 CTRP2; CTRP1 10.2915 16.355 6.4935 9.4392
Hs 888.Lu CTRP2 8.5284 12.9934 6.7208 11.8189
⏷ Show the Full List of 157 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 45 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 6.5713 11.4776 5.501 21.4873
JHOS-4 CTRP1 4.9349 7.0367 4.058 11.3195
OVMANA CTRP1 5.1057 7.4844 3.9844 11.2136
COV318 CTRP1 5.2019 6.3051 4.6553 4.9198
OC 314 CTRP2 5.6264 6.1312 5.6264 23.8535
RMUG-S CTRP1 6.8129 12.136 5.4659 40.3552
A2780 CTRP2; CTRP1 6.9391 9.8894 6.5176 16.6438
COV434 CTRP2; CTRP1 7.1118 9.4557 6.8485 14.9106
OAW28 CTRP2 7.2168 12.8372 5.5489 19.5968
TYK-nu CTRP2; CTRP1 7.4737 9.1864 7.3214 12.0996
OV-90 CTRP2; CTRP1 7.5101 10.2132 7.0092 13.1626
MCAS CTRP2 7.7105 11.577 6.6226 14.1327
TOV-21G CTRP2 7.839 10.8272 7.0914 11.933
SNU-119 CTRP2 7.92 11.8608 6.6974 13.3147
OVCAR-8 CTRP2; CTRP1 8.0448 9.1929 7.9429 8.1178
OVKATE CTRP1 8.1884 9.8931 7.8553 17.2143
OVSAHO CTRP2 8.2682 9.5717 8.0632 6.9843
RMG-I CTRP2; CTRP1 8.2832 13.6775 6.1633 14.6636
HEY A8 CTRP2; CTRP1 8.3238 11.0602 7.4693 9.1993
OVCAR-4 CTRP2; CTRP1 8.335 11.3332 7.353 9.676
DOV13 CTRP2 8.3367 10.5143 7.7361 8.0863
OVCAR-5 CTRP2 8.3398 9.1471 8.2759 5.9871
Caov-3 CTRP2; CTRP1 8.3836 9.3404 8.2693 5.9096
ONCO-DG-1 CTRP2 8.4021 10.1665 7.9591 7.0275
Kuramochi CTRP2 8.4446 12.46 6.907 11.2342
ES2 CTRP2 8.4582 12.8201 6.7425 11.8833
TOV-112D CTRP2 8.4642 12.3652 6.9715 10.9235
IGROV-1 CTRP2; CTRP1 8.4755 9.7283 8.2249 5.8173
OV56 CTRP2 8.483 8.9954 8.4628 4.879
JHOS-2 CTRP2 8.4982 14.7418 5.8273 15.5078
SNU-8 CTRP2 8.5056 9.0315 8.4811 4.7431
OV7 CTRP2; CTRP1 8.531 9.0992 8.496 4.6422
OAW42 CTRP2; CTRP1 8.5461 9.2298 8.4799 4.6529
JHOM-1 CTRP2; CTRP1 8.5483 9.0568 8.5231 4.4922
SNU-840 CTRP2; CTRP1 8.617 9.2761 8.5435 4.2082
JHOC-5 CTRP2; CTRP1 8.6246 9.0846 8.6005 3.9802
OVISE CTRP2 8.6781 9.3167 8.5959 3.803
FU-OV-1 CTRP2 8.7241 10.4904 8.1275 5.5523
COV644 CTRP2; CTRP1 8.7876 9.9255 8.4591 4.0766
SK-OV-3 CTRP2; CTRP1 8.834 14.7179 6.1333 13.5764
EFO-21 CTRP2; CTRP1 8.8791 9.6949 8.6542 3.0311
OVK18 CTRP2; CTRP1 8.9415 14.6575 6.2591 12.8726
COV362 CTRP2; CTRP1 8.9649 9.6987 8.7399 2.5037
EFO-27 CTRP2; CTRP1 9.2545 11.0631 8.3199 3.654
OVTOKO CTRP2 9.3092 16.0261 5.8806 13.6349
⏷ Show the Full List of 45 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SYO-1 CTRP2 8.5663 9.2527 8.4943 4.5088
