Details of the Drug-Related molecule(s) Interaction Atlas

General Information of DME (ID: DE4LYSA)

• DME Name: Cytochrome P450 3A4 (CYP3A4) DME Info
• Gene Name: CYP3A4

Molecule-Related Drug & Molecule List

637 Approved Drug(s) Transported by This DTP

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
Abiraterone acetate	DMANBZI	Prostate cancer	2C82.0	Approved	[1]
Acalabrutinib	DM7GCVW	leukaemia	2A60-2B33	Approved	[2]
Acenocoumarol	DMH75KV	Thrombosis	DB61-GB90	Approved	[3]
Acetaminophen	DMUIE76	Allergic rhinitis	CA08.0	Approved	[4]
Adinazolam	DMBHO9Y	Anxiety disorder	6B00-6B0Z	Approved	[5]
Albendazole	DMYZ57N	Echinococcus granulosus infectious disease		Approved	[6]
Alclometasone	DMAE84F	Exanthem		Approved	[7]
Aldosterone	DM9S2JW	Hypertension	BA00-BA04	Approved	[8]
Alectinib	DMP1I6Y	Lung cancer	2C25.0	Approved	[9]
Alfentanil	DMVO0UB	Anaesthesia	9A78.6	Approved	[10]
Aliskiren	DM1BV7W	Hypertension	BA00-BA04	Approved	[11]
Alitretinoin	DMME8LH	Kaposi sarcoma	2B57	Approved	[12]
Almotriptan malate	DMFG5ST	N. A.	N. A.	Approved	[13]
Alogliptin	DM8WI3R	Type-2 diabetes	5A11	Approved	[14]
Alosetron	DML2A03	Diarrhea-predominant irritable bowel syndrome	DD91.01	Approved	[15]
Alpelisib	DMEXMYK	Breast cancer	2C60-2C65	Approved	[16]
Alprazolam	DMC7XDN	Anxiety		Approved	[17]
Ambrisentan	DMD1QXW	Pulmonary arterial hypertension	BB01.0	Approved	[18]
Ambroxol	DMWJE9D	Bronchitis	CA20	Approved	[19]
Amcinonide	DMM1JL9	Exanthem		Approved	[20]
Amiodarone	DMUTEX3	Tachyarrhythmias	BC71	Approved	[21]
Amitriptyline	DMK7F9S	Depression	6A70-6A7Z	Approved	[22]
Amlodipine	DMBDAZV	Angina pectoris	BA40	Approved	[23]
Amprenavir	DMLMXE0	Human immunodeficiency virus infection	1C62	Approved	[24]
Anastrozole	DMNP60F	Breast cancer	2C60-2C65	Approved	[25]
Apixaban	DM89JLN	Thrombosis	DB61-GB90	Approved	[26]
Apremilast	DMTWS9E	Psoriasis vulgaris	EA90	Approved	[27]
Aprepitant	DM053KT	Depression	6A70-6A7Z	Approved	[28]
Argatroban	DMFI46A	Thrombosis	DB61-GB90	Approved	[29]
Aripiprazole	DM3NUMH	Bipolar I disorder		Approved	[30]
Armodafinil	DMGB035	Malignant glioma	2A00.0	Approved	[31]
ARN-509	DMT81LZ	Acute myeloid leukaemia	2A60	Approved	[32]
Artemether	DM48QOT	Malaria	1F40-1F45	Approved	[33]
Artemisinin	DMOY7W3	Malaria	1F40-1F45	Approved	[34]
Asenapine	DMSQZE2	Schizophrenia	6A20	Approved	[35]
Atazanavir	DMSYRBX	Human immunodeficiency virus infection	1C62	Approved	[36]
Atenolol	DMNKG1Z	Angina pectoris	BA40	Approved	[37]
Atorvastatin	DMF28YC	Acute coronary syndrome	BA41	Approved	[38]
Atovaquone	DMY4UMW	Fungal infection	1F29-1F2F	Approved	[39]
Avanafil	DM75CXN	Erectile dysfunction	HA01.1	Approved	[40]
Axitinib	DMGVH6N	Renal cell carcinoma	2C90	Approved	[41]
Azelastine	DMXTMBJ	Allergic conjunctivitis	9A60.02	Approved	[42]
Aztreonam	DMDNJHG	Bacterial infection	1A00-1C4Z	Approved	[43]
Baloxavir marboxil	DM1UV7F	Influenza virus infection	1E30-1E32	Approved	[44]
Baricitinib	DM4ONW5	Rheumatoid arthritis	FA20	Approved	[45]
BAY 80-6946	DMLOS5R	Follicular lymphoma	2A80	Approved	[46]
Beclomethasone	DMZPHIK	Allergic rhinitis	CA08.0	Approved	[47]
Bedaquiline	DM3906J	Drug-resistant tuberculosis		Approved	[48]
Benzphetamine	DMIJATC	Obesity	5B81	Approved	[49]
Bepridil	DM0RKS4	Chronic/stable angina	BA40.1	Approved	[50]
Betamethasone Valerate	DMMIAXO	Dermatological disease	DA24.Y	Approved	[51]
Bexarotene	DMOBIKY	Cutaneous T-cell lymphoma	2B01	Approved	[19]
Bezafibrate	DMZDCS0	Hypercholesterolaemia	5C80.0	Approved	[52]
Bicalutamide	DMZMSPF	Prostate cancer	2C82.0	Approved	[53]
Bimatoprost	DMX0E5B	Alopecia	ED70	Approved	[54]
Bisoprolol	DM3UZ95	Hypertension	BA00-BA04	Approved	[55]
BOCEPREVIR	DMBSHMF	Hepatitis C virus infection	1E51.1	Approved	[56]
Bortezomib	DMNO38U	Leukemia		Approved	[57]
Bosentan	DMIOGBU	Pulmonary arterial hypertension	BB01.0	Approved	[58]
Bosutinib	DMTI8YE	Blast phase chronic myelogenous leukemia, BCR-ABL1 positive		Approved	[59]
Brentuximab vedotin	DMWLC57	Hodgkin lymphoma	2B30	Approved	[60]
Brilinta	DMBR01X	Acute coronary syndrome	BA41	Approved	[61]
Brinzolamide	DMBAPFG	Ocular hypertension	9C61.01	Approved	[19]
Bromocriptine	DMVE3TK	Acromegaly	5A60.0	Approved	[62]
Bromperidol	DM24XYQ	Schizophrenia	6A20	Approved	[63]
Budesonide	DMJIBAW	Allergic rhinitis	CA08.0	Approved	[64]
Bupivacaine	DM4PRFC	Anaesthesia	9A78.6	Approved	[65]
Buprenorphine	DMPRI8G	Opioid dependence	6C43.2Z	Approved	[66]
Buspirone	DMBS632	Anxiety disorder	6B00-6B0Z	Approved	[67]
Busulfan	DMXYJ9C	Chronic myelogenous leukaemia	2A20.0	Approved	[68]
Cabazitaxel	DMPAZHC	Breast cancer	2C60-2C65	Approved	[69]
Cabergoline	DMQ4HIN	Hyperprolactinaemia	5A60.1	Approved	[70]
Cabozantinib	DMIYDT4	Medullary thyroid gland carcinoma		Approved	[71]
Caffeine	DMKBJWP	Allergic rhinitis	CA08.0	Approved	[72]
Calcitriol	DM8ZVJ7	Congenital alopecia	LC30	Approved	[73]
Canagliflozin	DMFRM1I	Non-insulin dependent diabetes	5A11	Approved	[74]
Cannabidiol	DM0659E	Dravet syndrome	8A61.11	Approved	[75]
Capsaicin	DMGMF6V	Back pain	ME84.Z	Approved	[76]
Carbamazepine	DMZOLBI	Epilepsy	8A60-8A68	Approved	[77]
Cariprazine	DMJYDVK	Bipolar disorder	6A60	Approved	[78]
Carvedilol	DMHTEAO	Chronic heart failure	BD1Z	Approved	[79]
Celecoxib	DM6LOQU	Dysmenorrhea	GA34.3	Approved	[80]
Cenobamate	DM8KLU9	Complex partial seizure	8A68.0	Approved	[81]
Cephalexin	DMD5JU8	Acute otitis media	AB00	Approved	[82]
Cerivastatin	DMXCM7H	Hyperlipidaemia	5C80	Approved	[38]
Cevimeline	DMWSMND	Sjogren syndrome	4A43.20	Approved	[83]
Chenodiol	DMQ8JIK	Cholelithiasis	DC11	Approved	[84]
Chloroquine	DMSI5CB	Malaria	1F40-1F45	Approved	[85]
Chlorpheniramine	DM5URA2	Allergic rhinitis	CA08.0	Approved	[86]
Chlorpromazine	DMBGZI3	Acute intermittent hepatic porphyria	5C58.11	Approved	[87]
Chlorzoxazone	DMCYVDT	Acute pain	MG31	Approved	[19]
Ciclesonide	DM2NA4K	Allergic rhinitis	CA08.0	Approved	[88]
Ciclosporin	DMAZJFX	Graft-versus-host disease	4B24	Approved	[89]
Cilostazol	DMZMSCT	Intermittent claudication	BD40.00	Approved	[90]
Cinacalcet	DMCX0K3	Hyperparathyroidism	5A51	Approved	[91]
Cinnarizine	DM7U5QJ	Meniere disease	AB31.0	Approved	[50]
Ciprofibrate	DMGC5DB	Hyperlipoproteinemia	5C80	Approved	[52]
Cisapride	DMY7PED	Gastroesophageal reflux disease	DA22.Z	Approved	[92]
Citalopram	DM2G9AE	Acute coronary syndrome	BA41	Approved	[93]
Clarithromycin	DM4M1SG	Acute maxillary sinusitis		Approved	[94]
Clevidipine butyrate	DMW4M97	Hypertension	BA00-BA04	Approved	[50]
