General Information of Drug (ID: DM08E9O)

Drug Name
Diazepam Drug Info
Synonyms
diazepam; Valium; 439-14-5; Diazemuls; Ansiolisina; Sibazon; Relanium; Faustan; Apaurin; Stesolid; Seduxen; Methyldiazepinone; Valitran; Tranqdyn; Seduksen; Relaminal; Quiatril; Quetinil; Dipezona; Diazetard; Diazepan; Calmpose; Tranimul; Tensopam; Serenack; Paranten; Kiatrium; Domalium; Condition; Bialzepam; Ansiolin; Unisedil; Stesolin; Serenamin; Ruhsitus; Renborin; Quievita; Tranquirit; Serenzin; Neurolytril; Liberetas; Diacepan; Ceregulart; Calmocitene; Bensedin; Atensine; Apozepam; Umbrium; Sonacon; Sedipam; Levium; Diapam; Atilen; Assival; Amiprol; Diazepam (intranasal, epilepsy)
Indication
Disease Entry ICD 11 Status REF
Alcohol withdrawal Approved [1]
Alcohol withdrawal delirium Approved [1]
Anxiety Approved [1]
Epilepsy 8A60-8A68 Approved [2]
Tetanus 1C13 Investigative [1]
Cross-matching ID
PubChem CID
3016
ChEBI ID
CHEMBL12
CAS Number
CAS 439-14-5
TTD Drug ID
DM08E9O
VARIDT Drug ID
DR00999
INTEDE Drug ID
DR0480
ACDINA Drug ID
D00190

Molecule-Related Drug Atlas

Molecule-Related Drug Atlas
Molecule Type:
DTT
DTP
DME
DOT
Drug Status:
Approved Drug(s)
Clinical Trial Drug(s)
Investigative Drug(s)
Drug(s) Targeting Translocator protein (TSPO)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Flunitrazepam DMGR5Z3 Insomnia 7A00-7A0Z Approved [19]
Oxazepam DMXNZM4 Alcohol withdrawal delirium Approved [20]
Midazolam DMXOELT Agitation 6A70.3 Approved [21]
Temazepam DM02A65 Insomnia 7A00-7A0Z Approved [21]
Flumazenil DMPCG2L Benzodiazepine overdose PC91 Approved [22]
Alprazolam DMC7XDN Anxiety Approved [19]
Clotiazepam DM59AZT Anxiety disorder 6B00-6B0Z Approved [23]
Quazepam DMY4D87 Insomnia 7A00-7A0Z Approved [21]
Eszopiclone DM8RZ9H Insomnia 7A00-7A0Z Approved [24]
Triazolam DMETYK5 Insomnia 7A00-7A0Z Approved [21]
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Drug(s) Transported By P-glycoprotein 1 (ABCB1)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Amoxicillin DMUYNEI Acute otitis media AB00 Approved [25]
Doxorubicin DMVP5YE Acute myelogenous leukaemia 2A41 Approved [26]
Methotrexate DM2TEOL Anterior urethra cancer Approved [27]
Folic Acid DMEMBJC Colorectal carcinoma Approved [28]
Fluorouracil DMUM7HZ Adenocarcinoma 2D40 Approved [27]
Cisplatin DMRHGI9 Adenocarcinoma 2D40 Approved [27]
Progesterone DMUY35B Amenorrhea GA20.0 Approved [4]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [27]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [29]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [30]
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Drug(s) Metabolized By Cytochrome P450 3A4 (CYP3A4)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Doxorubicin DMVP5YE Acute myelogenous leukaemia 2A41 Approved [31]
Progesterone DMUY35B Amenorrhea GA20.0 Approved [32]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [33]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [34]
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [35]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [36]
Etoposide DMNH3PG Acute myelogenous leukaemia 2A41 Approved [37]
Zidovudine DM4KI7O Human immunodeficiency virus infection 1C62 Approved [38]
Prasterone DM67VKL Chronic obstructive pulmonary disease CA22 Approved [32]
Verapamil DMA7PEW Angina pectoris BA40 Approved [13]