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 8.728 9.2144 8.6818 3.853
Cancer Drug Sensitivity Data Curated from 23 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Yamato-SS CTRP2 8.7623 9.1812 8.7281 3.0673
Aska-SS CTRP2 8.7641 9.1983 8.7256 3.071
TTC-709 CTRP2 6.2336 13.0546 4.4644 26.1068
G-401 CTRP2; CTRP1 6.3358 9.3874 6.022 20.228
A-204 CTRP2 6.6287 8.9505 6.4586 17.7618
SK-LMS-1 CTRP2 6.8671 11.051 5.9889 18.8282
Rh41 CTRP2 7.2256 9.5623 6.9376 14.2174
KYM-1 CTRP2 7.538 8.7586 7.4852 11.2903
TE 617.T CTRP2 7.8803 10.4767 7.287 11.0513
SK-UT-1 CTRP2 8.167 13.3782 6.2005 14.7492
BT-12 CTRP2 8.2497 10.7909 7.5221 9.1662
BT-16 CTRP2 8.3223 9.2785 8.2205 6.2407
RKN CTRP2; CTRP1 8.4002 9.0088 8.3718 5.4902
GCT CTRP2 8.4294 9.521 8.2552 5.7991
HT-1080 CTRP2; CTRP1 8.4303 12.8511 6.7045 12.1288
TE 441.T CTRP2 8.524 12.5185 6.9511 10.8757
MES-SA CTRP2 8.5466 9.0702 8.5182 4.4837
Rh18 CTRP2 8.5987 9.3434 8.5008 4.389
Tm87-16 CTRP2 8.6709 9.2506 8.609 3.7759
Hs 729.T CTRP2 8.7568 14.6245 6.113 13.8188
SW982 CTRP2 8.9037 9.4242 8.7981 2.3967
G-402 CTRP2 9.1433 14.6705 6.4204 11.7851
RD CTRP2 10.9044 19.3637 5.4626 12.4115
⏷ Show the Full List of 23 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H CTRP2; CTRP1 7.4085 10.6984 6.7023 14.6009
NCI-H2452 CTRP2 8.0087 10.0269 7.6097 9.4457
ACC-MESO-1 CTRP2 8.2374 15.0081 5.462 17.4998
NCI-H2052 CTRP2; CTRP1 8.4011 9.1007 8.3538 5.5199
IST-Mes1 CTRP2 8.5697 11.6992 7.3954 8.931
NCI-H28 CTRP2; CTRP1 8.6029 12.8443 6.8618 11.0736
MPP 89 CTRP2 8.6174 9.2794 8.5418 4.1821
JL-1 CTRP2 8.7169 9.0912 8.6984 3.3144
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 5 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
LNCaP clone FGC CTRP2 7.6314 10.2554 7.1191 12.3768
PaCa-3 CTRP2; CTRP1 8.4648 9.0222 8.4387 5.0207
DU145 CTRP2 8.5364 12.4022 7.0197 10.5638
VCaP CTRP2 8.607 10.1969 8.1519 5.7353
22Rv1 CTRP2 8.6879 14.0425 6.3426 13.0317
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-15 CTRP2 8.4222 11.9644 7.1285 10.3689
A-253 CTRP2 8.5798 10.6301 7.922 6.7363
Cancer Drug Sensitivity Data Curated from 33 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HGC-27 CTRP2 6.2984 7.9379 6.2686 19.4743
SNU-1 CTRP2 6.812 9.2173 6.59 16.7272
GSS CTRP2 6.9229 9.0572 6.7532 15.8009
ECC10 CTRP2 7.5125 8.4227 7.4988 11.3264
SNU-5 CTRP2 7.5237 9.9509 7.1234 12.66