Clindamycin	DM15HL8	Acne vulgaris	ED80	Approved	[95]
Clobazam - Lundbeck	DMW1OQ0	Anxiety disorder	6B00-6B0Z	Approved	[96]
Clofazimine	DMEBOFW	Crohn disease	DD70	Approved	[19]
Clofibrate	DMPC1J7	Dysbetalipoproteinemia	5C80.2	Approved	[52]
Clonazepam	DMTO13J	Absence epilepsy		Approved	[49]
Clonidine	DM6RZ9Q	Attention deficit hyperactivity disorder	6A05.Z	Approved	[97]
Clopidogrel	DMOL54H	Acute coronary syndrome	BA41	Approved	[38]
Clorazepate	DMC3JST	Alcohol withdrawal		Approved	[98]
Clotiazepam	DM59AZT	Anxiety disorder	6B00-6B0Z	Approved	[99]
Clotrimazole	DMMFCIH	Cutaneous candidiasis	1F23.14	Approved	[100]
Clozapine	DMFC71L	Schizophrenia	6A20	Approved	[101]
Cobicistat	DM6L4H2	Human immunodeficiency virus infection	1C62	Approved	[102]
Cocaine	DMSOX7I	Anaesthesia	9A78.6	Approved	[19]
Codeine	DMJX6ZG	Allergic rhinitis	CA08.0	Approved	[103]
Colchicine	DM2POTE	Acute gout flare	FA25.0	Approved	[104]
Conivaptan	DM1V329	Euvolemic hyponatremia	5C72	Approved	[105]
Conjugated Estrogens	DMLT0E1	Dyspareunia	GA12	Approved	[106]
Connexyn	DMF29Q5	Attention deficit hyperactivity disorder	6A05.Z	Approved	[107]
Corticotropin	DMP9TWZ	Cushing disease	5A70	Approved	[108]
Cortisone Acetate	DMG8K57	Acne vulgaris	ED80	Approved	[109]
Crizotinib	DM4F29C	Non-small-cell lung cancer	2C25.Y	Approved	[110]
Cyclandelate	DMO0R76	Dementia	6D80-6D86	Approved	[50]
Cyclobenzaprine	DM1YBRM	Depression	6A70-6A7Z	Approved	[111]
Cyclophosphamide	DM4O2Z7	Advanced cancer	2A00-2F9Z	Approved	[112]
Cytarabine	DMZD5QR	Acute lymphoblastic leukaemia	2A85	Approved	[113]
Dabrafenib	DMX6OE3	Melanoma	2C30	Approved	[114]
Daclatasvir	DMSFK9V	Hepatitis C virus infection	1E51.1	Approved	[115]
Dacomitinib	DMOH8VY	Non-small-cell lung cancer	2C25.Y	Approved	[116]
Dantrolene	DM1D8XY	Hyperthermia	MG26	Approved	[19]
Dapagliflozin	DM28UJG	Non-insulin dependent diabetes	5A11	Approved	[117]
Dapsone	DM4LT8A	Acne vulgaris	ED80	Approved	[118]
Darifenacin	DMWXLYZ	Overactive bladder	GC50.0	Approved	[119]
Darolutamide	DMV7YFT	Prostate cancer	2C82.0	Approved	[120]
Darunavir	DMN3GCH	Human immunodeficiency virus infection	1C62	Approved	[121]
Dasatinib	DMJV2EK	Blast phase chronic myelogenous leukemia, BCR-ABL1 positive		Approved	[122]
Daunorubicin	DMQUSBT	Acute monocytic leukemia		Approved	[123]
Deflazacort	DMV0RNS	Duchenne dystrophy	8C70	Approved	[124]
Delamanid	DMXE76K	Multi-drug resistant tuberculosis	MG52.00	Approved	[125]
Delavirdine	DM3NF5G	Human immunodeficiency virus infection	1C62	Approved	[126]
Desipramine	DMT2FDC	Attention deficit hyperactivity disorder	6A05.Z	Approved	[127]
Desogestrel	DM27U4Y	Contraception	QA21	Approved	[128]
Desonide	DMTP2NJ	Allergic rhinitis	CA08.0	Approved	[19]
Desoxycorticosterone Acetate	DMS0AFE	Discovery agent	N.A.	Approved	[129]
Desoxycorticosterone Pivalate	DMSA4B3	Addison disease	5A74.0	Approved	[129]
Desvenalfaxine succinate	DMJE6KO	Fibromyalgia	MG30.01	Approved	[130]
Dexamethasone	DMMWZET	Acute adrenal insufficiency		Approved	[131]
Dexamethasone sodium phosphate	DMIG8DW	Ataxia-telangiectasia	4A01.31	Approved	[131]
Dexlansoprazole	DM1DBV5	Erosive esophagitis	DA25.0	Approved	[132]
Dextromethorphan	DMUDJZM	Allergic rhinitis	CA08.0	Approved	[133]
Dextropropoxyphene	DM23HCX	Pain	MG30-MG3Z	Approved	[134]
Diazepam	DM08E9O	Alcohol withdrawal		Approved	[135]
Diclofenac	DMPIHLS	Chronic renal failure	GB61.Z	Approved	[136]
Diethylstilbestrol	DMN3UXQ	Gonorrheal vaginitis	GA02	Approved	[137]
Difluprednate	DMMFVB3	Ocular pain	MC18	Approved	[138]
Digitoxin	DMWVIGP	Arrhythmia	BC9Z	Approved	[139]
Digoxin	DMQCTIH	Arrhythmia	BC9Z	Approved	[140]
Dihydralazine	DMZIXU9	Hypertension	BA00-BA04	Approved	[141]
Dihydroergotamine	DM5IKUF	Cluster headache	8A81.0	Approved	[142]
Diltiazem	DMAI7ZV	Angina pectoris	BA40	Approved	[143]
Dirithromycin	DM0D9YJ	Bacterial infection	1A00-1C4Z	Approved	[144]
Disopyramide	DM5SYZP	Long QT syndrome	BC65.0	Approved	[145]
Disulfiram	DMCL2OK	Alcohol dependence	6C40.2	Approved	[146]
Docetaxel	DMDI269	Advanced cancer	2A00-2F9Z	Approved	[147]
Dofetilide	DMPN1TW	Sinus rhythm disorder	BC9Y	Approved	[148]
Dolasetron	DMMG26Z	Nausea	MD90	Approved	[149]
Dolutegravir	DMCZGRE	Human immunodeficiency virus infection	1C62	Approved	[150]
Domperidone	DMBDPY0	Gastrointestinal disease	DE2Z	Approved	[151]
Donepezil	DMIYG7Z	Advanced cancer	2A00-2F9Z	Approved	[152]
Dorzolamide	DMA17D0	Ocular hypertension	9C61.01	Approved	[19]
Doxapram	DMCYANK	Respiratory disease	CB40	Approved	[153]
Doxazosin	DM9PLRH	Benign prostatic hyperplasia	GA90	Approved	[154]
Doxepin	DMPI98T	Anxiety		Approved	[155]
Doxorubicin	DMVP5YE	Acute myelogenous leukaemia	2A41	Approved	[156]
Doxycycline	DM7ICNU	Acne vulgaris	ED80	Approved	[157]
Dronedarone	DMA8FS5	Angina pectoris	BA40	Approved	[158]
Drospirenone	DM1A9W3	Acne vulgaris	ED80	Approved	[159]
DU-176b	DMCIJBH	Atrial fibrillation	BC81.3	Approved	[160]
Dydrogesterone	DMAKIDV	Menstrual disorder	GA20.3	Approved	[161]
E-2007	DMJDYNQ	Diabetic neuropathy	8C0Z	Approved	[162]
Efavirenz	DMC0GSJ	Human immunodeficiency virus infection	1C62	Approved	[163]
Elbasvir	DMJLE18	Coronavirus Disease 2019 (COVID-19)	1D6Y	Approved	[164]
Eletriptan	DMW649X	Migraine	8A80	Approved	[38]
Eliglustat tartrate	DMSRZAO	Metabolic disorder	5C50-5D2Z	Approved	[38]
Elvitegravir	DMG9B1U	Human immunodeficiency virus infection	1C62	Approved	[165]
Emetine	DMCT2YF	Hepatitis virus infection	1E50-1E51	Approved	[166]
Enalapril	DMNFUZR	Congestive heart failure	BD10	Approved	[19]
Entrectinib	DMMPTLH	Non-small-cell lung cancer	2C25	Approved	[167]
Epinastine	DMX0K3Q	Allergic conjunctivitis	9A60.02	Approved	[168]
Eplerenone	DMF0NQR	Heart failure	BD10-BD13	Approved	[169]
Erdafitinib	DMI782S	Bladder cancer	2C94	Approved	[170]
Ergocalciferol	DMHO0AR	Hypoparathyroidism	5A50	Approved	[171]
Ergonovine	DM0VEC1	Postpartum haemorrhage	JA43	Approved	[172]
Ergotamine	DMKR3C5	Cluster headache	8A81.0	Approved	[173]
Ergotidine	DM78IME	Osteoarthritis	FA00-FA05	Approved	[174]
Eribulin	DM1DX4Q	Breast cancer	2C60-2C65	Approved	[175]
Erlotinib	DMCMBHA	Adrenal gland neoplasm		Approved	[59]
Erythromycin	DM4K7GQ	Acne vulgaris	ED80	Approved	[176]
Escitalopram	DMFK9HG	Major depressive disorder	6A70.3	Approved	[93]
Estazolam	DMZGXUM	Insomnia	7A00-7A0Z	Approved	[177]
Estradiol	DMUNTE3	Acne vulgaris	ED80	Approved	[178]
Estradiol Acetate	DM07U2A	Hormone replacement therapy	8E01	Approved	[179]
Estradiol Cypionate	DM27Z5T	Hormone replacement therapy	8E01	Approved	[179]