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Drug(s) Metabolized By Cytochrome P450 1A2 (CYP1A2)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Fluorouracil DMUM7HZ Adenocarcinoma 2D40 Approved [39]
Dinoprostone DMTYOPD Medical abortion JA00.1Z Approved [40]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [41]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [42]
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [43]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [44]
Etoposide DMNH3PG Acute myelogenous leukaemia 2A41 Approved [37]
Oxaliplatin DMQNWRD Adenocarcinoma 2D40 Approved [45]
Verapamil DMA7PEW Angina pectoris BA40 Approved [46]
Diclofenac DMPIHLS Chronic renal failure GB61.Z Approved [47]
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Drug(s) Metabolized By Cytochrome P450 3A5 (CYP3A5)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Doxorubicin DMVP5YE Acute myelogenous leukaemia 2A41 Approved [48]
Progesterone DMUY35B Amenorrhea GA20.0 Approved [49]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [50]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [12]
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [51]
Sulfasalazine DMICA9H Irritable bowel syndrome DD91.0 Approved [52]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [53]
Etoposide DMNH3PG Acute myelogenous leukaemia 2A41 Approved [54]
Verapamil DMA7PEW Angina pectoris BA40 Approved [55]
Sorafenib DMS8IFC Adenocarcinoma 2D40 Approved [12]
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Drug(s) Metabolized By Cytochrome P450 3A7 (CYP3A7)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Progesterone DMUY35B Amenorrhea GA20.0 Approved [56]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [12]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [12]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [12]
Prasterone DM67VKL Chronic obstructive pulmonary disease CA22 Approved [7]
Verapamil DMA7PEW Angina pectoris BA40 Approved [57]
Sorafenib DMS8IFC Adenocarcinoma 2D40 Approved [12]
Quinine DMSWYF5 Malaria 1F40-1F45 Approved [12]
Irinotecan DMP6SC2 Adenocarcinoma 2D40 Approved [12]
Metronidazole DMTIVEN Abscess Approved [58]
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Drug(s) Metabolized By Cytochrome P450 2C18 (CYP2C18)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Verapamil DMA7PEW Angina pectoris BA40 Approved [7]
Diclofenac DMPIHLS Chronic renal failure GB61.Z Approved [59]
Propofol DMB4OLE Anaesthesia 9A78.6 Approved [60]
Phenytoin DMNOKBV Epilepsy 8A60-8A68 Approved [7]
Tretinoin DM49DUI Acne vulgaris ED80 Approved [61]
Methadone DMTW6IU Advanced cancer 2A00-2F9Z Approved [62]
Dapsone DM4LT8A Acne vulgaris ED80 Approved [63]
Lidocaine DML4ZOT Anaesthesia 9A78.6 Approved [7]
Phenobarbital DMXZOCG Cluster headache 8A81.0 Approved [64]
Ifosfamide DMCT3I8 Adult central nervous system germ cell tumor Approved [65]
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Drug(s) Metabolized By Cytochrome P450 2C8 (CYP2C8)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Fluorouracil DMUM7HZ Adenocarcinoma 2D40 Approved [39]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [66]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [66]
Zidovudine DM4KI7O Human immunodeficiency virus infection 1C62 Approved [7]
Verapamil DMA7PEW Angina pectoris BA40 Approved [67]
Diclofenac DMPIHLS Chronic renal failure GB61.Z Approved [68]
Sorafenib DMS8IFC Adenocarcinoma 2D40 Approved [69]
Quinine DMSWYF5 Malaria 1F40-1F45 Approved [66]