KE-39 CTRP2 7.8291 9.753 7.5247 10.2722
MKN1 CTRP2 7.8663 10.9127 7.0812 11.9037
SNU-216 CTRP2 8.0444 9.333 7.9012 8.2407
NCI-N87 CTRP2 8.086 10.1049 7.6587 9.0452
SNU-16 CTRP2 8.1894 9.8266 7.8813 7.9003
GSU CTRP2 8.2612 8.9906 8.2246 6.4145
MKN7 CTRP2; CTRP1 8.2772 13.1711 6.4038 13.6762
Fu97 CTRP2; CTRP1 8.3124 10.9201 7.524 9.0041
MKN74 CTRP2; CTRP1 8.3287 12.2068 6.923 11.4297
23132/87 CTRP2 8.3411 10.1664 7.8967 7.4337
NUGC-3 CTRP2 8.3445 17.105 4.5166 20.6894
SNU-668 CTRP2 8.379 9.7445 8.1148 6.4772
AGS CTRP2; CTRP1 8.4646 9.0972 8.4242 5.1034
SNU-601 CTRP2 8.5126 9.1912 8.453 4.8215
SNU-719 CTRP2 8.5134 12.7657 6.8196 11.4436
ECC12 CTRP2 8.5181 19.5535 3.4474 23.6915
SH-10-TC CTRP2; CTRP1 8.5321 13.0873 6.6778 11.9883
HuG1-N CTRP2 8.6076 9.3246 8.5167 4.3038
NUGC-4 CTRP2; CTRP1 8.6096 9.506 8.4537 4.5354
Hs 746.T CTRP2 8.7359 9.3709 8.6397 3.4713
SNU-620 CTRP2 8.737 9.232 8.6865 3.2949
MKN45 CTRP2 8.8291 9.2776 8.7728 2.7037
KATO III CTRP2 8.9501 10.4272 8.37 4.0347
LMSU CTRP2 10.4163 15.8881 6.811 7.9303
IM95 CTRP2 12.484 34.9969 -1.0709 26.6808
SNU-1077 CTRP2 7.6676 11.5771 6.5797 14.4123
SNU-685 CTRP2 8.5109 12.6463 6.8762 11.2144
SNG-M CTRP2; CTRP1 8.6407 13.0661 6.7859 11.3072
⏷ Show the Full List of 33 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 12 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
8505C CTRP2 8.0308 12.0756 6.703 13.0257
FTC-133 CTRP2 8.4001 10.8846 7.6267 8.3735
CGTH-W-1 CTRP2 8.4258 11.8131 7.2055 10.0429
FTC-238 CTRP2 8.5227 13.4566 6.4866 12.7956
TT2609-C02 CTRP2 8.5663 10.3088 8.0596 6.2092
SW579 CTRP2 8.5876 14.2706 6.1406 14.0645
8305C CTRP2 8.6765 9.2482 8.6158 3.7343
TT CTRP2 8.909 15.7816 5.6666 15.2733
BHT-101 CTRP2 9.0615 10.6736 8.3477 3.8901
ML-1 [Human leukemia] CTRP2 9.2172 10.7155 8.4596 3.1089
CAL-62 CTRP2 9.3791 10.7309 8.5816 2.3021
B-CPAP CTRP2 9.4738 21.7633 3.1481 22.603
⏷ Show the Full List of 12 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Detroit 562 CTRP2 6.8198 9.613 6.48 17.1057
SNU-1214 CTRP2 7.6875 12.2149 6.3032 15.4687
YD-10B CTRP2 8.1103 12.2324 6.7041 12.833
HSC-3 CTRP2 8.1257 11.2646 7.1791 10.8605
HSC-4 CTRP2 8.2256 12.6355 6.6178 12.9187
HSC-2 CTRP2; CTRP1 8.2749 12.9846 6.4931 13.3168
SNU-46 CTRP2 8.3826 15.9883 5.1056 18.5161
PE/CA-PJ34 (clone C12) CTRP2 8.4244 12.3119 6.9609 11.0565
CAL-33 CTRP2 8.5034 9.5457 8.3252 5.3237