Estradiol Valerate	DM8MC6O	Hormone replacement therapy	8E01	Approved	[179]
Estramustine	DMWTAOI	Prostate cancer	2C82.0	Approved	[180]
Estrone	DM5T6US	Acne vulgaris	ED80	Approved	[181]
Estropipate	DMRMDWA	Hypogonadism	5A61.0	Approved	[182]
Eszopiclone	DM8RZ9H	Insomnia	7A00-7A0Z	Approved	[38]
Ethanol	DMDRQZU	Chronic pain	MG30	Approved	[19]
Ethchlorvynol	DM53IP1	Insomnia	7A00-7A0Z	Approved	[183]
Ethinyl Estradiol	DMODJ40	Acne vulgaris	ED80	Approved	[184]
Ethosuximide	DMDZ9LT	Epilepsy	8A60-8A68	Approved	[185]
Ethynodiol Diacetate	DMZM84R	Contraception	QA21	Approved	[186]
Etonogestrel	DMKA8J4	Contraception	QA21	Approved	[128]
Etoposide	DMNH3PG	Acute myelogenous leukaemia	2A41	Approved	[187]
Etoricoxib	DM6A4NW	Rheumatoid arthritis	FA20	Approved	[188]
Etravirine	DMGV8QU	Human immunodeficiency virus-1 infection	1C62	Approved	[189]
Everolimus	DM8X2EH	Advanced cancer	2A00-2F9Z	Approved	[190]
Exemestane	DM9HPW3	Hormonally-responsive breast cancer	2C60-2C65	Approved	[191]
Ezetimibe	DM7A8TW	Atherosclerosis	BD40	Approved	[192]
Famciclovir	DMJHLSD	Meniere disease	AB31.0	Approved	[193]
Fedratinib hydrochloride	DML2DCR	N. A.	N. A.	Approved	[194]
Felbamate	DM1V5ZS	Epilepsy	8A60-8A68	Approved	[195]
Felodipine	DMOSW35	Hypertension	BA00-BA04	Approved	[196]
Fenofibrate	DMFKXDY	Coronary atherosclerosis		Approved	[52]
Fentanyl	DM8WAHT	Analgesia	MB40.8	Approved	[197]
Fesoterodine fumarate	DM13495	Overactive bladder	GC50.0	Approved	[198]
Fexinidazole	DMOYE70	African trypanosomiasis	1F51	Approved	[199]
Finasteride	DMWV3TZ	Baldness, male pattern		Approved	[19]
Flibanserin	DM70DTN	Depression	6A70-6A7Z	Approved	[200]
Flucloxacillin	DMNUWST	Bacterial infection	1A00-1C4Z	Approved	[201]
Fludrocortisone	DMUDIR8	Addison disease	5A74.0	Approved	[19]
Flumethasone	DMUNG4A	Exanthem		Approved	[7]
Flunisolide	DMZSWQC	Allergic rhinitis	CA08.0	Approved	[202]
Flunitrazepam	DMGR5Z3	Insomnia	7A00-7A0Z	Approved	[203]
Fluocinolone Acetonide	DMG2KI4	Choroiditis		Approved	[202]
Fluocinonide	DM65KL8	Exanthem		Approved	[202]
Fluorometholone	DM2HKC4	Chronic obstructive pulmonary disease	CA22	Approved	[20]
Fluoxetine	DM3PD2C	Bipolar depression		Approved	[204]
Fluoxymesterone	DMUHCF1	Breast cancer	2C60-2C65	Approved	[205]
Fluprednisolone	DMZWBKG	Asthma	CA23	Approved	[206]
Flurandrenolide	DMHCI9S	Exanthem		Approved	[7]
Flurazepam	DMAL4G0	Insomnia	7A00-7A0Z	Approved	[207]
Fluspirilene	DMFO843	Schizophrenia	6A20	Approved	[50]
Flutamide	DMK0O7U	Prostate cancer	2C82.0	Approved	[208]
Fluticasone	DMGCSVF	Allergic rhinitis	CA08.0	Approved	[20]
Fluvastatin	DM4MDJY	Arteriosclerosis	BD40	Approved	[209]
Fosamprenavir	DM4W9B3	Human immunodeficiency virus infection	1C62	Approved	[210]
Fosphenytoin	DMOX3LB	Epilepsy	8A60-8A68	Approved	[211]
Fostamatinib	DM6AUHV	Immune thrombocytopenic purpura	3B64.13	Approved	[212]
Fulvestrant	DM0YZC6	Breast cancer	2C60-2C65	Approved	[213]
Galantamine	DMEO794	Alzheimer disease	8A20	Approved	[214]
Gefitinib	DM15F0X	Colon adenocarcinoma		Approved	[215]
Gemfibrozil	DMD8Q3J	Hyperlipidaemia	5C80	Approved	[52]
Gemtuzumab ozogamicin	DMJ2O7B	Acute myeloid leukaemia	2A60	Approved	[52]
Gepirone	DMGX5Q0	Major depressive disorder	6A70.3	Approved	[216]
Gestrinone	DMP0OVQ	Breast cancer	2C60-2C65	Approved	[217]
Gilteritinib	DMTI0ZO	Acute myeloid leukaemia	2A60	Approved	[218]
Glecaprevir	DM31YVO	N. A.	N. A.	Approved	[219]
Glibenclamide	DM8JXPZ	Diabetic complication	5A2Y	Approved	[38]
Glipizide	DMZA5PQ	Diabetic complication	5A2Y	Approved	[220]
Granisetron	DMIUW25	Malignant glioma	2A00.0	Approved	[221]
Grepafloxacin	DMGLX0T	Chronic bronchitis	CA20.1	Approved	[222]
Halaven	DM7JNTV	Breast cancer	2C60-2C65	Approved	[223]
Halcinonide	DMGLAX1	Exanthem		Approved	[224]
Halofantrine	DMOMK1V	Malaria	1F40-1F45	Approved	[225]
Haloperidol	DM96SE0	Delirium		Approved	[226]
Halothane	DM80OZ5	Anaesthesia	9A78.6	Approved	[227]
Hexobarbital	DMQ314B	Anaesthesia	9A78.6	Approved	[228]
Hydrocodone bitartrate	DMIAPBE	N. A.	N. A.	Approved	[229]
Hydrocortisone	DMGEMB7	Acne vulgaris	ED80	Approved	[230]
Hydromorphone	DMHP21E	Back pain	ME84.Z	Approved	[231]
Hydroquinone	DM6AVR4	Melasma	ED60.1	Approved	[232]
Hydroxyamphetamine	DMJAS3O	N. A.	N. A.	Approved	[233]
Hydroxychloroquine	DMSIVND	Chronic renal failure	GB61.Z	Approved	[234]
Hydroxyprogesterone	DMIKQH5	Solid tumour/cancer	2A00-2F9Z	Approved	[235]
Hydroxyzine	DMF8Y74	Allergic rhinitis	CA08.0	Approved	[236]
Ibrutinib	DMHZCPO	Mantle cell lymphoma	2A85.5	Approved	[237]
Ibuprofen	DM8VCBE	Dysmenorrhea	GA34.3	Approved	[238]
Idelalisib	DM602WT	Chronic lymphocytic leukaemia	2A82.0	Approved	[239]
Ifosfamide	DMCT3I8	Adult central nervous system germ cell tumor		Approved	[38]
Iloperidone	DM6AUFY	Schizophrenia	6A20	Approved	[240]
Imatinib	DM7RJXL	Acute lymphoblastic leukaemia	2A85	Approved	[241]
Imipramine	DM2NUH3	Depression	6A70-6A7Z	Approved	[127]
Imiquimod	DM1TMA3	Alopecia areata	ED70.2	Approved	[19]
Indacaterol	DMQJHR7	Chronic obstructive pulmonary disease	CA22	Approved	[242]
Indapamide	DMGN1PW	Edema	MG29	Approved	[243]
Indinavir	DM0T3YH	Human immunodeficiency virus infection	1C62	Approved	[38]
Ipriflavone	DM0IO13	Osteoporosis	FB83.0	Approved	[244]
Irbesartan	DMTP1DC	Diabetic kidney disease	GB61.Z	Approved	[245]
Irinotecan	DMP6SC2	Adenocarcinoma	2D40	Approved	[246]
Isavuconazonium	DMD45S9	N. A.	N. A.	Approved	[247]
Isosorbide Dinitrate	DMBI4JG	Anal fissure	DB50.0	Approved	[248]
Isosorbide Mononitrate	DMYLMU0	Angina pectoris	BA40	Approved	[248]
Isotretinoin	DM4QTBN	Acne vulgaris	ED80	Approved	[249]
Istradefylline	DM20VSK	Parkinson disease	8A00.0	Approved	[250]
Itraconazole	DMCR1MV	Aspergillosis	1F20	Approved	[251]
Ivabradine	DM0L594	Angina pectoris	BA40	Approved	[252]
Ivacaftor	DMZC1HS	Cystic fibrosis	CA25	Approved	[253]
Ivermectin	DMDBX5F	Intestinal strongyloidiasis due to nematode parasite	1F6B	Approved	[254]
Ixabepilone	DM2OZ3G	Breast cancer	2C60-2C65	Approved	[255]
Ketamine	DMT5HA4	Anaesthesia	9A78.6	Approved	[256]
Ketobemidone	DMM3L6Z	Pain	MG30-MG3Z	Approved	[257]
Ketoconazole	DMPZI3Q	Blastomycosis	1F22	Approved	[21]
Lansoprazole	DMXYLQ3	Gastric ulcer	DA60	Approved	[258]
Lapatinib	DM3BH1Y	Breast cancer	2C60-2C65	Approved	[259]
Lefamulin	DME6G97	Community-acquired pneumonia	CA40.Z	Approved	[260]
Leflunomide	DMR8ONJ	Arthritis	FA20	Approved	[261]
Lercanidipine	DMPWSEM	Hypertension	BA00-BA04	Approved	[262]