Mycophenolate mofetil DMPQAGE Hepatosplenic T-cell lymphoma Approved [70]
Propofol DMB4OLE Anaesthesia 9A78.6 Approved [60]
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Drug(s) Metabolized By Cytochrome P450 2C9 (CYP2C9)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Progesterone DMUY35B Amenorrhea GA20.0 Approved [71]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [72]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [73]
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [7]
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [74]
Zidovudine DM4KI7O Human immunodeficiency virus infection 1C62 Approved [7]
Verapamil DMA7PEW Angina pectoris BA40 Approved [75]
Diclofenac DMPIHLS Chronic renal failure GB61.Z Approved [76]
Estrone DM5T6US Acne vulgaris ED80 Approved [77]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [78]
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Drug(s) Metabolized By Cytochrome P450 2B6 (CYP2B6)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [79]
Verapamil DMA7PEW Angina pectoris BA40 Approved [7]
Diclofenac DMPIHLS Chronic renal failure GB61.Z Approved [80]
Estrone DM5T6US Acne vulgaris ED80 Approved [73]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [81]
Irinotecan DMP6SC2 Adenocarcinoma 2D40 Approved [82]
Propofol DMB4OLE Anaesthesia 9A78.6 Approved [83]
Nicotine DMWX5CO Lung cancer 2C25.0 Approved [84]
Phenytoin DMNOKBV Epilepsy 8A60-8A68 Approved [85]
Amitriptyline DMK7F9S Depression 6A70-6A7Z Approved [86]
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Drug(s) Metabolized By Mephenytoin 4-hydroxylase (CYP2C19)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Amoxicillin DMUYNEI Acute otitis media AB00 Approved [87]
Progesterone DMUY35B Amenorrhea GA20.0 Approved [71]
Tamoxifen DMLB0EZ Breast cancer 2C60-2C65 Approved [88]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [89]
Zidovudine DM4KI7O Human immunodeficiency virus infection 1C62 Approved [7]
Verapamil DMA7PEW Angina pectoris BA40 Approved [90]
Diclofenac DMPIHLS Chronic renal failure GB61.Z Approved [59]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [78]
Quinine DMSWYF5 Malaria 1F40-1F45 Approved [91]
Propofol DMB4OLE Anaesthesia 9A78.6 Approved [60]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Imatinib DM7RJXL Acute lymphoblastic leukaemia 2A85 Approved [13]
Etoposide DMNH3PG Acute myelogenous leukaemia 2A41 Approved [92]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [13]
Dapsone DM4LT8A Acne vulgaris ED80 Approved [13]
Ifosfamide DMCT3I8 Adult central nervous system germ cell tumor Approved [13]
Nateglinide DMLK2QH Diabetic complication 5A2Y Approved [13]
Thalidomide DM70BU5 Adult T-cell leukemia/lymphoma Approved [13]
Ketobemidone DMM3L6Z Pain MG30-MG3Z Approved [13]
Irbesartan DMTP1DC Diabetic kidney disease GB61.Z Approved [13]
Terbinafine DMI6HUW Fungal infection 1F29-1F2F Approved [13]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Meclofenamic acid DM05FXR Ankylosing spondylitis FA92.0 Approved [93]
Ciclosporin DMAZJFX Graft-versus-host disease 4B24 Approved [94]
Benzbromarone DMC3YUA Gout FA25 Approved [95]
Flufenamic Acid DMC8VNH Dysmenorrhea GA34.3 Approved [95]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [96]
Nitrazepam DMEGIQ6 Epilepsy 8A60-8A68 Approved [16]
Flunitrazepam DMGR5Z3 Insomnia 7A00-7A0Z Approved [16]
Chenodiol DMQ8JIK Cholelithiasis DC11 Approved [97]
Gamolenic acid DMQN30Z Allergy 4A80-4A85 Approved [98]
