Details of the Drug-Related molecule(s) Interaction Atlas

General Information of Drug (ID: DMTLRGZ)

Drug Name
SGC-CBP30 Drug Info
Synonyms
SGC-CBP30; 1613695-14-9; (s)-4-(1-(2-(3-chloro-4-methoxyphenethyl)-5-(3,5-dimethylisoxazol-4-yl)-1h-benzo[d]imidazol-1-yl)propan-2-yl)morpholine; 2-[2-(3-chloro-4-methoxyphenyl)ethyl]-5-(dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-1,3-benzodiazole; 2-[2-(3-Chloro-4-Methoxyphenyl)ethyl]-5-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-1-[(2s)-2-(Morpholin-4-Yl)propyl]-1h-Benzimidazole; 2LO; C28H33ClN4O3; GTPL7529; SCHEMBL17512896; CHEMBL3622373; AOB4800; MolPort-035-395-859; BDBM188519; EX-A2159; ZINC96170456; s7256
Indication
Disease Entry ICD 11 Status REF
Discovery agent N.A. Investigative [1]
Cross-matching ID
PubChem CID
72201027
TTD Drug ID
DMTLRGZ

Molecule-Related Drug Atlas

Molecule-Related Drug Atlas
Molecule Type:
DTT
DOT
Drug Status:
Clinical Trial Drug(s)
Patented Agent(s)
Investigative Drug(s)
Approved Drug(s)
Download the Complete Related Drug List
Drug(s) Targeting CREB-binding protein (CREBBP)
Drug Name Drug ID Indication ICD 11 Highest Status REF
C 82 DMEWXFK Scleroderma 4A42 Phase 1/2 [4]
CCS1477 DM9UZM1 Solid tumour/cancer 2A00-2F9Z Phase 1/2 [5]
PRI-724 DM0HTEF Acute myeloid leukaemia 2A60 Phase 1/2 [6]
FT-7051 DMCK3OI Prostate cancer 2C82.0 Phase 1 [7]
Pyrrolo-pyrrolone derivative 6 DMBW208 N. A. N. A. Patented [8]
I-CBP112 DMQX3W6 Discovery agent N.A. Investigative [9]
ischemin DMM2I9G Discovery agent N.A. Investigative [10]
⏷ Show the Full List of 7 Drug(s)
Drug(s) Targeting Histone acetyltransferase KAT6B (KAT6B)
Drug Name Drug ID Indication ICD 11 Highest Status REF
garcinol DM6B9ZG Discovery agent N.A. Investigative [11]
anacardic acid DMAS5BI Discovery agent N.A. Investigative [12]
I-CBP112 DMQX3W6 Discovery agent N.A. Investigative [13]
C646 DMCOQKH Discovery agent N.A. Investigative [14]
MG149 DM7V58G Discovery agent N.A. Investigative [15]
Drug(s) Affected By Interleukin-10 (IL10)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [16]
Nitric Oxide DM1RBYG Hypertension BA00-BA04 Approved [17]
Ribavirin DMEYLH9 Hepatitis C virus infection 1E51.1 Approved [18]
Methotrexate DM2TEOL Anterior urethra cancer Approved [19]
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [20]
Quercetin DM3NC4M Obesity 5B81 Approved [21]
Bisoprolol DM3UZ95 Hypertension BA00-BA04 Approved [22]
Tretinoin DM49DUI Acne vulgaris ED80 Approved [23]
Acetic Acid, Glacial DM4SJ5Y infection in the ear canal AA0Y Approved [24]
Isoniazid DM5JVS3 Latent tuberculosis infection Approved [25]
⏷ Show the Full List of 10 Drug(s)
Drug(s) Affected By Interleukin-17A (IL17A)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Methotrexate DM2TEOL Anterior urethra cancer Approved [26]
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [27]
Isoniazid DM5JVS3 Latent tuberculosis infection Approved [25]
Paroxetine DM5PVQE Anxiety disorder 6B00-6B0Z Approved [28]
Arsenic trioxide DM61TA4 Acute lymphoblastic leukaemia 2A85 Approved [29]
Calcitriol DM8ZVJ7 Congenital alopecia LC30 Approved [30]
Ethanol DMDRQZU Chronic pain MG30 Approved [31]
Arsenic DMTL2Y1 N. A. N. A. Approved [32]
Aspirin DM672AH Acute coronary syndrome BA41 Approved [33]
Resveratrol DM3RWXL Giant cell arteritis 4A44.2 Phase 3 [34]
⏷ Show the Full List of 10 Drug(s)
Drug(s) Affected By Interleukin-23 receptor (IL23R)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Methotrexate DM2TEOL Anterior urethra cancer Approved [35]
Tretinoin DM49DUI Acne vulgaris ED80 Approved [36]
(+)-JQ1 DM1CZSJ Testicular cancer 2C80 Phase 1 [37]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [38]
Glyphosate DM0AFY7 Malaria 1F40-1F45 Investigative [39]
NAPQI DM8F5LR Autoimmune disease 4A40-4A45 Investigative [40]
⏷ Show the Full List of 6 Drug(s)
Drug(s) Affected By Interleukin-22 (IL22)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [41]
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [42]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [43]
Dinoprostone DMTYOPD Medical abortion JA00.1Z Approved [44]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [38]
bisphenol A DM2ZLD7 Discovery agent N.A. Investigative [45]
⏷ Show the Full List of 6 Drug(s)
Drug(s) Affected By Interleukin-21 (IL21)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [27]
Folic Acid DMEMBJC Colorectal carcinoma Approved [46]
(+)-JQ1 DM1CZSJ Testicular cancer 2C80 Phase 1 [37]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [47]
Drug(s) Affected By T-box transcription factor TBX21 (TBX21)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Tretinoin DM49DUI Acne vulgaris ED80 Approved [48]
Dinoprostone DMTYOPD Medical abortion JA00.1Z Approved [44]
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [49]
Aspirin DM672AH Acute coronary syndrome BA41 Approved [50]
Budesonide DMJIBAW Allergic rhinitis CA08.0 Approved [51]
Urethane DM7NSI0 N. A. N. A. Phase 4 [52]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [38]
Formaldehyde DM7Q6M0 Discovery agent N.A. Investigative [53]
⏷ Show the Full List of 8 Drug(s)

Molecular Interaction Atlas of This Drug

Molecular Interaction Atlas
Download the Complete Interaction Atlas for Visualization in Cytoscape

Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
CREB-binding protein (CREBBP) TTFRCTK CBP_HUMAN Inhibitor [2]
Histone acetyltransferase KAT6B (KAT6B) TTH4VJL KAT6B_HUMAN Inhibitor [2]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Interleukin-10 (IL10) OTIRFRXC IL10_HUMAN Gene/Protein Processing [3]
Interleukin-17A (IL17A) OTY72FT2 IL17_HUMAN Gene/Protein Processing [3]
Interleukin-21 (IL21) OTABCY4W IL21_HUMAN Gene/Protein Processing [3]
Interleukin-22 (IL22) OTW31FU9 IL22_HUMAN Gene/Protein Processing [3]
Interleukin-23 receptor (IL23R) OTT6L7U8 IL23R_HUMAN Gene/Protein Processing [3]
T-box transcription factor TBX21 (TBX21) OT3UK5KE TBX21_HUMAN Gene/Protein Processing [3]

References

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