Letrozole	DMH07Y3	Estrogen-receptor positive breast cancer		Approved	[263]
Levobupivacaine	DM783CH	Anaesthesia	9A78.6	Approved	[264]
Levocetirizine dihydrochloride	DMW6ZJI	Allergic rhinitis	CA08.0	Approved	[265]
Levomethadyl acetate hydrochloride	DM429AE	N. A.	N. A.	Approved	[266]
Levomilnacipran	DMV26S8	Fibromyalgia	MG30.01	Approved	[]
Levothyroxine	DMHN027	Congenital hypothyroidism		Approved	[267]
LGX818	DMNQXV8	Melanoma	2C30	Approved	[268]
Lidocaine	DML4ZOT	Anaesthesia	9A78.6	Approved	[269]
LIDOFLAZINE	DMV23GL	Angina pectoris	BA40	Approved	[50]
Liotrix	DMSTXWR	N. A.	N. A.	Approved	[270]
Lisuride	DMCME17	Acromegaly	5A60.0	Approved	[271]
Lobeglitazone	DMHY3IP	Type-2 diabetes	5A11	Approved	[272]
LOMERIZINE	DME0TC8	Migraine	8A80	Approved	[50]
Lomitapide mesylate	DMLB4PE	N. A.	N. A.	Approved	[273]
Lonafarnib	DMGM2Z6	Hutchinson-Gilford progeria syndrome	LD2B	Approved	[274]
Loperamide	DMOJZQ9	Diarrhea	ME05.1	Approved	[275]
Lopinavir	DMITQS0	Human immunodeficiency virus infection	1C62	Approved	[276]
Loratadine	DMF3AN7	Allergy	4A80-4A85	Approved	[19]
Lorcaserin	DMG6OYJ	Obesity	5B81	Approved	[277]
Lorlatinib	DMICDLV	Non-small-cell lung cancer	2C25.Y	Approved	[278]
Losartan	DM72JXH	Diabetic kidney disease	GB61.Z	Approved	[19]
Loteprednol Etabonate	DM8QTJI	Eye inflammation	9A02	Approved	[279]
Lovastatin	DM9OZWQ	Arteriosclerosis	BD40	Approved	[280]
Loxapine	DM8AI9U	Bipolar disorder	6A60	Approved	[281]
Lumefantrine	DM29GAD	Malaria	1F40-1F45	Approved	[282]
Lurasidone hydrochloride	DMCVPXO	Schizophrenia	6A20	Approved	[283]
LY2835219	DM93VBZ	Breast cancer	2C60-2C65	Approved	[284]
Macitentan	DMP79A1	Cardiovascular disease	BA00-BE2Z	Approved	[285]
Maribavir	DM3GTAL	Cytomegalovirus infection	1D82	Approved	[286]
Marinol	DM70IK5	Anorexia nervosa cachexia	6B80	Approved	[38]
Mebendazole	DMO14SG	Ascariasis	1F62	Approved	[287]
Medroxyprogesterone	DMBGWPH	Solid tumour/cancer	2A00-2F9Z	Approved	[288]
Medrysone	DMJ90O5	Corneal abrasion	NA06.4	Approved	[20]
Mefloquine	DMWT905	Malaria	1F40-1F45	Approved	[289]
Megestrol	DMDH9KX	Breast cancer	2C60-2C65	Approved	[290]
Meloxicam	DM2AR7L	Arthritis	FA20	Approved	[291]
Meperidine	DMX4GND	Pain	MG30-MG3Z	Approved	[292]
Mephenytoin	DM5UGDK	Epilepsy	8A60-8A68	Approved	[293]
Meprednisone	DMTL9IP	Chronic obstructive pulmonary disease	CA22	Approved	[20]
Mestranol	DMG3F94	Contraception	QA21	Approved	[294]
Methadone	DMTW6IU	Advanced cancer	2A00-2F9Z	Approved	[295]
Methoxsalen	DME8FZ9	Cutaneous T-cell lymphoma	2B01	Approved	[296]
Methoxyflurane	DML0RAE	Anaesthesia	9A78.6	Approved	[297]
Methylergonovine	DMBEX4O	Spontaneous abortion	JA00.0	Approved	[173]
Methylprednisolone	DM4BDON	Acute adrenal insufficiency		Approved	[298]
Methyltestosterone	DMWLFGO	Advanced cancer	2A00-2F9Z	Approved	[299]
Metoclopramide	DMFA5MY	Nausea	MD90	Approved	[300]
Metoprolol	DMOJ0V6	Acute coronary syndrome	BA41	Approved	[301]
Metronidazole	DMTIVEN	Abscess		Approved	[302]
Mexiletine	DMCTE9R	Ventricular tachycardia	BC71	Approved	[303]
Mianserin	DMVKA4O	Depression	6A70-6A7Z	Approved	[267]
Miconazole	DMPMYE8	Cutaneous candidiasis	1F23.14	Approved	[304]
Midazolam	DMXOELT	Agitation	6A70.3	Approved	[305]
Midostaurin	DMI6E0R	Acute myeloid leukaemia	2A60	Approved	[306]
Mifepristone	DMGZQEF	Cushing disease	5A70	Approved	[307]
Mirabegron	DMS1GYT	Overactive bladder	GC50.0	Approved	[308]
Mirtazapine	DML53ZJ	Depression	6A70-6A7Z	Approved	[309]
MK-1439	DM215WE	Human immunodeficiency virus infection	1C62	Approved	[310]
Modafinil	DMYILBE	Malignant glioma	2A00.0	Approved	[19]
Momelotinib	DMF98Q0	Myelofibrosis	2A20.2	Approved	[311]
Mometasone	DM45OJN	Allergic asthma	CA23.0	Approved	[20]
Montelukast	DMD157S	Allergic asthma	CA23.0	Approved	[38]
Morphine	DMRMS0L	Advanced cancer	2A00-2F9Z	Approved	[312]
Mycophenolate mofetil	DMPQAGE	Hepatosplenic T-cell lymphoma		Approved	[313]
Naloxegol	DML0B41	Opioid-induced constipation	DB32.1	Approved	[314]
Nateglinide	DMLK2QH	Diabetic complication	5A2Y	Approved	[315]
Nefazodone	DM4ZS8M	Major depressive disorder	6A70.3	Approved	[316]
Nelfinavir mesylate	DMFX6G8	N. A.	N. A.	Approved	[38]
Nevirapine	DM6HX9B	Human immunodeficiency virus infection	1C62	Approved	[317]
Nicardipine	DMCDYW7	High blood pressure	BA00	Approved	[318]
Nicotine	DMWX5CO	Lung cancer	2C25.0	Approved	[319]
Nifedipine	DMSVOZT	Angina pectoris	BA40	Approved	[320]
Nilotinib	DM7HXWT	Chronic myelogenous leukaemia	2A20.0	Approved	[321]
Nimodipine	DMQ0RKZ	Cerebral vasospasm	BA85.Z	Approved	[19]
Nisoldipine	DM7ISKJ	Hypertension	BA00-BA04	Approved	[19]
Nitrazepam	DMEGIQ6	Epilepsy	8A60-8A68	Approved	[322]
Nitrendipine	DM21C09	Hypertension	BA00-BA04	Approved	[19]
Norethindrone acetate	DMDGCQP	N. A.	N. A.	Approved	[323]
Norgestimate	DMYP4XC	Acne vulgaris	ED80	Approved	[324]
Nortriptyline	DM4KDYJ	Depression	6A70-6A7Z	Approved	[325]
Oestradiol valerate and dienogest	DMZK0FQ	Contraception	QA21	Approved	[326]
Olaparib	DM8QB1D	Ovarian cancer	2C73	Approved	[327]
Olopatadine	DMKMWQG	Allergic conjunctivitis	9A60.02	Approved	[328]
Omeprazole	DM471KJ	Cystic fibrosis	CA25	Approved	[38]
Ondansetron	DMOTQ1I	Chemotherapy-induced nausea	MD90	Approved	[329]
OPC-34712	DMHG57U	Major depressive disorder	6A70.3	Approved	[330]
Ornidazole	DM6QHDJ	Amoebiasis	1A36	Approved	[331]
Orphenadrine citrate	DMFIQ20	N. A.	N. A.	Approved	[332]
Ospemifene	DMC4GEI	Dyspareunia	GA12	Approved	[333]
Oxatomide	DM1F42Z	Hay fever	CA08.00	Approved	[334]
Oxazepam	DMXNZM4	Alcohol withdrawal delirium		Approved	[335]
Oxybutynin hydrochloride	DMF2KLU	Urinary incontinence	MF50.2	Approved	[336]
Oxymorphone	DM65AGJ	Pain	MG30-MG3Z	Approved	[337]
Palbociclib	DMD7L94	Breast cancer	2C60-2C65	Approved	[338]
Paliperidone	DM7NPJS	Psychotic disorder	6A20-6A25	Approved	[339]
Palonosetron	DMBHMOX	Nausea	MD90	Approved	[340]
Panobinostat	DM58WKG	Chronic graft versus host disease		Approved	[341]
Pantoprazole	DMSVOCZ	Gastrinoma	2C10.1	Approved	[342]
Paramethadione	DMR5ZUP	Absence epilepsy		Approved	[343]
Paramethasone	DM6PR40	Inflammation	1A00-CA43.1	Approved	[20]
Paroxetine	DM5PVQE	Anxiety disorder	6B00-6B0Z	Approved	[344]
Pazopanib	DMF57DM	N. A.	N. A.	Approved	[345]
Pentamidine	DMHZJCG	African trypanosomiasis	1F51	Approved	[6]
Perazine	DM2AOTZ	Psychotic disorder	6A20-6A25	Approved	[346]
Pergolide mesylate	DM5GKOV	N. A.	N. A.	Approved	[70]
Perhexiline	DMINO7Z	Angina pectoris	BA40	Approved	[347]
Permethrin	DMZ0Q1G	Pediculus capitis infestation	1G00.0	Approved	[348]
