General Information of DTT (ID: TTJFY5U)

DTT Name Adenosine A3 receptor (ADORA3) DTT Info
UniProt ID
AA3R_HUMAN
Gene Name ADORA3

Molecule-Related Drug & Molecule List

Molecule-Related Drug List
Molecule Type:
DTT
DTP
DME
Drug Status:
Investigative Drug(s)
Discontinued Drug(s)
Clinical Trial Drug(s)
Preclinical Drug(s)
5 Clinical Trial Drug(s) Transported by This DTP
Drug Name Drug ID Indication ICD 11 Highest Status REF
IB-MECA DM9G5XD Psoriasis vulgaris EA90 Phase 3 [1], [2]
CF102 DMP56WJ Hepatocellular carcinoma 2C12.02 Phase 2 [3]
NITD609 DMQHBSX Malaria 1F40-1F45 Phase 2 [4]
Tonapofylline DMBH316 Acute and chronic heart failure BD1Z Phase 2 [5]
SCH-442416 DMQ2K1V N. A. N. A. Phase 1 [6]
------------------------------------------------------------------------------------
4 Discontinued Drug(s) Transported by This DTP
Drug Name Drug ID Indication ICD 11 Highest Status REF
BEMESETRON DMSPJX9 N. A. N. A. Discontinued in Phase 3 [7]
Dizocilpine DMMGYXR Cerebrovascular ischaemia 8B1Z Terminated [7]
Methylthioadenosine DMC8J6F Multiple sclerosis 8A40 Terminated [9]
METRIFUDIL DMS5CZ4 N. A. N. A. Terminated [10]
------------------------------------------------------------------------------------
3 Preclinical Drug(s) Transported by This DTP
Drug Name Drug ID Indication ICD 11 Highest Status REF
BAY 60-6583 DMTEJV1 Myocardial ischemia BA6Z Preclinical [8]
CF502 DMQSJ20 Inflammation 1A00-CA43.1 Preclinical [3]
CF602 DM0ULO2 Inflammation 1A00-CA43.1 Preclinical [3]
------------------------------------------------------------------------------------
209 Investigative Drug(s) Transported by This DTP
Drug Name Drug ID Indication ICD 11 Highest Status REF
(+)-BUTACLAMOL DMX6UYN Discovery agent N.A. Investigative [7]
(2R,3S)-3-(6-Amino-purin-9-yl)-nonan-2-ol DM852Z6 Discovery agent N.A. Investigative [11]
(E)-8-(3-chlorostyryl)-caffeine DMQT15Z Discovery agent N.A. Investigative [12]
(R,S)-PHPNECA DMQO71C Discovery agent N.A. Investigative [13]
(S)-PIA DM04BHI Discovery agent N.A. Investigative [14]
1,2-dihydro-2-oxoquinazoline-4-carboxyanilide DM542I9 Discovery agent N.A. Investigative [15]
1-(2-(diethylamino)quinazolin-4-yl)-3-phenylurea DMU5BOW Discovery agent N.A. Investigative [16]
1-Allyl-3,7-dihydro-purine-2,6-dione DML54H2 Discovery agent N.A. Investigative [17]
1-Benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione DMYGZ8V Discovery agent N.A. Investigative [18]
1-Benzyl-3-methyl-3,7-dihydro-purine-2,6-dione DMMRV21 Discovery agent N.A. Investigative [17]
1-Butyl-3,7-dihydro-purine-2,6-dione DMOE2ZV Discovery agent N.A. Investigative [17]
1-Cyclopentyl-3,7-dihydro-purine-2,6-dione DMEMQFH Discovery agent N.A. Investigative [17]
1-Phenethyl-3,7-dihydro-purine-2,6-dione DMA29SX Discovery agent N.A. Investigative [17]
1-phenyl-3-(2-(pyridin-2-yl)quinazolin-4-yl)urea DM9SKYC Discovery agent N.A. Investigative [16]
1-phenyl-3-(2-(pyridin-3-yl)quinazolin-4-yl)urea DMQKB6W Discovery agent N.A. Investigative [16]
1-phenyl-3-(3-(pyridin-2-yl)isoquinolin-1-yl)urea DMJNAX5 Discovery agent N.A. Investigative [16]
1-phenyl-3-(quinazolin-4-yl)urea DMZOEQY Discovery agent N.A. Investigative [16]