Indomethacin DMSC4A7 Bursitis Approved [95]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Doxorubicin DMVP5YE Acute myelogenous leukaemia 2A41 Approved [99]
Meclofenamic acid DM05FXR Ankylosing spondylitis FA92.0 Approved [100]
Levonorgestrel DM1DP7T Atypical endometrial hyperplasia Approved [101]
Desogestrel DM27U4Y Contraception QA21 Approved [101]
Salicyclic acid DM2F8XZ Acne vulgaris ED80 Approved [100]
Sulindac DM2QHZU Acute myelogenous leukaemia 2A41 Approved [100]
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [102]
Quercetin DM3NC4M Obesity 5B81 Approved [103]
Tretinoin DM49DUI Acne vulgaris ED80 Approved [104]
Glimepiride DM5FSJA Diabetic complication 5A2Y Approved [105]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Meclofenamic acid DM05FXR Ankylosing spondylitis FA92.0 Approved [100]
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [106]
Salicyclic acid DM2F8XZ Acne vulgaris ED80 Approved [107]
Sulindac DM2QHZU Acute myelogenous leukaemia 2A41 Approved [100]
Quercetin DM3NC4M Obesity 5B81 Approved [108]
Arsenic trioxide DM61TA4 Acute lymphoblastic leukaemia 2A85 Approved [109]
Aspirin DM672AH Acute coronary syndrome BA41 Approved [100]
Liothyronine DM6IR3P Congenital hypothyroidism Approved [110]
Testosterone DM7HUNW Hot flushes GA30 Approved [111]
Glibenclamide DM8JXPZ Diabetic complication 5A2Y Approved [105]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Progesterone DMUY35B Amenorrhea GA20.0 Approved [112]
Meclofenamic acid DM05FXR Ankylosing spondylitis FA92.0 Approved [100]
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [113]
Salicyclic acid DM2F8XZ Acne vulgaris ED80 Approved [100]
Sulindac DM2QHZU Acute myelogenous leukaemia 2A41 Approved [100]
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [114]
Glimepiride DM5FSJA Diabetic complication 5A2Y Approved [105]
Ethacrynic acid DM60QMR Edema MG29 Approved [113]
Aspirin DM672AH Acute coronary syndrome BA41 Approved [100]
Liothyronine DM6IR3P Congenital hypothyroidism Approved [110]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Penicillamine DM40EF6 Cystinuria 5C60.2 Approved [115]
Cannabidiol DM0659E Dravet syndrome 8A61.11 Approved [116]
Beta-carotene DM0RXBT Vitamin deficiency 5B55-5B71 Approved [117]
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [118]
Methotrexate DM2TEOL Anterior urethra cancer Approved [119]
Ceruletide DM2WE5K Caerulein stimulated gastric and pancreatic secretion 5A4Y Approved [120]
Dactinomycin DM2YGNW Adult kidney Wilms tumor Approved [121]
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [122]
Quercetin DM3NC4M Obesity 5B81 Approved [123]
obeticholic acid DM3Q1SM Primary biliary cholangitis DB96.1 Approved [124]
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Drug(s) Affected By Albumin (ALB)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [125]
Sulfamethoxazole DMB08GE Acute otitis media AB00 Approved [115]
Tolbutamide DM02AWV Advanced cancer 2A00-2F9Z Approved [126]
Sertraline DM0FB1J Coronary heart disease BA80.Z Approved [127]
Methimazole DM25FL8 Hyperthyroidism 5A02 Approved [128]
Imipramine DM2NUH3 Depression 6A70-6A7Z Approved [129]
Colchicine DM2POTE Acute gout flare FA25.0 Approved [130]
Methotrexate DM2TEOL Anterior urethra cancer Approved [131]
Quercetin DM3NC4M Obesity 5B81 Approved [132]
obeticholic acid DM3Q1SM Primary biliary cholangitis DB96.1 Approved [124]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Fulvestrant DM0YZC6 Breast cancer 2C60-2C65 Approved [133]