Perphenazine	DMA4MRX	Schizophrenia	6A20	Approved	[349]
PF-04449913	DMSB068	Chronic myelomonocytic leukaemia	2A40	Approved	[]
Phenelzine	DMHIDUE	Depression	6A70-6A7Z	Approved	[350]
Phenobarbital	DMXZOCG	Cluster headache	8A81.0	Approved	[351]
Phenprocoumon	DMDO279	Myocardial infarction	BA41-BA43	Approved	[352]
Phentermine	DMG60XN	Obesity	5B81	Approved	[353]
Phenytoin	DMNOKBV	Epilepsy	8A60-8A68	Approved	[354]
Pilocarpine	DMV9ADG	Glaucoma/ocular hypertension	9C61	Approved	[355]
Pimecrolimus	DMZLGRB	Atopic dermatitis	EA80	Approved	[356]
Pimozide	DMW83TP	Schizophrenia	6A20	Approved	[357]
Pinacidil	DMRADYL	High blood pressure	BA00	Approved	[358]
Pioglitazone	DMKJ485	Amyotrophic lateral sclerosis	8B60.0	Approved	[359]
Pipotiazine	DMC68DF	Schizophrenia	6A20	Approved	[360]
Podofilox	DMT2EJP	Condyloma	1A95	Approved	[361]
Polatuzumab vedotin	DMF6Y0L	Diffuse large B-cell lymphoma	2A81	Approved	[362]
Pomalidomide	DMTGBAX	Plasma cell myeloma	2A83.1	Approved	[363]
Ponatinib	DMYGJQO	Acute lymphoblastic leukaemia	2A85	Approved	[364]
Posaconazole	DMUL5EW	Aspergillosis	1F20	Approved	[365]
Pranlukast	DMYHDCA	Allergic rhinitis	CA08.0	Approved	[366]
Prasterone	DM67VKL	Chronic obstructive pulmonary disease	CA22	Approved	[367]
Prasugrel	DM7MT6E	Acute coronary syndrome	BA41	Approved	[368]
Pravastatin	DM6A0X7	Adult acute monocytic leukemia		Approved	[369]
Prazepam	DMEWC7N	Anxiety		Approved	[370]
Praziquantel	DMOU1PK	Flatworm infection	1F70-1F86	Approved	[371]
Prednicarbate	DMBUNVW	Exanthem		Approved	[372]
Prednisolone	DMQ8FR2	Acute adrenal insufficiency		Approved	[373]
Prednisone	DM2HG4X	Acute asthma	CA23	Approved	[298]
Pretomanid	DMDYA31	Tuberculosis	1B10-1B14	Approved	[374]
Primaquine	DMWQ16I	Malaria	1F40-1F45	Approved	[375]
Progesterone	DMUY35B	Amenorrhea	GA20.0	Approved	[367]
Proguanil	DMBL79I	Malaria	1F40-1F45	Approved	[376]
Promazine	DMZAL7W	Acute intermittent hepatic porphyria	5C58.11	Approved	[377]
Promegestone	DMK4S8I	Gynecological disease	GA6Z	Approved	[326]
Propafenone	DMPIBJK	Tachyarrhythmias	BC71	Approved	[378]
Propiverine	DMUWBIJ	Urinary incontinence	MF50.2	Approved	[379]
Propofol	DMB4OLE	Anaesthesia	9A78.6	Approved	[380]
Propranolol	DM79NTF	Angina pectoris	BA40	Approved	[228]
Pyrazinamide	DM4IF32	Meningeal tuberculosis		Approved	[381]
Quazepam	DMY4D87	Insomnia	7A00-7A0Z	Approved	[382]
Quetiapine	DM1N62C	Anorexia nervosa cachexia	6B80	Approved	[383]
Quinidine	DMLPICK	N. A.	N. A.	Approved	[384]
Quinine	DMSWYF5	Malaria	1F40-1F45	Approved	[385]
Rabeprazole	DMMZXIW	Bacterial infection	1A00-1C4Z	Approved	[386]
Raloxifene	DMDKF3M	Osteoporosis	FB83.0	Approved	[387]
Ramelteon	DM7IW9J	Insomnia	7A00-7A0Z	Approved	[388]
Ranolazine	DM0C9IL	Acute coronary syndrome	BA41	Approved	[389]
Reboxetine	DM26PRD	Depression	6A70-6A7Z	Approved	[390]
Regorafenib	DMHSY1I	Gastrointestinal stromal tumour	2B5B	Approved	[391]
Repaglinide	DM5SXUV	Diabetic complication	5A2Y	Approved	[315]
Ribociclib Succinate	DM9CIUW	Breast cancer	2C60-2C65	Approved	[392]
Rifabutin	DM1YBHK	Mycobacterium infection	1B10-1B21	Approved	[393]
Rifampicin	DM5DSFZ	Non-insulin dependent diabetes	5A11	Approved	[394]
Rifapentine	DMCHV4I	Pulmonary tuberculosis	1B10.Z	Approved	[395]
Rifaximin	DMW1TV2	Bacterial infection	1A00-1C4Z	Approved	[396]
Rilpivirine	DMJ0QOW	Human immunodeficiency virus infection	1C62	Approved	[397]
Rimexolone	DMTAREC	Arthritis	FA20	Approved	[398]
Riociguat	DMXBLMP	Chronic thromboembolic pulmonary hypertension		Approved	[399]
Risdiplam	DMIMF8J	Spinal muscular atrophy	8B61	Approved	[400]
Risperidone	DMN6DXL	Bipolar I disorder		Approved	[19]
Ritonavir	DMU764S	Human immunodeficiency virus infection	1C62	Approved	[401]
Rivaroxaban	DMQMBZ1	Deep vein thrombosis	BD71	Approved	[402]
Rofecoxib	DM3P5DA	Osteoarthritis	FA00-FA05	Approved	[38]
Roflumilast	DMPGHY8	Asthma	CA23	Approved	[403]
Rokitamycin	DMCZWOK	Bacterial infection	1A00-1C4Z	Approved	[404]
Rolapitant	DM8XP26	Chemotherapy-induced nausea	MD90	Approved	[405]
Romidepsin	DMT5GNL	Cutaneous T-cell lymphoma	2B01	Approved	[406]
Ropinirole	DMA6S1D	Parkinson disease	8A00.0	Approved	[407]
Ropivacaine	DMSPJG2	Anaesthesia	9A78.6	Approved	[408]
Rosiglitazone	DMILWZR	Chronic kidney disease	GB61	Approved	[409]
Rosuvastatin	DMMIQ7G	Arteriosclerosis	BD40	Approved	[410]
Rotigotine	DMP7X6Q	N. A.	N. A.	Approved	[70]
Rucaparib	DM9PVX8	Ovarian cancer	2C73	Approved	[]
Safinamide mesylate	DM0J2ZT	Parkinson disease	8A00.0	Approved	[411]
Salbutamol	DMN9CWF	Acute asthma	CA23	Approved	[19]
Salmeterol	DMIEU69	Allergic asthma	CA23.0	Approved	[412]
Saquinavir	DMG814N	Human immunodeficiency virus infection	1C62	Approved	[413]
Saxagliptin	DMGXENV	Type-2 diabetes	5A11	Approved	[414]
Selegiline Hydrochloride	DM3VR1L	Parkinson disease	8A00.0	Approved	[415]
Sertraline	DM0FB1J	Coronary heart disease	BA80.Z	Approved	[344]
Sevoflurane	DMC9O43	Anaesthesia	9A78.6	Approved	[297]
Sibutramine	DMFJTDI	Obesity	5B81	Approved	[416]
Sildenafil citrate	DMSWJ5X	N. A.	N. A.	Approved	[38]
SILODOSIN	DMJSBT6	Benign prostatic hyperplasia	GA90	Approved	[417]
Simeprevir	DMLUA9D	Chronic HCV-1 infection	1E51.1	Approved	[418]
Simvastatin	DM30SGU	Arteriosclerosis	BD40	Approved	[419]
Siponimod	DM2R86O	Multiple sclerosis	8A40	Approved	[420]
Sirolimus	DMGW1ID	Advanced cancer	2A00-2F9Z	Approved	[19]
Sitagliptin	DMGDKXN	Cystic fibrosis	CA25	Approved	[421]
Solifenacin	DMG592Q	Overactive bladder	GC50.0	Approved	[422]
Sonidegib phosphate	DM72409	N. A.	N. A.	Approved	[423]
Sorafenib	DMS8IFC	Adenocarcinoma	2D40	Approved	[424]
Stiripentol	DMMSDOY	Dravet syndrome	8A61.11	Approved	[425]
Sufentanil	DMU7YEL	Analgesia	MB40.8	Approved	[426]
Sulfadiazine	DMTW3R8	Rheumatic fever	1B40-1B42	Approved	[19]
Sulfamethoxazole	DMB08GE	Acute otitis media	AB00	Approved	[427]
Sulfinpyrazone	DMEV954	Gout	FA25	Approved	[428]
Sunitinib	DMCBJSR	Acute undifferentiated leukemia		Approved	[59]
Suvorexant	DM0E6S3	Insomnia	7A00-7A0Z	Approved	[429]
Tacrolimus	DMZ7XNQ	Graft-versus-host disease	4B24	Approved	[19]
Tadalafil	DMJZHT1	Benign prostatic hyperplasia	GA90	Approved	[430]
Tamoxifen	DMLB0EZ	Breast cancer	2C60-2C65	Approved	[431]
Tamsulosin	DM5QF9V	Benign prostatic hyperplasia	GA90	Approved	[432]
Tasimelteon	DMLOQ1V	Insomnia	7A00-7A0Z	Approved	[433]
Tasosartan	DMM13DI	Hypertension	BA00-BA04	Approved	[19]
Telaprevir	DMMRV29	Hepatitis C virus infection	1E51.1	Approved	[434]
Telithromycin	DMZ4P3A	Bacterial infection	1A00-1C4Z	Approved	[435]