1-Prop-2-ynyl-3,7-dihydro-purine-2,6-dione DMCBX7R Discovery agent N.A. Investigative [17]
1-Propyl-3,7-dihydro-purine-2,6-dione DML5J94 Discovery agent N.A. Investigative [17]
2'-Me-CCPA DMDFPGB Discovery agent N.A. Investigative [19]
2,5'-dichloro-5'-deoxy-N6-cyclopentyladenosine DMMESIU Discovery agent N.A. Investigative [20]
2,6,8-triphenyl-9H-purine DM4IFPQ Discovery agent N.A. Investigative [21]
2,6-bis(4-chlorophenyl)-9H-purine DMYQNK0 Discovery agent N.A. Investigative [21]
2,6-bis(4-methoxyphenyl)-9H-purine DMC2N80 Discovery agent N.A. Investigative [21]
2,6-bis(4-tolyl)-9H-purine DM41RZX Discovery agent N.A. Investigative [21]
2,6-diphenyl-1-deazapurine DMW2VZ1 Discovery agent N.A. Investigative [22]
2,6-diphenyl-8-(1-ethylpropyl)-1-deazapurine DMY3C78 Discovery agent N.A. Investigative [22]
2,6-diphenyl-8-ethyl-1-deazapurine DM0C8BW Discovery agent N.A. Investigative [22]
2,6-diphenyl-8-methyl-1-deazapurine DMI79FV Discovery agent N.A. Investigative [22]
2,6-diphenyl-8-tButyl-1-deazapurine DM6D1BQ Discovery agent N.A. Investigative [22]
2,6-diphenyl-9H-purine DM5SXYI Discovery agent N.A. Investigative [21]
2,6-dphenyl-8-propyl-1-deazapurine DM8F9KO Discovery agent N.A. Investigative [22]
2-(1H-benzo[d]imidazol-2-yl)quinoxaline DM0Y2P1 Discovery agent N.A. Investigative [23]
2-(1H-imidazo[4,5-c]pyridin-2-yl)quinoxaline DMXA20E Discovery agent N.A. Investigative [24]
2-(2''-indolylethyloxy)adenosine DMCLIN8 Discovery agent N.A. Investigative [25]
2-(3''(5''-chloro-indolyl)ethyloxy)adenosine DMD8Q3E Discovery agent N.A. Investigative [25]
2-(3''(7''-bromo-indolyl)ethyloxy)adenosine DMITEND Discovery agent N.A. Investigative [25]
2-(3''-(4''-bromo-indolyl)ethyloxy)adenosine DMXRHOY Discovery agent N.A. Investigative [25]
2-(3''-(5''-bromo-indolyl)ethyloxy)adenosine DMR8PGZ Discovery agent N.A. Investigative [25]
2-(3''-(5''-fluoro-indolyl)ethyloxy)adenosine DME3IN1 Discovery agent N.A. Investigative [25]
2-(3''-(5''-hydroxyindolyl)ethyloxy)adenosine DM6BIOP Discovery agent N.A. Investigative [25]
2-(3''-(5''-iodo-indolyl)ethyloxy)adenosine DMFP0IW Discovery agent N.A. Investigative [25]
2-(3''-(5''-methoxy-indolyl)ethyloxy)adenosine DMWA0MN Discovery agent N.A. Investigative [25]
2-(3''-(6''-bromo-indolyl)ethyloxy)adenosine DMGRC24 Discovery agent N.A. Investigative [25]
2-(3''-(6''-chloro-indolyl)ethyloxy)adenosine DML39UW Discovery agent N.A. Investigative [25]
2-(3''-(benzoimidazole-1''-yl)ethyloxy)adenosine DMLDOH6 Discovery agent N.A. Investigative [25]
2-(3''-(benzotriazole-1''-yl)ethyloxy)adenosine DM1KCUV Discovery agent N.A. Investigative [25]
2-(3''-indolylethyloxy)adenosine DMXRAE3 Discovery agent N.A. Investigative [25]
2-(3''-pyrrolylethyloxy)adenosine DMNCP8Y Discovery agent N.A. Investigative [25]
2-(4-chloro-1H-benzo[d]imidazol-2-yl)quinoxaline DM7BHYS Discovery agent N.A. Investigative [24]
2-(4-chlorophenyl)-6-phenyl-9H-purine DMAPWNR Discovery agent N.A. Investigative [21]
2-(4-ethylthiobenzimidazol-2-yl)quinoxaline DMTAVU5 Discovery agent N.A. Investigative [24]
2-(4-hydroxypent-1-yl)-N6-methoxyadenosine DM1C864 Discovery agent N.A. Investigative [26]