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [134]
obeticholic acid DM3Q1SM Primary biliary cholangitis DB96.1 Approved [124]
Tretinoin DM49DUI Acne vulgaris ED80 Approved [135]
Marinol DM70IK5 Anorexia nervosa cachexia 6B80 Approved [136]
Testosterone DM7HUNW Hot flushes GA30 Approved [137]
Acocantherin DM7JT24 Atrial fibrillation BC81.3 Approved [138]
Calcitriol DM8ZVJ7 Congenital alopecia LC30 Approved [137]
Ciclosporin DMAZJFX Graft-versus-host disease 4B24 Approved [139]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [96]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Arsenic trioxide DM61TA4 Acute lymphoblastic leukaemia 2A85 Approved [140]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [96]
Flunitrazepam DMGR5Z3 Insomnia 7A00-7A0Z Approved [141]
Arsenic DMTL2Y1 N. A. N. A. Approved [142]
GSK683699 DMTW79H Inflammatory bowel disease DD72 Phase 2 [143]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [144]
bisphenol A DM2ZLD7 Discovery agent N.A. Investigative [145]
Trichostatin A DM9C8NX Solid tumour/cancer 2A00-2F9Z Investigative [146]
TBPS DMFC3XP Discovery agent N.A. Investigative [147]
Muscimol DMNTF2O Discovery agent N.A. Investigative [141]
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Drug(s) Affected By Biglycan (BGN)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Isotretinoin DM4QTBN Acne vulgaris ED80 Approved [148]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [96]
Niclosamide DMJAGXQ Cestodes infection 1F70-1F76 Approved [149]
Dasatinib DMJV2EK Blast phase chronic myelogenous leukemia, BCR-ABL1 positive Approved [150]
Temozolomide DMKECZD Adenocarcinoma 2D40 Approved [151]
Dexamethasone DMMWZET Acute adrenal insufficiency Approved [152]
Decitabine DMQL8XJ Acute myelogenous leukaemia 2A41 Approved [153]
Cisplatin DMRHGI9 Adenocarcinoma 2D40 Approved [153]
Acetaminophen DMUIE76 Allergic rhinitis CA08.0 Approved [154]
Estradiol DMUNTE3 Acne vulgaris ED80 Approved [155]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Simvastatin DM30SGU Arteriosclerosis BD40 Approved [114]
Quercetin DM3NC4M Obesity 5B81 Approved [108]
Troglitazone DM3VFPD Diabetic complication 5A2Y Approved [156]
Arsenic trioxide DM61TA4 Acute lymphoblastic leukaemia 2A85 Approved [157]
Aspirin DM672AH Acute coronary syndrome BA41 Approved [158]
Ciclosporin DMAZJFX Graft-versus-host disease 4B24 Approved [94]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [159]
Hydrocortisone DMGEMB7 Acne vulgaris ED80 Approved [160]
Dexamethasone DMMWZET Acute adrenal insufficiency Approved [152]
Cupric Sulfate DMP0NFQ Fungal infection 1F29-1F2F Approved [161]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Selenium DM25CGV N. A. N. A. Approved [162]
Arsenic trioxide DM61TA4 Acute lymphoblastic leukaemia 2A85 Approved [163]
Hydroquinone DM6AVR4 Melasma ED60.1 Approved [164]
Acocantherin DM7JT24 Atrial fibrillation BC81.3 Approved [138]
Leflunomide DMR8ONJ Arthritis FA20 Approved [165]
Ciclosporin DMAZJFX Graft-versus-host disease 4B24 Approved [94]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [159]
Niclosamide DMJAGXQ Cestodes infection 1F70-1F76 Approved [149]
Temozolomide DMKECZD Adenocarcinoma 2D40 Approved [151]
Dexamethasone DMMWZET Acute adrenal insufficiency Approved [152]
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Drug(s) Affected By Fibromodulin (FMOD)