SCC-25 CTRP2 8.5048 9.5409 8.3285 5.3074
SNU-1041 CTRP2 8.5214 14.1429 6.1452 14.1879
BHY CTRP2 8.5606 12.8986 6.7968 11.4348
PE/CA-PJ49 CTRP2 8.5625 9.0506 8.5391 4.3602
SCC-9 CTRP2; CTRP1 8.5878 9.3144 8.4997 4.4558
PE/CA-PJ41 (clone D2) CTRP2 8.6111 9.1527 8.5703 4.098
CAL-27 CTRP2 8.6154 9.1547 8.5745 4.0699
BICR 18 CTRP2 8.7301 10.5617 8.099 5.6555
BICR 6 CTRP2 8.7347 9.251 8.6784 3.3312
YD-8 CTRP2 8.7421 9.7996 8.4686 4.1225
BICR 56 CTRP2 8.7581 9.1526 8.7305 3.0719
BICR 22 CTRP2 8.7601 9.4006 8.6547 3.346
BICR 16 CTRP2 8.8125 9.337 8.7344 2.8953
SNU-899 CTRP2 8.8379 12.6499 7.1676 9.3006
BICR 31 CTRP2 8.8389 16.3074 5.344 16.6544
FaDu CTRP2 8.8572 12.6148 7.202 9.1166
SNU-1066 CTRP2 9.1755 14.1864 6.6894 10.6137
PE/CA-PJ15 CTRP2 9.5666 16.6373 5.7854 13.5166
SNU-1076 CTRP2 12.8493 22.4853 5.3006 10.1574
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 24 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
KMBC-2 CTRP1 3.2515 5.004 3.1251 28.2819
RT-4 CTRP2; CTRP1 5.3658 8.5737 5.1691 26.2641
HT-1376 CTRP2; CTRP1 6.1823 10.5767 5.4512 22.7729
U-BLC1 CTRP2 7.1351 8.91 7.0191 14.1966
UM-UC-3 CTRP2; CTRP1 7.1648 10.123 6.6743 15.3804
5637 CTRP2; CTRP1 7.8676 13.9182 5.6581 17.5887
UM-UC-1 CTRP2 8.021 10.8822 7.2513 10.8292
253J CTRP2 8.2145 9.1115 8.148 6.8312
JMSU-1 CTRP2 8.2275 10.804 7.494 9.3349
HT-1197 CTRP2 8.3846 12.3949 6.8834 11.466
KU-19-19 CTRP2 8.3982 9.6199 8.1844 6.1565
TCCSUP CTRP2 8.4071 12.4235 6.8903 11.387
RT-112 CTRP2 8.4781 12.4834 6.9263 11.0797
BC-3C CTRP2 8.6466 9.1716 8.6043 3.8667
SCaBER CTRP2 8.698 12.5806 7.0778 9.9713
647V CTRP2 8.7779 9.1706 8.7478 2.9491
253J-BV CTRP2 8.7843 10.1878 8.3302 4.5789
639V CTRP2 8.8032 9.2929 8.7396 2.9026
CAL-29 CTRP2 8.8843 9.7743 8.6228 3.1452
J82 CTRP2 8.9165 14.9895 6.0687 13.6674
BFTC-905 CTRP2 8.9964 9.7071 8.7641 2.2983
SW1710 CTRP2 8.9971 12.563 7.3494 8.2119
T24 CTRP2 9.2879 14.8112 6.4704 11.2986
VM-CUB-1 CTRP2 9.4419 14.3743 6.8148 9.5858
⏷ Show the Full List of 24 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HeLa CTRP2 5.8148 6.1586 5.8148 22.5976

References

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2 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Target id: 696).
3 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Target id: 702).
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