2-(4-methoxyphenyl)-6-phenyl-9H-purine DMXTHOV Discovery agent N.A. Investigative [21]
2-(4-methyl-1H-benzo[d]imidazol-2-yl)quinoxaline DMDXIN1 Discovery agent N.A. Investigative [23]
2-(4-nitro-1H-benzo[d]imidazol-2-yl)quinoxaline DMBJICP Discovery agent N.A. Investigative [24]
2-(5-chloro-1H-benzo[d]imidazol-2-yl)quinoxaline DM0ZB89 Discovery agent N.A. Investigative [24]
2-(5-cyano-1-pent-1-ynyl)-N6-methoxyadenosine DMSIJ17 Discovery agent N.A. Investigative [26]
2-(hex-1-ynyl)-N6-methoxyadenosine DM7YLTS Discovery agent N.A. Investigative [26]
2-acetylaminoquinazoline-4-carboxyanilide DM0NJYZ Discovery agent N.A. Investigative [15]
2-aminoquinazoline-4-carboxy-(4-bromophenyl)amide DMJW4CS Discovery agent N.A. Investigative [15]
2-aminoquinazoline-4-carboxyanilide DMQJYX7 Discovery agent N.A. Investigative [15]
2-azido-N6-methyl-9-(beta-D-ribofuranosyl)adenine DMBSDIV Discovery agent N.A. Investigative [27]
2-benzoylaminoquinazoline-4-carboxyanilide DMGEFQP Discovery agent N.A. Investigative [15]
2-benzyl-2H-pyrazolo[3,4-c]quinolin-4(5H)-one DM6E04T Discovery agent N.A. Investigative [28]
2-chloro-2'-C-methyl-tecadenoson DMD3ZNP Discovery agent N.A. Investigative [29]
2-chloroadenosine DMYPQEW Discovery agent N.A. Investigative [12]
2-ethyl-4-(thiazol-2-yl)thieno[3,2-d]pyrimidine DMWCGE8 Discovery agent N.A. Investigative [30]
2-ethynyl-N6-methoxyadenosine DM2D78W Discovery agent N.A. Investigative [26]
2-Phenyl-2H-pyrazolo[4,3-c]quinoline DMAHI7G Discovery agent N.A. Investigative [31]
2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one DMQXCIK Discovery agent N.A. Investigative [32]
2-phenylethylyl-adenosine derivative DMW3F5C Discovery agent N.A. Investigative [33]
2-phenylpropoxyadenosine DMZQCEP Discovery agent N.A. Investigative [25]
2-tolyl-6-phenyl-9H-purine DM1HABS Discovery agent N.A. Investigative [21]
2-[(4-acetylphenyl)ethynyl]-N6-methoxyadenosine DMKC1GI Discovery agent N.A. Investigative [26]
2-[(4-fluorophenyl)ethynyl]-N6-methoxyadenosine DMTNQZU Discovery agent N.A. Investigative [26]
3-(3-chloro-1H-pyrazol-5-yl)quinoxalin-2(1H)-one DMI2RH1 Discovery agent N.A. Investigative [23]
3-Methyl-1-phenethyl-3,7-dihydro-purine-2,6-dione DMKYPUW Discovery agent N.A. Investigative [17]
3-noradamantyl-1,3-dipropylxanthine DMFHYAE Discovery agent N.A. Investigative [34]
4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one DMM9X0G Discovery agent N.A. Investigative [35]
4-Ethoxy-7-((E)-styryl)-furo[3,2-g]chromen-5-one DM8642Z Discovery agent N.A. Investigative [36]
4-Methoxy-2-phenyl-2H-pyrazolo[4,3-c]quinoline DM97B2G Discovery agent N.A. Investigative [31]
4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide DMFKN1M Discovery agent N.A. Investigative [37]
5,6,7-Trimethyl-2-p-tolyl-chromen-4-one DM6VPF4 Discovery agent N.A. Investigative [38]
5,7-dibromo-9H-pyrido[3,4-b]indol-6-ol DMZLOVB Discovery agent N.A. Investigative [39]
5,7-diphenyl-3H-imidazo[4,5-b]pyridin-2-ol DM4TIXY Discovery agent N.A. Investigative [22]
5-Butyl-8-phenyl-3H-[1,2,4]triazolo[5,1-i]purine DM2EPFZ Discovery agent N.A. Investigative [40]
6-ethylamino-2-(3''-indolyl)ethyloxy)adenosine DME4GBS Discovery agent N.A. Investigative [25]