Temazepam	DM02A65	Insomnia	7A00-7A0Z	Approved	[436]
Temsirolimus	DMS104F	Renal cell carcinoma	2C90	Approved	[86]
Tenapanor	DMCOZJY	Irritable bowel syndrome	DD91.0	Approved	[437]
Teniposide	DMLW57T	Acute lymphoblastic leukaemia	2A85	Approved	[438]
Tenofovir alafenamide	DMTQF4A	Hiv infectious disease		Approved	[439]
Tenofovir disoproxil fumarate	DMSY4ZG	Discovery agent	N.A.	Approved	[439]
Terbinafine	DMI6HUW	Fungal infection	1F29-1F2F	Approved	[38]
Testosterone cypionate	DMC1TEV	N. A.	N. A.	Approved	[440]
Theophylline	DMRJFN9	Bronchitis	CA20	Approved	[441]
Thiamylal	DMHDF7B	Anaesthesia	9A78.6	Approved	[442]
Thiotepa	DMIZKOP	Breast cancer	2C60-2C65	Approved	[443]
Tiagabine	DMKSQG0	Epilepsy	8A60-8A68	Approved	[444]
Tianeptine	DMYN8MA	Major depressive disorder	6A70.3	Approved	[445]
Tindamax	DM3OWT4	Bacterial infection	1A00-1C4Z	Approved	[446]
Tipranavir	DM8HJX6	Human immunodeficiency virus infection	1C62	Approved	[447]
Tofacitinib	DMBS370	Rheumatoid arthritis	FA20	Approved	[448]
Tolterodine	DMSHPW8	Overactive bladder	GC50.0	Approved	[449]
Tolvaptan	DMIWFRL	Autosomal dominant polycystic kidney disease	GB81	Approved	[450]
Topiramate	DM82Z30	Alcohol dependence	6C40.2	Approved	[451]
Toremifene	DMQYUWG	Breast cancer	2C60-2C65	Approved	[452]
TP-434	DM5A31S	Intra-abdominal infection	1A40	Approved	[453]
Trabectedin	DMG3Y89	Leiomyosarcoma	2B58	Approved	[454]
Tramadol	DMRQD04	Osteoarthritis	FA00-FA05	Approved	[455]
Tranilast	DME5Y64	Allergic rhinitis	CA08.0	Approved	[50]
Trazodone	DMK1GBJ	Depression	6A70-6A7Z	Approved	[456]
Tretinoin	DM49DUI	Acne vulgaris	ED80	Approved	[457]
Triamcinolone diacetate	DM7LRKD	N. A.	N. A.	Approved	[458]
Triazolam	DMETYK5	Insomnia	7A00-7A0Z	Approved	[459]
TRICLABENDAZOLE	DMPWGBR	Helminth infection	1F90.0	Approved	[460]
Trifarotene	DMOL793	Acne vulgaris	ED80	Approved	[461]
Trilostane	DMQZ9GF	Cushing disease	5A70	Approved	[462]
Trimebutine	DMPYQ7B	Irritable bowel syndrome	DD91.0	Approved	[50]
Trimethadione	DM0Q8MZ	Absence epilepsy		Approved	[343]
Trimethoprim	DMM7CHK	Acute otitis media	AB00	Approved	[19]
Trofosfamide	DMHB2C3	Non-hodgkin lymphoma	2B33.5	Approved	[463]
Troglitazone	DM3VFPD	Diabetic complication	5A2Y	Approved	[464]
Troleandomycin	DMUZNIG	Bacterial infection	1A00-1C4Z	Approved	[465]
Tropisetron	DMNSJ7V	Fibromyalgia	MG30.01	Approved	[149]
Udenafil	DM1IQRP	Erectile dysfunction	HA01.1	Approved	[466]
Ulipristal	DMBNI20	Contraception	QA21	Approved	[467]
Upadacitinib	DM32B5U	Rheumatoid arthritis	FA20	Approved	[468]
Valdecoxib	DMAY7H4	Osteoarthritis	FA00-FA05	Approved	[469]
Vandetanib	DMRICNP	Solid tumour/cancer	2A00-2F9Z	Approved	[470]
Vardenafil	DMTBGW8	Cystic fibrosis	CA25	Approved	[471]
Velpatasvir	DMGF8ZQ	N. A.	N. A.	Approved	[472]
Vemurafenib	DM62UG5	Melanoma	2C30	Approved	[473]
Venlafaxine	DMR6QH0	Anxiety disorder	6B00-6B0Z	Approved	[38]
Verapamil	DMA7PEW	Angina pectoris	BA40	Approved	[38]
Vilanterol	DMF5EK1	Chronic obstructive pulmonary disease	CA22	Approved	[474]
Vilazodone	DM4LECQ	Major depressive disorder	6A70.3	Approved	[475]
Vinblastine	DM5TVS3	Advanced cancer	2A00-2F9Z	Approved	[476]
Vincamine	DMK1ZOR	Cerebrovascular disease	8B2Z	Approved	[477]
Vincristine	DMINOX3	Acute lymphoblastic leukaemia	2A85	Approved	[478]
Vindesine	DMVR628	Acute lymphoblastic leukaemia	2A85	Approved	[479]
Vinorelbine	DMVXFYE	Advanced cancer	2A00-2F9Z	Approved	[477]
Vinpocetine	DMVN2E6	Ischemic stroke	8B11.5Z	Approved	[50]
Vismodegib	DM5IXKQ	Basal cell carcinoma	2C32	Approved	[480]
Vitamin A	DMJ2AH4	Night blindness	9D45	Approved	[481]
Vitamin D	DMWQUC9	N. A.	N. A.	Approved	[482]
Vitamin E	DMZC90K	Atherosclerosis	BD40	Approved	[483]
Vonoprazan	DMO6315	Helicobacter infection	DA42-DA63	Approved	[484]
Vorapaxar	DMA16BR	Myocardial infarction	BA41-BA43	Approved	[485]
Voriconazole	DMAOL2S	Aspergillosis	1F20	Approved	[486]
Vortioxetine	DM6F1PU	Major depressive disorder	6A70.3	Approved	[487]
Voxelotor	DMCS6M5	Sickle-cell disorder	3A51	Approved	[194]
Warfarin	DMJYCVW	Atrial fibrillation	BC81.3	Approved	[488]
Xatral	DMLHOA0	Benign prostatic hyperplasia	GA90	Approved	[489]
Yohimbine	DMJCP1Y	Erectile dysfunction	HA01.1	Approved	[490]
Zafirlukast	DMHNQOG	Asthma	CA23	Approved	[491]
Zalcitabine	DMH7MUV	Human immunodeficiency virus infection	1C62	Approved	[492]
Zaleplon	DMGFWSM	Insomnia	7A00-7A0Z	Approved	[493]
Ziconotide	DMSLJP4	Pain	MG30-MG3Z	Approved	[50]
Zidovudine	DM4KI7O	Human immunodeficiency virus infection	1C62	Approved	[494]
Zileuton	DMVRIC2	Allergic asthma	CA23.0	Approved	[38]
Ziprasidone	DMM58JY	Bipolar disorder	6A60	Approved	[495]
Zithromax	DMN4H2O	Syphilis infection	1A6Z	Approved	[19]
Zolpidem	DMWOSKJ	Insomnia	7A00-7A0Z	Approved	[496]
Zonisamide	DM0DTF7	Alcohol dependence	6C40.2	Approved	[497]
Zopiclone	DMPI6Z0	Insomnia	7A00-7A0Z	Approved	[498]
ZOTEPINE	DMF3VXA	Anxiety disorder	6B00-6B0Z	Approved	[499]
Icotinib hydrochloride	DM5GFIK	Non-small-cell lung cancer	2C25.Y	Registered	[500]
Aminophenazone	DMY2AH1	N. A.	N. A.	Phase 4	[501]
Azelnidipine	DMA12HL	Hypertension	BA00-BA04	Phase 4	[502]
Barnidipine	DMJSDBE	N. A.	N. A.	Phase 4	[503]
Beclabuvir	DMLKUG7	N. A.	N. A.	Phase 4	[504]
Benidipine	DMWNP6B	N. A.	N. A.	Phase 4	[505]
Brotizolam	DMGXD5T	N. A.	N. A.	Phase 4	[506]
Chlorphenamine	DM6C4YJ	Allergic rhinitis	CA08.0	Phase 4	[86]
Cibenzoline	DMBG0N4	N. A.	N. A.	Phase 4	[507]
Cyproterone acetate	DMLMOIJ	N. A.	N. A.	Phase 4	[326]
Dapoxetine	DMV6KFY	Premature ejaculation	HA03.0Z	Phase 4	[508]
Demegestone	DMV5KTJ	N. A.	N. A.	Phase 4	[509]
Dihydrocodeine	DMB0FWL	Allergic rhinitis	CA08.0	Phase 4	[510]
Ebastine	DMH21D9	N. A.	N. A.	Phase 4	[511]
Ergonovine maleate	DM9WPIH	N. A.	N. A.	Phase 4	[172]
Ethinylestradiol propanesulfonate	DM7ITZK	N. A.	N. A.	Phase 4	[512]
Etizolam	DM8TNX3	Anxiety disorder	6B00-6B0Z	Phase 4	[513]
Etoperidone	DMR7U8F	N. A.	N. A.	Phase 4	[514]
Gestodene	DM9R1YU	N. A.	N. A.	Phase 4	[515]
Grazoprevir	DM9BPLW	Hepatitis C	1E51	Phase 4	[516]
Ketazolam	DM170OH	N. A.	N. A.	Phase 4	[370]
Lacidipine	DMQP5I3	N. A.	N. A.	Phase 4	[517]
Levamlodipine	DM92S6N	Hypertension	BA00-BA04	Phase 4	[23]
Lynestrenol	DM82JP0	N. A.	N. A.	Phase 4	[323]
Medifoxamine	DM0UGYX	N. A.	N. A.	Phase 4	[19]
Mexazolam	DME1X96	N. A.	N. A.	Phase 4	[419]
Mosapride	DM2VOQ3	N. A.	N. A.	Phase 4	[518]
Nomegestrol	DMRP8XB	N. A.	N. A.	Phase 4	[326]
Otilonium	DMU1JVW	N. A.	N. A.	Phase 4	[50]
Parecoxib	DMIV8CT	N. A.	N. A.	Phase 4	[519]