Drug Name Drug ID Indication ICD 11 Highest Status REF
Hydrogen peroxide DM1NG5W Infectious disease 1A00-CA43.1 Approved [134]
Arsenic trioxide DM61TA4 Acute lymphoblastic leukaemia 2A85 Approved [163]
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [166]
Phenytoin DMNOKBV Epilepsy 8A60-8A68 Approved [167]
Doxorubicin DMVP5YE Acute myelogenous leukaemia 2A41 Approved [99]
Methotrexate DM2TEOL Anterior urethra cancer Approved [168]
Cisplatin DMRHGI9 Adenocarcinoma 2D40 Approved [168]
Urethane DM7NSI0 N. A. N. A. Phase 4 [169]
SNDX-275 DMH7W9X Breast cancer 2C60-2C65 Phase 3 [170]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [144]
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Drug Name Drug ID Indication ICD 11 Highest Status REF
Valproate DMCFE9I Epilepsy 8A60-8A68 Approved [159]
Flunitrazepam DMGR5Z3 Insomnia 7A00-7A0Z Approved [141]
Flumazenil DMPCG2L Benzodiazepine overdose PC91 Approved [171]
Decitabine DMQL8XJ Acute myelogenous leukaemia 2A41 Approved [172]
Methamphetamine DMPM4SK Anxiety Approved [173]
Benzo(a)pyrene DMN7J43 N. A. N. A. Phase 1 [174]
TBPS DMFC3XP Discovery agent N.A. Investigative [147]
bisphenol A DM2ZLD7 Discovery agent N.A. Investigative [145]
Trichostatin A DM9C8NX Solid tumour/cancer 2A00-2F9Z Investigative [146]
Manganese DMKT129 N. A. N. A. Investigative [175]
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Molecular Interaction Atlas of This Drug

Molecular Interaction Atlas

Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Translocator protein (TSPO) TTPTXIN TSPO_HUMAN Agonist [3]

Drug Transporter (DTP)
DTP Name DTP ID UniProt ID MOA REF
P-glycoprotein 1 (ABCB1) DTUGYRD MDR1_HUMAN Substrate [4]

Drug-Metabolizing Enzyme (DME)
DME Name DME ID UniProt ID MOA REF
Cytochrome P450 3A4 (CYP3A4) Main DME DE4LYSA CP3A4_HUMAN Substrate [5]
Cytochrome P450 2C9 (CYP2C9) DE5IED8 CP2C9_HUMAN Substrate [6]
Mephenytoin 4-hydroxylase (CYP2C19) Main DME DEGTFWK CP2CJ_HUMAN Substrate [7]
Cytochrome P450 1A2 (CYP1A2) DEJGDUW CP1A2_HUMAN Substrate [8]
Cytochrome P450 3A5 (CYP3A5) DEIBDNY CP3A5_HUMAN Substrate [9]
Cytochrome P450 2B6 (CYP2B6) DEPKLMQ CP2B6_HUMAN Substrate [10]
Cytochrome P450 2C8 (CYP2C8) DES5XRU CP2C8_HUMAN Substrate [11]
Cytochrome P450 3A7 (CYP3A7) DERD86B CP3A7_HUMAN Substrate [12]
Prostaglandin G/H synthase 1 (COX-1) DE073H6 PGH1_HUMAN Substrate [13]
Cytochrome P450 2C18 (CYP2C18) DEZMWRE CP2CI_HUMAN Substrate [14]

Drug Off-Target (DOT)
DOT Name DOT ID UniProt ID Interaction REF
Albumin (ALB) OTVMM513 ALBU_HUMAN Protein Interaction/Cellular Processes [15]
Aldo-keto reductase family 1 member C1 (AKR1C1) OTQKR4CM AK1C1_HUMAN Gene/Protein Processing [16]
Aldo-keto reductase family 1 member C2 (AKR1C2) OTQ2XMO3 AK1C2_HUMAN Gene/Protein Processing [16]
Aldo-keto reductase family 1 member C3 (AKR1C3) OTU2SXBA AK1C3_HUMAN Gene/Protein Processing [16]
Aldo-keto reductase family 1 member C4 (AKR1C4) OTW2MMOF AK1C4_HUMAN Gene/Protein Processing [16]
Biglycan (BGN) OT3AV6IF PGS1_HUMAN Gene/Protein Processing [17]
Collagen alpha-1(I) chain (COL1A1) OTI31178 CO1A1_HUMAN Gene/Protein Processing [17]
Collagen alpha-1(VII) chain (COL7A1) OT3MIRZJ CO7A1_HUMAN Gene/Protein Processing [17]
Fibromodulin (FMOD) OT9EJ5H8 FMOD_HUMAN Gene/Protein Processing [17]
Gamma-aminobutyric acid receptor subunit alpha-1 (GABRA1) OTC2W96H GBRA1_HUMAN Gene/Protein Processing [18]

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