6-guanidino-2-(3''-indolylethyloxy)adenosine DMM86PK Discovery agent N.A. Investigative [25]
6-Hydroxy-5,7-dimethyl-beta-carboline DM0CVTI Discovery agent N.A. Investigative [39]
8-Bromo-9-(3-hydroxypropyl)-9H-adenine DMA258T Discovery agent N.A. Investigative [41]
8-Bromo-9-(sec-butyl)-9H-adenine DMSQPFM Discovery agent N.A. Investigative [41]
8-Bromo-9-cyclobutyl-9H-adenine DMUTV76 Discovery agent N.A. Investigative [41]
8-Bromo-9-cyclohexyl-9H-adenine DMLVCON Discovery agent N.A. Investigative [41]
8-Bromo-9-cyclopentyl-9H-adenine DMCK0O1 Discovery agent N.A. Investigative [41]
8-bromo-9-isobutyl-9H-purin-6-amine DMZF3UN Discovery agent N.A. Investigative [42]
8-Bromo-9-isopropyl-9H-adenine DMIN9HC Discovery agent N.A. Investigative [41]
8-Hydroxy-5,7,9-trimethyl-delta-carboline DMG4W2C Discovery agent N.A. Investigative [39]
8-Hydroxy-7,9-dimethyl-delta-carboline DMFL46R Discovery agent N.A. Investigative [39]
8-PHENYL THEOPHYLLINE DMFGUCY Discovery agent N.A. Investigative [43]
8-propyl-2,6-diphenyl-9H-purine DMT6YUF Discovery agent N.A. Investigative [21]
9-Cyclopentyl-9H-adenine DMSGU2L Discovery agent N.A. Investigative [41]
9-Ethyl-8-phenylethynyl-9H-purin-6-ylamine DMRVS2D Discovery agent N.A. Investigative [44]
9H-purine derivative DMF1XLZ Discovery agent N.A. Investigative [7]
AB-MECA DMQPHFU Discovery agent N.A. Investigative [14]
ACN-1052 DM3E4QR Glaucoma/ocular hypertension 9C61 Investigative [45]
ATL802 DMYMCQA Discovery agent N.A. Investigative [46]
CIRSIMARITIN DMA3N9R Discovery agent N.A. Investigative [38]
CP608,039 DMTKO7P Discovery agent N.A. Investigative [47]
Cyclohexyl-(2-phenoxy-9H-purin-6-yl)-amine DM84ZX5 Discovery agent N.A. Investigative [48]
Cyclohexyl-(2-phenylsulfanyl-9H-purin-6-yl)-amine DMLREDJ Discovery agent N.A. Investigative [48]
Ethyl 5-benzoyl-4-phenylthiazol-2-ylcarbamate DMK4T5Y Discovery agent N.A. Investigative [5]
Flavone DMEQH6J Discovery agent N.A. Investigative [36], [38]
Galangin DM5TQ2O Discovery agent N.A. Investigative [38]
GNF-PF-2224 DM26UKN Discovery agent N.A. Investigative [49]
Hexanoic Acid (2,6-diphenylpyrimidin-4-yl)amide DMJOZYG Discovery agent N.A. Investigative [50]
I-ABA DMIJ2GV Discovery agent N.A. Investigative [51]
I-ABOPX DM5X0JS Discovery agent N.A. Investigative [51]
isobutylmethylxanthine DM46F5X Discovery agent N.A. Investigative [43]
KF26777 DMPBDW0 Discovery agent N.A. Investigative [52]
L-249313 DMEK65F Discovery agent N.A. Investigative [53]
LUF-5417 DMUPQED Discovery agent N.A. Investigative [5]
LUF-5433 DME4O5D Discovery agent N.A. Investigative [5]
LUF-5767 DMP08QO Discovery agent N.A. Investigative [50]
LUF-5816 DMQZDMH Discovery agent N.A. Investigative [22]
LUF-5833 DMDHUL8 Ischemia 8B10-8B11 Investigative [45]
LUF-5956 DMG4YWM Discovery agent N.A. Investigative [21]
LUF-5957 DMJFMH9 Discovery agent N.A. Investigative [21]
LUF-5962 DMR6LIE Discovery agent N.A. Investigative [21]
LUF-5978 DMCTM3L Discovery agent N.A. Investigative [22]
LUF-5980 DMGOIF5 Discovery agent N.A. Investigative [22]
LUF-5981 DMHO3XL Discovery agent N.A. Investigative [22]
MESULERGINE DMKGWAH Discovery agent N.A. Investigative [7]