Pinaverium	DM4OIMZ	N. A.	N. A.	Phase 4	[50]
Pregnenolone	DM6VFO1	Schizophrenia	6A20	Phase 4	[520]
Prenylamine	DM8PTSY	N. A.	N. A.	Phase 4	[50]
RUPATADINE	DMBPN7T	N. A.	N. A.	Phase 4	[521]
Tenofovir disoproxil	DM62IPN	N. A.	N. A.	Phase 4	[439]

120 Clinical Trial Drug(s) Transported by This DTP

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
5-methoxypsoralen	DME2A8X	Psoriasis vulgaris	EA90	Phase 3	[522]
ABT-263	DMNE56X	Myelofibrosis	2A20.2	Phase 3	[523]
ABT-761	DM3FIC2	Asthma	CA23	Phase 3	[524]
AL3818	DM3WP0N	Alveolar soft part sarcoma	2A60-2C35	Phase 3	[525]
Alisporivir	DM83EBP	Duchenne dystrophy	8C70	Phase 3	[526]
Anacetrapib	DMP2BFG	Arteriosclerosis	BD40	Phase 3	[527]
ARC029	DMYNJHI	Alzheimer disease	8A20	Phase 3	[528]
ASP-2151	DM5N1OB	Herpes simplex virus infection	1F00	Phase 3	[529]
Atrasentan	DMM74PK	Diabetic nephropathy	GB61.Z	Phase 3	[530]
Azimilide	DMUIBV8	Atrial fibrillation	BC81.3	Phase 3	[531]
Balaglitazone	DMXBHR6	Type-1 diabetes	5A10	Phase 3	[409]
BAY 86-9766	DMPW5SB	Solid tumour/cancer	2A00-2F9Z	Phase 3	[532]
Blonanserin	DM36C17	Schizophrenia	6A20	Phase 3	[533]
Carebastine	DMUVMWZ	Ocular allergy	4A81	Phase 3	[511]
CC-25430	DMV7WSN	N. A.	N. A.	Phase 3	[50]
Cediranib	DMWO5ZR	Peritoneal cavity cancer	2C51.Z	Phase 3	[534]
CHLORIDE	DM1TJXA	Solid tumour/cancer	2A00-2F9Z	Phase 3	[535]
Cilnidipine	DM1975O	High blood pressure	BA00	Phase 3	[536]
Cinitapride	DMEGFYD	Functional dyspepsia	DD90.3	Phase 3	[537]
Clomethiazole	DMSPN58	Stroke	8B20	Phase 3	[19]
Dalcetrapib	DMKNCVM	Acute coronary syndrome	BA41	Phase 3	[538]
Entresto	DMTWLXY	Acute myocardial infarction	BA41	Phase 3	[539]
Enzastaurin	DM5H0R9	Diffuse large B-cell lymphoma	2A81	Phase 3	[540]
Eperisone	DM1SMAI	Muscle spasm	MB47.3	Phase 3	[541]
Esketamine	DMVU687	Depression	6A70-6A7Z	Phase 3	[256]
Evacetrapib	DMCDZ15	Cardiovascular disease	BA00-BE2Z	Phase 3	[542]
Exatecan	DMCA7FN	Solid tumour/cancer	2A00-2F9Z	Phase 3	[543]
GLYCYRRHIZIN	DM8M2N3	Influenza virus infection	1E30-1E32	Phase 3	[544]
GTPL-9088	DMPS7U2	N. A.	N. A.	Phase 3	[545]
HE3286	DMB9U5E	Type-2 diabetes	5A11	Phase 3	[546]
HKI-272	DM6QOVN	Breast cancer	2C60-2C65	Phase 3	[547]
Iclaprim	DM7YNV9	Bacterial infection	1A00-1C4Z	Phase 3	[548]
Isavuconazole	DMSV12M	Candidemia	1F23.3Y	Phase 3	[549]
Jakafi	DMNORK8	Essential thrombocythemia	3B63.1Z	Phase 3	[550]
Karenitecin	DMCRGY4	Lung cancer	2C25.0	Phase 3	[551]
L-651582	DMWTPCA	Solid tumour/cancer	2A00-2F9Z	Phase 3	[50]
Laquinimod	DM3IWS8	Lupus	4A40	Phase 3	[552]
Linopirdine	DM0ZOGX	Cognitive impairment	6D71	Phase 3	[553]
LU AE58054	DMWGRQD	Schizophrenia	6A20	Phase 3	[554]
MANIDIPINE	DMJPGUA	N. A.	N. A.	Phase 3	[555]
MURAGLITAZAR	DMG3NFZ	N. A.	N. A.	Phase 3	[556]
Nabiximols	DMHKJ5I	Cancer related pain	MG30	Phase 3	[557]
Netupitant	DMEKAYI	Chemotherapy-induced nausea	MD90	Phase 3	[558]
Odanacatib	DM1EO3G	Osteoporosis	FB83.0	Phase 3	[559]
Plitidepsin	DMJ8AUE	Multiple myeloma	2A83	Phase 3	[560]
Pracinostat	DMTD7AB	Acute myeloid leukaemia	2A60	Phase 3	[561]
Rebamipide	DM2GHCR	Peptic ulcer	DA61	Phase 3	[562]
Remacemide	DM3YXP8	Pain	MG30-MG3Z	Phase 3	[563]
Rifalazil	DMYXOHV	Bacterial infection	1A00-1C4Z	Phase 3	[564]
Rivoglitazone	DMBY31K	Ocular inflammation	9C61.24	Phase 3	[409]
Rolofylline	DMSZPR3	Heart failure	BD10-BD13	Phase 3	[565]
Selinexor	DMBD4K3	Multiple myeloma	2A83	Phase 3	[566]
Semagacestat	DML83IW	Parkinson disease	8A00.0	Phase 3	[567]
TAK-875	DMIM5AP	Type-2 diabetes	5A11	Phase 3	[568]
Terodiline	DM4MZXE	Urinary incontinence	MF50.2	Phase 3	[50]
Triptolide	DMCMDVR	Autoimmune diabetes	5A10	Phase 3	[569]
Vicriviroc	DMMTW9K	Human immunodeficiency virus infection	1C62	Phase 3	[38]
Sarizotan	DMH7IPW	Rett syndrome	LD90.4	Phase 2/3	[570]
3,5-diiodothyropropionic acid	DML8M5T	Cardiovascular disease	BA00-BE2Z	Phase 2	[571]
9-AMINOCAMPTOTHECIN	DMQXYRG	Acquired immune deficiency syndrome	1C62.3	Phase 2	[572]
ABT-384	DM7XW5Y	Alzheimer disease	8A20	Phase 2	[573]
AZD2014	DMOEARH	Solid tumour/cancer	2A00-2F9Z	Phase 2	[574]
BC-3781 intravenous	DMY1UGV	Bacterial infection	1A00-1C4Z	Phase 2	[575]
BIIB014	DMH7RJ1	Parkinson disease	8A00.0	Phase 2	[576]
BMS 650032	DMQI43G	Hepatitis C virus infection	1E51.1	Phase 2	[577]
Carfentanil	DM7ADGX	N. A.	N. A.	Phase 2	[578]
Cenicriviroc	DM4V8WF	Human immunodeficiency virus infection	1C62	Phase 2	[579]
CP-122721	DMSWLM5	Major depressive disorder	6A70.3	Phase 2	[580]
Danoprevir	DM20MDU	Hepatitis C virus infection	1E51.1	Phase 2	[581]
Dexloxiglumide	DM52HUD	Pancreatic malfunction	DC30-DC3Z	Phase 2	[582]
EMIVIRINE	DMQH1NV	Human immunodeficiency virus infection	1C62	Phase 2	[583]
Famitinib	DMSFWT7	Solid tumour/cancer	2A00-2F9Z	Phase 2	[584]
Ferroquine	DMICMXE	Malaria	1F40-1F45	Phase 2	[585]
Gallopamil	DMXBR27	Asthma	CA23	Phase 2	[586]
GS-9620	DMG5C8D	Hepatitis B virus infection	1E51.0	Phase 2	[587]
HE3235	DMV50R1	Breast cancer	2C60-2C65	Phase 2	[588]
Impoyz	DMB1N6P	Scalp dermatosis		Phase 2	[589]
JNJ-37822681	DMV41P5	Schizophrenia	6A20	Phase 2	[590]
KNI-272	DMQZ5HF	Human immunodeficiency virus infection	1C62	Phase 2	[591]
Lersivirine	DMSEVBH	Human immunodeficiency virus infection	1C62	Phase 2	[592]
LY2603618	DMCXRZF	Pancreatic cancer	2C10	Phase 2	[593]
LY333531	DMGMC8H	Solid tumour/cancer	2A00-2F9Z	Phase 2	[594]
MB-07811	DM6JTSZ	Hyperlipidaemia	5C80	Phase 2	[595]
MSC1936369B	DMH1DYU	Colorectal cancer	2B91.Z	Phase 2	[596]
NCI-C50000	DMVQKB3	N. A.	N. A.	Phase 2	[50]
Netoglitazone	DM8H7OA	Non-alcoholic fatty liver disease	DB92	Phase 2	[409]
ONAPRISTONE	DMT6E5N	Breast cancer	2C60-2C65	Phase 2	[597]
PDX-101	DM6OC53	Plasma cell myeloma	2A83.1	Phase 2	[598]
PEG-SN38	DMX9ZM4	Breast cancer	2C60-2C65	Phase 2	[599]
Pradefovir	DM1O0DV	Hepatitis virus infection	1E50-1E51	Phase 2	[600]
PYRAZOLOACRIDINE	DMSOPAU	Colorectal cancer	2B91.Z	Phase 2	[381]
R-roscovitine	DMSH108	Non-small-cell lung cancer	2C25.Y	Phase 2	[601]
Sutezolid	DM2KQ71	Tuberculosis	1B10-1B1Z	Phase 2	[602]
Terguride	DMZNFPG	Pulmonary arterial hypertension	BB01.0	Phase 2	[603]
Tocopherol	DMBIJZ6	N. A.	N. A.	Phase 2	[604]
Trastuzumab emtansine	DMU1LXS	HER2-positive breast cancer	2C60-2C65	Phase 2	[144]
Vilaprisan	DME7VZD	Endometriosis	GA10	Phase 2	[605]
BRN-3122594	DMQKXSW	N. A.	N. A.	Phase 1/2	[20]
CC-223	DMMQYL9	Solid tumour/cancer	2A00-2F9Z	Phase 1/2	[606]
Dexamethasone palmitate	DMCMT4V	Choroidal neovascularization	9B76	Phase 1/2	[607]
GEA-6414	DM8J0MK	N. A.	N. A.	Phase 1/2	[50]