METHOCTRAMINE DMH2CKX Discovery agent N.A. Investigative [7]
MPC-MECA DMONDP1 Discovery agent N.A. Investigative [14]
MRE 2029F20 DMUK1PA Discovery agent N.A. Investigative [54]
MRE 3008F20 DM72US0 Discovery agent N.A. Investigative [14], [55]
MRE 3010F20 DMMFJA8 Discovery agent N.A. Investigative [14]
MRS-1220 DMT6JH9 Discovery agent N.A. Investigative [56]
MRS1041 DMBXKYR Discovery agent N.A. Investigative [36]
MRS1042 DMVT865 Discovery agent N.A. Investigative [36]
MRS1067 DMAEW9M Discovery agent N.A. Investigative [57]
MRS1088 DMSKWL7 Discovery agent N.A. Investigative [36]
MRS1093 DM801AO Discovery agent N.A. Investigative [36]
MRS1097 DMLOHAZ Discovery agent N.A. Investigative [58]
MRS1177 DMBXTPU Discovery agent N.A. Investigative [59]
MRS1186 DMGJ0IE Discovery agent N.A. Investigative [59]
MRS1191 DM9WX3C Discovery agent N.A. Investigative [45]
MRS1476 DMLQYN7 Discovery agent N.A. Investigative [60]
MRS1486 DMFJHMQ Discovery agent N.A. Investigative [60]
MRS1505 DM3Q5NO Discovery agent N.A. Investigative [60]
MRS1523 DM4AONZ Discovery agent N.A. Investigative [60]
MRS5151 DM1GUTC Discovery agent N.A. Investigative [61]
MRS5698 DMDF6WG Discovery agent N.A. Investigative [62]
MRS928 DMKJ9WM Discovery agent N.A. Investigative [36], [38]
N(6)-cyclohexyladenosine DMHINE0 Discovery agent N.A. Investigative [63]
N*2*-Benzyl-N*6*-cyclohexyl-9H-purine-2,6-diamine DM41TQB Discovery agent N.A. Investigative [48]
N*6*-Cyclohexyl-N*2*-ethyl-9H-purine-2,6-diamine DM1K2A4 Discovery agent N.A. Investigative [48]
N*6*-Cyclohexyl-N*2*-phenyl-9H-purine-2,6-diamine DM3C8PJ Discovery agent N.A. Investigative [48]
N*6*-Cyclooctyl-N*2*-phenyl-9H-purine-2,6-diamine DMCOPR3 Discovery agent N.A. Investigative [48]
N-(2,6-diphenylpyrimidin-4-yl)-3-methylbutyramide DM6HGK4 Discovery agent N.A. Investigative [50]
N-(2,6-diphenylpyrimidin-4-yl)acetamide DMQ0DMU Discovery agent N.A. Investigative [50]
N-(2,6-diphenylpyrimidin-4-yl)benzamide DMBW752 Discovery agent N.A. Investigative [50]
N-(2,6-diphenylpyrimidin-4-yl)butyramide DM5EF71 Discovery agent N.A. Investigative [50]
N-(2,6-diphenylpyrimidin-4-yl)isobutyramide DMWPZCS Discovery agent N.A. Investigative [50]
N-(2,6-diphenylpyrimidin-4-yl)propionamide DM89NGE Discovery agent N.A. Investigative [50]
N-(2-(furan-2-yl)-3,4'-bipyridin-6-yl)acetamide DMLTROU Discovery agent N.A. Investigative [64]
N-(4,5-diphenylpyrimidin-2-yl)acetamide DM34R10 Discovery agent N.A. Investigative [50]
N-(4,6-diphenylpyrimidin-2-yl)-4-chlorobenzamide DM1PSR7 Discovery agent N.A. Investigative [50]
N-(4,6-diphenylpyrimidin-2-yl)propionamide DMJZ2IP Discovery agent N.A. Investigative [50]
N-(5-Benzoyl-4-phenylthiazol-2-yl)benzamide DMTF8US Discovery agent N.A. Investigative [5]
N6-((+/-)-endo-norborn-2-yl)adenosine DM30KXV Discovery agent N.A. Investigative [20]
N6-(3-Iodobenzyl)-2'-O-methyladenosine DM2W9NO Discovery agent N.A. Investigative [65]
N6-cyclopentyladenosine DMD6AJO Discovery agent N.A. Investigative [66]
N6-methoxy-2-phenylethynyladenosine DMDG59X Discovery agent N.A. Investigative [26]
N6-methoxy-2-[(2-pyridinyl)ethynyl]adenosine DMSEL5W Discovery agent N.A. Investigative [26]