H3B-6545	DMIFCY2	Breast cancer	2C60-2C65	Phase 1/2	[608]
LS-172108	DMZNIAG	N. A.	N. A.	Phase 1/2	[609]
LY2940680	DMTJWIQ	Solid tumour/cancer	2A00-2F9Z	Phase 1/2	[610]
TG02	DMZFIGQ	Anaplastic astrocytoma	2A00.0	Phase 1/2	[611]
ABT-333	DM7TOWX	Hepatitis C virus infection	1E51.1	Phase 1	[612]
AZD-3839	DM72FOD	Alzheimer disease	8A20	Phase 1	[613]
CALANOLIDE A	DMQTUH8	Mycobacterium infection	1B10-1B21	Phase 1	[614]
Capravirine	DM9ERH1	Human immunodeficiency virus infection	1C62	Phase 1	[615]
Clemizole	DM4UAPD	Hepatitis C virus infection	1E51.1	Phase 1	[616]
GS-9883	DMMF5IE	N. A.	N. A.	Phase 1	[617]
H3B-6527	DMAYTRK	Hepatocellular carcinoma	2C12.02	Phase 1	[618]
ITX-5061	DM702MU	Human immunodeficiency virus-1 infection	1C62	Phase 1	[619]
LY-2811376	DM8LGWR	Alzheimer disease	8A20	Phase 1	[620]
Mibefradil	DMU9VDS	Glioblastoma multiforme	2A00.0	Phase 1	[621]
MLN8054	DMUANF3	Solid tumour/cancer	2A00-2F9Z	Phase 1	[622]
SAFINGOL	DMBGUDR	Psoriasis vulgaris	EA90	Phase 1	[623]
SC-20713	DM7GSLB	N. A.	N. A.	Phase 1	[186]
Teneligliptin	DMGJCDR	Type-2 diabetes	5A11	Phase 1	[624]
Tetrandrine	DMAOJBX	Sarcoma	2A60-2C35	Phase 1	[50]

38 Discontinued Drug(s) Transported by This DTP

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
Astemizole	DM2HN6Q	Allergic rhinitis	CA08.0	Withdrawn from market	[19]
FENDILINE	DMH6NG5	Coronary artery disease	BA80	Withdrawn from market	[50]
Methaqualone	DMW9NY0	Insomnia	7A00-7A0Z	Withdrawn from market	[625]
Phenacetin	DMRQAM0	Analgesia	MB40.8	Withdrawn from market	[626]
Roxithromycin	DMVMIK2	Bacterial infection	1A00-1C4Z	Withdrawn from market	[627]
Sertindole	DMMP65N	Schizophrenia	6A20	Withdrawn from market	[628]
Terfenadine	DM4KLPT	Allergy	4A80-4A85	Withdrawn from market	[141]
Zomepirac	DM7APNJ	Pain	MG30-MG3Z	Withdrawn from market	[629]
Epothilone B	DMM5ZX6	Solid tumour/cancer	2A00-2F9Z	Discontinued in Phase 3	[255]
GW873140	DMG6TS2	Human immunodeficiency virus-1 infection	1C62	Discontinued in Phase 3	[630]
Seletracetam	DM3IJMN	Epilepsy	8A60-8A68	Discontinued in Phase 3	[50]
Seratrodast	DMPNTDL	Allergic asthma	CA23.0	Discontinued in Phase 3	[631]
Octopamine	DMLQVTJ	Thrombosis	DB61-GB90	Discontinued in Phase 2a	[632]
Benzydamine	DMEQL9U	Chemotherapy or radiotherapy-induced mucositis	DA42-DA60	Discontinued in Phase 2	[633]
BMS-181101	DMT4VSE	Mood disorder	6A60-6E23	Discontinued in Phase 2	[634]
BMS-488043	DMRPU10	Human immunodeficiency virus infection	1C62	Discontinued in Phase 2	[635]
Dexniguldipine	DMLZIT2	Solid tumour/cancer	2A00-2F9Z	Discontinued in Phase 2	[50]
Ezlopitant	DMTUPZ2	Irritable bowel syndrome	DD91.0	Discontinued in Phase 2	[636]
FCP-3P1	DMTQLIJ	Arteriosclerosis	BD40	Discontinued in Phase 2	[23]
GW-766994	DMKC0J5	Asthma	CA23	Discontinued in Phase 2	[637]
Norcisapride	DMJSKUI	Gastroesophageal reflux disease	DA22.Z	Discontinued in Phase 2	[638]
Prednisolone sodium metazoate	DM082ZW	Inflammatory bowel disease	DD72	Discontinued in Phase 2	[639]
RS-8359	DMERM0K	Major depressive disorder	6A70.3	Discontinued in Phase 2	[640]
Tesmilifene	DMPB36I	Breast cancer	2C60-2C65	Discontinued in Phase 2	[641]
Torcetrapib	DMDHYM7	Hyperlipidaemia	5C80	Discontinued in Phase 2	[642]
Banoxantrone	DMK5I07	Acute lymphoblastic leukaemia	2A85	Discontinued in Phase 1	[643]
Mofarotene	DMKHEQL	Solid tumour/cancer	2A00-2F9Z	Discontinued in Phase 1	[644]
Roquinimex	DMMK42O	Rheumatoid arthritis	FA20	Discontinued in Phase 1	[645]
Vanoxerine	DMBQPA5	Cocaine addiction	6C45.2	Discontinued in Phase 1	[646]
VR-776	DMFQWNI	Premature ejaculation	HA03.0Z	Discontinued in Phase 1	[647]
Darodipine	DM160FM	Cerebrovascular ischaemia	8B1Z	Terminated	[50]
Dotarizine	DM6Q05K	Migraine	8A80	Terminated	[50]
Emopamil	DMW210B	Cerebrovascular ischaemia	8B1Z	Terminated	[50]
Flosequinan	DMY89KQ	Cardiovascular disease	BA00-BE2Z	Terminated	[651]
NIGULDIPINE	DMSPWMF	N. A.	N. A.	Terminated	[50]
Nimesulide	DMR1NMD	Metastatic colorectal cancer	2B91	Terminated	[50]
NSC-303812	DMEYMHB	N. A.	N. A.	Discontinued	[652]
WIN-55212-2	DMACBIW	N. A.	N. A.	Terminated	[50]

4 Preclinical Drug(s) Transported by This DTP

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
Oxycodone hydrochloride	DMCA7LN	Chronic pain	MG30	Application submitted	[648]
Ciglitazone	DMAPO0T	Pulmonary fibrosis	CB03.4	Preclinical	[409]
Organon	DMERWUC	Schizophrenia	6A20	Preclinical	[649]
VUFB-11502	DM7WFR0	N. A.	N. A.	Preclinical	[650]

31 Investigative Drug(s) Transported by This DTP

Drug Name	Drug ID	Indication	ICD 11	Highest Status	REF
(11-BETA)-11,21-DIHYDROXY-PREGN-4-ENE-3,20-DIONE	DMTPQ84	Discovery agent	N.A.	Investigative	[653]
6-Benzyloxy-9H-purin-2-ylamine	DMFI7A8	Discovery agent	N.A.	Investigative	[654]
agmatine	DMSBZ29	Discovery agent	N.A.	Investigative	[50]
Bencyclane	DM7H3VY	N. A.	N. A.	Investigative	[50]
Benzodiazepine	DM9H34M	Anxiety disorder	6B00-6B0Z	Investigative	[19]
Benzotetronic acid	DM4OKXI	N. A.	N. A.	Investigative	[655]
Benzyloxyresorufin	DM26SR7	N. A.	N. A.	Investigative	[656]
Butyrfentanyl	DM9X2FV	N. A.	N. A.	Investigative	[657]
Chlormadinone	DM64K0A	N. A.	N. A.	Investigative	[509]
Clorindione	DMLPXNC	N. A.	N. A.	Investigative	[658]
CTK1G9578	DMI3J0F	N. A.	N. A.	Investigative	[659]
CV-4093	DM983QP	Discovery agent	N.A.	Investigative	[555]
cyamemazine	DMZ6YPV	Discovery agent	N.A.	Investigative	[660]
Dexverapamil	DM9P4JW	N. A.	N. A.	Investigative	[50]
Dihydrostreptomycin	DMPDQSV	N. A.	N. A.	Investigative	[108]
Equilenin	DMHO56W	Discovery agent	N.A.	Investigative	[661]
Erythromycin salnacedin	DM0PHEW	Discovery agent	N.A.	Investigative	[176]
Ethyl biscoumacetate	DMR5Z2A	N. A.	N. A.	Investigative	[662]
Ethylmorphine	DM0YROF	Discovery agent	N.A.	Investigative	[663]
Imipramine oxide	DMZKABS	N. A.	N. A.	Investigative	[664]
Medazepam	DMNKSX3	N. A.	N. A.	Investigative	[665]
Medrogestone	DMNEAJG	N. A.	N. A.	Investigative	[666]
Mepacrine	DMU8L7C	Discovery agent	N.A.	Investigative	[667]
Miocamycin	DMDQK9G	N. A.	N. A.	Investigative	[668]
Niludipine	DM8OGMA	N. A.	N. A.	Investigative	[50]
Nordazepam	DMHAWYQ	N. A.	N. A.	Investigative	[669]
PARAOXON	DMN4ZKC	Discovery agent	N.A.	Investigative	[670]
Phenazone	DMCE985	Discovery agent	N.A.	Investigative	[38]
talinolol	DMRTD16	Discovery agent	N.A.	Investigative	[671]
taurochenodeoxycholic acid	DMEL9UT	Discovery agent	N.A.	Investigative	[672]
[3H]estrone-3-sulphate	DMGPF0N	Discovery agent	N.A.	Investigative	[182]

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