N6-methoxy-2-[(3-pyridinyl)ethynyl]-adenosine DMP7246 Discovery agent N.A. Investigative [26]
N6-methoxy-2-[(4-methoxyphenyl)ethynyl]adenosine DM8LR62 Discovery agent N.A. Investigative [26]
N6-methoxy-2-[(4-methylphenyl)ethynyl]adenosine DM1KA9R Discovery agent N.A. Investigative [26]
N6-methoxy-2-[(4-pentylphenyl)ethynyl]adenosine DMQ5K8R Discovery agent N.A. Investigative [26]
N6-methoxy-2-[(4-pyridinyl)ethynyl]adenosine DM9H3W8 Discovery agent N.A. Investigative [26]
N6-methoxy-2-[2-(trimethylsilyl)ethynyl]adenosine DMRBS50 Discovery agent N.A. Investigative [26]
NIPECOTIC ACID DMPV450 Discovery agent N.A. Investigative [7]
NSC-407228 DMKJWGP Discovery agent N.A. Investigative [38]
PENECA DMIDSJ9 Discovery agent N.A. Investigative [13]
PSB-10 DMXDWO7 Discovery agent N.A. Investigative [67]
PSB-11 DMGK2PC Discovery agent N.A. Investigative [68]
PSB36 DMBGM1E Discovery agent N.A. Investigative [69]
PSB603 DM6QERS Discovery agent N.A. Investigative [70]
R-N6-(phenylisopropyl)adenosine DM2N3BA Discovery agent N.A. Investigative [71], [25]
REVERSINE DMWDNOK Discovery agent N.A. Investigative [48]
sakuranetin DMUAQYZ Discovery agent N.A. Investigative [36]
SB-298 DMU2J3K Discovery agent N.A. Investigative [70]
Serotonin DMOFCRY Discovery agent N.A. Investigative [7]
TCPA DMTF4VI Discovery agent N.A. Investigative [72]
visnagin DMCSHE8 Discovery agent N.A. Investigative [36]
VUF-8504 DM8OTAG Discovery agent N.A. Investigative [16]
VUF-8507 DMQFWV7 Discovery agent N.A. Investigative [16]
VUF5574 DMUA751 Discovery agent N.A. Investigative [73]
xanthine amine congener DMGYVFD Discovery agent N.A. Investigative [14]
[1,2,4]triazolo[1,5-a]quinoxalin-4(5H)-one DMPV0QN Discovery agent N.A. Investigative [74]
[125I]AB-MECA DM8EQFL Discovery agent N.A. Investigative [14]
[125I]APNEA DM95A4Z Discovery agent N.A. Investigative [75]
[3H]CCPA DMHDGB3 Discovery agent N.A. Investigative [29]
[3H]HEMADO DMEO6AH Discovery agent N.A. Investigative [76]
[3H]kainate DMMK7XU Discovery agent N.A. Investigative [7]
[3H]NECA DMAO9SH Discovery agent N.A. Investigative [77], [78]
[3H]OSIP339391 DM4BY5J Discovery agent N.A. Investigative [42]
[3H]PSB-11 DMFDCJK Discovery agent N.A. Investigative [68]
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⏷ Show the Full List of 209 Investigative Drug(s)
Molecule Interaction Atlas

References

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11 Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors. J Med Chem. 1995 May 12;38(10):1720-35.
12 A binding site model and structure-activity relationships for the rat A3 adenosine receptor. Mol Pharmacol. 1994 Jun;45(6):1101-11.
13 N(6)-alkyl-2-alkynyl derivatives of adenosine as potent and selective agonists at the human adenosine A(3) receptor and a starting point for searching A(2B) ligands. J Med Chem. 2002 Jul 18;45(15):3271-9.
14 [(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors. Mol Pharmacol. 2000 May;57(5):968-75.
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16 Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. J Med Chem. 2006 Jul 13;49(14):4085-97.
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